Known Bioactives Library: Biomol ICCBL - 2012

ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3402 A03 Enzo Life Sciences SL-115 C16 Ceramide Bioactive lipids: Activates PKC zeta 3402 A04 Enzo Life Sciences L-120 C-PAF Bioactive lipids: PAF receptor agonist 3402 A05 Enzo Life Sciences SL-145 C8 Ceramine Bioactive lipids: Ceramide analog. Apoptosis inducer

3402 A06 Enzo Life Sciences PG-047 D12-Prostaglandin J2 Bioactive lipids: Bioactive prostaglandin 3402 A07 Enzo Life Sciences FA-021 (R)-(+)-Methandamide CNS receptor ligands: Cannabinoid CB1 receptor agonist 3402 A08 Enzo Life Sciences FA-009 Dihomo-gamma-linolenic acid Bioactive lipids: Polyunsaturated fatty acid 3402 A09 Enzo Life Sciences DM-200 1α,25-Dihydroxyvitamin D3 Nuclear receptor ligands: Vitamin D receptor agonist 3402 A10 Enzo Life Sciences SL-125 Dihydrosphingosine Bioactive lipids: Apoptosis inducer 3402 A11 Enzo Life Sciences DG-100 1,2-Didecanoyl-glycerol (10:0) Bioactive lipids: Activates PKC 3402 A12 Enzo Life Sciences GR-207 Diidolylmethane Nuclear receptor ligands: AHR agonist 3402 A13 Enzo Life Sciences DG-112 1,2-Dioctanoyl-SN-glycerol Bioactive lipids: Activates PKC 3402 A14 Enzo Life Sciences SL-205 DL-Dihydrosphingosine Lipid biosynthesis: Sphingosine kinase inhibitor 3402 A15 Enzo Life Sciences DG-115 1,2-Dioleoyl-glycerol (18:1) Bioactive lipids: Activates PKC 3402 A16 Enzo Life Sciences SL-210 DL-PDMP Lipid biosynthesis: Glucosylceramide synthase inhibitor 3402 A17 Enzo Life Sciences EE-11 (±)11(12)-Epoxyeicosatrienoic acid Bioactive lipids: Bioactive arachidonic acid metabolite 3402 A18 Enzo Life Sciences SL-215 DL-PPMP Lipid biosynthesis: Glucosylceramide synthase inhibitor 3402 A19 Enzo Life Sciences H-112 12(R)-HETE Bioactive lipids: Bioactive arachidonic acid metabolite 3402 A20 Enzo Life Sciences FA-002 Docosahexaenoic acid(22:6 n-3) Bioactive lipids: Polyunsaturated fatty acid 3402 A21 Enzo Life Sciences H-012 12(S)-HETE Bioactive lipids: Bioactive arachidonic acid metabolite 3402 A22 Enzo Life Sciences FA-012 Docosapentaenoic acid Bioactive lipids: Polyunsaturated fatty acid 3402 B03 Enzo Life Sciences AC-104 Bepridil·HCl Ion channel ligands: Calcium channels 3402 B04 Enzo Life Sciences GR-313 Lycorine Inhibitors: inhibits TNFalpha production 3402 B05 Enzo Life Sciences CA-415 Cyclopiazonic acid Ion channel ligands: Intracellular calcium 3402 B06 Enzo Life Sciences GR-316 10-hydroxycamptothecin Inhibitors: topoisomerase 1 inhibitor 3402 B07 Enzo Life Sciences AC-100 Dantrolene Ion channel ligands: Intracellular calcium 3402 B08 Enzo Life Sciences GR-308 Beta-lapachone Inhibitors: topoisomerase 1 inhibitor 3402 B09 Enzo Life Sciences KC-115 Diazoxide Ion channel ligands: Potassium channels 3402 B10 Enzo Life Sciences T-113 Parthenolide Inhibitors: IkappaB kinase inhibitor 3402 B11 Enzo Life Sciences CA-204 Dichlorobenzamil·HCl Ion channel ligands: Calcium channels 3402 B12 Enzo Life Sciences PI-102 MG-132 Protease inhibitors: Proteasome inhibitor 3402 B13 Enzo Life Sciences CA-205 Diltiazem·HCl Ion channel ligands: Calcium channels 3402 B14 Enzo Life Sciences EI-352 QNZ Inhibitors: NFkappaB inhibitor 3402 B15 Enzo Life Sciences KC-158 E-4031 Ion channel ligands: Potassium channels 3402 B16 Enzo Life Sciences GR-211 bezafibrate Nuclear receptor ligands: PPAR alpha agonist 3402 B17 Enzo Life Sciences CM-102 Fipronil Ion channel ligands: Misc. channels 3402 B18 Enzo Life Sciences IM-100 Cycloheximide-N-ethylethanoate Inhibitors: FKBP12 inhibitor 3402 B19 Enzo Life Sciences AC-130 Flecainide acetate Ion channel ligands: Sodium channels 3402 B20 Enzo Life Sciences A-165 Ascomycin (FK-520) Inhibitors: binds to FKBP inhibits calcineurin 3402 B21 Enzo Life Sciences AC-123 Flufenamic acid Ion channel ligands: Potassium channels 3402 B22 Enzo Life Sciences FR-100 U-74389G Inhibitors: superoxide/free-radical inhibitor 3402 C03 Enzo Life Sciences HP-012 12(S)-HPETE Bioactive lipids: Fatty acid hydroperoxide 3402 C04 Enzo Life Sciences FA-010 Docosatrienoic acid (22:3 n-3) Bioactive lipids: Polyunsaturated fatty acid 3402 C05 Enzo Life Sciences G-234 12-Methoxydodecanoic acid Bioactive lipids: Myristic acid analog 3402 C06 Enzo Life Sciences FA-024 Eicosa-5,8-dienoic acid (20:2 n-12) Bioactive lipids: Polyunsaturated fatty acid 3402 C07 Enzo Life Sciences HO-013 13(S)-HODE Bioactive lipids: Bioactive linoleic acid metabolite 3402 C08 Enzo Life Sciences FA-007 Eicosadienoic acid (20:2 n-6) Bioactive lipids: Polyunsaturated fatty acid 3402 C09 Enzo Life Sciences HP-013 13(S)-HPODE Bioactive lipids: Fatty acid hydroperoxide 3402 C10 Enzo Life Sciences FA-001 Eicosapentaenoic acid (20:5 n-3) Bioactive lipids: Polyunsaturated fatty acid 3402 C11 Enzo Life Sciences PG-048 13,14-Dihydro-PGE1 Bioactive lipids: Bioactive prostaglandin 3402 C12 Enzo Life Sciences FA-008 Eicosatrienoic acid (20:3 n-3) Bioactive lipids: Polyunsaturated fatty acid 3402 C13 Enzo Life Sciences GR-102 13-cis retinoic acid Nuclear receptor ligands: Retinoid receptor ligand 3402 C14 Enzo Life Sciences L-110 Enantio-PAF C16 Bioactive lipids: Negative control for PAF 13-Keto-octadeca-9Z,11E-dienoic 3402 C15 Enzo Life Sciences KO-013 Bioactive lipids: Bioactive linoleic acid metabolite acid 3402 C16 Enzo Life Sciences G-222 Farnesylthioacetic acid Bioactive lipids: Carboxymethylation inhibitor (±)14,15-Epoxyeicosa-5Z,8Z,11Z- 3402 C17 Enzo Life Sciences EE-14 Bioactive lipids: Bioactive arachidonic acid metabolite trienoic acid 3402 C18 Enzo Life Sciences RA-105 Fluprostenol Bioactive lipids: Prostaglandin FP receptor agonist 3402 C19 Enzo Life Sciences H-015 15(S)-HETE Bioactive lipids: Bioactive arachidonic acid metabolite 3402 C20 Enzo Life Sciences FA-006 Gamma-linolenic acid (18:3 n-6) Bioactive lipids: Polyunsaturated fatty acid 3402 C21 Enzo Life Sciences HP-015 15(S)-HPETE Bioactive lipids: Fatty acid hydroperoxide 3402 C22 Enzo Life Sciences LE-009 Leukotoxin A (9,10-EODE) Bioactive lipids: Bioactive linoleic acid metabolite 3402 D03 Enzo Life Sciences CA-225 Flunarizine·2HCl Ion channel ligands: Calcium channels 3402 D04 Enzo Life Sciences EI-207 Ebselen Inhibitors: glutathione peroxidase mimetic 3402 D05 Enzo Life Sciences AC-116 Fluspirilene Ion channel ligands: Potassium channels 3402 D06 Enzo Life Sciences CN-266 TRIM Inhibitors: bNOS/iNOS inhibitor 3402 D07 Enzo Life Sciences CA-245 FPL-64176 Ion channel ligands: Calcium channels 3402 D08 Enzo Life Sciences PD-195 Zardaverine Inhibitors: phosphodiesterase (PDE1/2) inhibitor 3402 D09 Enzo Life Sciences CA-422 6-Gingerol Ion channel ligands: Intracellular calcium 3402 D10 Enzo Life Sciences PD-190 Zaprinast Inhibitors: phosphodiesterase (PDE1) inhibitor 3402 D11 Enzo Life Sciences AC-120 Glipizide Ion channel ligands: Potassium channels 3402 D12 Enzo Life Sciences PD-185 Vinpocetine Inhibitors: phosphodiesterase (PDE1) inhibitor 3402 D13 Enzo Life Sciences KC-120 Glyburide Ion channel ligands: Potassium channels 3402 D14 Enzo Life Sciences PD-180 Trequinsin Inhibitors: phosphodiesterase (PDE3) inhibitor 3402 D15 Enzo Life Sciences NA-135 Grayanotoxin III Ion channel ligands: Sodium channels 3402 D16 Enzo Life Sciences PD-179 Siguazodan Inhibitors: phosphodiesterase (PDE3) inhibitor 3402 D17 Enzo Life Sciences CM-101 R(+)-IAA-94 Ion channel ligands: Misc. channels 3402 D18 Enzo Life Sciences PD-175 Rolipram Inhibitors: phosphodiesterase (PDE4 ) inhibitor 3402 D19 Enzo Life Sciences CA-207 L-cis-Diltiazem·HCl Ion channel ligands: Calcium channels

Biomol ICCBL - 2012 Page 1 of 6 Created 9/2015 ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3402 D20 Enzo Life Sciences EI-117 Ro 20-1724 Inhibitors: phosphodiesterase (PDE4 ) inhibitor

3402 D21 Enzo Life Sciences AC-128 Lidocaine·HCl·H2O Ion channel ligands: Sodium channels 3402 D22 Enzo Life Sciences PD-155 MY-5445 Inhibitors: phosphodiesterase (PDE5) inhibitor 3402 E03 Enzo Life Sciences PG-050 15-deoxy-Prostaglandin J2 Bioactive lipids: Bioactive prostaglandin 3402 E04 Enzo Life Sciences LE-012 Leukotoxin B (12,13-EODE) Bioactive lipids: Bioactive linoleic acid metabolite 3402 E05 Enzo Life Sciences K-015 15-Ketoicosatetraenoic acid Bioactive lipids: Bioactive arachidonic acid metabolite 3402 E06 Enzo Life Sciences LB-004 Leukotriene B4 Bioactive lipids: Leukotriene B4 receptor agonist

3402 E07 Enzo Life Sciences PG-021 16,16-Dimethyl-prostaglandin E2 Bioactive lipids: Prostaglandin EP receptor agonist 3402 E08 Enzo Life Sciences LC-004 Leukotriene C4 Bioactive lipids: CysLT receptor agonist 3402 E09 Enzo Life Sciences EI-103 17-Octadecynoic acid Lipid biosynthesis: Inhibits fatty acid omega oxidation 3402 E10 Enzo Life Sciences LD-004 Leukotriene D4 Bioactive lipids: CysLT receptor agonist

3402 E11 Enzo Life Sciences PG-042 17-Phenyl-trinor-prostaglandin E2 Bioactive lipids: Prostaglandin EP1 receptor agonist 3402 E12 Enzo Life Sciences LE-004 Leukotriene E4 Bioactive lipids: CysLT1 receptor agonist 3402 E13 Enzo Life Sciences L-134 1-Acyl-PAF Bioactive lipids: PAF agonist 3402 E14 Enzo Life Sciences FA-023 Linoleamide Endocannabinoids: Bioactive linoleic acid metabolite 1-Hexadecyl-2-arachidonoyl- 3402 E15 Enzo Life Sciences DG-140 Bioactive lipids: DAG analog glycerol 3402 E16 Enzo Life Sciences FA-014 Linoleic acid Bioactive lipids: Polyunsaturated fatty acid 3402 E17 Enzo Life Sciences L-106 1-Hexadecyl-2-methylglycero-3 PC Bioactive lipids: PAF receptor agonist 3402 E18 Enzo Life Sciences FA-005 Linolenic acid (18:3 n-3) Bioactive lipids: Polyunsaturated fatty acid 3402 E19 Enzo Life Sciences EI-150 1-Hexadecyl-2-O-acetyl-glycerol Bioactive lipids: Blocks DAG activation of PKC 3402 E20 Enzo Life Sciences LXA-004 Lipoxin A4 Bioactive lipids: Bioactive arachidonic acid metabolite 3402 E21 Enzo Life Sciences EI-149 1-Hexadecyl-2-O-methyl-glycerol Bioactive lipids: Blocks DAG activation of PKC 3402 E22 Enzo Life Sciences LP-101 L-NASPA Bioactive lipids: LPA agonist / antagonist 3402 F03 Enzo Life Sciences ALX-550-253 Loperamide·HCl Ion channel ligands: Calcium channels 3402 F04 Enzo Life Sciences EI-145 A-3 Kinase inhibitors: kinase inhibitor 3402 F05 Enzo Life Sciences AC-103 Methoxyverapimil·HCl Ion channel ligands: Calcium channels 3402 F06 Enzo Life Sciences G-200 Acetyl (N)-s-farnesyl-l-cysteine Inhibitors: farnesylation inhibitor 3402 F07 Enzo Life Sciences KC-125 Minoxidil Ion channel ligands: Potassium channels 3402 F08 Enzo Life Sciences GR-300 Actinomycin D Inhibitors: transcription inhibitor 3402 F09 Enzo Life Sciences KC-130 Minoxidil sulfate Ion channel ligands: Potassium channels 3402 F10 Enzo Life Sciences VR-101 Arvanil Ion channel ligands: Vaniloid receptor agonist 3402 F11 Enzo Life Sciences AC-108 Nicardipine·HCl Ion channel ligands: Calcium channels 3402 F12 Enzo Life Sciences EI-277 AG1478 Kinase inhibitors: Tyrosine kinase inhibitor. Broad spectrum 3402 F13 Enzo Life Sciences CA-210 Nifedipine Ion channel ligands: Calcium channels 3402 F14 Enzo Life Sciences EI-188 AG213 (Tyrphostin 47) Kinase inhibitors: EGF-R tyrosine kinase inhibitor 3402 F15 Enzo Life Sciences AC-134 Niflumic acid Ion channel ligands: Misc. channels 3402 F16 Enzo Life Sciences EI-229 AG-370 Kinase inhibitors: PDGF receptor kinase inhibitor 3402 F17 Enzo Life Sciences CA-216 Niguldipine Ion channel ligands: Calcium channels 3402 F18 Enzo Life Sciences EI-272 AG-490 Kinase inhibitors: JAK2 inhibitor 3402 F19 Enzo Life Sciences ALX-550-277 Nimodipine Ion channel ligands: Calcium channels 3402 F20 Enzo Life Sciences EI-258 AG-879 Kinase inhibitors: NGF receptor inhibitor 3402 F21 Enzo Life Sciences ALX-550-278 Nitrendipine Ion channel ligands: Calcium channels 3402 F22 Enzo Life Sciences A-150 Alamethicin Inhibitors: monovalent cation ionophore 3402 G03 Enzo Life Sciences L-108 1-Octadecyl-2-methylglycero-3 PC Bioactive lipids: Inhibits PI-specific PLC 3402 G04 Enzo Life Sciences RA-101 LY-171883 Bioactive lipids: Leukotriene D4 receptor antagonist 3402 G05 Enzo Life Sciences DG-125 1-Oleoyl 2-acetyl-glycerol Bioactive lipids: PKC activator 3402 G06 Enzo Life Sciences L-101 Lyso-PAF C16 Bioactive lipids: Inactive PAF metabolite 3402 G07 Enzo Life Sciences DG-135 1-Stearoyl-2-lineoyl-glycerol Bioactive lipids: PKC activator 3402 G08 Enzo Life Sciences LP-100 Lysophosphatidic acid·Na Bioactive lipids: LPA receptor antagonist 3402 G09 Enzo Life Sciences DG-130 1-stearoyl-2-arachidonyl-glycerol Bioactive lipids: PKC activator 3402 G10 Enzo Life Sciences SL-221 D-erythro-MAPP Lipid biosynthesis: Ceramidase inhibitor 3402 G11 Enzo Life Sciences DM-300 24,25-Dihydroxyvitamin D3 Nuclear receptor ligands: Vitamin D receptor ligand 3402 G12 Enzo Life Sciences SL-222 L-erythro-MAPP Lipid biosynthesis: Negative control for D-erythro-MAPP 3402 G13 Enzo Life Sciences DM-100 25-Dihydroxyvitamin D3 Nuclear receptor ligands: Vitamin D receptor ligand 3402 G14 Enzo Life Sciences FA-004 Mead acid (20:3 n-9) Bioactive lipids: Polyunsaturated fatty acid 3402 G15 Enzo Life Sciences FA-028 2-Arachidonoylglycerol Endocannabinoids: Cannabinoid CB1 receptor agonist 3402 G16 Enzo Life Sciences FA-027 Mead ethanolamide Endocannabinoids: Cannabinoid receptor agonist 3402 G17 Enzo Life Sciences G-231 2-Fluoropalmitic acid Bioactive lipids: Protein palmitoylation inhibitor 3402 G18 Enzo Life Sciences GR-106 Methoprene acid Nuclear receptor ligands: Retinoid RXR agonist 3402 G19 Enzo Life Sciences G-230 2-Hydroxymyristic acid Bioactive lipids: Protein myristoylation inhibitor 3402 G20 Enzo Life Sciences PG-052 Misoprostol, free acid Bioactive lipids: Prostaglandin EP receptor agonist 3402 G21 Enzo Life Sciences GR-103 4-hydroxyphenylretinamide Nuclear receptor ligands: Retinoid receptor agonist / apoptosis inducer 3402 G22 Enzo Life Sciences SL-105 N,N-Dimethylsphingosine Lipid biosynthesis: Sphingosine kinase inhibitor 3402 H03 Enzo Life Sciences AC-132 N-Phenylanthranilic acid Ion channel ligands: Misc. channels 3402 H04 Enzo Life Sciences EI-303 AG-1296 Kinase inhibitors: c-kit, FGF and PDGF kinase inhibitor 3402 H05 Enzo Life Sciences CM-100 NPPB Ion channel ligands: Misc. channels 3402 H06 Enzo Life Sciences PD-152 Milrinone Inhibitors: phosphodiesterase (PDE3) inhibitor 3402 H07 Enzo Life Sciences KC-127 NS-1619 Ion channel ligands: Potassium channels 3402 H08 Enzo Life Sciences GR-333 PRIMA-1 Inhibitors: p53 reactivator 3402 H09 Enzo Life Sciences KC-155 Paxilline Ion channel ligands: Potassium channels 3402 H10 Enzo Life Sciences EI-313 Ikarugamycin Inhibitors: inhibits clathrin coated pit mediated endocytosis 3402 H11 Enzo Life Sciences KC-131 PCO-400 Ion channel ligands: Potassium channels 3402 H12 Enzo Life Sciences AP-101 4-Amino-1,8-naphthalimide Inhibitors: PARP inhibitor 3402 H13 Enzo Life Sciences KC-157 Penitrem A Ion channel ligands: Potassium channels 3402 H14 Enzo Life Sciences G-400 3-aminobenzamide (3-ABA) Inhibitors: ADP ribose polymerase, apoptosis inhibitor 3402 H15 Enzo Life Sciences AC-131 Phenamil Ion channel ligands: Sodium channels 3402 H16 Enzo Life Sciences EI-308 17-Allylamino-geldanamycin Inhibitors: HSP-90 inhibitor

Biomol ICCBL - 2012 Page 2 of 6 Created 9/2015 ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3402 H17 Enzo Life Sciences AC-121 Phentolamine Ion channel ligands: Potassium channels 3402 H18 Enzo Life Sciences ST-102 Anisomycin Inhibitors: MAP kinase activator 3402 H19 Enzo Life Sciences AC-125 Phenytoin Ion channel ligands: Sodum channels 3402 H20 Enzo Life Sciences CC-101 Aphidicolin Inhibitors: DNA polymerase inhibitor 3402 H21 Enzo Life Sciences AC-109 Pimozide Ion channel ligands: Calcium channels 3402 H22 Enzo Life Sciences EI-175 Aristolochic acid Lipid biosynthesis: phospholipase A2 inhibitor 3402 I03 Enzo Life Sciences G-232 4-Oxatetradecanoic acid Bioactive lipids: Myristic acid analog 3402 I04 Enzo Life Sciences LEA-004 N-Acetyl-leukotriene E4 Bioactive lipids: Bioactive arachidonic acid metabolite 3402 I05 Enzo Life Sciences H-005 5(S)-HETE Bioactive lipids: Bioactive arachidonic acid metabolite 3402 I06 Enzo Life Sciences FA-029 N-arachidonoylglycine Endocannabinoids: FAAH inhibitor 3402 I07 Enzo Life Sciences HP-005 5(S)-HPETE Bioactive lipids: Fatty acid hydroperoxide 3402 I08 Enzo Life Sciences FA-030 N-linoleoylglycine Endocannabinoids: FAAH inhibitor 3402 I09 Enzo Life Sciences EE-56 5,6-Epoxyeicosatrienoic acid Bioactive lipids: Bioactive arachidonic acid metabolite 3402 I10 Enzo Life Sciences L-100 PAF C16 Bioactive lipids: PAF receptor agonist 3402 I11 Enzo Life Sciences ET-004 5,8,11,14-Eicosatetraynoic acid Bioactive lipids: Cyclooxygenase & lipoxygenase inhibitor 3402 I12 Enzo Life Sciences L-105 PAF C18 Bioactive lipids: PAF receptor agonist 3402 I13 Enzo Life Sciences ET-003 5,8,11-Eicosatriynoic acid Bioactive lipids: Lipoxygenase inhibitor 3402 I14 Enzo Life Sciences L-107 PAF C18:1 Bioactive lipids: PAF receptor agonist 3402 I15 Enzo Life Sciences K-005 5-Ketoeicosatetraenoic acid Bioactive lipids: 5-KETE receptor (R527) agonist 3402 I16 Enzo Life Sciences FA-018 Palmitylethanolamide Endocannabinoids: Cannabinoid CB2 receptor agonist 3402 I17 Enzo Life Sciences GR-206 6-Formylindolo [3,2-B] carbazole Bioactive lipids: AHR agonist 3402 I18 Enzo Life Sciences LP-103 Dipalmitoylphosphatidic acid Bioactive lipids: Activates MAP kinase cascade

3402 I19 Enzo Life Sciences PG-017 6-Keto-prostaglandin F1a Bioactive lipids: Bioactive prostaglandin

3402 I20 Enzo Life Sciences PG-001 Prostaglandin A1 Bioactive lipids: Bioactive prostaglandin 3402 I21 Enzo Life Sciences EI-112 7,7-Dimethyleicosadienoic acid Bioactive lipids: PLA2 inhibitor

3402 I22 Enzo Life Sciences PG-002 Prostaglandin A2 Bioactive lipids: Bioactive prostaglandin 3402 J03 Enzo Life Sciences AC-118 Pinacidil Ion channel ligands: Potassium channels 3402 J04 Enzo Life Sciences PD-150 8-methoxymethyl-IBMX Inhibitors: phosphodiesterase (PDE1) inhibitor 3402 J05 Enzo Life Sciences AC-127 Procainamide Ion channel ligands: Sodium channels 3402 J06 Enzo Life Sciences PD-149 MBCQ Inhibitors: phosphodiesterase (PDE5) inhibitor 3402 J07 Enzo Life Sciences AC-124 Propafenone Ion channel ligands: Potassium channels 3402 J08 Enzo Life Sciences G-235 B581 Inhibitors: farnesyltransferase inhibitor

3402 J09 Enzo Life Sciences AC-129 Quinidine·HCl·H2O Ion channel ligands: Sodium channels 3402 J10 Enzo Life Sciences GR-244 BADGE Nuclear receptor ligands: PPAR gamma antagonist

3402 J11 Enzo Life Sciences AC-122 Quinine·HCl·2H2O Ion channel ligands: Potassium channels 3402 J12 Enzo Life Sciences CM-110 Bafilomycin A1 Inhibitors: vaculolar ATPase inhibitor 3402 J13 Enzo Life Sciences NA-134 QX-314 Ion channel ligands: Sodium channels 3402 J14 Enzo Life Sciences CA-411 BAPTA-AM Inhibitors: cell permeable Ca++ chelator 3402 J15 Enzo Life Sciences CA-450 Ryanodine Ion channel ligands: Intracellular calcium 3402 J16 Enzo Life Sciences EI-315 Blebbistatin Inhibitors: Myosin II inhibitor 3402 J17 Enzo Life Sciences NA-116 SDZ-201106 Ion channel ligands: Sodium channels 3402 J18 Enzo Life Sciences CM-113 Bongkrekic acid Inhibitors: ANT inhibitor 3402 J19 Enzo Life Sciences CA-230 SKF-96365 Ion channel ligands: Calcium channels 3402 J20 Enzo Life Sciences AC-582 IB-MECA CNS receptor ligands: Adenosine receptor agonist 3402 J21 Enzo Life Sciences CA-260 Tetrandine Ion channel ligands: Calcium channels 3402 J22 Enzo Life Sciences G-405 Brefeldin A Inhibitors: ARF GEF inhibitor 3402 K03 Enzo Life Sciences EE-89 8,9-Epoxyeicosatrienoic acid Bioactive lipids: Bioactive arachidonic acid metabolite

3402 K04 Enzo Life Sciences PG-003 Prostaglandin B1 Bioactive lipids: Bioactive prostaglandin

3402 K05 Enzo Life Sciences PG-049 8-epi-Prostaglandin F2a Bioactive lipids: Thromboxane TP receptor agonist

3402 K06 Enzo Life Sciences PG-004 Prostaglandin B2 Bioactive lipids: Bioactive prostaglandin 3402 K07 Enzo Life Sciences HO-409 9(S)-HODE Bioactive lipids: Bioactive linoleic acid metabolite

3402 K08 Enzo Life Sciences PG-005 Prostaglandin D2 Bioactive lipids: Prostaglandin DP receptor agonist 3402 K09 Enzo Life Sciences HP-019 9(S)-HPODE Bioactive lipids: Fatty acid hydroperoxide

3402 K10 Enzo Life Sciences PG-006 Prostaglandin E1 Bioactive lipids: Prostaglandin EP receptor agonist 3402 K11 Enzo Life Sciences FA-025 9,10-Octadecenoamide Endocannabinoids: Endogenous sleep inducing lipid

3402 K12 Enzo Life Sciences PG-007 Prostaglandin E2 Bioactive lipids: Prostaglandin EP receptor agonist

3402 K13 Enzo Life Sciences PG-031 9a,11b-Prostaglandin F2 Bioactive lipids: Bioactive prostaglandin

3402 K14 Enzo Life Sciences PG-010 Prostaglandin F1a Bioactive lipids: Prostaglandin FP receptor agonist

3402 K15 Enzo Life Sciences PG-030 9b,11a-Prostaglandin F2 Bioactive lipids: Bioactive prostaglandin

3402 K16 Enzo Life Sciences PG-008 Prostaglandin F2a Bioactive lipids: Prostaglandin FP receptor agonist 3402 K17 Enzo Life Sciences GR-101 9-cis Retinoic acid Nuclear receptor ligands: Retinoid RXR agonist

3402 K18 Enzo Life Sciences PG-011 Prostaglandin I2 Bioactive lipids: Prostaglandin IP receptor agonist 3402 K19 Enzo Life Sciences EI-347 Dimethyloxaloylglycine Inhibitor: Prolyl-4-hydroxylase inhibitor

3402 K20 Enzo Life Sciences PG-033 Prostaglandin J2 Bioactive lipids: Bioactive prostaglandin 3402 K21 Enzo Life Sciences FA-011 Adrenic acid (22:4, n-6) Bioactive lipids: Polyunsaturated fatty acid 3402 K22 Enzo Life Sciences GR-100 All trans retinoic acid Nuclear receptor ligands: Retinoid RAR agonist 3402 L03 Enzo Life Sciences PE-180 Thapsigargin Ion channel ligands: Intracellular calcium 3402 L04 Enzo Life Sciences CN-252 Bromo-7-nitroindazole Inhibitors: NO synthase inhibitor 3402 L05 Enzo Life Sciences EI-110 TMB-8 Ion channel ligands: Intracellular calcium 3402 L06 Enzo Life Sciences CN-115 8-Bromo-cAMP Activators: PKA activator 3402 L07 Enzo Life Sciences KC-135 Tolazamide Ion channel ligands: Potassium channels 3402 L08 Enzo Life Sciences CN-205 8-Bromo-cGMP Activators: PKG activator 3402 L09 Enzo Life Sciences AC-117 Tolbutamide Ion channel ligands: Potassium channels 3402 L10 Enzo Life Sciences EI-168 Bumetanide Inhibitors: Na+K+Cl- cotransport inhibitor 3402 L11 Enzo Life Sciences KC-159 U-37883A Ion channel ligands: Potassium channels 5'-N-Ethylcarboxamidoadenosine 3402 L12 Enzo Life Sciences AC-601 CNS receptor ligands: adenosine receptor agonist (NECA) 3402 L13 Enzo Life Sciences N-701 U-50488 Ion channel ligands: Calcium channels 3402 L14 Enzo Life Sciences EI-304 BW-B 70C Lipid biosynthesis: 5 lipoxygenase inhibitor 3402 L15 Enzo Life Sciences ALX-550-306 Verapimil Ion channel ligands: Calcium channels 3402 L16 Enzo Life Sciences PI-126 CA-074-Me Protease inhibitors: Cathepsin B inhibitor

Biomol ICCBL - 2012 Page 3 of 6 Created 9/2015 ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3402 L17 Enzo Life Sciences NA-125 Veratridine Ion channel ligands: Sodium channels 3402 L18 Enzo Life Sciences EI-311 SB-415286 Kinase inhibitors: GSK3 beta inhibitor 3402 L19 Enzo Life Sciences AC-106 YS035 Ion channel ligands: Calcium channels 3402 L20 Enzo Life Sciences PI-101 Calpeptin Protease inhibitors: Calpain inhibitor 3402 L21 Enzo Life Sciences KC-170 ZM226600 Ion channel ligands: Potassium channels 3402 L22 Enzo Life Sciences EI-198 Calphostin C Kinase inhibitors: PKC inhibitor 3402 M03 Enzo Life Sciences G-221 N-Acetyl-S-geranyl-L-cysteine Bioactive lipids: Negative control for AGGC and AFC 3402 M04 Enzo Life Sciences EI-209 REV-5901 Lipid biosynthesis: 5-Lipoxygenase inhibitor N-acetyl-S-geranylgeranyl-L- 3402 M05 Enzo Life Sciences G-220 Bioactive lipids: ICMT inhibitor Cysteine 3402 M06 Enzo Life Sciences G-201 S-farnesyl-L-cysteine Bioactive lipids: MDR ATPase activator 3402 M07 Enzo Life Sciences CR-108 AM-251 CNS receptor ligands: Cannabinoid CB1 receptor antagonist 3402 M08 Enzo Life Sciences EI-155 Sphingosine Bioactive lipids: PKC inhibitor 3402 M09 Enzo Life Sciences GR-104 AM-580 Nuclear receptor ligands: Retinoid RAR agonist 3402 M10 Enzo Life Sciences RA-103 SQ-29548 Bioactive lipids: Thromboxane A2 antagonist 3402 M11 Enzo Life Sciences FA-026 Anandamide (18:2,n-6) Endocannabinoids: Cannabinoid receptor agonist 3402 M12 Enzo Life Sciences L-126 Tetrahydrocannabinol-7-oic acid Nuclear receptor ligands: PPAR gamma agonist 3402 M13 Enzo Life Sciences FA-019 Anandamide (20:3,n-6) Endocannabinoids: Cannabinoid receptor agonist 3402 M14 Enzo Life Sciences GR-105 TTNPB Nuclear receptor ligands: Retinoid RAR agonist 3402 M15 Enzo Life Sciences FA-017 Anandamide (20:4, n-6) Endocannabinoids: Cannabinoid receptor agonist 3402 M16 Enzo Life Sciences PG-023 U-46619 Bioactive lipids: Thromboxane TP receptor agonist 3402 M17 Enzo Life Sciences FA-020 Anandamide (22:4,n-6) Endocannabinoids: Cannabinoid receptor agonist 3402 M18 Enzo Life Sciences RA-102 U-75302 Bioactive lipids: Leukotriene B4 receptor antagonist 3402 M19 Enzo Life Sciences FA-022 Arachidonamide Endocannabinoids: Bioactive arachidonic acid metabolite 3402 M20 Enzo Life Sciences CR-105 WIN 55,212-2 mesylate CNS receptor ligands: Cannabinoid CB1/CB2 receptor agonist 3402 M21 Enzo Life Sciences FA-003 Arachidonic acid (20:4, n-6) Bioactive lipids: Polyunsaturated fatty acid 3402 M22 Enzo Life Sciences GR-200 WY-14643 Nuclear receptor ligands: PPAR alpha agonist 3402 N03 Enzo Life Sciences PI-122 Tosyl-Phe-CMK (TPCK) Protease inhibitors: Serine protease inhibitor 3402 N04 Enzo Life Sciences EI-192 Calyculin A Inhibitors: PP1, PP2A inhibitor 3402 N05 Enzo Life Sciences PI-113 Thiorphan Protease inhibitors: Neutral endopeptidase inhibitor 3402 N06 Enzo Life Sciences GR-301 Camptothecin Inhibitors: Topoisomerase 1 inhibitor 3402 N07 Enzo Life Sciences PI-112 Z-prolyl-prolinal Protease inhibitors: Prolyl endopeptidase inhibitor 3402 N08 Enzo Life Sciences PR-105 Cantharidin Inhibitors: PP2A inhibitor 3402 N09 Enzo Life Sciences PI-125 NapSul-Ile-Trp-CHO Protease inhibitors: Cathepsin L inhibitor 3402 N10 Enzo Life Sciences EI-125 E-Capsaicin Ion channel ligands: vanilloid receptor agonist 3402 N11 Enzo Life Sciences PI-110 3,4-dichloroisocoumarin Protease inhibitors: Granzyme B inhibitor 3402 N12 Enzo Life Sciences NK-101 Capsazepine Ion channel ligands: vanilloid receptor antagonist 3402 N13 Enzo Life Sciences PI-128 Boc-GVV-CHO Protease inhibitors: Gamma secretase inhibitor 3402 N14 Enzo Life Sciences S-107 Castanospermine Inhibitors: glucosidase inhibitor 3402 N15 Enzo Life Sciences EI-212 Bestatin Protease inhibitors: Aminopeptidase inhibitor 3402 N16 Enzo Life Sciences EI-127 Dipyridamole Inhibitors: cGMP phosphodiesterase inhibitor 3402 N17 Enzo Life Sciences PI-123 Ala-Ala-Phe-CMK Protease inhibitors: Tripeptidyl peptidase II inhibitor 3402 N18 Enzo Life Sciences CM-119 CGP-37157 Inhibitors: inhibitor of mitochondrial Na+Ca+2 exchange 3402 N19 Enzo Life Sciences PI-130 MDL-28170 Protease inhibitors: Calpain inhibitor 3402 N20 Enzo Life Sciences EI-225 Chelerythrine Kinase inhibitors: PKC inhibitor 3402 N21 Enzo Life Sciences P-120 Ac-Leu-Leu-Nle-CHO Protease inhibitors: Calpain inhibitor 3402 N22 Enzo Life Sciences FR-102 CAPE Inhibitors: Antioxidant/ NFkappa B inhibitor 3402 O03 Enzo Life Sciences L-102 Arachidonoyl-PAF Bioactive lipids: PAF precursor 3402 O04 Enzo Life Sciences AC-119 4-Aminopyridine Ion channel ligands: Potassium channels 3402 O05 Enzo Life Sciences CR-104 BML-190 Bioactive lipids: Cannabinoid CB1 inverse agonist 3402 O06 Enzo Life Sciences KC-141 5-Hydroxydecanoate Ion channel ligands: Potassium channels 3402 O07 Enzo Life Sciences SL-100 C2 Ceramide Bioactive lipids: Apoptosis inducer 3402 O08 Enzo Life Sciences AC-126 Aconitine Ion channel ligands: Sodium channels 3402 O09 Enzo Life Sciences SL-101 C2 Dihydroceramide Bioactive lipids: Negative control for C2 ceramide 3402 O10 Enzo Life Sciences AC-115 AM 92016·HCl Ion channel ligands: Potassium channels 3402 O11 Enzo Life Sciences SL-112 C8 Ceramide Bioactive lipids: Stimulates Cer-activated PK 3402 O12 Enzo Life Sciences AC-133 Amantadine·HCl Ion channel ligands: Misc. channels 3402 O13 Enzo Life Sciences SL-113 C8 Dihydroceramide Bioactive lipids: Negative control for C8 ceramide 3402 O14 Enzo Life Sciences CA-200 Amiloride·HCl Ion channel ligands: Calcium channels 3402 O15 Enzo Life Sciences PG-035 Carbacyclin Bioactive lipids: PPAR delta agonist 3402 O16 Enzo Life Sciences AC-105 Amiodarone·HCl Ion channel ligands: Calcium channels 3402 O17 Enzo Life Sciences GR-205 Ciglitazone Nuclear receptor ligands: PPAR gamma agonist 3402 O18 Enzo Life Sciences CA-100 A-23187 Ion channel ligands: Calcium ionophore 3402 O19 Enzo Life Sciences EI-160 Clofibrate Nuclear receptor ligands: PPAR alpha agonist 3402 O20 Enzo Life Sciences CA-410 (R)-(+)-BAY K-8644 Ion channel ligands: Calcium channels 3402 O21 Enzo Life Sciences RA-106 Cloprostenol Bioactive lipids: Prostaglandin FP receptor agonist 3402 O22 Enzo Life Sciences NA-103 Benzamil·HCl Ion channel ligands: Calcium channels 3402 P03 Enzo Life Sciences CM-123 2-methoxyantimycin A3 Inhibitors: Bcl-2/Bcl-XL ligand induces apoptosis 3402 P04 Enzo Life Sciences AC-183 Cimaterol CNS receptor ligands: adrenoceptor agonist (beta) 3402 P05 Enzo Life Sciences AC-1800 ABC294640 SK2 inhib. 3402 P06 Enzo Life Sciences PR-115 CinnGEL 2Me Inhibitors: PTP1B inhibitor 3402 P07 Enzo Life Sciences CM-115 Decylubiquinone Inhibitors: inhibits mitochondrial permeability pore opening 3402 P08 Enzo Life Sciences AC-136 Cirazoline CNS receptor ligands: adrenoreceptor agonist (alpha) 3402 P09 Enzo Life Sciences AP-301 Betulinic acid Inhibitors: induces mitochondrial permeability pore opening 3402 P10 Enzo Life Sciences AC-152 Clonidine CNS receptor ligands: adrenoreceptor agonist (alpha) 3402 P11 Enzo Life Sciences EI-240 Deprenyl Inhibitors: inhibits glyceraldehyde-3-phosphate dehydrogenase 3402 P12 Enzo Life Sciences D-107 Clozapine CNS receptor ligands: Dopamine antagonist 3402 P13 Enzo Life Sciences CN-268 1400W·2HCl Inhibitors: iNOS inhibitor 3402 P14 Enzo Life Sciences EI-135 Curcumin Inhibitors: NFkappaB inhibitor 3402 P15 Enzo Life Sciences SL-220 Fumonisin B1 Lipid biosynthesis: inhibits ceramide synthase 3402 P16 Enzo Life Sciences GR-310 Cycloheximide Inhibitors: protein synthesis inhibitor 3402 P17 Enzo Life Sciences AP-304 Triptolide Inhibitors: inhibits NFkappaB transcriptional activation 3402 P18 Enzo Life Sciences A-195 Cyclosporin A Inhibitors: calcineurin inhibitor 3402 P19 Enzo Life Sciences GR-336 Tanshinone IIA Inhibitors: AP-1 inhibitor 3402 P20 Enzo Life Sciences PR-100 Cypermethrin Inhibitors: calcineurin inhibitor

Biomol ICCBL - 2012 Page 4 of 6 Created 9/2015 ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3402 P21 Enzo Life Sciences CA-421 Nigericin Inhibitors: induces intracellular acidification 3402 P22 Enzo Life Sciences T-108 Cytochalasin B Inhibitors: F actin capper 3403 A03 Enzo Life Sciences T-109 Cytochalasin D Inhibitors: F actin capper 3403 A05 Enzo Life Sciences ST-330 D609 Lipid biosynthesis: PC-PLC inhibitor 3403 A07 Enzo Life Sciences EI-274 Damnacanthal Kinase inhibitors: p56lck inhibitor 3403 A09 Enzo Life Sciences CN-223 YC-1 Activators: GC stimulator / Hif-1 alpha inhibitor 3403 A11 Enzo Life Sciences A-230 Decoyinine Inhibitors: lowers GTP levels 1-Deoxymannojirimycin 3403 A13 Enzo Life Sciences S-109 Inhibitors: mannosidase inhibitor hydrochloride 3403 A15 Enzo Life Sciences S-110 1-Deoxynojirimycin Inhibitors: glucosidase inhibitor 3403 A17 Enzo Life Sciences EI-126 Dexamethasone Nuclear receptor ligands: corticosteroid 3403 A19 Enzo Life Sciences CN-125 Dibutyrylcyclic AMP Activators: PKA activator 3403 A21 Enzo Life Sciences CN-215 Dibutyrylcyclic GMP Activators: PKA activator 3403 B03 Enzo Life Sciences T-101 Nocodazole Inhibitors: tubulin inhibitor 3403 B05 Enzo Life Sciences ST-315 OBAA Inhibitors: phospholipase A2 inhibitor 3403 B07 Enzo Life Sciences EI-181 Okadaic acid Inhibitors: PP1 PP2A inhibitor 3403 B09 Enzo Life Sciences CM-111 Oligomycin A Inhibitors: Fo ATP synthase inhibitor 3403 B11 Enzo Life Sciences CC-200 Olomoucine Kinase inhibitors: CDK inhibitor 3403 B13 Enzo Life Sciences CM-109 Ouabain Inhibitors: Na+K+ATPase inhibitor 3403 B15 Enzo Life Sciences L-133 PCA 4248 Bioactive lipids: PAF antagonist 3403 B17 Enzo Life Sciences EI-360 PD 98059 Kinase inhibitors: MEK inhibitor 3403 B19 Enzo Life Sciences EI-306 SU-4312 Kinase inhibitors: VEGF-R (Flk-1) tyrosine kinase 3403 B21 Enzo Life Sciences PI-120 Pepstatin Protease inhibitors: protease inhibitor 3403 C03 Enzo Life Sciences GR-234 GW-9662 Nuclear receptor ligands: PPAR gamma antagonist 3403 C05 Enzo Life Sciences D-100 6,7-ADTN CNS receptor ligands: Dopamine agonist 3403 C07 Enzo Life Sciences FR-110 Hinokitiol Inhibitors: Iron chelator 3403 C09 Enzo Life Sciences CN-240 Diphenyleneiodonium Inhibitors: flavoprotein inhibitor 3403 C11 Enzo Life Sciences CA-420 2,5-Ditertbutylhydroquinone Ion channel ligands: ER Ca++ ATPase inhibitor 3403 C13 Enzo Life Sciences GR-319 Doxorubicin Inhibitors: topoisomerase II inhibitor, induces apoptosis 3403 C15 Enzo Life Sciences EI-231 DRB (Benzimidazole) Kinase inhibitors: CKII inhibitor 3403 C17 Enzo Life Sciences FR-107 MnTBAP chloride Inhibitors: SOD mimetic 3403 C19 Enzo Life Sciences CA-302 E6 berbamine Inhibitors: calmodulin inhibitor 3403 C21 Enzo Life Sciences PI-107 E-64-d Protease inhibitors: calpain/cathepsin inhibitor 3403 D03 Enzo Life Sciences AP-100 6(5H)-Phenanthridinone Inhibitors: PARP inhibitor 3403 D05 Enzo Life Sciences PE-160 Phorbol 12-myristate 13-acetate Activators: PKC activator 3403 D07 Enzo Life Sciences GR-325 Pifithrin-α Inhibitors: p53 inhibitor 3403 D09 Enzo Life Sciences GR-233 CITCO Nuclear receptor ligands: Const. androstane receptor (CAR) agonist 3403 D11 Enzo Life Sciences EI-219 Piroxicam Lipid biosynthesis: COX1 inhibitor 3403 D13 Enzo Life Sciences GR-334 Cyclopamine Inhibitors: Hedgehog pathway inhibitor 3403 D15 Enzo Life Sciences EI-275 PP1 Protease inhibitors: src family trosine kinase inhibitor 3403 D17 Enzo Life Sciences AC-146 Prazocin CNS receptor ligands: adrenoreceptor agonist 3403 D19 Enzo Life Sciences AP-401 Propidium iodide Inhibitors: DNA intercalator 3403 D21 Enzo Life Sciences AR-107 (S)-(-)-propranolol·HCl CNS receptor ligands: adrenoceptor antagonist (beta) Inhibitors: Phosphodiesterase (PDE2) inhibitor/adenosine deaminase 3403 E03 Enzo Life Sciences PD-129 EHNA inhibitor 3403 E05 Enzo Life Sciences S-620 Pregnenolone-16α-carbonitrile Nuclear receptor ligands: PXR/SXR agonist 3403 E07 Enzo Life Sciences BL-093 Estradiol Nuclear receptor ligands: estrogen 3403 E09 Enzo Life Sciences GR-307 Etoposide Inhibitors: topoisomerase II inhibitor 3403 E11 Enzo Life Sciences CM-120 FCCP Inhibitors: mitochondrial uncoupler 3403 E13 Enzo Life Sciences CN-100 Forskolin Activators: Adenylate cyclase activator 3403 E15 Enzo Life Sciences EI-280 Geldanamycin Inhibitors: HSP90 inhibitor 3403 E17 Enzo Life Sciences ALX-350-006 Genistein Kinase inhibitors: Tyrosine kinase inhibitor 3403 E19 Enzo Life Sciences EI-283 Ro 31-8220 Kinase inhibitors: PKC inhibitor 3403 E21 Enzo Life Sciences EI-300 GM6001 Protease inhibitors: broad spectrum MMP inhibitor 3403 F03 Enzo Life Sciences GR-312 Puromycin·2HCl Inhibitors: protein synthesis inhibitor 3403 F05 Enzo Life Sciences EI-314 SB-431542 Kinase inhibitors: ALK4, ALK5, ALK7 inhibitor 3403 F07 Enzo Life Sciences EI-305 SP-600125 Kinase inhibitors: JNK inhibitor

3403 F09 Enzo Life Sciences AC-1142 Quercetin·2H2O Kinase inhibitors: kinase inhibitor (plus other) 3403 F11 Enzo Life Sciences A-275 Rapamycin Inhibitors: FRAP inhibitor 3403 F13 Enzo Life Sciences AM-100 Cyclo [Arg-Gly-Asp-D-Phe-Val] Inhibitors: integrin inhibitor 3403 F15 Enzo Life Sciences ST-300 RHC-80267 Lipid biosynthesis: DAG lipase inhibitor 3403 F17 Enzo Life Sciences PR-112 RK-682 Inhibitors: VHR phosphatase inhibitor 3403 F19 Enzo Life Sciences CC-205 Roscovitine Kinase inhibitors: CDK inhibitor 3403 F21 Enzo Life Sciences ALX-350-075 Rottlerin Kinase inhibitors: PKC delta inhibitor 3403 G03 Enzo Life Sciences EI-269 Go6976 Kinase inhibitors: PKC inhibitor 3403 G05 Enzo Life Sciences EI-287 Nimesulide Lipid biosynthesis: Cox 2 inhibitor 3403 G07 Enzo Life Sciences EI-148 H7 Kinase inhibitors: kinase inhibitor 3403 G09 Enzo Life Sciences EI-196 H-89 Kinase inhibitors: PKA inhibitor 3403 G11 Enzo Life Sciences EI-195 H9 Kinase inhibitors: kinase inhibitor 3403 G13 Enzo Life Sciences EI-233 HA1077 Kinase inhibitors: inhibitor of Rho-dependent kinases 3403 G15 Enzo Life Sciences EI-184 HA-1004 Kinase inhibitors: kinase inhibitor 3403 G17 Enzo Life Sciences EI-273 HBDDE Kinase inhibitors: PKC inhibitor 3403 G19 Enzo Life Sciences AC-764 Histamine CNS receptor ligands: Histamine receptor agonist 3403 G21 Enzo Life Sciences EI-248 HNMPA-(AM)3 Kinase inhibitors: Insulin receptor TK inhibitor 3403 H03 Enzo Life Sciences PR-110 RWJ-60475-(AM)3 Inhibitors: CD45 phosphatase inhibitor 3403 H05 Enzo Life Sciences EI-286 SB 203580 Kinase inhibitors: Suppressor of MAPKAP kinase-2 3403 H07 Enzo Life Sciences EI-294 SB 202190 Kinase inhibitors: MAP kinase inhibitor 3403 H09 Enzo Life Sciences CC-207 Indirubin-3'-monoxime Kinase inhibitors: GSK-3beta inhibitor 3403 H11 Enzo Life Sciences CC-206 Indirubin Kinase inhibitors: GSK-3beta inhibitor 3403 H13 Enzo Life Sciences NS-820 Serotonin CNS receptor ligands: serotonin receptor agonist 3403 H15 Enzo Life Sciences FR-104 Resveratrol Activators: SIRT1 activator

Biomol ICCBL - 2012 Page 5 of 6 Created 9/2015 ICCB-L ICCB-L Vendor Vendor ID Compound Name Compound description Plate Well 3403 H17 Enzo Life Sciences GR-331 Splitomycin Inhibitors: sir2p inhibitor 3403 H19 Enzo Life Sciences EI-297 PP2 Kinase inhibitors: Src family tyrosine kinase inhibitor 3403 H21 Enzo Life Sciences EI-271 Piceatannol Kinase inhibitors: Syk inhibitor Hoechst 33342·3HCl 3403 I03 Enzo Life Sciences GR-303 Inhibitors: DNA minor groove binder (BisBenzimide) 3403 I05 Enzo Life Sciences C-117 (-)-Huperzine A Inhibitors: acetylcholinesterase inhibitor 3403 I07 Enzo Life Sciences GR-230 24(S)-hydroxycholesterol Nuclear receptor ligands: LXR agonist 3403 I09 Enzo Life Sciences GR-332 ICRF-193 Inhibitors: topo II inhibitor that does not cause DNA breaks 3403 I11 Enzo Life Sciences EI-131 Indomethacin Lipid biosynthesis: cyclooxygenase inhibitor 3403 I13 Enzo Life Sciences CA-201 Ionomycin Ion channel ligands: Ca++ ionophore 3403 I15 Enzo Life Sciences PD-140 IBMX Inhibitors: PDE inhibitor (broad spec), adenosineR agonist 3403 I17 Enzo Life Sciences EI-309 NSC-95397 Inhibitors: CDC25 phosphatase inhibitor 3403 I19 Enzo Life Sciences BL-169 Juglone Inhibitors: PIN1 inhibitor 3403 I21 Enzo Life Sciences EI-152 K252A Kinase inhibitors: Kinase inhibitor (Broad spectrum) 3403 J03 Enzo Life Sciences CN-140 SQ22536 Inhibitors: adenylate cyclase inhibitor 3403 J05 Enzo Life Sciences T-112 Alrestatin Inhibitors: aldose reductase inhibitor 3403 J07 Enzo Life Sciences EI-156 staurosporine Kinase inhibitors: kinase inhibitor - non-selective 3403 J09 Enzo Life Sciences S-112 swainsonine Inhibitors: protein glycosylation inhibitor 3403 J11 Enzo Life Sciences S-650 Tamoxifen Nuclear receptor ligands: estrogen antagonist 3403 J13 Enzo Life Sciences T-104 Taxol = Paclitaxel Inhibitors: microtubule stabilizer 3403 J15 Enzo Life Sciences EI-253 RG-14620 Kinase inhibitors: EGF-R tyrosine kinase inhibitor 3403 J17 Enzo Life Sciences T-115 Thalidomide Inhibitors: TNFalpha synthesis inhibitor 3403 J19 Enzo Life Sciences CN-257 Thiocitrulline [L-Thiocitrulline] Inhibitors: bNOS inhibitor 3403 J21 Enzo Life Sciences EI-246 GF-109203X Kinase inhibitors: PKC inhibitor 3403 K03 Enzo Life Sciences EI-230 KN-62 Kinase inhibitors: CaM kinase II inhibitor 3403 K05 Enzo Life Sciences EI-199 KT-5720 Kinase inhibitors: PKA inhibitor 3403 K07 Enzo Life Sciences G-242 L-744,832 Inhibitors: Ras farnesyltransferase inhibitor 3403 K09 Enzo Life Sciences CN-255 Furoxan Activators: NO donor 3403 K11 Enzo Life Sciences T-110 Latrunculin B Inhibitors: Actin inhibitor 3403 K13 Enzo Life Sciences EI-185 Lavendustin A Kinase inhibitors: Tyrosine kinase inhibitor EGF-R) 3403 K15 Enzo Life Sciences CC-202 N9-Isopropylolomoucine Kinase inhibitors: CDC-2 kinase inhibitor 3403 K17 Enzo Life Sciences PI-118 Leupeptin Protease inhibitors: protease inhibitor 3403 K19 Enzo Life Sciences EI-278 BAY 11-7082 Inhibitors: Inhibits IKK kinase activation 3403 K21 Enzo Life Sciences PR-113 Tyrphostin-8 Inhibitors: Calcineurin inhibitor 3403 L03 Enzo Life Sciences EI-267 Tyrphostin AG-825 Kinase inhibitors: HER-1,2 tyrosine kinase inhibitor 3403 L05 Enzo Life Sciences NA-136 Kavain (+/-) Ion channel ligands: voltage-dependent Na channel inhibitor 3403 L07 Enzo Life Sciences AP-300 TPEN Inhibitors: cell permable heavy metal chelator 3403 L09 Enzo Life Sciences GR-309 Trichostatin-A Inhibitors: histone deacetylase inhibitor 3403 L11 Enzo Life Sciences CA-310 Trifluoperazine Inhibitors: calmodulin inhibitor-possibly only at high concentrations! 3403 L13 Enzo Life Sciences CC-104 Tunicamycin Inhibitors: glycosylation inhibitor 3403 L15 Enzo Life Sciences PI-143 Nafamostat mesylate Inhibitors: Serine protease inhibitor 3403 L17 Enzo Life Sciences EI-263 Tyrphostin AG-126 Kinase inhibitors: tyrosine kinase inhibitor 3403 L19 Enzo Life Sciences EI-190 Tyrphostin 1 Inhibitors: Calcineurin inhibitor 3403 L21 Enzo Life Sciences EI-215 Tyrphostin 9 Kinase inhibitors: PDGF-R tyrosine kinase inhibitor 3403 M03 Enzo Life Sciences CN-242 L-NAME Inhibitors: NO synthesis inhibitor 3403 M05 Enzo Life Sciences ST-420 LY-294002 Lipid biosynthesis: PI-3-Kinase inhibitor 3403 M07 Enzo Life Sciences CN-200 LY-83583 Inhibitors: Inhibits NO-activation of guanylate cyclase 3403 M09 Enzo Life Sciences EI-293 5-Iodotubercidin Kinase inhibitors: ERK-2 inhibitor 3403 M11 Enzo Life Sciences EI-177 Manoalide Lipid biosynthesis: Phospholipase A2 inhibitor 3403 M13 Enzo Life Sciences G-236 Manumycin A Inhibitors: ras farnesylation inhibitor 3403 M15 Enzo Life Sciences G-410 Mastoparan Activators: activates heterotrimeriuc GTPases 3403 M17 Enzo Life Sciences FR-103 MCI-186 Inhibitors: antioxidant, cytoprotectant 3403 M19 Enzo Life Sciences PI-129 Gliotoxin Protease inhibitors: Inhibitor of 20S-proteasome chymotrypsin activity 3403 M21 Enzo Life Sciences EI-295 LFM-A13 Kinase inhibitors: BTK inhibitor 3403 N03 Enzo Life Sciences ST-391 U73122 Lipid biosynthesis: PLC inhibitor 3403 N05 Enzo Life Sciences EI-282 U-0126 Kinase inhibitors: MEK inhibitor 3403 N07 Enzo Life Sciences KC-140 Valinomycin Ion channel ligands: K+ ionophore 3403 N09 Enzo Life Sciences T-116 Vinblastine Inhibitors: tubulin inhibitor 3403 N11 Enzo Life Sciences CA-320 W7 Inhibitors: calmodulin antagonist 3403 N13 Enzo Life Sciences ST-415 Wortmannin Lipid biosynthesis: PI-3Kinase, other kinases inhibitor 3403 N15 Enzo Life Sciences EI-299 Y-27632 Kinase inhibitors: ROCK inhibitor 3403 N17 Enzo Life Sciences AC-161 Yohimbine CNS receptor ligands: Adrenoreceptor antagonist (alpha) 3403 N19 Enzo Life Sciences ZW-9170 Z-Leu3-VS Protease inhibitors: Proteasome inhibitor 3403 N21 Enzo Life Sciences EI-298 ZM336372 Kinase inhibitors: Raf inhibitor 3403 O03 Enzo Life Sciences CC-103 Methotrexate CNS receptor ligands: DHFR inhibitor 3403 O05 Enzo Life Sciences C-114 (±)-Epibatidine CNS receptor ligands: nicotinic cholinergic agonist 3403 O07 Enzo Life Sciences G-226 Mevinolin (Lovastatin) Lipid biosynthesis: Inhibitor HMG-CoA reductase 3403 O09 Enzo Life Sciences GR-311 Mitomycin C Inhibitors: cross links DNA 3403 O11 Enzo Life Sciences EI-197 ML7 Kinase inhibitors: kinase inhibitor 3403 O13 Enzo Life Sciences EI-153 ML9 Kinase inhibitors: kinase inhibitor 3403 O15 Enzo Life Sciences GR-322 Monastrol Inhibitors: Eg5 inhibitor 3403 O17 Enzo Life Sciences EI-307 GW-5074 Kinase inhibitors: cRAF1 kinase inhibitor 3403 O19 Enzo Life Sciences A-248 Monensin sodium Ion channel ligands: Na+ ionophore 3403 O21 Enzo Life Sciences A-235 FK-506 Inhibitors: FKBP ligand 3403 P03 Enzo Life Sciences P-416 Z-VAD(OMe)-FMK Protease inhibitors: Caspase inhibitor (broad spectrum) 3403 P05 Enzo Life Sciences EI-261 NS-398 Lipid biosynthesis: Cox-2 inhibitor 3403 P07 Enzo Life Sciences EI-216 AA-861 Lipid biosynthesis: 5-lipoxygenase inhibitor 3403 P09 Enzo Life Sciences A-249 Mycophenolic acid Inhibitors: Inosine-5'-monophosphate dehydrogenase inhibitor 3403 P11 Enzo Life Sciences CT-115 Shikonin Inhibitors: Apoptosis inducer, p53 dependent 3403 P13 Enzo Life Sciences AC-1557 2-APB Inhibitors: IP3 receptor blocker 3403 P15 Enzo Life Sciences EI-211 CDC Lipid biosynthesis: 12-Lipoxygenase inhibitor 3403 P17 Enzo Life Sciences G-237 Cerulenin Lipid biosynthesis: Fatty acid biosynthesis inhibitor 3403 P19 Enzo Life Sciences CA-305 Phenoxybenzamine Inhibitors: Calmodulin antagonist 3403 P21 Enzo Life Sciences T-126 Wiskostatin Inhibitors: N-WASP inhibitor

Biomol ICCBL - 2012 Page 6 of 6 Created 9/2015