Tech Help: Email: [email protected] | Toll Free: 800.891.9699 (US Only) | Enzyme Inhibitors Enzymes are biological catalysts that drive various reactions within a cell. They are required for nearly every function of a living cell/organism from digestion of food to the synthesis of DNA. Enzymes are usually very specific as to which reactions they catalyze and the substrates that are involved. Enzyme activity can be modulated by different classes of molecules. Enzyme Inhibitors are molecules that bind to the enzyme and decrease or completely stop their function. Since blocking the activity of an enzyme can have profound effects on the downstream cellular events sometimes with pathological or disease consequences, enzyme inhibition is a crucial component of new drug design. The discovery of new and potent enzyme inhibitors and developing better classes of inhibitors constitutes a dynamic branch of biochemical and pharmacological research in the area of Diabetes, Cancer, HIV and many more. BioVision offers a comprehensive collection of more than 800 enzyme inhibitors covering all the core biological/pharmacological research areas. ACAT (Acyl-CoA cholesteryl Acyl Transferase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Arecoline hydrobromide B1824 100 mg, 500 mg 300-08-3 Endostatin, human recombinant 4759 20 μg, 100 μg, 1 mg N/A Avasimibe 9506 5 mg, 25 mg 166518-60-1 Endostatin, human recombinant 4799 100 μg, 1 mg N/A Naringenin 1772 250 mg, 1 g 480-41-1 Fumagillin 2368 1 mg, 5 mg 23110-15-8 Pellitorine 2053 1 mg, 5 mg 18836-52-7 Isoxanthohumol 2529 5 mg, 25 mg 70872-29-6 Penicillide B1245 250 µg, 1 mg 55303-92-9 2-Methoxyestradiol 2166 5 mg, 25 mg 362-07-2 Pyripyropene A B1910 500 µg, 1 mg 147444-03-9 SKLB610 2610 5 mg, 25 mg 1125780-41-7 Terpendole C 2214 250 µg, 1 mg 156967-65-6 Thiabendazole 2161 1 g 148-79-8 TMP-153 B1181 10 mg, 50 mg 128831-46-9 Tranilast 1876 10 mg, 50 mg 53902-12-8 ACC (Acetyl-CoA Carboxylase) Inhibitors Angiotensin Receptor Antagonists Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. ACC2 Inhibitor 1717 1 mg, 5 mg N/A BIBS39 B1071 5 mg, 25 mg 133085-33-3 CP-640186 9422 5 mg, 25 mg 591778-68-6 EXP-3174 9672 5 mg, 25 mg 124750-92-1 CP-640186 hydrochloride B1254 5 mg, 25 mg 591778-70-0 Losartan potassium 2750 50 mg, 250 mg 124750-99-8 Valsartan 2004 25 mg, 100 mg, 500 mg 137862-53-4 ACE (Angiotensin-Converting Enzyme) Inhibitors Product Name Cat. No. Size CAS. No. Arginase Inhibitors ACE2 Inhibitor, DX600 9687 100 µg, 500 µg, 1 mg N/A Product Name Cat. No. Size CAS. No. Captopril B1187 1 g, 5 g 62571-86-2 BEC 2359 1 mg, 5 mg 63107-40-4 Adenylase Cyclase Inhibitors Aromatase Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. 2',5'-Dideoxyadenosine 2770 5 mg, 25 mg 6698-26-6 Exemestane 9473 5 mg, 25 mg 107868-30-4 KH7 2350 5 mg, 25 mg 330676-02-3 ATPase Inhibitors PACAP (human, chicken, mouse, ovine, B1562 100 μg, 500 μg 143748-18-9 porcine, rat) (6-38) Product Name Cat. No. Size CAS. No. SQ 22536 2019 5 mg, 25 mg 17318-31-9 Bafilomycin A1 1829 50 µg, 250 µg 88899-55-2 (-)-Blebbistatin 2406 1 mg, 5 mg 856925-71-8 AKR (Aldo-Keto Reductase) Inhibitors (+)-Blebbistatin 2407 1 mg, 5 mg 1177356-70-5 Product Name Cat. No. Size CAS. No. (±)-Blebbistatin 2405 5 mg, 25 mg 674289-55-5 AKR1C3 Inhibitor I 2403 5 mg, 25 mg N/A Bufalin 2509 10 mg, 50 mg 465-21-4 AKR1C3 Inhibitor II 2404 5 mg, 25 mg N/A Autophagy Inhibitors AKR1C3 Inhibitor III 2424 5 mg, 25 mg N/A Product Name Cat. No. Size CAS. No. Androgen Receptor Antagonists ATM Kinase Inhibitor, KU-55933 1685 5 mg 587871-26-9 Product Name Cat. No. Size CAS. No. Bafilomycin A1 1829 50 µg, 250 µg 88899-55-2 ARN-509 9535 5 mg, 25 mg 956104-40-8 Chloroquine Diphosphate 1825 100 mg, 500 mg 50-63-5 MDV-3100 9479 10 mg, 50 mg 915087-33-1 EZSolution™ Gö 6976 1785 500 µg 136194-77-9 ODM-201 9668 5 mg, 25 mg 1297538-32-9 Gö 6976 1711 500 µg 136194-77-9 Angiogenesis Inhibitors 3-Methyladenine 2249 25 mg, 100 mg 5142-23-4 Spautin-1 2037 5 mg, 25 mg 1262888-28-7 Product Name Cat. No. Size CAS. No. Angiostatin Human 4919 100 μg, 500 μg N/A Bcl-2 (B-cell 2) Inhibitors Angiostatin K1-3, human recombinant 4920 20 μg, 100 μg, 1 mg N/A Product Name Cat. No. Size CAS. No. BIBF1120 2167 5 mg, 25 mg 928326-83-4 A-1155463 B1821 5 mg, 25 mg 1235034-55-5 Borrelidin 2367 250 µg, 1 mg 7184-60-3 A-1210477 B1826 5 mg, 25 mg 1668553-26-1 Castanospermine 2293 10 mg, 50 mg 79831-76-8 A-1331852 B1948 5 mg, 25 mg 1430844-80-6

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 2 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. ABT-263 2467 5 mg, 25 mg 923564-51-6 110044-82-1 DiscoveryPak™ Calpain Inhibitors Set 136632-32-1 ABT-737 2463 5 mg, 25 mg 852808-04-9 (Containing Cat. No. 1834, 1835, 1506, S228 1 Set 133410-84-1 AT-101 2380 5 mg, 25 mg 90141-22-3 2195, 1906) 88191-84-8 BCl-2 Inhibitor GX15-070 2040 5 mg 803712-67-6 179528-45-1 MDL 28170 2195 10 mg, 50 mg 88191-84-8 BCl-2 Inhibitor, ABT-199 2253 1 mg, 5 mg 1257044-40-8 1257044-40-8 PD 150,606 1906 5 mg, 25 mg 179528-45-1 DiscoveryPak™ Bcl2 Inhibitors Set 923564-51-6 (Containing Cat. No. 2253, 2467, 2463, S229 1 Set 852808-04-9 Caspase & Granzyme B Inhibitors 2380, 2040) 90141-22-3 Product Name Cat. No. Size CAS. No. 803712-67-6 Ac-DEVD-CHO B1951 1 mg, 5 mg 169332-60-9 BDA366 B1827 5 mg, 25 mg 1909226-00-1 inhibitor 2783 5 mg, 25 mg 54135-60-3 BH3I-1 B1277 5 mg, 25 mg 300817-68-9 AZ10417808 2786 1 mg, 5 mg 331645-84-2 CC-122 B1650 5 mg, 25 mg 1015474-32-4 Biotin-DEVD-FMK 1124 20 µl (10 mM) N/A CID-5721353 B1275 5 mg, 25 mg 301356-95-6 Biotin-IETD-FMK 1121 20 µl (10 mM) N/A HA14-1 B1832 5 mg, 25 mg 65673-63-4 Biotin-VAD-FMK 1123 20 µl (10 mM) 1135688-15-1 Pyridoclax B1817 1 mg, 5 mg 1651890-44-6 Biotin-VDVAD-FMK 1032 20 µl (10 mM) N/A S63845 B1819 250 μg, 1 mg 1799633-27-4 Boc-D-FMK 1160 1 mg, 5 mg 187389-53-3 TW-37 2789 5 mg, 25 mg 877877-35-5 Caspase Family Inhibitor Set K107 5 x 25 µl N/A WEHI-539 B1818 5 mg, 25 mg 1431866-33-9 Caspase Family Inhibitor Set II K108 7 x 25 µl N/A BMP (Bone Morphogenetic Protein) Inhibitors Caspase Family Inhibitor Set III K210 8 x 25 µl N/A Product Name Cat. No. Size CAS. No. Caspase Family Inhibitor Set IV K220 12 x 25 µl N/A DMH-1 9542 5 mg, 25 mg 1206711-16-1 Caspase Inhibitor Boc-D-FMK 1120 20 µl (10 mM) 187389-53-3 EZSolution™ LDN193189 2092 5 mg 1062368-24-4 Caspase-1 Inhibitor Z-YVAD-FMK 1012 20 µl (10 mM), 100 µl (2 mM) N/A LDN193189 1995 5 mg, 25 mg 1062368-24-4 Caspase-10 Inhibitor AEVD-FMK 1112 20 µl (10 mM), 100 µl (2 mM) 1135688-47-9 Caspase-12 Inhibitor Z-ATAD-FMK 1079 20 µl (10 mM), 100 µl (2 mM) N/A Bone Resorption Inhibitors Caspase-13 Inhibitor LEED-FMK 1115 20 µl (10 mM), 100 µl (2 mM) N/A Product Name Cat. No. Size CAS. No. Caspase-2 Inhibitor Z-VDVAD-FMK 1073 20 µl (10 mM), 100 µl (2 mM) N/A Alendronate sodium 2168 50 mg, 250 mg 121268-17-5 Caspase-3 Inhibitor Q-DEVD-Oph 1175 1 mg, 3 mg, 5 mg N/A Pamidronate disodium 1884 50 mg, 250 mg 57248-88-1 Caspase-3 Inhibitor Z-DEVD-FMK 1009 20 µl (10 mM), 100 µl (2 mM) 210344-95-9 Zoledronic acid hydrate 2653 10 mg, 50 mg 165800-06-6 Caspase-3 inhibitor, Z-DQMD-FMK 2782 1 mg, 5 mg N/A Bromodomain Inhibitors Caspase-3/7 Inhibitor 2780 1 mg, 5 mg 220509-74-0 Caspase-4 Inhibitor Z-LEVD-FMK 1108 20 µl (10 mM), 100 µl (2 mM) N/A Product Name Cat. No. Size CAS. No. Caspase-5 Inhibitor Z-WEHD-FMK 1100 20 µl (10 mM), 100 µl (2 mM) N/A BAZ2-ICR B1865 5 mg, 25 mg 1665195-94-7 Caspase-6 Inhibitor Z-VEID-FMK 1011 20 µl (10 mM), 100 µl (2 mM) N/A BI-7273 B1879 5 mg, 25 mg 1883429-21-7 Caspase-8 Inhibitor Z-IETD-FMK 1064 20 µl (10 mM), 100 µl (2 mM) N/A BI-9564 B1880 5 mg, 25 mg 1883429-22-8 Caspase-8 Inhibitor, Q-IETD-Oph 1176 1 mg, 3 mg, 5 mg N/A Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4 Caspase-9 Inhibitor Z-LEHD-FMK 1074 20 µl (10 mM), 100 µl (2 mM) N/A Bromosporine 2652 1 mg, 5 mg 1619994-69-2 Caspase-9 Inhibitor, Q-LEHD-Oph 1177 1 mg, 3 mg, 5 mg N/A CPI-0610 B1201 5 mg, 25 mg 1380087-89-7 Caspase-Family Inhibitor Z-VAD-FMK 1010 20 µl (10 mM), 100 µl (2 mM) 187389-52-2 CPI-203 9404 1 mg, 5 mg 1446144-04-2 EMAP-II Inhibitor Z-ASTD-FMK 1127 20 µl (10 mM) N/A GSK-2801 9553 5 mg, 25 mg 1619994-68-1 FITC-DEVD-FMK 9499 100 Assays N/A I-BET151 2220 1 mg, 5 mg 1300031-49-5 FITC-IETD-FMK 9533 100 Assays N/A I-BET726 B1569 5 mg, 25 mg 1300031-52-0 FITC-LEHD-FMK 9534 100 Assays N/A I-BET762 2628 1 mg, 5 mg 1260907-17-2 FITC-VAD-FMK 9497 100 Assays N/A I-CBP112 9405 1 mg, 5 mg N/A FITC-VDVAD-FMK 9498 100 Assays N/A EZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4 FMK Negative Control 1122 20 µl (10 mM), 100 µl (2 mM) 197855-65-5 (-)-JQ1 2384 1 mg 1268524-71-5 Granzyme B Inhibitor Ac-IEPD-CHO 1119 1 mg N/A Mivebresib B1564 5 mg, 25 mg 1445993-26-9 Granzyme B Inhibitor Z-AAD-CH2Cl 1128 20 µl (10 mM) N/A MS436 2680 5 mg, 25 mg 1395084-25-9 Ivachtin 2788 1 mg, 5 mg 745046-84-8 OF-1 9592 5 mg, 25 mg 919973-83-4 Pan-caspase inhibitor, Q-VD(OMe)-Oph 2787 1 mg, 5 mg N/A OTX015 2651 1 mg, 5 mg 202590-98-5 EZSolution™ Q-DEVD-Oph 1178 1 mg N/A PFI-1 2203 1 mg, 5 mg 1403764-72-6 EZSolution™ Q-VD-Oph 1173 1 mg 1135695-98-5 PFI-3 2895 5 mg, 25 mg 1819363-80-8 Q-VD-OPh 1170 1 mg, 3 mg, 5 mg 1135695-98-5 RVX-208 9408 1 mg, 5 mg 1044870-39-4 EZSolution™ Q-VD-OPh, Negative Control 1174 1 mg N/A SGC-CBP30 9554 5 mg, 25 mg 1613695-14-9 QVD-OPh Negative Control 1171 1 mg, 3 mg, 5 mg N/A Calpain Inhibitors VX-765 2781 5 mg, 25 mg 273404-37-8 Product Name Cat. No. Size CAS. No. Z-AEVD-FMK B1162 1 mg, 5 mg 1135688-47-9 EZSolutioin™ Calpain Inhibitor I, ALLN 2544 5 mg 110044-82-1 Z-ATAD-FMK 1152 1 mg, 5 mg N/A Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1 Z-DEVD-FMK 1143 1 mg, 5 mg 210344-95-9 Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1 Z-FA-FMK 1986 1 mg, 5 mg 105637-38-5 Calpain Inhibitor Z-LLY-FMK 1125 20 µl (10 mM) 133410-84-1 Z-IETD-FMK 1148 1 mg, 5 mg N/A Calpain Inhibitor, Z-LLY-FMK B1506 250 μg, 1 mg 133410-84-1 Z-LEHD-FMK 1149 1 mg, 5 mg N/A 2 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 3 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Z-LEVD-FMK 1144 1 mg, 5 mg N/A Nimesulide 2777 1 g, 5 g 51803-78-2 Z-VAD-FMK 1140 1 mg, 5 mg 187389-52-2 Parecoxib Sodium B1989 10 mg, 50 mg 198470-85-8 Z-VDVAD-FMK 1142 1 mg, 5 mg N/A Robenacoxib B1990 5 mg, 25 mg 220991-32-2 Z-VEID-FMK 1146 1 mg, 5 mg N/A Rofecoxib B1982 10 mg, 50 mg 162011-90-7 Z-YVAD-FMK 1141 1 mg, 5 mg N/A Valdecoxib B1991 5 mg, 25 mg 181695-72-7 Cathepsin Inhibitors DNA Ligase Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Balicatib 2596 5 mg, 25 mg 354813-19-7 L-189 9674 5 mg, 25 mg 64232-83-3 Cathepsin B&L Inhibitor Z-Phe-Phe-FMK 1126 20 µl (10 mM) N/A L-67 9633 5 mg, 25 mg 325970-71-6 Cathepsin G Inhibitor 1982 1 mg 429676-93-7 DPP-4 (Dipeptidyl Peptidase-4 ) Inhibitors Odanacatib B1617 5 mg, 25 mg 603139-19-1 Tanshinone IIA-Sulfonic Sodium B1902 5 mg, 25 mg 69659-80-9 Product Name Cat. No. Size CAS. No. Z-FA-FMK 1986 1 mg, 5 mg 105637-38-5 Alogliptin benzoate 9656 50 mg, 250 mg 850649-62-6 Diprotin A 2191 5 mg, 25 mg 90614-48-5 CDc42 Inhibitors Diprotin B 2192 5 mg, 25 mg 90614-49-6 Product Name Cat. No. Size CAS. No. DPP IV Inhibitor, K 579 1963 1 mg, 5 mg 440100-64-1 ML141 2267 5 mg, 25 mg 71203-35-5 DPP IV Inhibitor, NVP DPP 728 1964 1 mg, 5 mg 247016-69-9 MLS-573151 1929 5 mg, 25 mg 10179-57-4 DPPIV Inhibitor, P32/98 2571 5 mg, 25 mg 136259-20-6 ZCL278 2466 5 mg, 25 mg 587841-73-4 668270-12-0 DiscoveryPak™ DPP-IV Inhibitors Set 361442-04-8 Cell Adhesion Inhibitors (Containing Cat. No. 2240, 9528, 1757, K890 5 Inhibitors 654671-77-9 2798, 2188) 1029877-94-8 Product Name Cat. No. Size CAS. No. 274901-16-5 K-7174 dihydrochloride 9478 5 mg, 25 mg 191089-60-8 Linagliptin 2240 50 mg, 250 mg 668270-12-0 CETP (Cholesteryl Ester Transfer Protein) MK-3102 9599 1 mg, 5 mg 1226781-44-7 Inhibitors Saxagliptin 9528 50 mg, 250 mg 361442-04-8 Sitagliptin Monohydrate 1757 100 mg, 1 g 654671-77-9 Product Name Cat. No. Size CAS. No. Teneligliptin B1932 10 mg, 50 mg 760937-92-6 EZSolution™ 2531 1 mg 875446-37-0 Trelagliptin succinate 2798 5 mg, 25 mg 1029877-94-8 Anacetrapib 2418 1 mg, 5 mg 875446-37-0 Vildagliptin 2188 10 mg, 50 mg 274901-16-5 875446-37-0 DiscoveryPak™ CETP Inhibitors Set 211513-37-0 (Containing Cat. No. 2418, 2419, 2558, S225 1 Set DUBs (Deubiquitinating Enzymes) & Related 1186486-62-3 2420) 262352-17-0 Inhibitors EZSolution ™ 2532 1 mg 211513-37-0 Product Name Cat. No. Size CAS. No. Dalcetrapib 2419 1 mg, 5 mg 211513-37-0 DUB Inhibitor, NSC-632839 2570 5 mg, 25 mg 157654-67-6 2558 5 mg, 25 mg 1186486-62-3 DUB Inhibitor, PR-619 2302 5 mg, 25 mg 2645-32-1 Sclerotiorin 2334 250 µg, 1 mg 549-23-5 HBX-41108 9608 5 mg, 25 mg 924296-39-9 EZSolution™ 2533 5 mg 262352-17-0 LDN-57444 2016 5 mg, 25 mg 668467-91-2 Torcetrapib 2420 5 mg, 25 mg 262352-17-0 ML-323 2658 5 mg, 25 mg 1572414-83-5 Chloride Channel Blockers NSC-687852 2021 5 mg, 25 mg 1009817-63-3 Spautin-1 2037 5 mg, 25 mg 1262888-28-7 Product Name Cat. No. Size CAS. No. USP14 Inhibitor, IU1 1845 5 mg, 25 mg 314245-33-5 CaCCinh-A01 B2014 5 mg, 25 mg 407587-33-1 USP7/USP47 Inhibitor, P 22077 2301 5 mg, 25 mg 1247819-59-5 CFTR Inhibitor-172 2487 1 mg, 5 mg 307510-92-5 WP-1130 2014 5 mg, 25 mg 856243-80-6 CLP-290 B1282 5 mg, 25 mg 1181083-81-7 Cholesterol Transport Inhibitors FAAH (Fatty Acid Amide Hydrolase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. FAAH Inhibitor, PF-622 1928 5 mg, 25 mg 898235-65-9 9468 25 mg, 100 mg 163222-33-1 JNJ-1661010 2413 5 mg, 25 mg 681136-29-8 U-18666A 9469 5 mg, 25 mg 3039-71-2 JZL195 B1064 5 mg, 25 mg 1210004-12-8 COX (Cyclooxygenase) Inhibitors EZSolution™ MAFP 2811 5 mg 188404-10-6 Product Name Cat. No. Size CAS. No. FAS (Fatty Acid Synthase) Inhibitors Celecoxib 1574 100 mg, 1 g 169590-42-5 Product Name Cat. No. Size CAS. No. Cimicoxib B1984 5 mg, 25 mg 265114-23-6 Cerulenin 1579 5 mg, 50 mg 17397-89-6 Deracoxib B1985 10 mg, 50 mg 169590-41-4 DPVP B1243 1 mg 223386-36-5 DuP-697 B1517 5 mg, 25 mg 88149-94-4 FAS Inhibitor, C75 1547 1 mg 191282-48-1 Etoricoxib B1983 10 mg, 50 mg 202409-33-4 GSK-2194069 B1571 5 mg, 25 mg 1332331-21-1 Firocoxib B1986 5 mg, 25 mg 189954-96-9 α-Mangostin B1059 10 mg, 50 mg 6147-11-1 6-Gingerol 2507 5 mg, 25 mg 23513-14-6 Loganin B1161 10 mg, 50 mg 18524-94-2 Ferroptosis Inhibitors Lumiracoxib B1987 5 mg, 25 mg 220991-20-8 Product Name Cat. No. Size CAS. No. Mavacoxib B1988 5 mg, 25 mg 170569-88-7 Ferrostatin-1 2230 5 mg, 25 mg 347174-05-4

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 4 FPT (Farnesyl Protein Transferase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Andrastin A, Aspergillus fumigatus 2149 250 µg, 1 mg 174232-42-9 (-)-Epigallocatechin gallate 1841 50 mg 989-51-5 Arglabin 9691 1 mg, 5 mg 84692-91-1 Garcinol 2088 5 mg, 25 mg 78824-30-3 FTI-277 hydrochloride 2874 5 mg, 25 mg 180977-34-8 Plumbagin 2290 50 mg, 250 mg 481-42-5 L-778123 hydrochloride 9638 10 mg, 50 mg 253863-00-2 Remodelin 9411 5 mg, 25 mg 949912-58-7 Lonafarnib B1616 5 mg, 25 mg 193275-84-2 HDAC (Histone Deacetylase) Inhibitors Manumycin A 2333 1 mg, 5 mg 52665-74-4 Product Name Cat. No. Size CAS. No. Tipifarnib, Free base 2296 1 mg, 5 mg 192185-72-1 ACY-1215 2629 5 mg, 25 mg 1316214-52-4 Glucosidase Inhibitors ACY-775 B2011 5 mg, 25 mg 1375466-18-4 Product Name Cat. No. Size CAS. No. Apicidin 1601 1 mg 183506-66-3 Castanospermine 2293 10 mg, 50 mg 79831-76-8 AR-42 (HDAC-42) 2716 1 mg, 5 mg 935881-37-1 Conduritol B Epoxide 9574 5 mg, 25 mg 6090-95-5 BG-45 B1866 5 mg, 25 mg 926259-99-6 Miglitol 2335 5 mg, 25 mg 72432-03-2 BML210 B1128 5 mg, 25 mg 537034-17-6 GLUT1 (Glucose Transporter) Inhibitors BRD-73954 9596 5 mg, 25 mg 1440209-96-0 CAY10683 B1051 5 mg, 25 mg 1477949-42-0 Product Name Cat. No. Size CAS. No. CBHA 2284 5 mg, 10 mg 174664-65-4 BAY-876 B1572 5 mg, 25 mg 1799753-84-6 Chidamide 2261 1 mg, 5 mg 743420-02-2 Fasentin B1576 5 mg, 25 mg 392721-37-8 CI-994 1742 10 mg, 50 mg 112522-64-2 Naringenin 1772 250 mg, 1 g 480-41-1 Citarinostat B1560 5 mg, 25 mg 1316215-12-9 Resveratrol 1758 100 mg, 500 mg 501-36-0 CUDC-101 1966 5 mg, 25 mg 1012054-59-9 Rubusoside B1574 5 mg, 25 mg 64849-39-4 Depudecin 2087 100 µg 139508-73-9 STF-31 9585 5 mg, 25 mg 724741-75-7 Droxinostat 9570 5 mg, 25 mg 99873-43-5 WZB117 B1573 5 mg, 25 mg 1223397-11-2 Elevenostat B1893 1 mg N/A Glutamate Receptor Antagonists FK228 2447 1 mg 128517-07-7 HC Toxin 2728 500 µg, 1 mg 83209-65-8 Product Name Cat. No. Size CAS. No. 183506-66-3 LY-341495 2875 1 mg, 5 mg 201943-63-7 DiscoveryPak™ HDAC Inhibitor Set 58880-19-6 (Containing Cat. No. 1601, 1606, 1607, K851 6 Inhibitors 251456-60-7 Glutamate Uptake Inhibitors 1608, 1647) 1716-12-7 1069-66-5 Product Name Cat. No. Size CAS. No. 112522-64-2 Evans Blue Tetrasodium 2586 1 g 314-13-6 404950-80-7 Rose bengal 2587 100 mg, 500 mg 632-69-9 DiscoveryPak™ HDAC Inhibitor Set II 149647-78-9 (Containing Cat. No. 1742, 1612, 1604, K876 7 Inhibitors 38937-66-5 2202, 1605, 1606, 1984) 287383-59-9 Glycolysis Inhibitors 58880-19-6 Product Name Cat. No. Size CAS. No. 537049-40-4 6-Aminonicotinamide B1047 100 mg, 500 mg 329-89-5 ITF2357 9431 1 mg, 5 mg 732302-99-7 3-Bromopyruvic acid B1045 100 mg, 500 mg 1113-59-3 ITSA-1 2089 5 mg, 25 mg 200626-61-5 2-Deoxy-D-Glucose B1048 100 mg, 500 mg 154-17-6 JNJ-26481585 9612 5 mg, 25 mg 875320-29-9 Lonidamine B1058 10 mg, 50 mg 50264-69-2 LAQ824 2634 1 mg, 5 mg 404951-53-7 Oxythiamine Chloride Hydrochloride B1046 100 mg, 500 mg, 1 g 614-05-1 LMK-235 B1642 5 mg, 25 mg 1418033-25-6 Shikonin B1056 10 mg, 50 mg 517-89-5 M344 1607 1 mg 251456-60-7 MC-1568 B1085 5 mg, 25 mg 852475-26-4 GST (Glutathione S-Transferase) Inhibitors MGCD0103 2633 10 mg, 50 mg 726169-73-9 Product Name Cat. No. Size CAS. No. MS-275 (Entinostat, SNDX-275) 1590 1 mg, 5 mg 209783-80-2 Ezatiostat 2608 5 mg, 25 mg 168682-53-9 NCH 51 B1130 5 mg, 25 mg 848354-66-5 GST Inhibitor-1 (Cibacron Blue 3G-A, 1555R 1 g 84166-13-2 Sodium Salt) Nexturastat A 2098 1 mg 1403783-31-2 GST Inhibitor-2 (Ethacrynic acid)) 1556 1 g 58-54-8 NKL 22 (MDK-4154) B1133 10 mg, 50 mg 537034-15-4 Nullscript 2186 1 mg, 5 mg 300816-11-9 GTPase Inhibitors Oxamflatin 2250 1 mg, 5 mg 151720-43-3 Product Name Cat. No. Size CAS. No. Panobinostat (LBH589) 1612 1 mg, 5 mg, 25 mg 404950-80-7 BQU57 9576 5 mg, 25 mg 1637739-82-2 PCI 34051 2251 5 mg, 25 mg 950762-95-5 CID-1067700 2688 5 mg, 25 mg 314042-01-8 PXD101 2480 5 mg, 25 mg 414864-00-9 RBC8 B1136 5 mg, 25 mg 361185-42-4 Pyroxamide 2189 5 mg, 25 mg 382180-17-8 Guanylate Cyclase Inhibitors RGFP966 2818 5 mg, 25 mg 1396841-57-8 Product Name Cat. No. Size CAS. No. SAHA 1604 1 mg, 5 mg 149647-78-9 SB 939 2285 1 mg, 5 mg 929016-96-6 LY-83583 B1314 5 mg, 25 mg 91300-60-6 SBHA 2202 50 mg, 250 mg 38937-66-5 HAT (Histone Acetyltransferase) Inhibitors 4SC-202 B1230 5 mg, 25 mg 1186222-89-8 Product Name Cat. No. Size CAS. No. Scriptaid 1605 1 mg 287383-59-9 Anacardic Acid 1849 5 mg, 25 mg 16611-84-0 Sodium butyrate 1609 1 g 156-54-7 C646, p300/CBP Inhibitor 1948 1 mg, 5 mg 328968-36-1 Sodium 4-phenylbutyrate 1608 100 mg, 1 g 1716-12-7 Curcumin, Curcuma longa (High Purity) 1850 10 mg, 50 mg 458-37-7 Splitomicin 1610 5 mg 5690-03-9 EML-425 B1882 5 mg, 25 mg 1675821-32-5 TC-H 106 B1148 10 mg, 50 mg 937039-45-7

4 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 5 HMG-CoA (3-Hydroxy-3-Methylglutaryl Coenzyme Product Name Cat. No. Size CAS. No. A) Inhibitors TMP-195 B1860 5 mg, 25 mg 1314891-22-9 Product Name Cat. No. Size CAS. No. TMP269 2679 5 mg, 25 mg 1314890-29-3 2278 10 mg, 50 mg 134523-00-5 EZSolution™ Trichostatin A 2271 1 mg 58880-19-6 (R,R)-Hymeglusin B1244 500 µg, 1 mg 29066-42-0 Trichostatin A 1606 1 mg 58880-19-6 1692 50 mg, 250 mg 75330-75-5 Tubacin 1984 250 µg, 1 mg 537049-40-4 1694 50 mg, 250 mg 73573-88-3 Tubastatin A 1724 1 mg, 5 mg 1239262-52-2 EZSolution™ 2806 5 mg 287714-41-4 UF 010 B1146 10 mg, 50 mg 537672-41-6 Rosuvastatin 1955 5 mg, 25 mg 287714-41-4 Valproic Acid, Sodium Salt 1647 200 mg 1069-66-5 1693 50 mg, 250 mg 79902-63-9 Hh (Hedgehog) Signaling Pathway Antagonists Hsp (Heat Shock Protein) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. BMS-833923 9547 5 mg, 25 mg 1059734-66-5 EZSolution™ 17-AAG 9495 1 mg 75747-14-7 BODIPY-Cyclopamine 2160 50 µg, 250 µg 334658-24-1 17-AAG 1774 1 mg, 5 mg 75747-14-7 CUR-61414 2743 5 mg, 25 mg 334998-36-6 17-DMAG hydrochloride 1776 1 mg, 5 mg 467214-21-7 EZSolution™ Cyclopamine 2545 5 mg 4449-51-8 AT-13387 B1961 5 mg, 25 mg 912999-49-6 Cyclopamine 1578 5 mg 4449-51-8 BIIB 021 2291 5 mg, 25 mg 848695-25-0 Cyclopamine tartrate 2518 1 mg, 5 mg 1178510-81-0 CUDC-305 9653 1 mg, 5 mg 1061318-81-7 Cyclopamine-KAAD 1910 50 µg 306387-90-6 Ganetespib (STA-9090) 9459 5 mg, 25 mg 888216-25-9 GANT58 1812 5 mg, 25 mg 64048-12-0 Geldanamycin 1564 1 mg, 5 mg 30562-34-6 GANT61 1892 5 mg 500579-04-4 KRIBB11 B1567 5 mg, 25 mg 342639-96-7 EZSolution™ GDC-0449 2539 5 mg 879085-55-9 Novobiocin Sodium Salt B1526 1 g, 5 g 1476-53-5 GDC-0449 1890 5 mg, 25 mg 879085-55-9 NVP-AUY922 1591 1 mg, 5 mg 747412-49-3 Hh Signaling Pathway Antagonist 1659 1 mg 330796-24-2 PU-H71 (Not Available for Sale in the U.S.) 9649 10 mg, 50 mg 873436-91-0 HPI-1 2410 5 mg, 25 mg 599150-20-6 PU-WS13 9442 5 mg, 25 mg 1454619-14-7 1987 50 mg, 100 mg, 500 mg, 1 g 84625-61-6 Radicicol B1533 1 mg, 5 mg 12772-57-5 Jervine 2357 1 mg, 5 mg 469-59-0 Sulfamethoxazole B1534 5 g, 25 g 723-46-6 JK 184 1726 1 mg 315703-52-7 XL888 2654 1 mg, 5 mg 1149705-71-4 LDE-225 2892 5 mg, 25 mg 956697-53-3 IDO (Indoleamine 2,3-Dioxygenase) Inhibitors LDE-225 diphosphate 2893 5 mg, 25 mg 1218778-77-8 Product Name Cat. No. Size CAS. No. LY-2940680 9604 5 mg, 25 mg 1258861-20-9 BMS-986205 B1839 5 mg, 25 mg 1923833-60-6 MK-4101 B1255 5 mg, 25 mg 935273-79-3 IDO Pathway inhibitor 2746 50 mg, 250 mg 110117-83-4 Robotnikinin 1923 1 mg 1132653-79-2 IDO1 Inhibitor I 2745 5 mg, 25 mg 914471-09-3 SANT-1 1978 1 mg, 5 mg 304909-07-7 INCB-024360 9477 5 mg, 25 mg 1204669-58-8 SANT-2 1976 1 mg, 5 mg 329196-48-7 Menadione 2747 500 mg, 1 g 58-27-5 Smo Antagonist, SA1 2154 2 mg, 5 mg N/A NLG919 9407 5 mg, 25 mg 1402836-58-1 Smo Antagonist, SA10 2159 2 mg, 5 mg N/A Smo Antagonist, SA9 2155 2 mg, 5 mg N/A KMO (Kynurenine 3-Monoxygenase) Inhibitors Tomatidine hydrochloride 1893 25 mg 6192-62-7 Product Name Cat. No. Size CAS. No. HIF (Hypoxia-Inducible Factor) Inhibitors JM6 1913 5 mg, 25 mg 1008119-83-2 Product Name Cat. No. Size CAS. No. Ro 61-8048 1912 5 mg, 25 mg 199666-03-0 BAY 87-2243 B1878 5 mg, 25 mg 1227158-85-1 LDH (Lactate Dehydrogenase) Inhibitors Chetomin 2180 1 mg 1403-36-7 Product Name Cat. No. Size CAS. No. Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7 Galloflavin 2672 5 mg, 25 mg 568-80-9 KC7F2 9641 10 mg, 50 mg 927822-86-4 (±)-Gossypol 2579 50 mg, 250 mg 303-45-7 PT-2385 B1920 5 mg, 25 mg 1672665-49-4 Sodium Oxamate 2580 1 g, 5 g 565-73-1 PX 12 2217 5 mg, 25 mg 141400-58-0 PX-478 hydrochloride B1033 5 mg, 25 mg 685898-44-6 Lipase Inhibitors HIF-PH (Hypoxia-Inducible Factor Prolyl Product Name Cat. No. Size CAS. No. Hydroxylase) Inhibitors Orlistat B1020 50 mg, 250 mg 96829-58-2 XEN445 2681 5 mg, 25 mg 1515856-92-4 Product Name Cat. No. Size CAS. No. BAY 85-3934 9597 5 mg, 25 mg 1154028-82-6 LO (Lipoxygenase) Inhibitors DMOG 2216 5 mg, 25 mg 89464-63-1 Product Name Cat. No. Size CAS. No. FG-4592 9681 5 mg, 25 mg 808118-40-3 NDGA 2581 100 mg, 500 mg 500-38-9 GSK1278863 B1107 1 mg, 5 mg 960539-70-2 MAO (Monoamine oxidase) Inhibitors IOX2 9451 5 mg, 25 mg 931398-72-0 Product Name Cat. No. Size CAS. No. JNJ-42041935 B1072 5 mg, 25 mg 1193383-09-3 Clorgyline hydrochloride 2622 10 mg, 50 mg 17780-75-5 HIV Integrase Inhibitors Harmine 2561 50 mg, 250 mg 442-51-3 Product Name Cat. No. Size CAS. No. Moclobemide 9561 10 mg, 50 mg 71320-77-9 Elvitegravir 9465 5 mg, 25 mg 697761-98-1 Pargyline hydrochloride 2618 500 mg, 1 g 306-07-0 GSK1349572 2288 5 mg, 25 mg 1051375-16-6 Rasagiline mesylate 2237 50 mg, 250 mg 161735-79-1

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 6 MDM2 (Murine Double Minute 2) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. AMG-232 9556 1 mg, 5 mg 1352066-68-2 LLY-507 B1111 1 mg, 5 mg 1793053-37-8 CGM097 B1820 1 mg, 5 mg 1313363-54-0 Lomeguatrib 2224 5 mg, 25 mg 192441-08-0 JNJ-26854165 2479 5 mg, 25 mg 881202-45-5 MAK-683 B1972 5 mg, 25 mg 1951408-58-4 MI-773 9610 1 mg, 5 mg 1303607-60-4 MI-2 B1835 5 mg, 25 mg 1271738-62-5 MX69 B1568 5 mg, 25 mg 1005264-47-0 MI-3 B1834 5 mg, 25 mg 1271738-59-0 Nutlin-3 1842 1 mg, 5 mg 548472-68-0 Nanaomycin A 2790 1 mg, 5 mg 52934-83-5 Nutlin-3b B1227 1 mg, 5 mg 675576-97-3 OICR-9429 B1256 5 mg, 25 mg 1801787-56-3 EZSolution™ RG7388 B1504 1 mg 1229705-06-9 PFI-2 B1259 5 mg, 25 mg 1627676-59-8 RG7388 2577 1 mg, 5 mg 1229705-06-9 RG 108 1679 10 mg, 30 mg 48208-26-0 RO8994 B1830 5 mg, 25 mg 1309684-94-3 Ryuvidine B1808 1 mg, 5 mg 265312-55-8 YH239-EE B1229 5 mg, 25 mg 1364488-67-4 SGC0946 2448 5 mg, 25 mg 1561178-17-3 MDR (Multidrug Resistance) Inhibitors SGI-1027 2726 5 mg, 25 mg 1020149-73-8 TC-E 5003 B1177 10 mg, 50 mg 17328-16-4 Product Name Cat. No. Size CAS. No. UNC0379 9588 5 mg, 25 mg 1620401-82-2 Elacridar 2792 5 mg, 25 mg 143664-11-3 UNC0631 2605 5 mg, 25 mg 1320288-19-4 HM-30181 B1285 5 mg, 25 mg 849675-66-7 UNC0638 1933 1 mg, 5 mg 1255580-76-7 KS-176 B1272 5 mg, 25 mg 1253452-78-6 UNC0642 2862 5 mg, 25 mg 1481677-78-4 MK-571 2691 5 mg, 25 mg 115104-28-4 UNC0646 2606 5 mg, 25 mg 1320288-17-2 MK-571 sodium 2692 5 mg, 25 mg 115103-85-0 UNC1999 2449 5 mg, 25 mg 1431612-23-5 NSC-23925 2686 5 mg, 25 mg 858474-14-3 WDR5 0103 B1125 10 mg, 50 mg 890190-22-4 Tariquidar 2853 10 mg, 50 mg 206873-63-4 Zebularine 2225 1 mg, 5 mg 3690-10-6 Verapamil hydrochloride 2861 1 g, 5 g 152-11-4 Zosuquidar trihydrochloride 9488 5 mg, 25 mg 167465-36-3 Microtubule Inhibitors Methyltransferase Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. ABT751 2836 5 mg, 25 mg 141430-65-1 Colchicine 1519 1 g 64-86-8 A-366 2859 1 mg, 5 mg 1527503-11-2 Combretastatin A4 2239 10 mg, 50 mg 117048-59-6 AMI-1 1943 5 mg, 25 mg 20324-87-2 CW069 9507 10 mg, 50 mg 1594094-64-0 AMI-5 2300 50 mg, 250 mg 17372-87-1 Cytochalasin D B1176 1 mg, 5 mg 22144-77-0 5-Aza-2'-deoxycytidine 1754 10 mg, 50 mg 2353-33-5 D-64131 B1066 10 mg, 50 mg 74588-78-6 AZ-505 ditrifluoroacetate B1883 1 mg, 5 mg 1035227-44-1 2232 10 mg, 50 mg 114977-28-5 EZSolution™ BIX 01294 2661 5 mg 935693-62-2 ELR-510444 9433 5 mg, 25 mg 1233948-35-0 BIX 01294 1678 5 mg, 25 mg 935693-62-2 Epothilone B 2012 1 mg, 5 mg 152044-54-7 BRD4770 9525 5 mg, 25 mg 1374601-40-7 Epothilone D 9559 1 mg, 5 mg 189453-10-9 Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4 Maytansinol B2015 5 mg, 25 mg 57103-68-1 C7280948 B1153 10 mg, 50 mg 587850-67-7 EZSolution™ Nocodazole B1874 5 mg 31430-18-9 Chaetocin 2283 500 µg 28097-03-2 Nocodazole 2185 10 mg, 50 mg 31430-18-9 EZSolution™ 3-Deazaneplanocin A 2409 1 mg 102052-95-9 1567 25 mg 33069-62-4 3-Deazaneplanocin A 2060 250 µg, 1 mg 102052-95-9 518-28-5, Podophyllotoxin 2767 50 mg, 250 mg 3-Deazaneplanocin A hydrochloride 2444 250 µg, 1 mg 120964-45-6 4354-76-1 2'-Deoxy-5-fluorocytidine 2387 50 mg, 250 mg 10356-76-0 Pseudolaric Acid B 2512 1 mg, 5 mg 82508-31-4 5’-Deoxy-5’-methylthioadenosine BA1053 10 mg, 50 mg 2457-80-9 Thiocolchicine 2213 5 mg, 25 mg 2730-71-4 DNA methylation inhibitor, Dichlone 2860 500 mg, 1 g 117-80-6 Vinblastine Sulfate 1959 5 mg, 25 mg 143-67-9 EED-226 B1845 5 mg, 25 mg 2083627-02-3 Vinorelbine Tartrate 1957 5 mg, 25 mg 125317-39-7 Ellagic Acid B1154 100 mg, 500 mg 476-66-4 EPZ004777 2381 1 mg, 5 mg 1338466-77-5 MIF (Migration Inhibitory Factor) Antagonists EZSolution™ EPZ005687 2375 2 mg 1396772-26-1 Product Name Cat. No. Size CAS. No. EPZ011989 B1221 5 mg, 25 mg 1598383-40-4 MIF-Antagonist, ISO-1 1895 5 mg 478336-92-4 EPZ-015666 9410 1 mg, 5 mg 1616391-65-1 MIF antagonist, p425 2158 1 g 2610-05-1 EPZ015866 (GSK591) B1216 5 mg, 25 mg 1616391-87-7 EZSolution™ EPZ-5676 2427 1 mg 1380288-87-8 Mitochondrial Division Inhibitors EPZ-5676 2382 1 mg, 5 mg 1380288-87-8 Product Name Cat. No. Size CAS. No. EZSolution™ EPZ-6438 2428 5 mg 1403254-99-8 Mdivi -1 2441 5 mg, 25 mg 338967-87-6 EPZ-6438 2383 5 mg, 25 mg 1403254-99-8 EZH2 Inhibitor, EPZ005687 2364 2 mg, 10 mg 1396772-26-1 Mitochondrial Electron Transport Chain EZSolution™ GSK126 2366 1 mg 1346574-57-9 Inhibitors GSK126 2282 1 mg, 5 mg 1346574-57-9 Product Name Cat. No. Size CAS. No. EZSolution™ GSK343 2365 1 mg N/A Antimycin A 2247 10 mg, 50 mg 1397-94-0 GSK343 2281 1 mg, 5 mg 1346704-33-3 Atpenin A5 (Synthetic) 2210 250 µg, 1 mg 119509-24-9 GSK-503 9538 5 mg, 25 mg 1346572-63-1 Cyantraniliprole B1648 5 mg, 25 mg 736994-63-1 HLCL-61 hydrochloride B1209 5 mg, 25 mg 586395-74-6 Phenformin hydrochloride 1889 100 mg, 1 g 834-28-6 EZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4 Rotenone 2248 250 mg, 1 g 83-79-4

6 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 7 MMP (Matrix Metalloproteinase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Atpenin A5 (Synthetic) 2210 250 µg 119509-24-9 MRT67307 B1604 5 mg, 25 mg 1190378-57-4 EZSolution™ Batimastat 2540 1 mg 130370-60-4 NF-κB Inhibitor, SN50 2506 500 µg, 1 mg 213546-53-3 Batimastat (MMP Inhibitor) 1704 1 mg, 5 mg 130370-60-4 Parthenolide 1868 10 mg, 50 mg 20554-84-1 Disulfiram 2308 50 mg, 250 mg 97-77-8 PDTC 1676 100 mg 5108-96-3 Doxycycline hyclate 2209 100 mg, 500 mg 24390-14-5 PS-1145 9671 5 mg, 25 mg 431898-65-6 GM 6001 1799 1 mg 142880-36-2 Rocaglamide 1863 100 µg 84573-16-0 Marimastat 1790 1 mg, 5 mg 154039-60-8 Sauchinone 2312 1 mg, 5 mg 177931-17-8 Minocycline Hydrochloride B1525 50 mg, 250 mg 13614-98-7 SC-514 2442 5 mg, 25 mg 354812-17-2 MMP-13 inhibitor 2392 5 mg, 25 mg 307002-71-7 STO-609 B1609 5 mg, 25 mg 52029-86-4 MMP-9 Inhibitor 1981 500 µg 1177749-58-4 TPCA-1 2431 5 mg, 25 mg 507475-17-4 MMP-III Inhibitor, NNGH 2569 5 mg, 25 mg 161314-17-6 Triptolide 1761 1 mg, 5 mg 38748-32-2 NSC 405020 2682 5 mg, 25 mg 7497-07-6 NLRP3 (NOD-Like Receptor Pyrin domain- TAPI-0 2067 1 mg 143457-40-3 containing protein 3) Inflammasome Inhibitors EZSolution™ TAPI-1 2537 1 mg 171235-71-5 TAPI-1 2068 1 mg 171235-71-5 Product Name Cat. No. Size CAS. No. TAPI-2 2069 1 mg 187034-31-7 Arglabin 9691 1 mg, 5 mg 84692-91-1 WAY-170523 9607 1 mg, 5 mg 307002-73-9 Isoliquiritigenin 2528 5 mg, 25 mg 961-29-5 MCC950 (Free base) B1031 1 mg, 5 mg 210826-40-7 MPO (Myeloperoxidase) Inhibitors MCC950 sodium 9686 1 mg, 5 mg 256373-96-3 Product Name Cat. No. Size CAS. No. Myeloperoxidase Inhibitor 1977 100 mg, 500 mg 5351-17-7 NOS (Nitric Oxide Synthase) Inhibitors NAALADase (N-Acetylated-Alpha-Linked-Acidic Product Name Cat. No. Size CAS. No. Bakuchiol 2494 1 mg, 5 mg 10309-37-2 Dipeptidase) Inhibitors Bardoxolone B1170 5 mg, 25 mg 218600-44-3 Product Name Cat. No. Size CAS. No. 3-Bromo-7-nitroindazole 2361 10 mg, 50 mg 74209-34-0 NAALDase Inhibitor, PMPA 2478 5 mg, 25 mg 173039-10-6 Curvularin 9694 1 mg, 5 mg 10140-70-2 Nampt (Nicotinamide Phosphoribosyltransferase) Diphenyleneiodonium chloride 2358 5 mg 4673-26-1 L-NAME hydrochloride 2356 100 mg, 500 mg, 1 g 51298-62-5 Inhibitors L-NMMA acetate 2348 5 mg, 25 mg, 100 mg 53308-83-1 Product Name Cat. No. Size CAS. No. 7-Nitroindazole 2360 50 mg, 250 mg 2942-42-9 CHS-828 2044 5 mg, 25 mg 200484-11-3 1400W dihydrochloride 2055 5 mg, 25 mg 214358-33-5 FK-866 1914 1 mg, 5 mg 658084-64-1 Nampt-IN-1 B1171 5 mg, 25 mg 1698878-14-6 Nuclear Export Inhibitors STF-118804 9552 5 mg, 25 mg 894187-61-2 Product Name Cat. No. Size CAS. No. STF-31 9585 5 mg, 25 mg 724741-75-7 EZSolution™ Leptomycin B 1814 25 µg 87081-35-4 Necroptosis and Necrosis Inhibitors PAD (Protein Arginine Deiminase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. EZSolution™ Nec-1s 2535 1 mg N/A GSK-106 hydrochloride B1036 500 µg, 1 mg 1652591-82-6 Nec-1s 2263 1 mg, 5 mg 852391-15-2 GSK-121 trifluoroacetate B1034 500 µg, 1 mg 1652591-80-4 Necrosis Inhibitor, Necrox-2 2228 1 mg, 5 mg N/A GSK-199 hydrochloride B1037 500 µg, 1 mg 1549811-53-1 Necrosis Inhibitor, Necrox-5 2229 1 mg, 5 mg 1383718-29-3 GSK-484 hydrochloride B1035 500 µg, 1 mg 1652591-81-5 Necrostatin-1 1864 5 mg, 25 mg 4311-88-0 PCSK9 (Proprotein Convertase Subtilisin Kexin 9) Necrostatin-5 1865 5 mg, 25 mg 337349-54-9 Inhibitors Necrostatin-7 1866 5 mg, 25 mg 351062-08-3 EZSolution™ Necrosulfonamide, Sterile- Product Name Cat. No. Size CAS. No. B1220 10 mg 1360614-48-7 Filtered SBC-110736 B1304 5 mg, 25 mg 1629166-02-4 Necrosulfonamide 9635 10 mg, 50 mg 1360614-48-7 PDE (Phosphodiesterase) Inhibitors NF-KB (Nuclear Factor-kappa B) Pathway Product Name Cat. No. Size CAS. No. Inhibitors 2352 5 mg, 25 mg 608141-41-9 Product Name Cat. No. Size CAS. No. 2560 5 mg, 25 mg 68550-75-4 Andrographolide 2389 50 mg, 250 mg 5508-58-7 2393 5 mg, 25 mg 73963-72-1 BAY 11-7082 1867 10 mg, 50 mg 19542-67-7 EHNA hydrochloride 2265 5 mg, 25 mg 58337-38-5 Berbamine dihydrochloride 2520 100 mg, 500 mg 6078-17-7 GSK-356278 B1292 5 mg, 25 mg 720704-34-7 BMS-345541 (Free base) B1907 1 mg, 5 mg 445430-58-0 IBMX 1714 100 mg 28822-58-4 Celastrol 1940 5 mg, 25 mg 34157-83-0 B1327 5 mg, 25 mg 50847-11-5 CHS-828 2044 5 mg, 25 mg 200484-11-3 2163 5 mg, 25 mg 78415-72-2 Dimethyl Fumarate 9660 100 mg, 500 mg 624-49-7 PF-04447943 B1264 5 mg, 25 mg 1082744-20-4 Honokiol 1762 10 mg, 50 mg 35354-74-6 9676 50 mg, 250 mg 74150-27-9 4'-Hydroxychalcone B1921 250 mg, 1 g 2657-25-2 RO 20-1724 2042 50 mg, 250 mg 29925-17-5 IKK16 B1087 5 mg, 25 mg 1186195-62-9 2675 10 mg, 50 mg 162401-32-3 ML130 1974 5 mg, 25 mg 799264-47-4 (R,S)- 2010 5 mg 61413-54-5 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 8 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. citrate 2872 10 mg, 50 mg 171599-83-0 Pifithrin-α, Cyclic, hydrobromide 2270 5 mg 511296-88-1 TAK-063 B1067 10 mg, 50 mg 1238697-26-1 Pifithrin-α 1554 10 mg 63208-82-2 Vesnarinone B2008 5 mg, 25 mg 81840-15-5 1715 25 mg 37762-06-4 Poly (ADP-ribose) Polymerase (PARP) Inhibitors Product Name Cat. No. Size CAS. No. 15-PGDH (15-hydroxy Prostaglandin ABT-888 1620 1 mg, 5 mg 912445-05-7 Dehydrogenase) Inhibitors AG-014699 phosphate 2890 1 mg, 5 mg 459868-92-9 Product Name Cat. No. Size CAS. No. BMN-673 B1861 1 mg, 5 mg 1207456-01-6 β-Glycyrrhetinic acid 9586 1 g 471-53-4 EZSolution™ DPQ 2866 5 mg 129075-73-6 SW-033291 9584 5 mg, 25 mg 459147-39-8 DPQ 1899 1 mg, 5 mg 129075-73-6 DR2313 1771 1 mg, 5 mg 284028-90-6 Phosphatase Inhibitors Iniparib 1968 5 mg, 25 mg 160003-66-7 Product Name Cat. No. Size CAS. No. 1,5-Isoquinolinediol 2415 10 mg, 50 mg 5154-02-9 Bakuchiol 2494 1 mg, 5 mg 10309-37-2 ME-0328 2751 5 mg, 25 mg 1445251-22-8 bpV(phen) 1793 5 mg 42494-73-5 MK-4827 9462 5 mg, 25 mg 1038915-60-4 bpV(pic) 1794 5 mg 148556-27-8 MK-4827 (Tosylate) B2003 5 mg, 25 mg 1038915-73-9 BVT948 B1810 1 mg, 5 mg 39674-97-0 NU 1025 2351 1 mg, 5 mg 90417-38-2 Calyculin A 1562 25 µg 101932-71-2 Olaparib 1952 5 mg, 25 mg 763113-22-0 Cantharidin 2510 10 mg, 50 mg 56-25-7 Phenformin hydrochloride 1889 100 mg, 1 g 834-28-6 Cyclosporine A 1522 100 mg, 1 g 59865-13-3 PJ-34 hydrochloride 2319 1 mg, 5 mg 344458-15-7 Cytostatin sodium B1240 250 µg 457070-06-3 FK-506 1563 1 mg, 10 mg 104987-11-3 PPAR (Peroxisome Proliferator-Activated Fostriecin sodium B1241 10 µg 87860-39-7 Receptor) Antagonists GSK2830371 2578 1 mg, 5 mg 1404456-53-6 Product Name Cat. No. Size CAS. No. IQ-1 1663 1 mg 331001-62-8 Astaxanthin 9698 5 mg, 25 mg 472-61-7 Microcystin-LR 1840 100 µg, 500 µg 101043-37-2 GSK-0660 2897 5 mg, 25 mg 1014691-61-2 Nodularin 2094 50 µg 118399-22-7 GSK-3787 2400 5 mg, 25 mg 188591-46-0 NSC-663284 B1809 1 mg, 5 mg 383907-43-5 GW 9662 1697 5 mg 22978-25-2 NSC-87877 2687 10 mg, 50 mg 56990-57-9 GW-6471 9453 1 mg, 5 mg 880635-03-0 Okadaic acid 1543 25 µg, 100 µg 78111-17-8 EZSolution™ GW 9662 9651 5 mg 22978-25-2 Okadaic acid, Ammonium Salt 1766 25 µg, 100 µg 155716-06-6 PPARγ Antagonist, G3335 1979 10 mg, 25 mg 36099-95-3 Okadaic acid, Potassium Salt 1765 25 µg, 100 µg 155751-72-7 SR1664 9432 1 mg, 5 mg 1338259-05-4 Okadaic acid, Sodium Salt 1764 25 µg, 100 µg 209266-80-8 T0070907 2095 5 mg 313516-66-4 (-)-p-Bromotetramisole oxalate 1901 5 mg, 25 mg 62284-79-1 EZBlock™ Phosphatase Inhibitor Cocktail PPI (Protein-Protein Interaction) Inhibitors K273 1 ml, Set (5 x 1 ml) N/A I (50X) Product Name Cat. No. Size CAS. No. EZBlock™ Phosphatase Inhibitor Cocktail II K275 1 ml, Set (5 x 1 ml) N/A ABT-263 2467 5 mg, 25 mg 923564-51-6 EZBlock™ Phosphatase Inhibitor Cocktail K276 1 ml, Set (5 x 1 ml) N/A III AT-406 B1829 5 mg, 25 mg 1071992-99-8 EZBlock™ Phosphatase Inhibitor Cocktail K282 1 ml, Set (5 x 1 ml) N/A BCl-2 Inhibitor, ABT-199 2253 1 mg, 5 mg 1257044-40-8 IV Birinapant 2597 1 mg, 5 mg 1260251-31-7 EZBlock™ Phosphatase Inhibitor Cocktail K298 1 vial, Set (5 x 1 vial) N/A XI Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4 PRL-3 Inhibitor B1825 5 mg, 25 mg 893449-38-2 CPI-203 9404 1 mg, 5 mg 1446144-04-2 Rubratoxin A B1239 250 µg , 500 µg 22467-31-8 GDC-0152 B1602 5 mg, 25 mg 873652-48-3 SHP099 hydrochloride B1308 5 mg, 25 mg 1801747-11-4 GDC-0917 B1918 1 mg, 5 mg 1446182-94-0 Sodium orthovanadate 9470 1 g, 5 g 13721-39-6 I-BET151 2220 1 mg, 5 mg 1300031-49-5 Sodium orthovanadate, Activated 9471 5 ml 13721-39-6 I-BET726 B1569 5 mg, 25 mg 1300031-52-0 Tautomycin B1237 10 µg, 50 µg 109946-35-2 I-BET762 2628 1 mg, 5 mg 1260907-17-2 EZBlock™ Universal Protease and \ K283 2 vials, 10 vials N/A EZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4 Phosphatase Inhibitor Cocktail EZBlock™ Universal Protease and (-)-JQ1 2384 1 mg 1268524-71-5 K284 1 ml, Set (5 x 1 ml) N/A Phosphatase Inhibitor Cocktail , EDTA-Free LCL161 B1601 5 mg, 25 mg 1005342-46-0 Phospholipase Inhibitors Lifitegrast B1917 5 mg, 25 mg 1025967-78-5 MS436 2680 5 mg, 25 mg 1395084-25-9 Product Name Cat. No. Size CAS. No. OTX015 2651 1 mg, 5 mg 202590-98-5 Darapladib B1265 5 mg, 25 mg 356057-34-6 PFI-1 2203 1 mg, 5 mg 1403764-72-6 FIPI 9593 5 mg, 25 mg 939055-18-2 RG-7112 B1919 1 mg, 5 mg 939981-39-2 LY315920 2666 1 mg, 5 mg 172732-68-2 EZSolution™ RG7388 B1504 1 mg 1229705-06-9 U-73122 B1887 5 mg, 25 mg 112648-68-7 RG7388 2577 1 mg, 5 mg 1229705-06-9 U-73343 B1888 5 mg, 25 mg 142878-12-4 RVX-208 9408 1 mg, 5 mg 1044870-39-4 p53 Inhibitors Protease Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. NSC 66811 2009 5 mg 6964-62-1 Abametapir 9665 100 mg, 500 mg 1762-34-1

8 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 9 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. AEBSF.HCl 1644 200 mg, 1 g 30827-99-7 (-)-Epigallocatechin gallate 1841 50 mg 989-51-5 Alvelestat B1653 5 mg, 25 mg 848141-11-7 Epoxomicin 2190 50 µg, 250 µg 134381-21-8 Antipain dihydrochloride 2834 5 mg, 25 mg 37682-72-7 2157 100 mg, 500 mg 43210-67-9 Aprotinin 4690 5 mg, 100 mg, 1 g 9087-70-1 Lactacystin (Natural) 2434 200 µg 133343-34-7 Argatroban 9670 10 mg, 50 mg 141396-28-3 Lactacystin (Synthetic) 1709 200 µg 133343-34-7 Batimastat (MMP Inhibitor) 1704 1 mg, 5 mg 130370-60-4 EZSolution™ MG-115 2144 1 mg N/A Bestatin 1733 25 mg, 100 mg 58970-76-6 MG-115 1831 1 mg, 5 mg N/A Bestatin hydrochloride 9630 5 mg, 25 mg 65391-42-6 EZSolution™ MG-132 1791 5 mg 133407-82-6 Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5 MG-132 1703 5 mg, 25 mg 133407-82-6 E-64 1739 5 mg, 25 mg 66701-25-5 ONX-0914 2555 5 mg, 25 mg 960374-59-8 Elastase Inhibitor 1922 5 mg 111682-13-4 Oprozomib 2386 5 mg, 25 mg 935888-69-0 Elastase Inhibitor, SPCK 1921 5 mg 65144-34-5 P5091 2277 5 mg, 25 mg 882257-11-6 Elastatinal 9629 5 mg, 25 mg 51798-45-9 EZSolution™ PS-341 2145 1 mg 179324-69-7 Enfuvirtide Acetate 2440 1 mg 914454-00-5 PS-341 1846 1 mg, 5 mg 179324-69-7 GGACK Dihydrochloride 1847 5 mg N/A VR23 B1515 5 mg, 25 mg 1624602-30-7 Lactacystin (Synthetic) 1709 200 µg 133343-34-7 Leupeptin, hemisulfate (Microbial) 1648 25 mg, 50 mg, 100 mg 103476-89-7 Protein Kinase Inhibitors Lopinavir 2241 50 mg, 250 mg 192725-17-0 Akt (thymoma viral proto-oncogene 1) Inhibitors EZSolution™ MG-132 1791 5 mg 133407-82-6 Product Name Cat. No. Size CAS. No. MG-132 1703 5 mg, 25 mg 133407-82-6 Afuresertib hydrochloride B1848 5 mg, 25 mg 1047645-82-8 Nafamostat Mesylate 1760 10 mg, 50 mg 82956-11-4 Akt Inhibitor (10-NCP) 2338 1 mg, 5 mg 925681-41-0 Pepstatin A 1732 25 mg, 100 mg 26305-03-3 Akt Inhibitor, Isozyme-Selective 1708 1 mg 612847-09-3 PMSF 1548 5 g, 25 g 329-98-6 Akt-I-1 B1610 1 mg, 5 mg 473382-39-7 PPACK Dihydrochloride 1848 5 mg N/A Cordycepin 2078 10 mg, 50 mg 73-03-0 EZBlock™ Protease Inhibitor Cocktail, GDC-0068 2667 1 mg, 5 mg 1001264-89-6 K272 1 ml, 5 ml, Set (5 x 1 ml) N/A EDTA-Free GSK-2110183 B1089 1 mg, 5 mg 1047644-62-1 EZBlock™ Protease Inhibitor Cocktail II K277 Set (5 x 1 vial) N/A GSK-690693 2272 5 mg, 25 mg 937174-76-0 EZBlock™ Protease Inhibitor Cocktail II, K394 1 vial, Set (5 x 1 vial) N/A Animal-Free Miransertib B1931 5 mg, 25 mg 1313881-70-7 Set (1 vial of lyophilized cocktail MK-2206 1888 500 µg, 1 mg 1032350-13-2 EZBlock™ Protease Inhibitor Cocktail III K278 N/A + 1 ml DMSO) Perifosine (KRX-0401) 1592 5 mg, 25 mg 157716-52-4 EZBlock™ Protease Inhibitor Cocktail IV K279 1 ml, Set (5 x 1 ml) N/A 371242-69-2 EZBlock™ Protease Inhibitor Cocktail IX K294 1 ml, Set (5 x 1 ml) N/A DiscoveryPak™ PI 3-Kinase Inhibitor Set 154447-36-6 EZBlock™ Protease Inhibitor Cocktail V, (Containing Cat. No. 1661, 1667, 1728, K856 5 Inhibitors 371935-74-9 K290 1 vial, Set (5 x 1 vial) N/A EDTA-Free 1780, 1781) 648450-29-7 EZBlock™ Protease Inhibitor Cocktail VI, 663619-89-4 K291 1 vial, Set (5 x 1 vial) N/A General Use PHT-427 2465 10 mg, 50 mg 1191951-57-1 EZBlock™ Protease Inhibitor Cocktail VII K292 1 ml, Set (5 x 1 ml) N/A SC66 1870 10 mg, 50 mg 871361-88-5 EZBlock™ Protease Inhibitor Cocktail VIII K293 1 ml, Set (5 x 1 ml) N/A SH-5 1818 500 µg 701976-54-7 EZBlock™ Protease Inhibitor Cocktail VIII, K395 1 vial, Set (5 x 1 vial) N/A SH-6 1819 500 µg 701976-54-7 DMSO-Free Triciribine 1707 1 mg 35943-35-2 EZBlock™ Protease Inhibitor Cocktail X, K297 1 vial, Set (5 x 1 vial) N/A EDTA-Free EZBlock™ Protease Inhibitor Cocktail XII, ALK (Anaplastic Lymphoma Kinase) Inhibitors K221 1 vial, Set (5 x 1 vial) N/A EDTA-free, Animal-free Product Name Cat. No. Size CAS. No. EZBlock™ Protease Inhibitor Cocktail XIII, K222 1 vial, Set (5 x 1 vial) N/A EZSolution™ A83-01, Sterile-Filtered 1989 1 ml 909910-43-6 EDTA & Animal-Free A 83-01 1725 1 mg 909910-43-6 EZBlock™ Protease Inhibitor Cocktail XIV K223 1 vial, Set (5 x 1 vial) N/A ASP-3026 B1296 5 mg, 25 mg 1097917-15-1 EZBlock™ Protease Inhibitor Cocktail XV K393 1 vial, Set (5 x 1 vial) N/A AZD-3463 2371 5 mg, 25 mg 1356962-20-3 Protease Inhibitor Cocktail K271 1 Kit N/A Belizatinib (TSR-011) B2028 5 mg, 25 mg 1357920-84-3 Simeprevir B1173 5 mg, 25 mg 923604-59-5 EZBlock™ Universal Protease and (AP26113) 9675 5 mg, 25 mg 1197953-54-0 K283 2 vials, 10 vials N/A Phosphatase Inhibitor Cocktail Brigatinib analog B2025 5 mg, 25 mg 1197958-12-5 EZBlock™ Universal Protease and K284 1 ml, Set (5 x 1 ml) N/A CH5424802 2867 5 mg, 25 mg 1256580-46-7 Phosphatase Inhibitor Cocktail , EDTA-Free Vicriviroc Malate 1599 1 mg, 5 mg 541503-81-5 1934 5 mg, 25 mg 877399-52-5 Ensartinib B1946 5 mg, 25 mg 1365267-27-1 Proteasome Inhibitors B1324 5 mg, 25 mg 1108743-60-7 Product Name Cat. No. Size CAS. No. GSK-1838705A B2026 1 mg, 5 mg 1116235-97-2 Aclacinomycin A hydrochloride B1905 1 mg, 5 mg 75443-99-1 LDK-378 B1928 5 mg, 25 mg 1032900-25-6 Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1 NVP-TAE684 1683 5 mg 761439-42-3 Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1 PF-06463922 B1169 10 mg, 50 mg 1454846-35-5 Carfilzomib 2385 5 mg, 25 mg 868540-17-4 SU-5416 9491 5 mg, 25 mg 204005-46-9 Celastrol 1940 5 mg, 25 mg 34157-83-0 TPX-0005 B2027 5 mg, 25 mg 2058227-19-1 CEP-18770 2433 5 mg, 25 mg 847499-27-8 AMPK (AMP-activated protein Kinase) Inhibitors Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5 Product Name Cat. No. Size CAS. No. Clioquinol 2454 1 g, 5 g 130-26-7 EZSolution™ Dorsomorphin 2547 5 mg 866405-64-3

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 10 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Dorsmorphin dihydrochloride 2835 5 mg, 25 mg 1219168-18-9 ONO-4059 analog B1897 5 mg, 25 mg 1351635-67-0 Dorsomorphin 1686 5 mg 866405-64-3 RN486 9678 1 mg, 5 mg 1242156-23-5 ATM (Ataxia Telangiectasia Mutated ) Kinase Inhibitors TP-0903 9590 5 mg, 25 mg 1341200-45-0 2+ Product Name Cat. No. Size CAS. No. CaM (Ca /calmodulin-dependent) Kinase Inhibitors ATM Kinase Inhibitor, KU-55933 1685 5 mg 587871-26-9 Product Name Cat. No. Size CAS. No. AZD-0156 B1305 5 mg, 25 mg 1821428-35-6 Berbamine dihydrochloride 2520 100 mg, 500 mg 6078-17-7 Ku-60019 9572 5 mg, 25 mg 925701-49-1 2013 500 µg, 1 mg 99533-80-9 ATR (Ataxia Telangiectasia & Rad3-related) Inhibitors KN-62 2495 1 mg, 5 mg 127191-97-3 KN-92 hydrochloride B1643 5 mg, 25 mg 1431698-47-3 Product Name Cat. No. Size CAS. No. KN-92 phosphate B1644 5 mg, 25 mg 1135280-28-2 AZ20 B1724 1 mg, 5 mg 1233339-22-4 KN-93 2524 250 µg, 1 mg 139298-40-1 AZD-6738 B1167 5 mg, 25 mg 1352226-88-0 KN-93, Water-Soluble 1909 1 mg, 5 mg 1188890-41-6 BAY-1895344 hydrochloride B1962 5 mg, 25 mg 1876467-74-1 STO-609 B1609 5 mg, 25 mg 52029-86-4 CGK733 B1725 5 mg, 25 mg 905973-89-9 ETP-46464 2457 5 mg, 25 mg 1345675-02-6 CDC7 (Cell Division Cycle 7 Homolog) Inhibitors VE-821 B1723 5 mg, 25 mg 1232410-49-9 Product Name Cat. No. Size CAS. No. VE-822 2840 5 mg, 25 mg 1232416-25-9 BMS-863233 hydrochloride 2598 5 mg, 25 mg 1169562-71-3 PHA-767491(HCl) B1639 5 mg, 25 mg 845714-00-3 Aurora Kinase Inhibitors Product Name Cat. No. Size CAS. No. CDK (Cyclin-Dependent Kinases) Inhibitors 656820-32-5 B1638 5 mg, 25 mg 160098-96-4 Product Name Cat. No. Size CAS. No. AMG-900 B1343 5 mg, 25 mg 945595-80-2 Alsterpaullone 1897 1 mg, 5 mg 237430-03-4 AT9283 2432 5 mg, 25 mg 896466-04-9 AMG-925 B1959 5 mg, 25 mg 1401033-86-0 Aurora Kinase B Inhibitor (AZD1152-HQPA) 1583 5 mg, 25 mg 722544-51-6 Aminopurvalanol A 2205 1 mg, 5 mg 220792-57-4 CCT-129202 B1934 1 mg, 5 mg 942947-93-5 AT-7519 hydrochloride 2816 5 mg, 25 mg 902135-91-5 CCT-137690 B195 5 mg, 25 mg 1095382-05-0 Bohemine B1040 10 mg, 50 mg 189232-42-6 CYC-116 B1936 5 mg, 25 mg 693228-63-6 Butyrolactone I 1690 200 µg 87414-49-1 Danusertib B1937 5 mg, 25 mg 827318-97-8 CVT-313 B1137 5 mg, 25 mg 199986-75-9 ENMD-2076 B1938 5 mg, 25 mg 934353-76-1 Dinaciclib 9537 5 mg, 25 mg 779353-01-4 GSK-1070916 B1939 5 mg, 25 mg 942918-07-2 Flavopiridol 2090 1 mg, 5 mg 146426-40-6 Hesperadin B1940 5 mg, 25 mg 422513-13-1 Kenpaullone 1904 1 mg 142273-20-9 JNJ-7706621 B1941 1 mg, 5 mg 443797-96-4 LY-2835219 B1039 10 mg, 50 mg 1231930-82-7 MK-5108 B1344 5 mg, 25 mg 1010085-13-8 MSC-2530818 B1975 1 mg, 5 mg 1883423-59-3 MK-8745 B1942 5 mg, 25 mg 885325-71-3 NG52 9420 5 mg, 25 mg 212779-48-1 MLN-8054 B1943 5 mg, 25 mg 869363-13-3 NU6102 2313 1 mg, 5 mg 444722-95-6 MLN8237 2718 5 mg, 25 mg 1028486-01-2 ON-013100 B1276 5 mg, 25 mg 865783-95-5 PF-03814735 B1257 5 mg, 25 mg 942487-16-3 PD-0332991 2843 5 mg, 25 mg 571190-30-2 PHA-680632 B1944 5 mg, 25 mg 398493-79-3 PD-0332991 isethionate 9480 5 mg, 25 mg 827022-33-3 Reversine 1851 1 mg, 5 mg 656820-32-5 RGB-286638, free base 2886 5 mg, 25 mg 784210-88-4 SNS-314 2446 5 mg, 25 mg 1057249-41-8 (LEE011) 9481 5 mg, 25 mg 1211441-98-3 TAK-901 B1945 5 mg, 25 mg 934541-31-8 (R)-Perharidine-1 2615 1 mg, 5 mg 1133437-80-5 TC-S 7010 B1203 5 mg, 25 mg 1158838-45-9 RO-3306 2039 1 mg, 5 mg 872573-93-8 EZSolution™ Tozasertib 1803 25 mg 639089-54-6 Roscovitine 1950 1 mg, 5 mg 186692-46-6 Tozasertib (VX-680, MK-0457, VX6) 1595 25 mg, 100 mg 639089-54-6 SNS-032 9490 5 mg, 25 mg 345627-80-7 Tripolin A 2307 1 mg, 5 mg 1148118-92-6 TG003 1905 5 mg, 25 mg 300801-52-9 ZM 447439 2018 1 mg, 5 mg 331771-20-1 THZ1 (Free base) 9664 5 mg, 25 mg 1604810-83-4 THZ1 hydrochloride 9544 5 mg, 25 mg 1604810-83-4 Axl Receptor Inhibitors 10Z-Hymenialdisine 2212 250 µg, 1 mg 82005-12-7 Product Name Cat. No. Size CAS. No. BMS-777607 2455 5 mg, 25 mg 1025720-94-8 Chk (Checkpoint Kinase) Kinase Inhibitor R428 9591 5 mg, 25 mg 1037624-75-1 Product Name Cat. No. Size CAS. No. SGI-7079 B1202 5 mg, 25 mg 1239875-86-5 AZD-7762 9414 5 mg, 25 mg 860352-01-8 TP-0903 9590 5 mg, 25 mg 1341200-45-0 CCT244747 9575 5 mg, 25 mg 1404095-34-6 BTK (Bruton’s Tyrosine Kinase) Inhibitors Chk2 Inhibitor 1702 1 mg 516480-79-8 Product Name Cat. No. Size CAS. No. CK (Casein kinase) Inhibitors B1193 5 mg, 25 mg 1420477-60-6 Product Name Cat. No. Size CAS. No. AVL-292 (Spebrutinib) 9413 5 mg, 25 mg 1202757-89-8 Apigenin 2508 25 mg, 100 mg 520-36-5 BTK Inhibitor, CNX-774 2600 5 mg, 25 mg 1202759-32-7 BMS-582949 B1704 1 mg, 5 mg 623152-17-0 BTK Inhibitor, PCI-32765 2298 5 mg, 25 mg 936563-96-1 CX-4945 2459 5 mg, 25 mg 1009820-21-6 CGI-1746 9647 5 mg, 25 mg 910232-84-7 D4476 1770 1 mg, 5 mg 301836-43-1 LFM-A13 2414 5 mg, 25 mg 244240-24-2 IC261 9669 5 mg, 25 mg 186611-52-9 ONO-4059 B1283 5 mg, 25 mg 1351636-18-4 LH-846 9423 10 mg, 50 mg 639052-78-1

10 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 11 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. OSI-930 B1712 5 mg, 25 mg 728033-96-3 GSK-3β Inhibitor, TWS119 1655 2 mg, 5 mg 601514-19-6 Pexmetinib B1711 5 mg, 25 mg 945614-12-0 IM-12 2822 5 mg, 25 mg 1129669-05-1 PH-797804 B1707 5 mg, 25 mg 586379-66-0 Kenpaullone 1904 1 mg 142273-20-9 SB239063 B1699 5 mg, 25 mg 193551-21-2 Leucettine L41 2617 1 mg, 5 mg 1112978-84-3 TA-01 B1214 5 mg, 25 mg 1784751-18-3 LY-2090314 B1043 5 mg, 25 mg 603288-22-8 TA-02 B1215 5 mg, 25 mg 1784751-19-4 PKC-9 B1755 5 mg N/A C-Met (Mesenchymal-Epithelial Transition Factor) Kinase Ro 31-8220 methanesulfonate 1946 1 mg, 5 mg 138489-18-6 Inhibitors SB 216763 1769 1 mg, 5 mg 280744-09-4 Product Name Cat. No. Size CAS. No. SB-415286 B1954 5 mg, 25 mg 264218-23-7 Altiratinib 9563 5 mg, 25 mg 1345847-93-9 TDZD-8 2854 5 mg, 25 mg 327036-89-5 AMG-208 2553 5 mg, 25 mg 1002304-34-8 Tideglusib 9601 5 mg, 25 mg 865854-05-3 BMS-777607 2455 5 mg, 25 mg 1025720-94-8 JAK (Janus Kinases) Inhibitors Crizotinib 1934 5 mg, 25 mg 877399-52-5 Product Name Cat. No. Size CAS. No. Carbozantinib 1935 5 mg, 25 mg 849217-68-1 ABT-494 B1947 5 mg, 25 mg 1310726-60-3 SU 11274 1938 5 mg, 25 mg 658084-23-2 AZD1480 2315 1 mg, 5 mg 935666-88-9 9476 5 mg, 25 mg 849217-64-7 2842 10 mg, 50 mg 1187594-09-7 Golvatinib 2655 5 mg, 25 mg 928037-13-2 Baricitinib phosphate 2841 10 mg, 50 mg 1187595-84-1 JNJ-38877605 B2063 5 mg, 25 mg 943540-75-8 BMS-911543 2630 1 mg, 5 mg 1271022-90-2 PF-04217903 B2062 5 mg, 25 mg 956905-27-4 Cedrulatinib 2803 5 mg, 25 mg 1198300-79-6 PHA-665752 B2057 5 mg, 25 mg 477575-56-7 CP-690550 1622 5 mg, 25 mg 477600-75-2 B1546 5 mg, 25 mg 905854-02-6 CP-690550 citrate 9428 5 mg, 25 mg 540737-29-9 DNA-PK (DNA-dependent Protein Kinase) Inhibitors Cyt387 2316 1 mg, 5 mg 1056634-68-4 Product Name Cat. No. Size CAS. No. Decernotinib (VX-509) B1260 5 mg, 25 mg 944842-54-0 Compound 401 1657 5 mg 168425-64-7 2871 10 mg, 50 mg 1206161-97-8 KU-0060648 B1115 5 mg, 25 mg 881375-00-4 GLPG0634 Analog B1836 5 mg, 25 mg 1206101-20-3 EZSolution™ NU-7441 B1875 5 mg 503468-95-9 INCB39110 B1894 5 mg, 25 mg 1334298-90-6 NU-7441 B1117 5 mg, 25 mg 503468-95-9 935666-88-9 1187594-09-7 DYRK (Dual-specificity Tyrosine Phosphorylation-regulated 1271022-90-2 DiscoveryPak™ JAK Inhibitors Set 477600-75-2 Kinase) Inhibitors (Containing Cat. No. 2315, 2842, 2630, S236 9 Inhibitors 1056634-68-4 Product Name Cat. No. Size CAS. No. 1622, 2316, 2871, 2139, 1853, 1809) 1206161-97-8 941678-49-5 Leucettine L41 2617 1 mg, 5 mg 1112978-84-3 202475-60-3 FAK (Focal Adhesion Kinase) Inhibitors 857064-38-1 133550-30-8 Product Name Cat. No. Size CAS. No. 477600-75-2 PF-562271 besylate B1253 5 mg, 25 mg 939791-38-5 PathwayReady™ JAK/STAT Signaling 111358-88-4 Inhibitor Panel 1260247-42-4 K864 8 Inhibitors Y15 B1252 10 mg, 50 mg 4506-66-5 (Containing Cat. No. 1570, 1622, 1805, 501919-59-1 1792, 1775, 1809, 1887, 1778) 857064-38-1 GSK (Glycogen Synthase Kinases) Inhibitors 2062-78-4 Product Name Cat. No. Size CAS. No. N/A Alsterpaullone 1897 1 mg, 5 mg 237430-03-4 LY-2784544 B1914 5 mg, 25 mg 1229236-86-5 1-Azakenpaullone 1944 1 mg, 5 mg 676596-65-9 MS-1020 1911 1 mg 1255516-86-9 Bikinin 2034 10 mg, 50 mg 188011-69-0 PF-03394197 2883 5 mg, 25 mg 1208319-26-9 BIO 1673 1 mg 667463-62-9 , Free base 2139 5 mg, 25 mg 941678-49-5 Bisindolylmaleimide I 1945 1 mg, 5 mg 133052-90-1 SAR-20347 B1290 5 mg, 25 mg 1450881-55-6 Bisindolylmaleimide I hydrochloride 1947 1 mg, 5 mg 176504-36-2 TG101348 2314 1 mg, 5 mg 936091-26-8 Ezsolution™ CHIR-98014 2639 1 mg 556813-39-9 Tyrphostin AG 490 1570 5 mg 133550-30-8 CHIR-98014 2595 1 mg, 5 mg 556813-39-9 WHI-P131 1853 5 mg, 25 mg 202475-60-3 CHIR 99021 1677 5 mg, 25 mg 252917-06-9 WHI-P154 2659 5 mg, 25 mg 211555-04-3 EZSolution™ CHIR99021 1748 5 mg 252917-06-9 WP1066 1809 5 mg, 25 mg 857064-38-1 EZSolution™ CHIR99021 trihydrochloride, B1219 1 ml 1782235-14-6 Sterile-Filtered JNK (c-Jun N-terminal Kinase) Inhibitors CHIR 99021 trihydrochloride B1199 5 mg, 25 mg 1782235-14-6 Product Name Cat. No. Size CAS. No. CP21R7 B1563 5 mg, 25 mg 125314-13-8 AS 602801 B1687 5 mg, 25 mg 848344-36-5 EZSolution™ CHIR99021, Sterile-Filtered 1991 1 ml 252917-06-9 AS601245 2162 1 mg, 5 mg 345987-15-7 EZSolution™ Necrosulfonamide, Sterile- BI-78D3 B1686 5 mg, 25 mg 883065-90-5 B1220 10 mg 1360614-48-7 Filtered DB07268 B1134 10 mg, 50 mg 929007-72-7 GSK-3 Inhibitor, AR-A014418 1953 2 mg, 5 mg 487021-52-3 IQ-1S B1279 5 mg, 25 mg 1421610-21-0 237430-03-4 188011-69-0 JNK-IN-7 B1695 1 mg, 5 mg 1408064-71-0 252917-06-9 DiscoveryPak™ GSK-3 Inhibitors Set JNK-IN-8 2729 5 mg, 25 mg 1410880-22-6 556813-39-9 (Containing Cat. No. 1897, 2034, 1677, S237 8 Inhibitors 487021-52-3 L-JNK Peptide Inhibitor I 7011 50 µl N/A 2595, 1953, 1655, B1043, 9601) 601514-19-6 EZSolution™ SP600125 9541 5 mg 129-56-6 603288-22-8 SP600125 1669 5 mg 129-56-6 865854-05-3 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 12 MLCK (Myosin Light Chain Kinase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. TCS JNK 5a B1688 5 mg, 25 mg 312917-14-9 ML-7 hydrochloride B2000 10 mg, 50 mg 110448-33-4 LRRK2 (Leucine-Rich Repeat Kinase 2) Inhibitors MLK (Mixed Lineage Kinase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. CZC-54252 hydrochloride 9567 10 mg, 50 mg 1191911-27-9 GNE-3511 B1341 5 mg, 25 mg 1496581-76-0 GSK2578215A 2845 5 mg, 25 mg 1285515-21-0 LY364947 2646 1 mg, 5 mg 396129-53-6 HG-10-012-01 2604 5 mg, 25 mg 1351758-81-0 URMC-099 9443 5 mg, 25 mg 1229582-33-5 JH-II-127 9632 5 mg, 25 mg 1700693-08-8 mTOR (mammalian Target Of Rapamycin) Inhibitors PF-06447475 9447 5 mg, 25 mg 1527473-33-1 Product Name Cat. No. Size CAS. No. MAP (Mitogen-Activated Protein) Kinase-MEK Inhibitors A-674563 B1761 5 mg, 25 mg 552325-73-2 Product Name Cat. No. Size CAS. No. AZD-2014 9449 5 mg, 25 mg 1009298-59-2 APS-2-79 B1696 5 mg, 25 mg 2002381-31-7 AZD-5363 B1762 5 mg, 25 mg 1143532-39-1 AZD6244 2234 5 mg, 25 mg 606143-52-6 AZD8055 2340 1 mg, 5 mg 1009298-09-2 AZD8330 B1693 5 mg, 25 mg 869357-68-6 BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7 BAY 43-9006 1594 25 mg, 100 mg 475207-59-1 BI-D1870 1924 1 mg, 5 mg 501437-28-1 BI-847325 B1589 5 mg, 25 mg 1207293-36-4 BX-517 B1764 5 mg, 25 mg 850717-64-5 BIX02189 2670 1 mg, 5 mg 1094614-85-3 BX795 B1766 5 mg, 25 mg 702675-74-9 B1689 5 mg, 25 mg 934660-93-2 BX-912 B1765 5 mg, 25 mg 702674-56-4 DEL-22379 B1680 5 mg, 25 mg 181223-80-3 CCT128930 B1763 1 mg, 5 mg 885499-61-6 Doramapimod 1954 5 mg, 25 mg 285983-48-4 Deforolimus 1587 5 mg, 25 mg 572924-54-0 FR180204 B1683 5 mg, 25 mg 865362-74-9 1917 5 mg, 25 mg 159351-69-6 GDC-0623 B1690 5 mg, 25 mg 1168091-68-6 GDC-0084 B1656 5 mg, 25 mg 1382979-44-3 GSK-1120212 1960 1 mg, 5 mg 871700-17-3 GSK-2126458 1961 1 mg, 5 mg 1086062-66-9 LY2228820 B1702 5 mg, 25 mg 862507-23-1 INK-128 9527 5 mg, 25 mg 1224844-38-5 212631-79-3 LY 303511 B1734 1 mg, 5 mg 154447-38-8 167869-21-8 PathwayReady™ MAP Kinase Signaling LY3023414 B1759 5 mg, 25 mg 1386874-06-1 152121-47-6 Inhibitor Panel K862 7 Inhibitors 475207-59-1 mTOR Inhibitor, Ku-0063794 1779 1 mg, 5 mg 938440-64-3 (Containing Cat. No. 1585, 1666, 1712, 109511-58-2 1594, 1669, 1789, 1669) mTOR Inhibitor, WYE-132 2256 500 µg, 1 mg 1144068-46-1 208260-29-1 129-56-6 mTOR Inhibitor, WYE-23 2257 500 µg, 1 mg 1062169-46-3 MEK-162 2254 5 mg, 25 mg 606143-89-9 mTOR Inhibitor, WYE-28 2255 500 µg, 1 mg 1062172-60-4 Pamapimod B1700 1 mg, 5 mg 449811-01-2 OSI-027 2372 5 mg, 25 mg 936890-98-1 PD 169316 B1703 5 mg, 25 mg 152121-53-4 OXA-01 2695 5 mg, 25 mg 936889-68-8 EZSolution™ PD 98059 1783 5 mg 167869-21-8 371242-69-2 DiscoveryPak™ PI 3-Kinase Inhibitor Set 154447-36-6 PD 98059 1666 5 mg 167869-21-8 (Containing Cat. No. 1661, 1667, 1728, K856 5 Inhibitors 371935-74-9 EZSolution™ PD-0325901, Sterile-Filtered 1990 1 ml 391210-10-9 1780, 1781) 648450-29-7 663619-89-4 PD-0325901 1643 2 mg, 5 mg, 25 mg 391210-10-9 PP242 1658 1 mg 1092351-67-1 EZSolution™ PD184352 1871 1 mg 212631-79-3 Prodigiosin 2311 250 µg, 1 mg 82-89-3 PD184352 1585 1 mg, 5 mg, 25 mg 212631-79-3 EZSolution™ Rapamycin 1746 5 mg 53123-88-9 PD318088 B1697 1 mg, 5 mg 391210-00-7 Rapamycin 1568 5 mg, 50 mg 53123-88-9 Pimasertib B1698 5 mg, 25 mg 1236699-92-5 (CCI-779, Torisel) 1600 5 mg, 25 mg 162635-04-3 Refametinib B1889 5 mg, 25 mg 923032-37-5 EZSolution™ Torin 1 2353 5 mg 1222998-36-8 SB 202190 2493 5 mg, 25 mg 152121-30-7 Torin 1 2273 5 mg, 25 mg 1222998-36-8 EZSolution™ SB 203580 1786 1 mg 152121-47-6 EZSolution™ Torin 2 2354 5 mg 1223001-51-1 SB 203580 1712 1 mg, 5 mg 152121-47-6 Torin 2 2274 5 mg, 25 mg 1223001-51-1 SCH772984 B1682 5 mg, 25 mg 942183-80-4 Uprosertib B1760 5 mg, 25 mg 1047634-65-0 Skepinone-L B1110 1 mg, 5 mg 1221485-83-1 VPS34 inhibitor B1754 5 mg 1383716-40-2 SKF-86002 2894 5 mg, 25 mg 72873-74-6 WAY-600 B1731 1 mg, 5 mg 1062159-35-6 SL327 B1694 5 mg, 25 mg 305350-87-2 WYE-354 B1732 5 mg, 25 mg 1062169-56-5 TAK-715 B1701 5 mg, 25 mg 303162-79-0 WYE-687 B1730 5 mg, 25 mg 1062161-90-3 TAK-733 2460 5 mg, 25 mg 1035555-63-5 XL388 B1733 1 mg, 5 mg 1251156-08-7 7,3',4'-Trihydroxyisoflavone 1886 25 mg, 100 mg 485-63-2 U0126 1668 5 mg 109511-58-2 PDK1 (Phosphoinositide-Dependent Kinase 1) Inhibitors VRT752271 B1679 5 mg, 25 mg 869886-67-9 Product Name Cat. No. Size CAS. No. VX-11e B1681 5 mg, 25 mg 896720-20-0 GSK-2334470 B1555 5 mg, 25 mg 1227911-45-6 VX-702 1598 1 mg, 5 mg 745833-23-2 OSU-03012 2295 5 mg, 25 mg 742112-33-0 VX-745 2812 5 mg, 25 mg 209410-46-8 SGK-1 inhibitor B1757 5 mg N/A XMD17-109 B1685 5 mg, 25 mg 1435488-37-1 PI 3-Kinase (Phosphoinositide 3-Kinase) Inhibitors XMD8-92 B1684 5 mg, 25 mg 1234480-50-2 10Z-Hymenialdisine 2212 250 µg, 1 mg 82005-12-7 Product Name Cat. No. Size CAS. No. A66 B1654 5 mg, 25 mg 1166227-08-2 Acalisib B1666 5 mg, 25 mg 870281-34-8

12 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 13 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Alpelisib B1271 5 mg, 25 mg 1217486-61-7 ZSTK474 1597 25 mg, 100 mg 475110-96-4 AMG319 B1663 5 mg, 25 mg 1608125-21-8 PI3K-mTOR (Phosphoinositide 3Kinase-mTOR) Inhibitors APY-0201 9564 5 mg, 25 mg 1232221-74-7 Product Name Cat. No. Size CAS. No. AS 604850 2339 1 mg, 5 mg 648449-76-7 AS-252424 B1611 5 mg, 25 mg 900515-16-4 AS-041164 B1870 5 mg, 25 mg 6318-41-8 BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7 AZD-6482 B1143 5 mg, 25 mg 1173900-33-8 BGT226 B1719 1 mg, 5 mg 1245537-68-1 AZD-8186 B1027 5 mg, 25 mg 1627494-13-6 CP-466722 B1722 1 mg, 5 mg 1080622-86-1 AZD8835 B1661 5 mg, 25 mg 1620576-64-8 CZ415 B1726 5 mg, 25 mg 1429639-50-8 BAG 956 2456 5 mg, 25 mg 853910-02-8 GDC-0349 B1729 1 mg, 5 mg 1207360-89-1 BAY 80-6946 B1267 5 mg, 25 mg 1032568-63-0 GDC-0941 Dimethanesulfonate 9618 10 mg, 50 mg 957054-33-0 BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7 GDC-0980 2668 1 mg, 5 mg 1032754-93-0 CAL-101 (GS-1101) 2613 5 mg, 25 mg 870281-82-6 GNE 477 B1657 5 mg, 25 mg 1032754-81-6 CH5132799 B1669 5 mg, 25 mg 1007207-67-1 GNE-317 B1716 5 mg, 25 mg 1394076-92-6 CNX-1351 B1673 5 mg, 25 mg 1276105-89-5 HS-173 B1627 5 mg, 25 mg 1276110-06-5 CUDC-907 B1675 5 mg, 25 mg 1339928-25-4 P529 2462 5 mg, 25 mg 914913-88-5 CZC24832 B1676 5 mg, 25 mg 1159824-67-5 PF-04691502 2289 5 mg, 25 mg 1013101-36-4 GDC-0032 9573 5 mg, 25 mg 1282512-48-4 PF-05212384 9461 10 mg, 50 mg 1197160-78-3 GDC-0326 B1655 5 mg, 25 mg 1282514-88-8 PF-4989216 B1659 5 mg, 25 mg 1276553-09-3 GDC-0941 1623 1 mg, 5 mg 957054-30-7 PKI-402 B1727 1 mg, 5 mg 1173204-81-3 GSK-1059615 9450 5 mg, 25 mg 958852-01-2 PKI-402 B1715 1 mg, 5 mg 173204-81-3 GSK-2126458 1961 1 mg, 5 mg 1086062-66-9 PQR-309 B1300 5 mg, 25 mg 1225037-39-7 GSK2292767 B1660 5 mg, 25 mg 1254036-66-2 TG100713 B1717 5 mg, 25 mg 925705-73-3 GSK2636771 2793 5 mg, 25 mg 1372540-25-4 VS-5584 9603 1 mg, 5 mg 1246560-33-7 IC87114 1661 1 mg 371242-69-2 XL765 2551 5 mg, 25 mg 934493-76-2 IPI-145 2445 5 mg, 25 mg 1201438-56-3 IPI-549 B1971 5 mg, 25 mg 1693758-51-8 PIM (Proto-oncogene proviral Integration site for Moloney EZSolution™ LY294002 1747 5 mg 154447-36-6 murine virus) Kinase Inhibitors LY 294002 1667 5 mg, 25 mg 154447-36-6 Product Name Cat. No. Size CAS. No. MTX-211 B1968 5 mg, 25 mg 1952236-05-3 AZD1208 2719 1 mg, 5 mg 1204144-28-4 NVP-BKM120 2619 5 mg, 25 mg 944396-07-0 CX-6258 2851 5 mg, 25 mg 1202916-90-2 PI-103 1728 1 mg, 5 mg 371935-74-9 , Dihydrate 1773 250 mg, 1 g 6151-25-3 PI-3065 B1674 5 mg, 25 mg 955977-50-1 SGI-1776 2554 5 mg, 25 mg 1025065-69-3 PI3K-α Inhibitor B1869 5 mg, 25 mg 371943-05-4 SMI-4a 2211 5 mg 327033-36-3 PI3-Kγ Inhibitor, AS-605240 1780 1 mg, 5 mg 648450-29-7 TCS PIM-1 1 2848 10 mg, 50 mg 491871-58-0 612847-09-3 XL765 2551 5 mg, 25 mg 934493-76-2 915019-65-7 154447-36-6 PKD (Protein Kinase D) Inhibitors PathwayReady™ PI3-K/Akt/mTOR 938440-64-3 Signaling Inhibitor Panel 371935-74-9 Product Name Cat. No. Size CAS. No. (Containing Cat. No. 1708, 1626, 1667, K857 11 Inhibitors 648450-29-7 CID-2011756 2607 5 mg, 25 mg 638156-11-3 1779, 1728, 1780, 1658, 1568, 1781, 1707, 1092351-67-1 1670) 53123-88-9 CID-755673 2660 5 mg, 25 mg 521937-07-5 663619-89-4 CRT0066101 B1847 1 mg, 5 mg 1883545-60-5 35943-35-2 kb NB 142-70 9566 5 mg, 25 mg 1233533-04-4 19545-26-7 371242-69-2 PKG (Protein Kinase G) Inhibitors DiscoveryPak™ PI 3-Kinase Inhibitor Set 154447-36-6 (Containing Cat. No. 1661, 1667, 1728, K856 5 Inhibitors 371935-74-9 Product Name Cat. No. Size CAS. No. 1780, 1781) 648450-29-7 H-7 dihydrochloride 9543 5 mg, 25 mg 108930-17-2 663619-89-4 PIK-293 B1658 5 mg, 25 mg 900185-01-5 KT5823 2164 50 µg, 250 µg 126643-37-6 PIK-294 2614 5 mg, 25 mg 900185-02-6 PLK (Polo Like Kinase) Inhibitors PIK75 B1668 5 mg, 25 mg 372196-77-5 Product Name Cat. No. Size CAS. No. PIK-90 B1671 5 mg, 25 mg 677338-12-4 BI-2536 2370 5 mg, 25 mg 755038-02-9 PIK-93 B1670 5 mg, 25 mg 593960-11-3 BI 6727 2222 1 mg, 5 mg 755038-65-4 PX-866 1965 1 mg, 5 mg 502632-66-8 CFI-400945 B1287 5 mg, 25 mg 1338806-76-0 SAR-260301 B1263 5 mg, 25 mg 1260612-13-2 GSK461364 2287 5 mg, 25 mg 929095-18-1 Serabelisib B1930 5 mg, 25 mg 1268454-23-4 HMN-214 B1646 5 mg, 25 mg 173529-46-9 SF-2523 B1858 1 mg, 5 mg 1174428-47-7 Rigosertib 9482 5 mg, 25 mg 1225497-78-8 TG100-115 B1667 5 mg, 25 mg 677297-51-7 Ro3280 B1175 5 mg, 25 mg 1062243-51-9 TGR-1202 B1284 5 mg, 25 mg 1532533-67-7 SBE13 hydrochloride 2847 10 mg, 50 mg 1052532-15-6 TGX-115 1660 1 mg 351071-62-0 Wortmannin, Penicillium funiculosum 1670 1 mg 19545-26-7 TGX-221 1781 1 mg, 5 mg 663619-89-4 Wortmannin, Penicillium funiculosum 1670 1 mg 19545-26-7 Protein Kinase C Inhibitors XL-147 9401 5 mg, 25 mg 956958-53-5 Product Name Cat. No. Size CAS. No. YM201636 2045 1 mg, 5 mg 371942-69-7 Bisindolylmaleimide I 1945 1 mg, 5 mg 133052-90-1 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 14 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Bisindolylmaleimide I hydrochloride 1947 1 mg, 5 mg 176504-36-2 BIBW2992 (Tovok) 1616 1 mg, 5 mg 439081-18-2 Calphostin C 2611 50 µg, 100 µg 121263-19-2 BIBX-1382 9463 5 mg, 25 mg 196612-93-8 Cercosporin 9684 250 µg, 1 mg 35082-49-6 BLU9931 9639 5 mg, 25 mg 1538604-68-0 Chelerythrine chloride 2064 5 mg 3895-92-9 BLZ-945 B1651 5 mg, 25 mg 953769-46-5 D-erythro-Sphingosine 2425 5 mg, 25 mg 123-78-4 BMS-536924 B1908 1 mg, 5 mg 468740-43-4 Enzastaurin (LY317615) 1619 1 mg, 5 mg 170364-57-5 BMS-599626 1614 1 mg, 5 mg 873837-23-1 EZSolution™ Gö 6976 1785 500 µg 136194-77-9 BMS-754807 2631 1 mg, 5 mg 1001350-96-4 Gö 6976 1711 500 µg 136194-77-9 BMS-777607 2455 5 mg, 25 mg 1025720-94-8 EZSolution™ Gö 6983 9540 1 mg 133053-19-7 BMX-IN-1 B1330 5 mg, 25 mg 1431525-23-3 Gö 6983 9539 1 mg, 5 mg 133053-19-7 (SKI-606) 1584 5 mg, 25 mg 380843-75-4 H-7 dihydrochloride 9543 5 mg, 25 mg 108930-17-2 Brigatinib (AP26113) 9675 5 mg, 25 mg 1197953-54-0 Hypericin 2526 1 mg, 5 mg 548-04-9 Brivanib B1325 1 mg, 5 mg 649735-46-6 K252a 2013 500 µg, 1 mg 99533-80-9 Brivanib Alaninate B1326 1 mg, 5 mg 649735-63-7 LY-333,531 hydrochloride 2156 250 µg, 1 mg 169939-93-9 BTK Inhibitor, CNX-774 2600 5 mg, 25 mg 1202759-32-7 PKC412 2052 1 mg, 5 mg 120685-11-2 BTK Inhibitor, PCI-32765 2298 5 mg, 25 mg 936563-96-1 PKC-9 B1755 5 mg N/A (CI-1033, PD-183805) 1617 5 mg, 50 mg 289499-45-2 Ro 31-8220 methanesulfonate 1946 1 mg, 5 mg 138489-18-6 Carbozantinib 1935 5 mg, 25 mg 849217-68-1 EZSolution™ 1745 100 µg 62996-74-1 (AZD2171) 1613 1 mg, 5 mg 288383-20-0 Staurosporine 1048 100 µg, 1 mg 62996-74-1 CGI-1746 9647 5 mg, 25 mg 910232-84-7 Tamoxifen citrate 1551 1 g 54965-24-1 CH5183284 B1649 5 mg, 25 mg 1265229-25-1 CH5424802 2867 5 mg, 25 mg 1256580-46-7 Protein Tyrosine Kinase Inhibitors CL-387785 2826 10 mg, 50 mg 194423-06-8 Product Name Cat. No. Size CAS. No. CO-1686 () 2794 5 mg, 25 mg 1374640-70-6 EZSolution™ A83-01, Sterile-Filtered 1989 1 ml 909910-43-6 CP-673451 B1337 1 mg, 5 mg 343787-29-1 A 83-01 1725 1 mg 909910-43-6 CP-690550 1622 5 mg, 25 mg 477600-75-2 AAL-993 2740 2 mg, 10 mg 269390-77-4 CP-724714 B1333 5 mg, 25 mg 537705-08-1 ABL-001 B1949 1 mg, 5 mg 1492952-76-7 9679 5 mg, 25 mg 670220-88-9 ABT-869 1615 1 mg, 5 mg 796967-16-3 Crizotinib 1934 5 mg, 25 mg 877399-52-5 AC710 2884 5 mg, 25 mg 1351522-04-7 CTx-0294885 9435 5 mg, 25 mg 1439934-41-4 ACTB-1003 B2016 5 mg, 25 mg 939805-30-8 CUDC-101 1966 5 mg, 25 mg 1012054-59-9 AEE-788 9658 1 mg, 5 mg 497839-62-0 CZC-8004 B1868 5 mg, 25 mg 916603-07-1 AG 1478 1800 5 mg, 25 mg 175178-82-2 Damnacanthal B1094 1 mg, 5 mg 477-84-9 AG-1296 2376 5 mg 146535-11-7 EZSolution™ 2029 25 mg 302962-49-8 Altenusin, Penicillium sp. 2146 1 mg, 5 mg 31186-12-6 Dasatinib (BMS-354825, Sprycel) 1586 25 mg, 100 mg 302962-49-8 Altiratinib 9563 5 mg, 25 mg 1345847-93-9 DDR1-IN-1 B1331 5 mg, 25 mg 1449685-96-4 AMG-208 2553 5 mg, 25 mg 1002304-34-8 Dovitinib B1614 5 mg, 25 mg 405169-16-6 AMG-47a 2825 5 mg, 25 mg 882663-88-9 Dovitinib lactate B1615 5 mg, 25 mg 915769-50-5 AMG-925 B1959 5 mg, 25 mg 1401033-86-0 EAI-045 B1247 5 mg, 25 mg 1942114-09-1 AMG-Tie2 B1612 5 mg, 25 mg 870223-96-4 133550-30-8 Amuvatinib 9458 5 mg, 25 mg 850879-09-3 612847-09-3 289499-45-2 ANA-12 2878 10 mg, 50 mg 219766-25-3 184475-35-2 388082-78-8 Anomalin A 2151 1 mg 548740-86-9 PathwayReady™ EGFR Signaling Inhibitor 154447-36-6 Panel (Free base) B1613 5 mg, 25 mg 811803-05-1 167869-21-8 (Containing Cat. No. 1570, 1708, 1617, K863 14 Inhibitors Apatinib mesylate B1608 5 mg, 25 mg 1218779-75-9 172889-27-9 1589, 1624, 1667, 1666, 1767, 1712, 1594, 152121-47-6 ASP-3026 B1296 5 mg, 25 mg 1097917-15-1 1775, 1789, 1568) 475207-59-1 AT9283 2432 5 mg, 25 mg 896466-04-9 501919-59-1 AVL-292 (Spebrutinib) 9413 5 mg, 25 mg 1202757-89-8 208260-29-1 53123-88-9 (AG-013736) 1581 5 mg, 25 mg 319460-85-0 129-56-6 AZ-5104 9441 10 mg, 50 mg 1421373-98-9 289499-45-2 DiscoveryPak™ EGFR Tyrosine Kinase 183319-69-9 AZD-3463 2371 5 mg, 25 mg 1356962-20-3 Inhibitor Set K858 5 Inhibitors 184475-35-2 (Containing Cat. No. 1617, 1588, 1589, AZD-3759 9609 5 mg, 25 mg 1626387-80-1 388082-78-8 1624, 1656) AZD-4547 9403 5 mg, 25 mg 1035270-39-3 153436-54-5 EMD-1214063 B1297 5 mg, 25 mg 1100598-32-0 AZD-8931 9659 5 mg, 25 mg 848942-61-0 Emodin 1875 25 mg, 100 mg 518-82-1 AZD-9291 2674 5 mg, 25 mg 1421373-65-0 Ensartinib B1946 5 mg, 25 mg 1365267-27-1 AZD-9291 mesylate B1899 5 mg, 25 mg 1421373-66-1 Entrectinib B1324 5 mg, 25 mg 1108743-60-7 Bafetinib B1172 5 mg, 25 mg 859212-16-1 , Free Base 2048 100 mg, 1 g 183321-74-6 EZSolution™ BAY 43-9006 2031 25 mg 475207-59-1 EW-7197 B1191 1 mg, 5 mg 1352608-82-2 BAY 43-9006 1594 25 mg, 100 mg 475207-59-1 FIIN-2 9577 5 mg, 25 mg 1633044-56-0 BAY 43-9006, Free base 2142 25 mg, 100 mg 284461-73-0 Foretinib 9476 5 mg, 25 mg 849217-64-7 Bay 61-3606 Hydrochloride 1796 1 mg, 5 mg 732983-37-8 Fostamatinib Disodium 1936 1 mg, 5 mg 1025687-58-4 BIBF1120 2167 5 mg, 25 mg 928326-83-4

14 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 15 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Fruquintinib B1979 5 mg, 25 mg 1194506-26-7 Pelitinib (EKB-569) 2676 5 mg, 25 mg 257933-82-7 EZSolution™ 2030 5 mg 184475-35-2 PF-04554878 2888 5 mg, 25 mg 1073154-85-4 Gefitinib 1589 5 mg, 25 mg 184475-35-2 PF-06463922 B1169 10 mg, 50 mg 1454846-35-5 Genistein 1533 10 mg, 100 mg 446-72-0 PF299804 2678 5 mg, 25 mg 1110813-31-4 Genistin 1535 10 mg 529-59-9 PF-431396 2844 5 mg, 25 mg 717906-29-1 B1294 5 mg, 25 mg 1254053-43-4 PF-573228 2819 10 mg, 50 mg 869288-64-2 GNF-2 2470 5 mg, 25 mg 778270-11-4 Piceatannol 2072 5 mg, 25 mg 10083-24-6 GNF-5 B1329 5 mg, 25 mg 778277-15-9 Picropodophyllotoxin 2765 1 mg, 5 mg 477-47-4 Golvatinib 2655 5 mg, 25 mg 928037-13-2 PLX-3397 9617 10 mg, 50 mg 1029044-16-3 GS-9973 2669 1 mg, 5 mg 1229208-44-9 PND-1186 2823 5 mg, 25 mg 1061353-68-1 GSK1904529A 2286 5 mg, 25 mg 1089283-49-7 2712 10 mg, 50 mg 943319-70-8 GSK2256098 B1224 5 mg, 25 mg 1224887-10-8 Poziotinib 9519 10 mg, 50 mg 1092364-38-9 EZSolution™ GW2580 2549 5 mg 870483-87-7 PP1 1927 1 mg, 5 mg 172889-26-8 GW2580 1740 5 mg, 25 mg 870483-87-7 PP2 1767 1 mg, 5 mg 172889-27-9 GW-786034 1916 5 mg, 25 mg 444731-52-6 PP3 1797 10 mg, 50 mg 5334-30-5 GW788388 2820 10 mg, 50 mg 452342-67-5 2008 1 mg, 5 mg 950769-58-1 GZD824 2795 5 mg, 25 mg 1257628-77-5 R428 9591 5 mg, 25 mg 1037624-75-1 H3B-6527 B1647 5 mg, 25 mg 1702259-66-2 9613 10 mg, 50 mg 926037-48-1 Harmine 2561 50 mg, 250 mg 442-51-3 Rebastinib (DCC-2036) B1619 5 mg, 25 mg 1020172-07-9 Herbimycin A 2748 100 µg, 1 mg 70563-58-5 319460-85-0 289499-45-2 Hypericin 2526 1 mg, 5 mg 548-04-9 DiscoveryPak™ 184475-35-2 Mesylate (CGP-57148B, STI-571) 1625 100 mg, 1 g 220127-57-1 (RTK) Inhibitor Set 870483-87-7 K859 8 Inhibitors Imatinib, Free base 2141 100 mg, 1 g 152459-95-5 (Containing Cat. No. 1581, 1617, 1589, 388082-78-8 1740, 1624, 1675, 1674, 1611) 219580-11-7 IPI-549 B1971 5 mg, 25 mg 1693758-51-8 301836-41-9 ITD-1 2879 10 mg, 50 mg 1099644-42-4 341031-54-7 JAK Inhibitor, Pyridone 6 2534 500 µg, 1 mg 457081-03-7 2891 5 mg, 25 mg 755037-03-7 133550-30-8 Regorafenib monohydrate B1621 5 mg, 25 mg 1019206-88-2 477600-75-2 PathwayReady™ JAK/STAT Signaling EZSolution™ RepSox 2641 5 mg 446859-33-2 111358-88-4 Inhibitor Panel K864 8 Inhibitors 1260247-42-4 RN486 9678 1 mg, 5 mg 1242156-23-5 (Containing Cat. No. 1570, 1622, 1805, 501919-59-1 Saracatinib (AZD0530) 1582 5 mg, 25 mg 379231-04-6 1792, 1775, 1809, 1887) 857064-38-1 SB1518 () 2450 1 mg, 5 mg 937272-79-2 2062-78-4 JNJ-10198409 B1078 5 mg, 25 mg 627518-40-5 EZSolution™ SB-431542 1872 1 mg 301836-41-9 Ki 8751 2677 5 mg, 25 mg 228559-41-9 EZSolution™ SB-431542, Sterile-Filtered 1992 1 ml 301836-41-9 KRN-633 2839 5 mg, 25 mg 286370-15-8 SB-431542 1674 1 mg, 5 mg 301836-41-9 KW-2449 hydrochloride B1208 5 mg, 25 mg 1000669-72-6 EZSolution™ SB-525334 2881 5 mg 356559-20-1 Ditosylate (Tykerb, Tyverb, SB-525334 2880 5 mg, 25 mg 356559-20-1 1624 25 mg, 100 mg 388082-78-8 GW-572016) SD208 2885 5 mg, 25 mg 627536-09-8 EZSolution™ Lapatinib Ditosylate 2807 10 mg 388082-78-8 SSR128129E B1165 5 mg, 25 mg 848318-25-2 Lapatinib, Free base 2138 25 mg, 100 mg 231277-92-2 STK-321130 B2006 5 mg, 25 mg 923562-23-6 B1157 5 mg, 25 mg 417716-92-8 SU 11274 1938 5 mg, 25 mg 658084-23-2 LFM-A13 2414 5 mg, 25 mg 244240-24-2 SU 1498 1836 1 mg, 5 mg 168835-82-3 , Free base 2294 5 mg, 25 mg 867160-71-2 SU 16f B1081 5 mg, 25 mg 251356-45-3 LY-2109761 9605 5 mg, 25 mg 700874-71-1 SU 6668 1931 5 mg, 25 mg 252916-29-3 LY-2157299 9475 5 mg, 25 mg 700874-72-2 SU-5214 B1307 5 mg, 25 mg 186611-04-1 LY-2874455 9532 5 mg, 25 mg 1254473-64-7 EZSolution™ SU-5402 2017 500 µg 215543-92-3 LY364947 2646 1 mg, 5 mg 396129-53-6 SU-5402 1645 500 µg, 1 mg 215543-92-3 2007 5 mg, 25 mg 790299-79-5 EZSolution™ SU-5416 9492 5 mg 204005-46-9 meta-Topolin B1298 50 mg, 250 mg 75737-38-1 SU-5416 9491 5 mg, 25 mg 204005-46-9 MK-1775 2373 5 mg, 25 mg 955365-80-7 SU-5614 9643 5 mg, 25 mg 1055412-47-9 2022 5 mg, 25 mg 453562-69-1 EZSolution™ Malate 1804 25 mg 341031-54-7 MTX-211 B1968 5 mg, 25 mg 1952236-05-3 Sunitinib Malate (Sutent) 1611 25 mg, 100 mg, 1 g 341031-54-7 Naquotinib B1317 5 mg, 25 mg 448232-80-1 Sunitinib, Free base 2097 25 mg, 100 mg, 1 g 557795-19-4 2023 5 mg, 25 mg 698387-09-6 Syk Inhibitor 1983 1 mg, 5 mg 622387-85-3 1750 25 mg, 100 mg 641571-10-0 TAE-226 9436 5 mg, 25 mg 761437-28-9 NVP-AEW541 B1335 5 mg, 25 mg 475489-16-8 TAK 165 1951 5 mg, 25 mg 366017-09-6 NVP-BGJ398 2855 5 mg, 25 mg 872511-34-7 Tandutinib 2024 5 mg, 25 mg 387867-13-2 NVP-BHG712 2464 5 mg, 25 mg 940310-85-0 Tie2 Kinase Inhibitor B1338 5 mg, 25 mg 948557-43-5 NVP-TAE684 1683 5 mg 761439-42-3 Tivantinib B1546 5 mg, 25 mg 905854-02-6 B1218 5 mg, 25 mg 1353550-13-6 B1545 5 mg, 25 mg 475108-18-0 PD 153035 Hydrochloride 1656 2 mg 153436-54-5 B1542 5 mg, 25 mg 356068-94-5 PD 173074 1675 1 mg 219580-11-7 TP-0903 9590 5 mg, 25 mg 1341200-45-0

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 16 Syk (Spleen Tyrosine Kinase) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. TX1-85-1 B1313 5 mg, 25 mg 1603845-32-4 Bay 61-3606 Hydrochloride 1796 1 mg, 5 mg 732983-37-8 Tyrphostin AG 1295 1571 5 mg 71897-07-9 Cedrulatinib 2803 5 mg, 25 mg 1198300-79-6 Tyrphostin AG 490 1570 5 mg 133550-30-8 Fostamatinib Disodium 1936 1 mg, 5 mg 1025687-58-4 UNC-2025 B1262 5 mg, 25 mg 1429881-91-3 GS-9973 2669 1 mg, 5 mg 1229208-44-9 1370261-96-3, UNC2881 2837 5 mg, 25 mg 1493764-08-1 P505-15 9583 5 mg, 25 mg 1370261-97-4 1751 25 mg, 100 mg 443913-73-3 Piceatannol 2072 5 mg, 25 mg 10083-24-6 Varlitinib 2656 5 mg, 25 mg 845272-21-1 PRT-060318 B1911 5 mg, 25 mg 1194961-19-7 Vatalanib Dihydrochloride 2025 5 mg, 25 mg 212141-51-0 Syk Inhibitor 1983 1 mg, 5 mg 622387-85-3 Vatalanib, Free Base 2026 5 mg, 25 mg 212141-54-3 SYK Inhibitor, R406 9682 5 mg, 25 mg 841290-80-0 WH-4-023 2827 10 mg, 50 mg 837422-57-8 WHI-P131 1853 5 mg, 25 mg 202475-60-3 Other Protein Kinase Inhibitors EZSolution™ WP1066 2546 5 mg 857064-38-1 Product Name Cat. No. Size CAS. No. WZ4002 2461 5 mg, 25 mg 1213269-23-8 APY29 2591 5 mg, 25 mg 1216665-49-4 XL019 2609 5 mg, 25 mg 945755-56-6 AS-2444697 Hydrochloride B1585 5 mg, 25 mg 1287665-60-4 XL-228 2632 1 mg, 5 mg 898280-07-4 AT-13148 B1144 5 mg, 25 mg 1056901-62-2 Raf Kinase Inhibitors AZ-3146 B1145 5 mg, 25 mg 1124329-14-1 BAY-1217389 B1295 5 mg, 25 mg 1554458-53-5 Product Name Cat. No. Size CAS. No. Cercosporamide 9662 100 µg, 500 µg 131436-22-1 AZ 628 B1713 5 mg, 25 mg 878739-06-1 CGP-57380 9661 1 mg, 5 mg 522629-08-9 B-Raf Inhibitor 1 2599 5 mg, 25 mg 1093100-40-3 Compound 43 B1758 5 mg N/A CCT196969 B1752 5 mg 1163719-56-9 CPD5 B1750 5 mg N/A CCT241161 B1753 5 mg 1163719-91-2 CZC-54252 hydrochloride 9567 10 mg, 50 mg 1191911-27-9 CEP-32496 9615 5 mg, 25 mg 1188910-76-0 FRAX597 B1890 1 mg, 5 mg 1286739-19-2 DP-4978 B1288 5 mg, 25 mg 1454682-72-4 GNE-7915 B1342 5 mg, 50 mg 1351761-44-8 GDC0879 B1340 5 mg, 25 mg 905281-76-7 GNF-5837 B1339 5 mg, 25 mg 1033769-28-6 GDC0994 B1629 5 mg, 25 mg 1453848-26-4 GNF-7 B1139 5 mg, 25 mg 839706-07-9 Gossypin 2374 50 mg, 250 mg 652-78-8 GSK180736A B1628 5 mg, 25 mg 817194-38-0 GSK-2118436 mesylate 2800 5 mg, 25 mg 1195768-06-9 GSK2578215A 2845 5 mg, 25 mg 1285515-21-0 GW-5074 2412 5 mg, 25 mg 220904-83-6 GSK-2606414 9467 5 mg, 25 mg 1337531-36-8 L-779450 B1709 5 mg, 25 mg 303727-31-3 GSK-2656157 9466 5 mg, 25 mg 1337532-29-2 MLN2480 B1706 5 mg, 25 mg 1096708-71-2 GSK-583 B1301 5 mg, 25 mg 1346547-00-9 1029872-54-5, PLX-4032 2235 5 mg, 25 mg 918504-65-1 EZSolution™ GSK'872 B1501 5 mg 1346546-69-7 PLX-4720 2813 5 mg, 25 mg 918505-84-7 GSK'872 2673 5 mg, 25 mg 1346546-69-7 PLX-7904 B1249 5 mg, 25 mg 1393465-84-3 GW-441756 B1147 5 mg, 25 mg 504433-23-2 RAF265 2856 5 mg, 25 mg 927880-90-8 HG-10-012-01 2604 5 mg, 25 mg 1351758-81-0 RO5126766 B1705 5 mg, 25 mg 946128-88-7 HG-9-91-01 B1849 1 mg, 5 mg 1456858-58-4 SB-590885 B1708 5 mg, 25 mg 405554-55-4 HTH-01-015 2887 5 mg, 25 mg 1613724-42-7 TAK-632 2473 5 mg, 25 mg 1228591-30-7 IPA-3 2647 5 mg, 25 mg 42521-82-4 ZM 336372 1789 1 mg, 5 mg 208260-29-1 IRAK-1/4 Inhibitor 9578 5 mg, 25 mg 509093-47-4 Kobe0065 B1714 5 mg, 25 mg 436133-68-5 ROCK (Rho-associated protein Kinase) Inhibitors Kobe2602 B1710 5 mg, 25 mg 454453-49-7 Product Name Cat. No. Size CAS. No. LDK-378 B1928 5 mg, 25 mg 1032900-25-6 Fasudil, Monohydrochloride 1787 10 mg, 50 mg 105628-07-7 LIMKi 3 B1095 5 mg, 25 mg 1338247-35-0 GSK-269962 9654 5 mg, 25 mg 850664-21-0 LJH685 B1232 5 mg, 25 mg 1627710-50-2 EZSolution™ GSK429286A 2640 1 mg 864082-47-3 LJI-308 B1233 5 mg, 25 mg 1627709-94-7 GSK429286A 2637 1 mg, 5 mg 864082-47-3 LY-2584702 9445 5 mg, 25 mg 1082949-68-5 Hydroxyfasudil Hydrochloride B1559 5 mg, 25 mg 155558-32-0 MPI-0479605 9589 5 mg, 25 mg 1246529-32-7 RKI-1313 B1092 5 mg, 25 mg 1342276-76-9 Mps1-IN-1 B1603 5 mg, 25 mg 1125593-20-5 RKI-1447 2472 5 mg, 25 mg 1342278-01-6 NQDI-1 9645 10 mg, 50 mg 175026-96-7 ROCK Inhibitor (Rockout) 2342 5 mg, 25 mg 7272-84-6 OTS-964 B1964 5 mg, 25 mg 1338545-07-5 (S)-H-1152 dihydrochloride B1106 1 mg, 5 mg 451462-58-1 OTSSP167 B1065 5 mg, 25 mg 1431697-89-0 EZSolution™ Thiazovivin 1736 1 mg 1226056-71-8 PF-06447475 9447 5 mg, 25 mg 1527473-33-1 EZSolution™ Thiazovivin, Sterile-Filtered 1993 1 ml 1226056-71-8 PF-06650833 B1558 5 mg, 25 mg 1817626-54-2 Thiazovivin 1681 1 mg, 5 mg 1226056-71-8 PF-4708671 9460 10 mg, 50 mg 1255517-76-0 EZSolution™ Y-27632 1784 5 mg 146986-50-7 SBI-0206965 9580 5 mg, 25 mg N/A EZSolution™ Y-27632, Sterile-Filtered 1994 1 ml 146986-50-7 Selonsertib B1312 5 mg, 25 mg 1448428-04-3 Y-27632, dihydrochloride 1596 1 mg, 5 mg, 50 mg 146986-50-7 SL0101 B1895 5 mg, 25 mg 77307-50-7 ZINC00881524 B1840 5 mg, 25 mg 557782-81-7 SR7826 B1096 1 mg, 5 mg 1219728-20-7 SRPK (Serine-arginine-Rich Protein Kinase) Inhibitors T5601640 B1097 1 mg, 5 mg 924473-59-6 Product Name Cat. No. Size CAS. No. TGR5-Receptor-Agonist B1635 5 mg, 25 mg 1197300-24-5 SRPIN340 2458 5 mg, 25 mg 218156-96-8

16 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 17 PTEN (Phosphatase & Tensin Homolog) Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. 842133-18-0 bpV(phen) 1793 5 mg 42494-73-5 DiscoveryPak™ SGLT-2 Inhibitors Set 461432-26-8 (Containing Cat. No. B1597, 9452, 2877, S235 4 Inhibitors bpV(pic) 1794 5 mg 148556-27-8 864070-44-0 B1896) SF1670 2774 1 mg, 5 mg 345630-40-2 1210344-57-2 VO-OHpic, Trihydrate 1801 5 mg, 25 mg 476310-60-8 SIRT (Sirtuin) Inhibitors Rac1 Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Cambinol 1653 10 mg 14513-15-6 EHop-016 9595 5 mg, 25 mg 1380432-32-5 4-Hydroxynonenal 2083 1 mg, 5 mg 75899-68-2 NSC 23766 1941 1 mg, 5 mg 733767-34-5 Hyperforin. DCHA 2153 500 µg, 1 mg 238074-03-8 Inauhzin 9555 5 mg, 25 mg 309271-94-1 Renin Inhibitors Salermide 1873 5 mg, 25 mg 1105698-15-4 Product Name Cat. No. Size CAS. No. SIRT1 Inhibitor, EX-527 1652 10 mg 49843-98-3 Rat renin inhibitor peptide 2557 1 mg, 5 mg N/A SIRT2 Inhibitor 1857 5 mg, 25 mg 420831-40-9 Renin Inhibitor 2084 5 mg, 25 mg 173334-58-2 SIRT2 Inhibitor, AGK2 1651 10 mg 304896-28-4 SAH (S-Adenosyl-l-Homocysteine) hydrolase SIRT2 Inhibitor, B2 2085 5 mg 115687-05-3 Sirtinol 2062 1 mg, 5 mg 410536-97-9 Inhibitors Hexasodium Salt 1874 50 mg, 250 mg 129-46-4 Product Name Cat. No. Size CAS. No. Tenovin-1 9400 5 mg, 25 mg 380315-80-0 3-Deazaadenosine 2771 1 mg, 5 mg 6736-58-9 SK (Sphingosine Kinase) Inhibitors EZSolution™ 3-Deazaneplanocin A 2409 1 mg 102052-95-9 3-Deazaneplanocin A 2060 250 µg, 1 mg 102052-95-9 Product Name Cat. No. Size CAS. No. 3-Deazaneplanocin A hydrochloride 2444 250 µg, 1 mg 120964-45-6 ABC294640 B1231 5 mg, 25 mg 915385-81-8 Sphingosine Kinase Inhibitor, SKI-I 2046 5 mg, 25 mg 306301-68-8 SCD1 (Stearoyl-CoA Desaturase 1) Inhibitors Sphingosine Kinase Inhibitor, SKI-II 2047 5 mg, 25 mg 312636-16-1 Product Name Cat. No. Size CAS. No. MF-438 B1178 5 mg, 25 mg 921605-87-0 Smad Inhibitors PluriSIn 1 2471 10 mg, 50 mg 91396-88-2 Product Name Cat. No. Size CAS. No. EZSolution™ SCD1 Inhibitor 2548 1 mg N/A Smad3 Inhibitor, SIS3 2227 1 mg, 5 mg 521984-48-5 SCD1 Inhibitor 1716 1 mg, 5 mg 103229-33-6 Sodium Channel Modulators Secretase Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Aconitine 2423 10 mg, 50 mg 302-27-2 Beta-Secretase Inhibitor I 7501 1 mg N/A Ambroxol hydrochloride 9688 100 mg, 500 mg 23828-92-4 Beta-Secretase Inhibitor II 7502 1 mg N/A Veratridine 2422 5 mg, 25 mg 71-62-5 BMS-299897 9606 5 mg, 25 mg 290315-45-6 SREBP (Sterol Regulatory Element-Binding BMS-708163 B1622 5 mg, 25 mg 1146699-66-2 Proteins) Activation Inhibitors Compound 34 1898 200 µg, 1 mg N/A Compound E 1949 250 µg, 1 mg 209986-17-4 Product Name Cat. No. Size CAS. No. Compound W 2208 50 mg, 250 mg 173550-33-9 Betulin 1942 5 mg, 25 mg 473-98-3 EZSolution™ DAPT 2663 5 mg 208255-80-5 Fatostatin 2035 5 mg, 25 mg 298197-04-3 DAPT 1855 5 mg 208255-80-5 Xanthohumol 2258 5 mg, 25 mg 6754-58-1 DBZ 1649 1 mg, 5 mg 209984-56-5 Stat Inhibitors IMR-1 B1131 5 mg, 25 mg 310456-65-6 Product Name Cat. No. Size CAS. No. L-685, 458 1713 250 µg 292632-98-5 Cryptotanshinone 2429 5 mg, 25 mg 35825-57-1 LY-411575 2648 1 mg, 5 mg 209984-57-6 Galiellactone 2623 100 µg, 500 µg 133613-71-5 LY2811376 B1606 5 mg, 25 mg 1194044-20-6 133550-30-8 LY2886721 2299 5 mg, 25 mg 1262036-50-9 477600-75-2 MK-0752 B1980 1 mg, 5 mg 471905-41-6 PathwayReady™ JAK/STAT Signaling 111358-88-4 Inhibitor Panel 26305-03-3 K864 8 Inhibitors MK-8931 B1315 1 mg, 5 mg 1286770-55-5 (Containing Cat. No. 1570, 1622, 1805, 2062-78-4 RO4929097 2011 1 mg, 5 mg 847925-91-1 1732, 1887, 1775, 1778, 1809) 501919-59-1 N/A Semagacestat 2430 1 mg, 5 mg 425386-60-3 857064-38-1 SGLT-2 (Sodium Glucose Co-Transporter 2) 1805 500 µg, 1 mg 111358-88-4 LLL12 1792 5 mg, 25 mg N/A Inhibitors MS-1020 1911 1 mg 1255516-86-9 Product Name Cat. No. Size CAS. No. 1826 100 mg, 500 mg 50-65-7 Bexgliflozin (EGT1442) B1929 1 mg, 5 mg 1118567-05-7 Pimozide 1887 50 mg, 250 mg 2062-78-4 Canagliflogin B1597 10 mg, 50 mg 842133-18-0 Resveratrol 1758 100 mg, 500 mg 501-36-0 Dapagliflozin 9452 10 mg, 50 mg 461432-26-8 SH-4-54 B1637 5 mg, 25 mg 1456632-40-8 Empagliflozin 2877 10 mg, 50 mg 864070-44-0 STA-21 2626 250 µg, 1 mg 28882-53-3 Ertugliflozin B1896 5 mg, 25 mg 1210344-57-2 Stat3 Activation Inhibitor, SPI 1813 2 mg N/A Ipragliflozin B1926 5 mg, 25 mg 761423-87-4 EZSolution™ Stat3 Inhibitor I, S3I-201 2541 5 mg 501919-59-1 LX-4211 9623 5 mg, 25 mg 1018899-04-1 Stat3 Inhibitor I, S3I-201 1775 5 mg, 25 mg 501919-59-1

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 18 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. Stat3 Peptide Inhibitor, Cell-Permeable 1778 1 mg, 5 mg N/A Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1 Stat5 Inhibitor 9484 1 mg, 5 mg 285986-31-4 Carfilzomib 2385 5 mg, 25 mg 868540-17-4 Stattic 2625 5 mg, 25 mg 19983-44-9 Celastrol 1940 5 mg, 25 mg 34157-83-0 SUMOYlation Inhibitors CEP-18770 2433 5 mg, 25 mg 847499-27-8 Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5 Product Name Cat. No. Size CAS. No. Clioquinol 2454 1 g, 5 g 130-26-7 Anacardic Acid 1849 5 mg, 25 mg 16611-84-0 DBeQ 1858 5 mg, 25 mg 177355-84-9 Ginkgolic acid C15:1 9523 5 mg, 25 mg 22910-60-7 DUB Inhibitor, NSC-632839 2570 5 mg, 25 mg 157654-67-6 TACE Inhibitors Eeyarestatin I 9602 5 mg, 25 mg 412960-54-4 (-)-Epigallocatechin gallate 1841 50 mg 989-51-5 Product Name Cat. No. Size CAS. No. Fenbendazole 2157 100 mg, 500 mg 43210-67-9 TAPI-0 2067 1 mg 143457-40-3 Ginkgolic acid C15:1 9523 5 mg, 25 mg 22910-60-7 TAPI-1 2068 1 mg 171235-71-5 HBX-41108 9608 5 mg, 25 mg 924296-39-9 TAPI-2 2069 1 mg 187034-31-7 Lactacystin (Synthetic) 1709 200 µg 133343-34-7 Tankyrase Inhibitors LDN-57444 2016 5 mg, 25 mg 668467-91-2 Product Name Cat. No. Size CAS. No. MDBN 2033 10 mg, 50 mg 1485-00-3 AZ-6102 B1200 5 mg, 25 mg 1645286-75-4 MG-115 1831 1 mg, 5 mg 133407-86-0 JW55 2612 5 mg, 25 mg 664993-53-7 MG-132 1703 5 mg, 25 mg 133407-82-6 MN64 B1127 10 mg, 50 mg 92831-11-3 MLN-4924 2566 500 µg 905579-51-3 XAV939 1727 1 mg 284028-89-3 NMS-873 9600 5 mg, 25 mg 1418013-75-8 NSC-687852 2021 5 mg, 25 mg 1009817-63-3 Thioredoxin inhibitors NSC-697923 B1091 5 mg, 25 mg 343351-67-7 Product Name Cat. No. Size CAS. No. ONX-0914 2555 5 mg, 25 mg 960374-59-8 Auranofin 2219 10 mg, 50 mg 34031-32-8 Oprozomib 2386 5 mg, 25 mg 935888-69-0 PX 12 2217 5 mg, 25 mg 141400-58-0 P5091 2277 5 mg, 25 mg 882257-11-6 Topoisomerase Inhibitors PS-341 1846 1 mg, 5 mg 179324-69-7 PYR-41 1925 5 mg, 25 mg 418805-02-4 Product Name Cat. No. Size CAS. No. SMER-3 2514 5 mg, 25 mg 67200-34-4 Camptothecin 1039 1 ml, 50 mg, 500 mg 7689-03-4 Spautin-1 2037 5 mg, 25 mg 1262888-28-7 Doxorubicin.HCl 1527 5 mg 25316-40-9 (±)-Thalidomide 2020 10 mg, 50 mg 50-35-1 Ellipticine 9579 5 mg, 25 mg 519-23-3 TAME Hydrochloride 2050 100 mg, 500 mg, 1 g 1784-03-8 Epirubicin Hydrochloride 1753 5 mg, 25 mg 56390-09-1 TCID 2204 5 mg, 25 mg 30675-13-9 Etoposide 1043 10 µl, 25 mg, 250 mg 33419-42-0 USP14 Inhibitor, IU1 1845 5 mg, 25 mg 314245-33-5 Etoposide phosphate 2896 10 mg, 50 mg 117091-64-2 VR23 B1515 5 mg, 25 mg 1624602-30-7 10-Hydroxycamptothecin B1995 25 mg, 100 mg 19685-09-7 WP-1130 2014 5 mg, 25 mg 856243-80-6 Irinotecan Hydrochloride 1752 50 mg, 250 mg 100286-90-6 β-Lapachone 2262 5 mg, 25 mg 4707-32-8 VCP-p97 (Valosin-Containing Protein-p97) Mitoxantrone 1885 50 mg, 250 mg 65271-80-9 Inhibitors Pixantrone maleate 1958 5 mg, 25 mg 144675-97-8 Product Name Cat. No. Size CAS. No. 518-28-5, Podophyllotoxin 2767 50 mg, 250 mg 4354-76-1 CB5083 B1032 5 mg, 25 mg 1542705-92-9 SW-044248 B1135 5 mg, 25 mg 522650-83-5 DBeQ 1858 5 mg, 25 mg 177355-84-9 TAS-103 B1841 5 mg, 25 mg 174634-08-3 Eeyarestatin I 9602 5 mg, 25 mg 412960-54-4 Topotecan hydrochloride B2050 10 mg, 50 mg 119413-54-6 MDBN 2033 10 mg, 50 mg 1485-00-3 Ubiquitin Activating Enzyme E1 Inhibitor ML-240 B1142 5 mg, 25 mg 1346527-98-7 NMS-873 9600 5 mg, 25 mg 1418013-75-8 Product Name Cat. No. Size CAS. No. PYR-41 1925 5 mg, 25 mg 418805-02-4 Wnt (Wingless Phenotype in Drosophila) Ubiquitin Ligase (E3) Inhibitors Signaling Inhibitors Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. CRT Inhibitor, iCRT5 1896 5 mg, 25 mg N/A NSC 146109 hydrochloride 1907 5 mg 59474-01-0 FH535 2657 5 mg, 25 mg 108409-83-2 NSC 66811 2009 5 mg 6964-62-1 ICG-001 2275 5 mg, 25 mg 847591-62-2 NSC-687852 2021 5 mg, 25 mg 1009817-63-3 IQ-1 1663 1 mg 331001-62-8 PRT4165 B1054 5 mg, 25 mg 31083-55-3 IWP-2 1962 5 mg, 25 mg 686770-61-6 SKPin C1 2343 5 mg, 25 mg 432001-69-9 IWP-3 2349 1 mg, 5 mg 687561-60-0 SMER-3 2514 5 mg, 25 mg 67200-34-4 IWP-4 2650 1 mg, 5 mg 686772-17-8 (±)-Thalidomide 2020 10 mg, 50 mg 50-35-1 JW55 2612 5 mg, 25 mg 664993-53-7 TCID 2204 5 mg, 25 mg 30675-13-9 KY02111 2264 5 mg, 25 mg 1118807-13-8 Ubiquitin Proteasome Pathway Inhibitors LGK974 2645 1 mg, 5 mg 1243244-14-5 Product Name Cat. No. Size CAS. No. PNU-74654 B1837 5 mg, 25 mg 113906-27-7 Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1 QS11 1680 5 mg 944328-88-5

18 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 19 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. WIKI-4 B1630 5 mg, 25 mg 838818-26-1 Agistatin B B1021 1 mg, 5 mg 144096-46-8 EZSolution™ Wnt Antagonist, C59 9493 1 mg 1243243-89-1 Agistatin D B1022 1 mg, 5 mg 144096-47-9 Wnt Antagonist, C59 2063 1 mg, 5 mg 1243243-89-1 Agistatin E B1023 1 mg, 5 mg 144096-48-0 XAV939 1727 1 mg 284028-89-3 AHU-377 9520 5 mg, 25 mg 149709-62-6 Other Inhibitors AM-095 9581 5 mg, 25 mg 1228690-36-5 AM-095 Sodium B1225 5 mg, 25 mg 1345614-59-6 Cancer Stem cell Inhibitors Amidepsine A, Humcola sp. 2147 500 µg, 1 mg 169181-28-6 Product Name Cat. No. Size CAS. No. Amidepsine D, Humcola sp. 2148 500 µg, 1 mg 79786-34-8 A37 B1577 5 mg, 25 mg 896795-60-1 Andrastin A, Aspergillus fumigatus 2149 250 µg, 1 mg 174232-42-9 BRD7116 B1578 5 mg, 25 mg 329059-55-4 Apilimod mesylate B1129 5 mg, 25 mg 870087-36-8 Cancer Cell Stemness Inhibitor I 2476 5 mg, 25 mg 83280-65-3 Apixaban B1855 10 mg, 50 mg 503612-47-3 Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7 Aprepitant 9531 10 mg, 50 mg 170729-80-3 Galiellactone 2623 100 µg, 500 µg 133613-71-5 B1186 10 mg, 50 mg 129722-12-9 GDC-0084 B1656 5 mg, 25 mg 1382979-44-3 AT 56 2592 5 mg, 25 mg 162640-98-4 GNE 477 B1657 5 mg, 25 mg 1032754-81-6 AT-406 B1829 5 mg, 25 mg 1071992-99-8 ITE B1579 5 mg, 25 mg 448906-42-1 Atazanavir B1901 5 mg, 25 mg 198904-31-3 ML239 2696 5 mg, 25 mg 1378872-36-6 Atglistatin B1864 5 mg, 25 mg 1469924-27-3 ML243 2515 5 mg, 25 mg 1426576-80-8 Aurantimycin A 9692 1 mg, 5 mg 162478-50-4 PF-4989216 B1659 5 mg, 25 mg 1276553-09-3 Avibactam sodium 9569 5 mg, 25 mg 1192491-61-4 PND-1186 2823 5 mg, 25 mg 1061353-68-1 AX-024 hydrochloride B2013 5 mg, 25 mg 1704801-24-0 Pamaote B1593 5 mg, 25 mg 3546-41-6 AZD-1283 2838 5 mg, 25 mg 919351-41-0 Salinomycin Sodium B1584 25 mg, 100 mg 55721-31-8 AZD-1981 9611 5 mg, 25 mg 802904-66-1 SC-26196 B1580 5 mg, 25 mg 218136-59-5 AZD-4635 B2012 5 mg, 25 mg 1321514-06-0 Thioridazine Hydrochloride B1581 1 g, 5 g 130-61-0 AZD-5069 B2053 5 mg, 25 mg 878385-84-3 TY-52156 B1582 5 mg, 25 mg 934369-14-9 Azeliragon B1152 5 mg, 25 mg 603148-36-3 Verteporfin B1583 5 mg, 25 mg 129497-78-5 BAY 57-1293 2556 5 mg, 25 mg 348086-71-5 VS-5584 9603 1 mg, 5 mg 1246560-33-7 BD 1047 dihydrobromide B1069 10 mg, 50 mg 138356-21-5 Protein Synthesis Inhibitors Bedaquiline 9598 5 mg, 25 mg 843663-66-1 Product Name Cat. No. Size CAS. No. B1913 5 mg, 25 mg 738606-46-7 Betulin 1942 5 mg, 25 mg 473-98-3 Anisomycin 1549 10 mg 22862-76-6 Birinapant 2597 1 mg, 5 mg 1260251-31-7 Aurodox 2317 1 mg 12704-90-4 BMS-303141 2821 10 mg, 50 mg 943962-47-8 (-)-6-Azauridine 2’, 3’,5’-triacetate B1025 50 mg, 250 mg 2169-64-4 Bongkrekic Acid, Triammonium Salt 1820 100 µg 11076-19-0 6-Azauridine B1024 100 mg, 500 mg 54-25-1 Bosentan B1857 1 mg, 5 mg 147536-97-8 Blasticidin S Hydrochloride 1859 25 mg, 100 mg 3513-03-9 BQ-123 Sodium Salt B1552 1 mg, 5 mg 136553-81-6 Clindamycin hydrochloride 2627 10 mg, 50 mg 21462-39-5 BQ-610 B1553 1 mg, 5 mg 141595-53-1 Cycloheximide 1041 1 ml, 1 g, 5 g 66-81-9 BQ-788 Sodium Salt B1554 500 μg, 1 mg 156161-89-6 Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7 BTZ043 B1206 5 mg, 25 mg 1161233-85-7 Erythromycin 9619 5 g , 25 g 114-07-8 BV6 B1332 5 mg, 25 mg 1001600-56-1 G418 Sulfate 1557 1 g, 5 g, 25 g 108321-42-2 680C91 2292 5 mg, 25 mg 163239-22-3 Kanamycin Sulfate, USP 2498 5 g, 25 g 25389-94-0 Capsaicin 2521 50 mg, 250 mg 404-86-4 Kirromycin B1236 1 mg, 5 mg 50935-71-2 Catharanthine 1749 100 mg, 1 g 2468-21-5 Neomycin sulfate 9620 25 g, 100 g 1405-10-3 CB-839 B1179 5 mg, 25 mg 1439399-58-2 Nourseothricin sulfate 2882 50 mg, 100 mg, 500 mg, 1 g 96736-11-7 CBL0137 B2036 5 mg, 25 mg 1197996-80-7 Paromomycin Sulfate B1528 1 g, 5 g 1263-89-4 CCF-642 B2009 5 mg, 25 mg 346640-08-2 EZSolution™ Puromycin Dihydrochloride 1861 100 mg 58-58-2 25 mg, 100 mg, 250 mg, 9434 5 mg, 25 mg 5 mg, 25 mg 285986-88-1 Puromycin Dihydrochloride 1860 58-58-2 500 mg, 1 g Ceralifimod B1289 5 mg, 25 mg 891859-12-4 Roxithromycin 9621 1 g, 5 g 80214-83-1 CFTR Inhibitor, GlyH-101 2863 5 mg, 25 mg 328541-79-3 Streptomycin Sulfate 2517 50 g, 100 g, 500 g 3810-74-0 CH-223191 2723 5 mg, 25 mg 301326-22-7 Tetracycline Hydrochloride B1535 10 g, 50 g 64-75-5 CHD-5 2693 5 mg, 25 mg 289494-16-2 Thiostrepton 9677 50 mg, 250 mg 1393-48-2 Chetomin 2180 1 mg 1403-36-7 Tildipirosin 9673 1 mg, 5 mg 328898-40-4 CHIR-090 B1852 5 mg, 25 mg 728865-23-4 Protein Transport Inhibitors Chloroquine Diphosphate 1825 100 mg, 500 mg 50-63-5 Chlorpromazine Hydrochloride B1992 100 mg, 500 mg 69-09-0 Product Name Cat. No. Size CAS. No. CHR2797 2720 5 mg, 25 mg 238750-77-1 EZCell™ Protein Transport Inhibitor 20350-15-6 Cocktail (500X) K932 500 µl CHS-828 2044 5 mg, 25 mg 200484-11-3 28636-21-7 (Containing Cat. No. 1560, 1808) CID 2745687 1969 5 mg, 25 mg 264233-05-8 Other Inhibitors CID-5951923 2690 5 mg, 25 mg 749872-43-3 Product Name Cat. No. Size CAS. No. Cladribine B2037 5 mg, 25 mg 4291-63-8 A-803467 2559 5 mg, 25 mg 944261-74-9 Congo Red 2588 100 mg, 500 mg 573-68-0 Acivicin B1028 1 mg, 5 mg 42228-92-2 CPI-444 B1970 5 mg, 25 mg 1202402-40-1

Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 20 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. CPI-613 9464 10 mg, 50 mg 95809-78-2 L-67 9633 5 mg, 25 mg 325970-71-6 CT-2584 B1182 5 mg, 25 mg 166981-13-1 L-DON B1955 5 mg, 25 mg 157-03-9 Curcubitacin E B1592 1 mg, 5 mg 18444-66-1 Lamotrigine B1234 10 mg, 50 mg 84057-84-1 CWHM-12 B1251 5 mg, 25 mg 1564286-55-0 Lasofoxifene tartrate 9680 5 mg, 25 mg 190791-29-8 DiscoveryPak™ Cytochlor-THU Set 32387-56-7 K955 2 Radiosensitizers LCL161 B1601 5 mg, 25 mg 1005342-46-0 (Containing Cat. No. 2833, 1671) 18771-50-1 Leelamine hydrochloride 2717 5 mg, 25 mg 16496-99-4 Cytochlor 2833 5 mg, 25 mg 32387-56-7 2876 5 mg, 25 mg 182431-12-5 DBeQ 1858 5 mg, 25 mg 177355-84-9 LY404187 2698 5 mg, 25 mg 211311-95-4 Decylubiquinone 2099 1 mg, 10 mg 55486-00-5 Macitentan B1856 5 mg, 25 mg 441798-33-0 DG051 B1105 1 mg, 5 mg 929916-05-2 Madrasin B1278 5 mg, 25 mg 374913-63-0 DHEA 2172 100 mg, 500 mg 53-43-0 Mambalgin-1 2421 50 µg, 100 µg N/A DMOG 2216 5 mg, 25 mg 89464-63-1 Maraviroc B2044 5 mg, 25 mg 376348-65-1 Dofetilide B1189 5 mg, 25 mg 115256-11-6 6-Mercaptopurine (monohydrate) B2039 50 mg, 250 mg 50-44-2 Dynasore 1900 5 mg, 25 mg 304448-55-3 MDV-3100 9479 10 mg, 50 mg 915087-33-1 E-7046 B1966 5 mg, 25 mg 1369489-71-3 Mifepristone 1561 50 mg 84371-65-3 Edoxaban Tosylate 2714 5 mg, 25 mg 480449-71-6 Mirin B1075 10 mg, 50 mg 1198097-97-0 Eliglustat B1217 5 mg, 25 mg 491833-29-5 MK-1439 B1250 5 mg, 25 mg 1338225-97-0 Embelin B1600 5 mg, 25 mg 550-24-3 ML-354 9415 5 mg, 25 mg 89159-60-4 Entacapone B1190 10 mg, 50 mg 130929-57-6 ML161 2689 5 mg, 25 mg 423735-93-7 Epalrestat 2397 5 mg, 25 mg 82159-09-9 MPEP hydrochloride B1151 10 mg, 50 mg 219911-35-0 Eptifibatide 2439 1 mg 188627-80-7 3-Nitropropionic acid 2093 50 mg, 250 mg 504-88-1 Ethynylcytidine B1266 5 mg, 25 mg 180300-43-0 2-Nitro-5-thiothiocyanatobenzoic acid B1316 50 mg, 250 mg 30211-77-9 (R)-(+)-Etomoxir B1104 1 mg, 5 mg 124083-20-1 NS-3763 B1814 5 mg, 25 mg 70553-45-6 Evans Blue Tetrasodium 2586 1 g 314-13-6 NS6180 B1640 5 mg, 25 mg 353262-04-1 Ezatiostat 2608 5 mg, 25 mg 168682-53-9 NSC-207895 B1228 5 mg, 25 mg 58131-57-0 10058-F4 2739 5 mg, 25 mg 403811-55-2 NSC-348884 B1204 5 mg, 25 mg 81624-55-7 Fatostatin 2035 5 mg, 25 mg 298197-04-3 NVS-SM1 B1844 5 mg, 25 mg 1562338-42-4 FCCP 2398 5 mg, 25 mg 370-86-5 ODQ 2051 10 mg, 50 mg 41443-28-1 Felbamate B2004 10 mg, 50 mg 25451-15-4 ONO 1078 B1099 5 mg, 25 mg 103177-37-3 Fevipiprant B1588 5 mg, 25 mg 872365-14-5 OSMI-1 B1916 5 mg, 25 mg 1681056-61-0 Fidaxomicin 2832 1 mg, 5 mg 873857-62-6 Ozanimod B1196 5 mg, 25 mg 1306760-87-1 FITM B1859 1 mg, 5 mg 932737-65-0 PBTZ169 B1205 5 mg, 25 mg 1377239-83-2 FK-866 1914 1 mg, 5 mg 658084-64-1 PD-1/PD-L1 Inhibitor 1 B1213 5 mg, 25 mg 1675201-83-8 FLI-06 2603 5 mg, 25 mg 313967-18-9 PD-1/PD-L1 Inhibitor 2 B1050 5 mg, 25 mg 1675203-84-5 Fosaprepitant 9529 10 mg, 50 mg 172673-20-0 PD-123319 ditrifluoroacetate 9640 5 mg, 25 mg 130663-39-7 FPS-ZM1 B1933 5 mg, 25 mg 945714-67-0 Pellitorine 2053 1 mg, 5 mg 18836-52-7 Fulvestrant B1863 5 mg, 25 mg 129453-61-8 Pemetrexed B1862 50 mg, 250 mg 137281-23-3 Fusicoccin B1625 1 mg, 2 mg 20108-30-9 Pentostatin B2038 5 mg, 25 mg 53910-25-1 FX1 B2010 5 mg, 25 mg 1426138-42-2 Perampanel B2066 5 mg, 25 mg 380917-97-5 Ganciclovir 1918 50 mg, 250 mg, 1 g 82410-32-0 PF-04418948 B1168 5 mg, 25 mg 1078166-57-0 GBR-12935 B1998 10 mg, 50 mg 76778-22-8 PF-06291874 B2001 5 mg, 25 mg 1393124-08-7 GDC-0152 B1602 5 mg, 25 mg 873652-48-3 PF-3274167 B1026 5 mg, 25 mg 900510-03-4 DiscoveryPak™ Gemcitabine-THU Set 122111-03-9 K841 2 Modulators (Containing Cat. No. 1759, 1671) 18771-50-1 PF-8380 B1927 1 mg, 5 mg 1144035-53-9 Geodin 9685 1 mg, 5 mg 427-63-4 Phloretin 9625 100 mg, 500 mg 60-82-2 GIBH-130 B2071 5 mg, 25 mg 1252608-59-5 Pimecrolimus 1593 5 mg, 25 mg 137071-32-0 GKT-137831 9444 5 mg, 25 mg 1218942-37-0 PK 11195 2054 10 mg, 50 mg 85532-75-8 GLPG-1690 B1850 5 mg, 25 mg 1628260-79-6 3PO B2018 10 mg, 50 mg 13309-08-5 Glutaminase C-IN-1 (968) B1198 5 mg, 25 mg 311795-38-7 9526 10 mg, 50 mg 171228-49-2 GSK-961081 B1590 5 mg, 25 mg 743461-65-6 Prasugrel 9472 10 mg, 50 mg 150322-43-3 GSK1325756 B1103 1 mg, 5 mg 954126-98-8 PSI-7977 2715 5 mg, 25 mg 1190307-88-0 GSK2190915 B1891 1 mg, 5 mg 936350-00-4 PTC-124 9421 10 mg, 50 mg 775304-57-9 GSK2330672 B1102 1 mg, 5 mg 1345982-69-5 PTC-209 B1055 5 mg, 25 mg 315704-66-6 GW 4869 dihydrocloride 2417 1 mg, 5 mg 6823-69-4 QNZ46 B2007 5 mg, 25 mg 1237744-13-6 GYY 4137 1908 5 mg, 25 mg 106740-09-4 R162 B1180 5 mg, 25 mg 64302-87-0 HA 130 B1192 5 mg, 25 mg 1229652-21-4 RAD140 B1211 10 mg, 50 mg 1182367-47-0 Heptelidic Acid 2215 250 µg, 1 mg 74310-84-2 Retro-2 2516 5 mg, 25 mg 1429192-00-6 Itaconic acid 2576 1 g, 5 g 97-65-4 RI-1 B1823 5 mg, 25 mg 415713-60-9 Ivabradine Hydrochloride B1595 10 mg, 50 mg 148849-67-6 Rivaroxaban B1854 10 mg, 50 mg 366789-02-8 JNJ-31020028 9648 5 mg, 25 mg 1094873-14-9 RK-33 B1273 5 mg, 25 mg 1070773-09-9 K858 B1073 10 mg, 50 mg 72926-24-0 Ro 48-8071 fumarate B1042 10 mg, 50 mg 189197-69-1 Ki 16425 9545 5 mg, 25 mg 355025-24-0 RQ-002303078 9636 10 mg, 50 mg 1254205-52-1

20 Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 21 Product Name Cat. No. Size CAS. No. Product Name Cat. No. Size CAS. No. RSV-604 B1846 5 mg, 25 mg 676128-63-5 trans-ISRIB B1906 5 mg, 25 mg 1597403-47-8 S0859 9425 5 mg, 25 mg 1019331-10-2 EZSolution™ Triacsin C 9683 100 µg, 500 µg 76896-80-5 Salubrinal 1980 5 mg 405060-95-9 Triapine B1174 10 mg, 50 mg 143621-35-6 SB-715992 2468 5 mg, 25 mg 336113-53-2 Triclopidine hydrochloride B1141 50 mg, 250 mg 53885-35-1 SB-742457 9568 5 mg, 25 mg 607742-69-8 Trifluorothymidine B1126 10 mg, 50 mg 70-00-8 SM-164 B1816 250 μg, 1 mg 957135-43-2 Triflupromazine hydrochloride B1993 100 mg, 500 mg 1098-60-8 Suplatast tosylate 2624 10 mg, 50 mg 94055-76-2 Troviridine B1212 10 mg, 50 mg 149488-17-5 Suvorexant B1321 5 mg, 25 mg 1030377-33-3 Tunicamycin 2802 5 mg, 25 mg 11089-65-9 Syrosingopine B1323 1 mg, 5 mg 84-36-6 U-104 9631 5 mg, 25 mg 178606-66-1 T-5224 9546 5 mg, 25 mg 530141-72-1 U-93631 B1851 5 mg, 25 mg 152273-12-6 TAS-301 9644 10 mg, 50 mg 193620-69-8 UK-371804 B1843 5 mg, 25 mg 256477-09-5 TCS OX2 29 B1838 5 mg, 25 mg 372523-75-6 UK-5099 B1952 5 mg, 25 mg 56396-35-1 Tenofovir disoproxil fumarate 1920 5 mg, 25 mg 202138-50-9 UMI-77 B1108 5 mg, 25 mg 518303-20-3 EZSolution™ Tetrahydrouridine 2355 25 mg 18771-50-1 XAV939 1727 1 mg 284028-89-3 Tetrahydrouridine 1671 10 mg, 25 mg 18771-50-1 YK-4-279 2846 5 mg, 25 mg 1037184-44-3 TG6-10-1 9646 5 mg, 25 mg 1415716-58-3 YM-90709 B1074 10 mg, 50 mg 163769-88-8 Thapsigargin 1558 1 mg 67526-95-8 YM155 2310 5 mg, 25 mg 781661-94-7 Thiabendazole 2161 1 g 148-79-8 (Z)-4-Hydroxytamoxifen B1114 5 mg, 25 mg 68047-06-3 Tiplaxtinin B1634 5 mg, 25 mg 393105-53-8 Z-VRPR-FMK B1238 250 µg, 1 mg 1381885-28-4 TM-5275 Sodium salt B1884 5 mg, 25 mg 1103926-82-4 Zanamivir B1900 10 mg, 50 mg 139110-80-8 Tranilast 1876 10 mg, 50 mg 53902-12-8

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