Adooq Bioscience Kinase Inhibitors Catalog 2014-2015

Adooq Bioscience

Innovation through Bioscience

Kinase Inhibitors Catalog 2014-2015

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Who We Are Australia Sapphire Bioscience Pty. Ltd. Austria Hölzel Diagnostika Handels GmbH www.sapphirebioscience.com www.hoelzel-biotech.com [email protected] [email protected] Tel: 1800 062 088 Fax: +61296981022 Tel: +49(0)221-1260266 Fax: +49(0)221-1260267 Adooq Bioscience is one of the world leading suppliers of high-performance life- Canada Cedarlane China Shenzhen Minn Bolin Bio-Tech Co., Ltd. science reagents and reference compounds for the research fields. Now, Adooq www.cedarlanelabs.com www.mbolin-lktlabs.com/cn has more than 4200 products with validated biological and pharmacological [email protected] [email protected] Tel: +1(289)288-0001 Fax: +1(289)288-0020 Tel: +86-755-2510-6053 Fax: +86-755-2510-6053 activities, and an unique collection of over 2000 inhibitors on HDAC, PI3K, China Guangzhou Whiga Technology ltd. China ADVANCED TECH. & IND. CO., LTD. Apoptosis and more signaling pathways in stock. www.whiga.com.cn www.advtechind.com [email protected] [email protected] Tel: +862084224519 Fax: +862084224925 Tel: +852-23902293 Fax: +852-27898314

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Cathepsin 34 Progesterone Receptors 44 Histone demethylases 34 Renin-angiotensin-aldosterone system (RAAS) 45 Stem Cell Differentiation 34 Androgen Receptors 45 Contents PPAR 45 GSK-3 / Wnt / Hedgehog...... 35 Liver X receptors (LXRs) 45 Aromatase 46 Apoptosis...... 1 PI3K / Akt / mTOR...... 20 γ-Secretase 35 Retinoic Acid Receptors 46 Bcl-2 Family 1 Akt 20 Hedgehog 35 Glucocorticoid receptors 46 Caspase 1 Ferroptosis 20 Wnt 35 p53 1 PI3-Kinase (PI3K) 20 β-catenin 36 GSK-3 36 Transferases...... 46 TNF-α 1 mTOR 22 IAP 1 PDK1 23 Smoothened 36 Glucocorticoid receptors 46 RasGAP (Ras- P21) 2 Vitamin D Receptors 46 PERK 2 Transporters...... 37 GnRH receptor 46 Receptor Tyrosine Kinases...... 23 GPR 46 EGFR/HER2 23 ATPase 37 Phosphorylases 46 Angiogenesis...... 2 DNA-dependent protein kinase (DNA-PK) 23 Multidrug Transporters 37 Methyltransferases 47 EGFR / HER2 2 Ribosomal S6 protein kinases (RSK) 23 Sodium-dependent Glucose Cotransporter (SGLT) 37 Protein Prenyltransferases 47 MDM2 2 FGFR 24 Monocarboxylate transporters (MCT) 37 FPTase 47 Apoptosis Inducers 2 PDGFR 24 Neurotransmitter Transporters 38 Histone Methyltransferase 47 FGFR 3 VEGFR 24 AMPA receptor 38 Histone Acetyltransferases 47 PDGFR 3 Type 1 insulin-like growth factor receptor (IGF-1R) 24 DNA Methyltransferases 47 VEGFR 3 FLT3 (FMS-like tyrosine kinase 3) 25 Ion Channels...... 38 Vascular Disrupting Agent (VDA) 4 c-MET 25 Calcium Channels 38 Ubiquitin...... 48 HIF 5 ALK 25 P-gp 38 BCR-ABL 26 activating enzyme E1 48 CRM1 38 E3 ubiquitin ligase 48 MAPK...... 5 FAK 26 Ligand-gated Ion Channels 38 SRC 26 DUB 48 MEK/ERK 5 Sodium Channels 39 c-Kit 27 5-alpha-reductase 5 Potassium Channels 39 Spleen tyrosine kinase (Syk) 27 Others...... 48 Antiangiogenics 5 Chloride Channels 39 Tie-2 27 p38-MAPK 6 Cystic Fibrosis Transmembrane Regulator (CFTR) 39 Other inhibitors 48 Bone Morphogenetic Proteins (BMP) 28 JNK/c-Jun 6 Transient Receptor Potential Channels 40 p97 48 Bruton's tyrosine kinase 28 Raf 6 Carbonic Anhydrase 54 AMPK / Insulin Receptor...... 40 Cholinesterase 54 NF-kB/IkB...... 28 Casein Kinase 2 54 Cell Cycle...... 7 AMPK 40 NF-kB 28 Soluble guanylyl cyclase (sGC) 54 Checkpoint Kinase 7 Axl 28 Reagents 54 cyclin-dependent kinases (CDKs) 8 ATM / ATR...... 40 Tyrosine kinase 28 Integrin Receptors 54 Checkpoint Control Kinases 9 Trk Receptors 28 ATM 40 Toll-like Receptors 54 Aurora Kinase 9 Cytokines 29 NMDA Receptors 40 Beta-secretase (BACE) 54 PARP 9 IKK 29 ATR 40 LRRK2 54 Polo-like kinases (PLKs) 10 MELK 54 Rho-Kinase (ROCKs) 10 7-TM Receptors...... 41 β-lactamase 55 Topoisomerase 11 JAK / Stat...... 29 Gluconeogenesis 55 Microtubules 11 JAK 29 5-HT Receptors 41 Cholinesterases 55 Synthases / Synthetases 12 Stat 29 Adrenergic Receptors 41 Aldose Reductase 55 RNA/DNA Polymerase 12 Pim Kinase 29 Acetylcholine Muscarinic Receptors 42 Nitric Oxide Signaling 55 Telomerase 12 Histamine Receptors 42 Adenylyl Cyclase 55 Ligases 12 TGF-β / Smad...... 30 Dopamine Receptors 42 IDH1 55 Reverse Transcriptase 12 Opioid Receptors 42 LSD1 inhibitor 55 TGF-β / Smad Inhibitors 30 GABA Receptors 42 Protein Kinase C (PKC) 30 Casein Kinase 1 55 Cell Metabolism...... 13 Purinergic (P2Y) Receptors 42 Lipoxygenase 55 Metabotropic glutamate receptors (mGluR) 43 Sigma-1 receptor 55 Cytochrome P450 13 Proteases...... 30 Angiotensin Receptors 43 Mitosis 13 Caspase 30 Melatonin Receptors 43 -Amyloid 14 β Protein Kinase A 30 Peptide Receptors 43 Phosphodiesterases (PDEs) 14 Protein kinase D (PKD) 30 Smoothened Receptors 43 Hydroxylases 14 Proteasome 30 Chemokine Receptors (CCR5) 43 Dihydrofolate reductase (DHFR) 15 HCV Protease 31 G Protein 43 Dehydrogenases 15 HIV Protease 32 Platelet-Activating Factor (PAF) Receptors 43 Cyclooxygenase (COX) 15 Heat Shock Proteins (HSP) 32 Endothelin Receptors 43 Antimetabolite 16 Aminopeptidase 33 P2X Receptor 43 Histone Deacetylase (HDAC) 16 Integrase 33 LPA Receptor 43 Sir2-like Family Deacetylases (sirtuins) 17 Dipeptidyl Peptidase IV (DPP-4) 33 Prostanoid Receptors 43 Monoamine Oxidase (MAO) 17 Thrombin 33 Adenosine Receptors 44 Factor Xa 17 Angiotensin-Converting Enzyme (ACE) 33 Cannabinoid Receptors 44 Kinesin Spindle Protein 18 Matrix Metalloprotease 33 Neurotensin Receptors 44 DNA, RNA and Protein Synthesis 18 Other Proteases 33 CYP17 18 MMP 34 Endocrinology / Hormones...... 44 Phospholipases 19 Lipid Metabolism 19 Pregnane X Receptors 44 FAAH 19 Epigenetics...... 34 Estrogen Receptors 44 CETP 19 Bromodomain 34 Leukotriene receptor 44 DNA Methyltransferases 19 Orexin Receptors 44 HMG-CoA Reductase 19 Stem Cells...... 34 Somatostatin Receptors 44 Neuronal Metabolism 19 NK1 Receptors 44 Stem Cell Proliferation 34 IDO 19 Protease-Activated Receptors (PAR) 44

YM155 is a novel small molecule survivin suppressant with an IC50 of 0.54 nM for the inhibition of survivin promoter activity. MDM2 Apoptosis *Available package size: 5,10,25,100mg A10657 Nutlin-3 A11163 AT-406 A11179 NSC-207895 (XI-006) VX-765 is a novel Caspase-1 inhibitor,which is an enzyme that A11928 LCL-161 A11501 Nutlin 3a Bcl-2 Family controls the generation of two cytokines, IL-1b and IL-18. A12738 Birinapant (TL32711) A11502 Nutlin 3b A10022 ABT-263 (Navitoclax) *Available package size: 5,10,50,100mg A13582 MDM2 Inhibitor A10255 ABT-737 RasGAP (Ras- P21) A11090 PAC-1 A11944 Apoptosis Activator 2 A10935 Tipifarnib (Zarnestra) A12373 Z-VAD-FMK A11225 Pluripotin (SC-1) A13070 LY573636 (Tasisulam) A11930 PF-3758309 p53

A10491 JNJ 26854165 MDM2 antagonist Nutlin-3 is a potent inducer of apoptosis. *Available package size: 5,25,50,100mg

PF-3758309 is a small-molecule p21-activated kinase inhibitor Apoptosis Inducers ABT-737 is a pan-Bcl-2 inhibitor. IC50 values ranged from 192 nM (the inhibiting oncogenic signaling and tumor growth. A10582 Methylprednisolone *Available package size: 5,10,25,50mg A11279 FK866 *Available package size: 5,10,50,100mg pre-B cell line Hal-01) to <10 μM (Nalm-6, K562 and HL-60). A13750 Hypothemycin A11635 Cyclophosphamide monohydrate A10665 Obatoclax mesylate (GX15-070) JNJ-26854165 is one of p53-activating agents and synergizes with A11988 Gambogic acid A10955 TW-37 AraC or doxorubicin to induce p53-mediated apoptosis and may provide a novel therapeutic approach for the treatment of acute PERK A11448 HA14-1 leukemias. A12500 ABT-199 *Available package size: 5,10,50,100mg A12792 GSK2606414 A12743 BM-1074 A11931 RITA (NSC 652287) A13577 GSK2656157 A12823 Sabutoclax A11943 Tenovin-1 A13816 ISRIB (trans-isomer) A12907 BAM 7 A12305 Tenovin-6 A13578 AT101 A12449 Pifithrin-u A12450 Pifithrin-beta A12451 Pifithrin-alpha Angiogenesis A12930 NSC 319726 A13581 PRIMA-1 EGFR / HER2 A13727 Tenovin-3 A10043 AEE788 TNF-α A10047 AG-490 A10522 Lenalidomide (CC-5013) AT101, the R-(-) enantiomer of Gossypol acetic acid, binds with Bcl- A10743 Pomalidomide (CC-4047) A11957 Bay 11-7821 inhibit BIR3 domain and BID. 2, Bcl-xL and Mcl-1 with Ki of 0.32 μM, 0.48 μM and 0.18 μM; does not A11973 Necrostatin-1 BIBW2992 (Afatinib) is tyrosine kinase inhibitor (TKI) that *Available package size: 10,25,50,100mg A12748 QNZ irreversibly inhibits human epidermal growth factor receptor 2 (Her2) and epidermal growth factor receptor (EGFR) kinases. Caspase IAP AG-490 is a selective inhibitor of EGF receptor tyrosine kinase (IC50 *Available package size: 5,10,25,100mg A10984 VX-765 *Available package size: 10,50,100,200mg A10362 Erlotinib Hydrochloride A11002 YM155 values are 2 and 13.5 μM for EGFR and ErbB2 respectively). A10422 Gefitinib (Iressa) A10053 Tyrphostin AG 879 A10514 Lapatinib Ditosylate A10062 AST-6 A10612 Mubritinib (TAK 165) A10116 AZD8931 A10638 Neratinib (HKI-272) A10141 BIBW2992 (Afatinib) A10678 OSI-420 A10210 Chrysophanic acid (Chrysophanol) A10702 PD153035 (HCl salt) A10211 Canertinib (CI-1033) A10706 Pelitinib (EKB-569) A10242 CP-724714

A10990 WZ3146 A12650 PKC 412 A10049 Albendazole TSU-68 (SU-6668) is an inhibitor of RTKs involved in VEGF, bFGF and PDGF signaling, which inhibits endothelial cell proliferation. A10991 WZ4002 A10101 Tivozanib (AV-951) *Available package size: 5,10,50,100mg A10992 WZ8040 A10103 Axitinib A11022 AG-1478 (Tyrphostin AG-1478) A10137 Bibf1120 (Vargatef) A10963 Vandetanib (ZD6474) A11027 Arry-380 A10967 Vatalanib (PTK787) 2HCl Base A10996 XL184 free base (Cabozantinib)

PKC 412 is a broad spectrum protein kinase inhibitor. Inhibits BIBF1120 (Vargatef) is a novel triple angiokinase inhibitor that inhibits three growth factor receptors simultaneously: VEGFR, PDGF 1, Flt3, Cdk1/B, PKA, c-Kit, c-Fgr, c-Src, VEGFR1 and EGFR. Displays XL184 free base (Cabozantinib) is a small molecule designed to conventional PKC isoforms (α, β, γ), PDFRβ, VEGFR2, Syk, PKCη, Flk- and FGFR. potent antitumor activity. inhibit multiple receptor tyrosine kinases, specifically MET and *Available package size: 5,10,50,100mg *Available package size: 5,10,25mg VEGFR2. ARRY-380 is an ErbB-2 inhibitor that selectively binds to and inhibits A10162 Brivanib alaninate (BMS-582664) the phosphorylation of ErbB-2, resulting in growth inhibition and A12867 CGP-52411 *Available package size: 5,10,50,100mg A10185 Cediranib (AZD2171) death of ErbB-2-expressing tumor cells. A12868 ARRY-543 A11396 E-7050 (Golvatinib) A10204 Chloroxine *Available package size: 5,10,50,100mg A13588 Tyrphostin AG 183 A11496 Motesanib (AMG706) A10248 CYC116 A11028 AV-412 A13681 AZD-9291 A11557 SU14813 A10254 Brivanib (BMS-540215) A11051 PF299804 A13718 Icotinib Hydrochloride A11772 CP-547632 A11057 XL647 A13755 CNX-2006 A11954 ZM 323881 hydrochloride A11155 AST-1306 A13825 Icotinib A11955 ZM 306416 hydrochloride A11158 ARRY334543 A12027 (-)-Catechin gallate A11209 BMS 599626 (AC480) FGFR A12437 SU 5416 (Semaxinib) A11236 TAK-285 A10703 PD173074 A11075 AZD4547 Brivanib (BMS-540215) is a VEGFR -2 inhibitor with an IC50 of 25 A11159 BGJ398 (NVP-BGJ398) nM and Ki of 26 nM. A11244 LY 2874455 *Available package size: 5,10,50,200mg A10259 Imatinib (Gleevec) PDGFR SU 5416 is an inhibitor of vascular endothelial growth factor receptor A10340 E7080 (Lenvatinib) (VEGFR) that also inhibits other tyrosine kinases KIT, MET, FLT3 and A10504 KRN 633 RET. TAK-285 is an investigational HER2/EGFR inhibitor that penetrates A10880 Sunitinib Malate *Available package size: 10,25,50,100mg the CNS in Rats with an Intact Blood Brain Barrier (BBB). A10903 Telatinib (BAY 57-9352) *Available package size: 5,10,25,50mg A13234 SKLB1002 A11052 Crenolanib (CP-868596) A13377 SAR131675 A11263 BMS-690514 A11350 CP-673451 A13465 SKLB610 A11334 BIBX 1382 A11581 Toceranib (PHA 291639, SU 11654) A13966 TPT-260 (Dihydrochloride)

E7080 is a multi-kinase inhibitor that inhibits both VEGFR2 and VEGFR3 kinases. *Available package size: 5,10,50,100mg Toceranib is a kinase inhibitor with both antitumor and antiangiogenic activity through inhibition of KIT, vascular endothelial A10495 Kaempferol A10502 Ki8751 *Available package size: 5,10,25,50mg TPT-260 is a thiophene thiourea derivative. BIBX 1382 is a cell-permeable pyrimido-pyrimidine compound that growth factor receptor 2, and PDGFRβ. A10608 Motesanib Diphosphate (AMG-706) acts as a potent, reversible, ATP-competitive, and highly selective A10699 Pazopanib Hydrochloride (GW786034) *Available package size: 5,10,25,50mg inhibitor of EGFR. A11753 MK-2461 A10893 Taxifolin *Available package size: 5,10,25mg A11978 Delphinidin chloride A10953 TSU-68 (SU6668) Vascular Disrupting Agent (VDA) A11407 Apatinib (YN968D1) A10324 DMXAA (ASA404) A11558 SU-5402 VEGFR

A11752 Lapatinib (free base) A10025 Linifanib (ABT-869) A11948 AP26113 A11949 AG-17 Linifanib (ABT-869) is a structurally novel, potent inhibitor of RTK, VEGF and PDGF with IC50 of 0.2, 2, 4, and 7 nM for human endothelial A12448 Butein *Available package size: 5,10,50,100mg cells, PDGFR-β, KDR, and CSF-1R, respectively.

DMXAA (ASA404) is a tumor-vascular disrupting agent (tumor-VDA) A11441 GDC-0973 that attacks the blood supply of a cancerous tumor to cause tumor 5-alpha-reductase downstream activation of MAPKAP kinase-2 and heat shock protein regression. A11493 MEK162 (ARRY-438162) 27.SB 203580 is a specific inhibitor of p38α and p38β which suppresses *Available package size: 5,25,50,100mg A10037 Aciclovir (Acyclovir) A11794 VRT752271 *Available package size: 25,50,100,200mg A10188 Cefditoren pivoxil A12002 Arctigenin A10976 Vinorelbine (Navelbine) A10654 NPI-2358 (Plinabulin) A10338 Dutasteride (Avodart) A12505 TCS ERK 11e (VX-11e) A10982 VX-702 HIF A10387 Finasteride A12824 SCH772984 A10983 VX-745 A10631 Nefiracetam (Translon) A11078 PH-797804 A10012 2-Methoxyestradiol A11221 PD 169316 A11237 FG-4592 Antiangiogenics A11321 Skepinone-L A11562 SB 239063 A12601 Combretastatin A4 A11582 TAK-715 A12021 Asiaticoside SCH772984 is a novel, specific inhibitor of ERK-1/2 with IC50 of 4 nM A12408 ML-3043 and 1 nM, respectively. A12770 Talmapimod (SCIO-469) *Available package size: 5,10,25,50mg

FG-4592 is a novel hypoxia inducible factor prolyl hydroxylase A12866 Refametinib (RDEA-119, BAY 86-9766) inhibitor, in CKD anemia. A13135 Kobe0065 *Available package size: 10,25,50,100mg A13272 RO4987655 A11924 IOX 2 A13420 GDC0994 A12883 FM19G11 Combretastatin A4 is an antitumor, anti-angiogenic and antimetastatic agent, in vitro and in vivo. Inhibits tubulin polymerization. A14019 RO5126766 A12921 HIF-C2 Talmapimod (SCIO-469) is a selective, ATP-competitive p38 inhibitor *Available package size: 10,25,50,100mg A12978 BAY 87-2243 *Available package size: 10,25,50,100mg (IC50 = 9 nM for p38α in vitro). JNK/c-Jun RO5126766, also known as CH5126766, is a protein kinase inhibitor MAPK specific for the Raf and MEK mitogen-activated protein kinases A10860 SP600125 (MAPKs) with potential anti-neoplastic activity. A11296 AS 602801 (Bentamapimod) *Available package size: 5,10,25mg MEK/ERK A10257 AZD6244 (Selumetinib) A11352 CC-401 A10453 Honokiol A11969 TCS JNK 5a A10089 AS703026 A10704 PD318088 p38-MAPK A10115 AZD8330 A10705 PD98059 A10092 Asiatic acid A10150 BIX02188 A10148 Doramapimod (BIRB-796) A10151 BIX 02189

TCS JNK 5a is a highly selective inhibitor of JNK2 and JNK3 (pIC50 values are 6.7, 6.5, <5.0 and <4.8 for JNK3, JNK2, JNK1 and p38?? PD98059 is an equipotent antagonist of the aryl hydrocarbon respectively). receptor and inhibitor of mitogen-activated protein kinase kinase. *Available package size: 10,25,50mg *Available package size: 10,50,100,200mg A12749 JNK-IN-8

BIX02188 is a potent and selective inhibitor of MEK5. A10957 U0126-EtOH *Available package size: 5,10,50,100mg A11029 GSK1120212 (JTP-74057, Trametinib) Doramapimod (BIRB 796) is a small molecule inhibitor of p38 Raf MAPK,which plays a critical role in regulating the production of A10212 PD184352 (CI-1040) A11040 TAK-733 proinflammatory cytokines. A10001 Sorafenib (Nexavar) A10256 PD0325901 A11247 RO4927350 *Available package size: 5,10,50,100mg A10002 PLX-4720 A10545 LY2228820 A10420 GDC-0879 A10823 SB 202190 A10661 NVP-BHG712 A10824 SB 203580 A10739 PLX4032 (Vemurafenib)

PD0325901 is MEK inhibitor and non-competitive with ATP, Kiapp of RO4927350 is a potent and highly selective non-ATP-competitive 1 nM against activated MEK1 and MEK2. MEK1/2 inhibitor. *Available package size: 5,10,25,100mg *Available package size: 5,10,25,50mg

A11436 GW 5074 SNS-032 (BMS-387032) is a highly selective and potent inhibitor RO5185426. PLX4032 is a B-raf inhibitor with an IC50 of 44 nM. of cyclin-dependent kinases (Cdks) 2, 7, and 9, with in vitro growth PLX4032 (Vemurafenib) also known as RG7204, Vemurafenib, R7204; A12578 Kobe2602 *Available package size: 10,50,100,200mg inhibitory effects and ability to induce apoptosis in malignant B cells. A12739 PF-04880594 *Available package size: 5,10,50,100mg A10773 RAF265 (CHIR-265) A12891 Diazepinomicin A11045 Flavopiridol HCl A13226 LGX 818 A11047 PHA-848125 (Milciclib) SCH900776 is an agent targeting cell cycle checkpoint kinase 1 (Chk1) A11105 AZD5438 with potential radiosensitization and chemosensitization activities. A11129 Dinaciclib (SCH 727965) *Available package size: 5,10,25,50mg A11154 BMS-265246 A13403 ZCL-278 A11164 PHA-767491 A13575 BML-277 A11190 R547 RAF265 (CHIR-265) is an oral, highly selective RAF and VEGFR kinase A11220 Kenpaullone inhibitor, which is to control or normalize VEGFR-2 along with the LGX818 is an orally available Raf kinase inhibitor with potential inhibition of B-raf and c-Raf mutation to prevent cancers. cyclin-dependent kinases (CDKs) antineoplastic activity. *Available package size: 5,10,25,50mg *Available package size: 1,5,10,25mg A10093 AT7519

A10774 Raf265 derivative A13323 TAK-632 A10829 SB590885 A13525 L-779450 A11063 AZ628 A11077 ZM 336372 A11240 MLN2480 (BIIB-024) lessKenpaullone effect other is a kinases. potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), A11333 BRAF inhibitor CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much *Available package size: 10,50,100mg A11381 Dabrafenib (GSK2118436A) AT7519 is an inhibitor of multiple cyclin-dependent kinases (CDKs), which may result in cell cycle arrest, induction of apoptosis, and A11313 AT7519 HCl inhibition of tumor cell proliferation. A11347 CGP60474 *Available package size: 5,25,50,100mg A12352 Purvalanol B A10163 BS-181 HCl A12438 NU 6102 A10390 Flavopiridol (Alvocidib) A12742 BAY 1000394 A12989 LY2835219 A13454 SB1317 (TG-02) Dabrafenib is a potent and selective inhibitor of B-RAF protein kinase carrying V600E mutation, currently in clinical trial. A13547 P276-00 *Available package size: 5,25,50,100mg

Flavopiridol (Alvocidib) is a cyclin-dependent kinase inhibitor under clinical development for the treatment of chronic lymphocytic Cell Cycle leukemia. *Available package size: 5,10,25,50mg A10494 JNJ-7706621 Checkpoint Kinase A10701 PD 0332991 HCl P276-00, a novel cyclin-dependent inhibitor induces G1-G2 arrest, A10113 AZD7762 shows antitumor activity on cisplatin-resistant cells and significant in vivo efficacy in tumor models. A10599 MK-1775 *Available package size: 5,10,25mg

A13549 LEE011

CHIR-124 is a novel and potent Chk1 inhibitor (IC50: 0.32 nM and A13677 BMS-863233 (XL-413) 697 nM for Chk1 and Chk2 respectively). *Available package size: 5,10,25,100mg PD 0332991 HCl is an orally available pyrido-pyrimidine-derived cyclin-dependent kinase (CDK) inhibitor with potential antineoplastic A11108 CCT241533 activity. MK-1775 is a potent and selective Wee1 kinase inhibitor in vitro and A11167 SCH 900776 (MK-8776) *Available package size: 5,10,25,50mg in vivo. A10716 PHA-793887 A11520 PF 477736 *Available package size: 5,10,25,50mg A10806 Roscovitine (Seliciclib) A12703 SCH900776 BMS-863233, also known as XL-413, is an orally bioavailable cell A10850 SNS-032 (BMS-387032) division cycle 7 homolog (CDC7) kinase inhibitor with potential A11036 LY2603618 (IC-83) antineoplastic activity. A11046 CHIR-124 *Available package size: 5,10,25,50mg

A13721 TG003

AG-014699 (Rucaparib) is a PARP inhibitor that inhibits poly(ADP- A10135 BI6727 (Volasertib) ribose) polymerase (PARP) is a key enzyme in DNA repair. Checkpoint Control Kinases A10442 GSK461364 *Available package size: 5,25,50,100mg A10452 HMN-214 A11036 LY2603618 (IC-83) A10046 AG14361 A10673 ON-01910 A11108 CCT241533 A10111 Olaparib (AZD2281)

VX-680 is a potent and selective small-molecule inhibitor of the A10164 BSI-201 (Iniparib) Aurora Kinase Aurora kinases. *Available package size: 25,50,100,250mg A10004 MLN8237 (Alisertib) A11009 ZM-447439 A11066 AMG 900

A11067 TAK-901 ON-01910 is selectively cytotoxic for chronic lymphocytic leukemia BSI-201 is a potent inhibitor of PARP-1 and has been shown to cross A11081 CCT137690 cells through a dual mechanism of action involving PI3K/AKT the blood-brain barrier. inhibition and induction of oxidative stress. A11168 GSK1070916 *Available package size: 10,50,100,200mg *Available package size: 5,10,50,100mg A11171 PF-03814735 A11410 MK-5108 (VX-689) A10475 INO-1001 A11146 TAK-960 MLN8237 (Alisertib) is a selective Aurora kinase A inhibitor with a A10909 Tenofovir Disoproxil Fumarate median IC50 of 61 nM. A11026 MK-4827 *Available package size: 5,10,50,200mg

A10095 AT9283 A10100 Aurora A Inhibitor I A10109 AZD1152-HQPA (Barasertib) TAK-960 is a novel, orally available, selective inhibitor of polo-like MK-5108, also known as VX-689, is a competitive inhibitor of the kinase 1, shows broad-spectrum preclinical antitumor activity. ATP-binding site of aurora A kinase. MK-4827 is a novel potent, orally bioavailable PARP-1 and PARP-2 *Available package size: 5,10,50,100mg inhibitor. *Available package size: 5,10,50,100mg A11438 GW843682X *Available package size: 5,10mg A13250 Reversine A12429 MLN 0905 A13396 MK-8745 A11243 BMN673 A13245 RO3280

PARP Rho-Kinase (ROCKs) AZD 1152-HQPA is a highly potent and selective inhibitor of Aurora B, with Ki values to be 0.36 (Aurora B) and 1369 nM (Aurora A) A10019 A-966492 A10381 Fasudil HCl (HA-1077) respectively and has a high specificity versus a panel of 50 other kinases. *Available package size: 5,10,50,200mg A10184 CCT129202 BMN-673 is an orally bioavailable inhibitor of the nuclear enzyme A10248 CYC116 poly(ADP-ribose) polymerase (PARP) with potential antineoplastic A10448 Hesperadin activity.

A-966492 displayed high potency against the poly(ADP-ribose) *Available package size: 5,10,25,50mg Fasudil HCl is a cyclic nucleotide-dependent protein kinase inhibitor polymerase-1 (PARP-1) enzyme with a K(i) of 1 nM and an EC(50) of A12393 AZD-2461 1 nM in a whole cell assay. *Available package size: 250,500mg A12665 PJ 34 hydrochloride and Rho-associated kinase inhibitor (IC50 = 10.7 μM). *Available package size: 5,10,50,100mg A10441 GSK429286A A12750 UPF 1069 A10928 Thiazovivin A10026 ABT-888 (Veliparib) A13731 JW 55

Polo-like kinases (PLKs)

A10134 BI 2536 Hesperadin is a human Aurora B inhibitor with an IC50 of 40 nM for the prevention of the phosphorylation of substrate. ABT-888(Veliparib) is a potential anti-cancer drug acting as a PARP Thiazovivin is a selective inhibitor of Rho-associated kinase (ROCK). *Available package size: 5,10,50,100mg inhibitor. *Available package size: 5,10,25,50mg A10601 MLN8054 *Available package size: 10,50,100,200mg A10714 PHA-680632 A11001 Y-27632 dihydrochloride A10045 AG-014699 (Rucaparib) A10715 Danusertib (PHA-739358) A10851 SNS-314 BI 2536 is a selective inhibitor of Plk1, which inhibits Plk1 enzyme activity at low nanomolar concentrations. A10981 VX-680 (MK-0457, Tozasertib) *Available package size: 5,10,50,100mg

Y-27632 is a Rho-Associated Coil Kinase (ROCK) inhibitor that A10740 Podophyllotoxin CYT997 is a novel anti-cancer vascular disrupting agent (VDA). A13827 CK-636 increases the cloning efficiency of human embryonic stem cells In vitro, CYT997 is shown to potently inhibit the proliferation of (hESCs). A10939 Topotecan HCl (Hycamtin) vascular endothelial growth factor-stimulated human umbilical *Available package size: 5,10,25,50mg vein endothelial cells (IC(50) 3.7 ± 1.8 nM) and cause significant Synthases / Synthetases morphological changes at 100 nM, including membrane blebbing. A11610 Y-33075 A10050 Alendronate sodium hydrate *Available package size: 5,10,50,100mg A12348 GSK 269962 A10776 Raltitrexed (Tomudex) A10326 Docetaxel (Taxotere) A12546 NSC 23766 A12992 HQL-79 A10359 Epothilone A A12674 SR 3677 dihydrochloride A13583 1400W Dihydrochloride A10360 Epothilone B (EPO906)

Topotecan HCl (Hycamtin) is a chemotherapeutic agent that is a topoisomerase inhibitor. RNA/DNA Polymerase *Available package size: 50,100,200mg A10908 Tenofovir (Viread) A11231 Exatecan mesylate A11115 Abacavir A11120 Abacavir sulfate A11590 T-705 (Favipiravir) SR 3677 dihydrochloride is a potent and selective Rho-kinase inhibitor (IC50 values are 3 and 56 nM for ROCK-II and ROCK-I respectively). Epothilone B is a macrolide that causes the formation of bundles of *Available package size: 10,25,50,100mg intracellular microtubules in non-mitotic cells, induces the formation of hyperstable tubulin polymers, and arrests cell cycling in mitosis. A12740 EHop-016 *Available package size: 2,5,10,25mg A13067 RKI-1447 T-705, a substituted pyrazine compound, has been found to exhibit potent anti-influenza virus activity in vitro and in vivo. Exatecan mesylate inhibits topoisomerase I activity by stabilizing the A10689 Paclitaxel (Taxol) cleavable complex between topoisomerase I and DNA and inhibiting *Available package size: 10,25,50,100mg religation of DNA breaks, thereby inhibiting DNA replication and triggering apoptotic cell death. A13239 Actinomycin D *Available package size: 10,25,50,100mg A13274 Delavirdine mesylate RKI-1447 is a potent inhibitor of the Rho-associated ROCK kinases with anti-invasive and antitumor activities in breast cancer. A11861 Flumequine *Available package size: 5,10,25,50mg A11902 Pefloxacin mesylate Telomerase A13785 HA-1077 dihydrochloride A11997 (S)-10-Hydroxycamptothecin A10140 BIBR 1532 A12011 SN 38 Topoisomerase

A10041 Adriamycin Paclitaxel (Taxol) is a mitotic inhibitor that stabilizes microtubules and as a result, interferes with the normal breakdown of microtubules A10071 Amonafide (AS1413) during cell division. BIBR 1532 is a selective telomerase inhibitor (IC50 values are 93, A10174 Camptothecin *Available package size: 10,50,100,200mg > 100000 and > 100000 nM for human telomerase, human RNA A10194 Cerubidine polymerase I and human RNA polymerase II + III respectively). SN 38 is the active metabolite of irinotecan (an analog of A10740 Podophyllotoxin A10345 Epirubicin Hydrochloride *Available package size: 10,50,100,200mg camptothecin - a topoisomerase I inhibitor). A10973 Vincristine sulfate A10373 Etoposide (VP-16) A10240 Costunolide *Available package size: 50,100,250mg A10975 Vinflunine Tartrate A10465 Idarubicin HCl A11999 Betulinic acid A12663 Amrubicin A11412 Epothilone D A13093 Amsacrine A13059 Beta-Lapachone A13206 GENZ-644282

Microtubules Ligases A10024 ABT-751 A10238 Colchicine A10884 TAME A10264 CYT997 Idarubicin is an anthracycline antibiotic that is an anti-leukemia Epothilone D improves microtubule density, axonal integrity, and Reverse Transcriptase agent with higher DNA binding capacity and greater cytotoxicity than cognition in a transgenic mouse model of tauopathy. daunorubicin. *Available package size: 1,2,5,10mg *Available package size: 5,10,50,100mg A11449 Ixabepilone A10039 Adefovir dipivoxil A10477 Irbesartan (Avapro) A11617 Vinblastine A10349 Emtricitabine A10478 Irinotecan A12591 Cevipabulin (TTI-237) A10639 Nevirapine (Viramune) A10479 Irinotecan HCl Trihydrate (Campto) A12804 Eribulin Mesylate A10908 Tenofovir (Viread) A10596 Mitoxantrone Hydrochloride A13081 Fosbretabulin disodium (CA4P) A10609 Moxifloxacin HCl A13219 Nocodazole A10735 Pirarubicin A13735 CW069

A12587 Dapivirine A13366 Mephenytoin A12667 Lersivirine (UK-453061) A13367 Methoxyresorufin

β-Amyloid

A10312 Dimebon dihydrochloride Tenofovir is in a class of medications called nucleoside reverse A12647 Ro 90-7501 transcriptase inhibitors (NRTIs). It works by decreasing the amount Apremilast, a novel PDE4 inhibitor, inhibits spontaneous production of HIV in the blood. Lersivirine (UK-453,061) is a next-generation nonnucleoside reverse Phosphodiesterases (PDEs) of tumour necrosis factor-alpha from human rheumatoid synovial *Available package size: 10,25,50,100mg transcriptase inhibitor, active against wild-type HIV-1 and several cells and ameliorates experimental arthritis. nonnucleoside reverse transcriptase inhibitor-resistant strains. A10909 Tenofovir Disoproxil Fumarate A10216 Cilomilast (SB-207499) *Available package size: 2,5,10,25mg *Available package size: 5,10,25,50mg A11115 Abacavir A11326 Bay 60-7550 A11120 Abacavir sulfate Mitosis A12550 Zardaverine A12443 MK-1439 A12619 Avanafil A13872 INH1 A12776 AN2728 A13121 PF-04447943 Cilomilast is orally active and acts as a selective Phosphodiesterase-4 A13722 Deltarasin-HCl inhibitor with antiinflammatory effects that target bronchoconstriction, mucus hypersecretion, and airway remodeling associated with COPD. *Available package size: 5,10,50,100mg A10217 Cilostazol A10449 Hesperetin MK-1439 is a non-nucleoside reverse transcriptase inhibitor. A10464 Icariin *Available package size: 5,10,25,50mg A10541 Luteolin A10592 Milrinone (Primacor) A10733 Pimobendan (Vetmedin) interaction and thus impairing oncogenic KRAS signalling. Deltarasin is a novel small molecule inhibiting the KRAS PDEδ Cell Metabolism *Available package size: 5,10,25mg

Cytochrome P450 Hydroxylases A10485 Isotretinoin A10020 Abiraterone (CB-7598) A10542 LX 1606 Hippurate Pimobendan (Vetmedin) is a calcium sensitizer with positive TAK-700 (Orteronel) is an oral, non-steroidal androgen synthesis inotropic and vasodilator effects. It is also a selective inhibitor of inhibitor that selectively inhibits the 17,20 lyase enzyme. phosphodiesterase III (PDE3). *Available package size: 5,10,50,100mg *Available package size: 5,10,50,100mg

A11058 Abiraterone Acetate (CB7630) A10804 Roflumilast A11138 TOK-001 (Galeterone) A10805 Rolipram A10965 Vardenafil (CYP17A1), an enzyme which is expressed in testicular, adrenal, and A11019 Ibudilast (KC-404) prostaticAbiraterone tumor (CB-7598) tissues. inhibits 17 α-hydroxylase/C17,20 lyase LX 1606 hippurate is an orally bioavailable, small-molecule, *Available package size: 5,10,50,100mg tryptophan hydroxylase (TPH) inhibitor with potential A10081 Apigenin antiserotonergic activity. A10102 Avasimibe (CI-1011) *Available package size: 5,10,50,100mg A10120 Baicalein TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor. A10637 Nepicastat (free base) (SYN-117) A10200 Chloramphenicol *Available package size: 5,10,50,100mg A10234 Clotrimazole Ibudilast, a pharmacologic phosphodiesterase inhibitor, prevents A10498 Ketoconazole A11144 TH-302 human immunodeficiency Virus-1 Tat-Mediated activation of microglial cells. A10578 Methoxsalen (Oxsoralen) A11277 Cobicistat(GS-9350) *Available package size: 10,50,100mg A10625 Naringenin A11481 Luliconazole A11865 Hydroxyflutamide A10853 Sodium Danshensu A11073 GSK256066 A11977 TMS A10978 Voriconazole (Vfend) A11191 PF-2545920 A12544 PF 4981517 A11044 TAK-700 (Orteronel) A11289 Apremilast (CC 10004) Nepicastat is an inhibitor of dopamine beta-hydroxylase, an enzyme A13361 ABT that catalyzes the conversion of dopamine to norepinephrine. A13365 3-Cyano-7-ethoxycoumarin *Available package size: 5,10,50,100mg

A11172 Nepicastat hydrochloride A11183 PF-3845 Cyclooxygenase (COX) Histone Deacetylase (HDAC) A11785 LX 1606 A10030 Acetaminophen A10122 Belinostat (PXD101) A12833 Ro 61-8048 A10090 Asaraldehyde (Asaronaldehyde) A13363 Metyrapone A10193 Celecoxib A13998 DMOG A10304 Diclofenac sodium NS-398 is a COX-2 inhibitor used in the study of the function of A10382 Febuxostat (TEI-6720) cyclooxygenases. Dihydrofolate reductase (DHFR) A10461 Ibuprofen (Advil) *Available package size: 10,25,50,100mg Belinostat (PXD101) is a HDAC inhibitor that inhibits HDAC activity A10462 Ibuprofen Lysine (NeoProfen) A10021 Methotrexate (Abitrexate) A13244 Bromfenac sodium in HeLa cell extracts with an IC50 of 27 nM. A10474 Indomethacin (Indocid, Indocin) A10655 NSC 131463 (DAMPA) A13332 FK 3311 *Available package size: 10,50,100,200mg A10623 Naproxen sodium A10707 Pemetrexed (Alimta) A13342 Valdecoxib A10720 Phenylbutazone A10179 Carbamazepine A12796 Trimetrexate A13572 Parecoxib A10736 Piroxicam (Feldene) A10246 CUDC-101 Antimetabolite

A10177 Capecitabine (Xeloda)

Trimetrexate is a quinazoline derivative. It is a dihydrofolate reductase inhibitor. Piroxicam is an effective and potent inhibitor of prostaglandin CUDC-101 is a novel compound which inhibits multiple targets, which *Available package size: 5,10,25,50mg synthesis and a Cox-1 and Cox-2 inhibitor. is designed to inhibit HDAC, EGFR and Her2. *Available package size: 250,500mg *Available package size: 10,50,100,200mg Dehydrogenases A10749 Pravadoline (WIN 48098) A10337 Droxinostat Capecitabine is a prodrug, that is enzymatically converted to A10780 Ranolazine A10878 Sulindac (Clinoril) A10488 ITF2357 (Givinostat) 5-fluorouracil in the tumor, where it inhibits DNA synthesis and slows A11292 Alvimopan (ADL 8-2698) A11403 MK-8245 growth of tumor tissue. A10492 JNJ-26481585 A11464 Iguratimod (T 614) A11682 Gimeracil *Available package size: 1,5g A10516 LAQ824 (NVP-LAQ824) A11686 Flunixin meglumine A11786 CPI-613 A10183 Carmofur A11692 Acemetacin (Emflex) A10223 Cladribine A11693 Tolfenamic acid A10251 Flupirtine maleate A11694 Nimesulide A11695 Lornoxicam (Xefo) A11697 Licofelone

LAQ824 (NVP-LAQ824) is a potent novel histone deacetylase CPI-613 is a racemic mixture of the enantiomers of a synthetic alpha- inhibitor with significant activity against multiple myeloma. lipoic lipoic acid analogue with potential chemopreventive and *Available package size: 10,50,100mg antineoplastic activities. *Available package size: 5,10,25,50mg Flupirtine maleate is a Non-opioid analgesic with muscle relaxant A10518 LBH589 (Panobinostat) properties. A10560 MC1568 A12385 CGP 3466B maleate *Available package size: 10,25,100mg A12442 Brequinar A10286 Daphnetin A12902 AGI-5198 (IDH-C35) A10292 Decitabine Licofelone is a dual COX/LOX inhibitor, being considered as a treatment for osteoarthritis. It may reduce the gastrointestinal toxicity associated with other non-steroidal anti-inflammatory drugs, which only inhibit COX (cyclooxygenase). Licofelone is the first drug to inhibit both. MC1568 is a member of HDAC inhibitors that inhibits the histone deacetylase class II by modifying the genetic expression of various *Available package size: 5,10,50,100mg important genes of cell cycle mostly at G1 phase, resulting in the death of breast cancer cells by apoptosis. A11906 Phenacetin *Available package size: 10,25,50,100mg Decitabine is a hypomethylating agent.It hypomethylates DNA by AGI-5198, also know as IDH-C35, is the a very potent and selective A11918 Rofecoxib (Vioxx) inhibiting DNA methyltransferase. mutant IDH1 inhibitor that was shown to potential anticancer A11986 ATB-337 A10586 MGCD0103 (Mocetinostat) activity. *Available package size: 10,25,50,100mg A12434 (S)-(+)-Flurbiprofen A10611 MS-275 (Entinostat) *Available package size: 5,10,25,50mg A13116 NS-398 A10395 Fludarabine Phosphate (Fludara) A10700 PCI-24781 A10764 Pyroxamide (NSC 696085) A12903 AGI-6780 A10396 Fludarabine (Fludara) A10830 SB939 A12925 JK 184 A10947 Trichostatin-A (TSA)

A10954 Tubacin EX 527 is a potent and selective SIRT1 class III histone deacetylase A10158 BMS-740808 A11065 CX-5461 enzyme inhibitor A10979 Vorinostat (SAHA) A10800 Rivaroxaban (Xarelto) *Available package size: 5,10,25,100mg A11037 AR-42 (HDAC-42) A12411 Rivaroxaban Diol A11042 Tubastatin A HCl A10785 Resveratrol A12518 Betrixaban A11152 PCI-34051 A10862 SRT1720 A12870 Razaxaban A12871 Letaxaban (TAK-442) A13878 ABT333 CX-5461 is a first-in-class non-genotoxic small molecule targeted inhibitor of RNA polymerase I (Pol I) that activates the p53 pathway without causing DNA damage. Kinesin Spindle Protein *Available package size: 5,10,50,100mg PCI-34051 is a specific and potent histone deacetylase 8 (HDAC8) A10486 Ispinesib (SB-715992) A11147 CCT239065 inhibitor, with >200-fold selectivity over the other HDAC isoforms. *Available package size: 10,25,50,100mg A11179 NSC-207895 (XI-006) A11803 Azithromycin (Zithromax) A11153 CUDC-907 A11804 Adenine sulfate A11920 Romidepsin (FK228 ,Depsipeptide) A12326 INNO-206 (Aldoxorubicin) A11940 ACY-1215 (Rocilinostat) A11964 CI994 (Tacedinaline) SRT1720 is an inhibitor developed intended as a small-molecule activator of the sirtuin subtype SIRT1. *Available package size: 5,10,50,200mg

A12527 Inauhzin Ispinesib (SB-715992) is a potent inhibitor of kinesin spindle protein, A12904 AK-7 a kinesin motor protein essential for the formation of a bipolar mitotic spindle and cell cycle progression through mitosis. Aldoxorubicin, also known as INNO-206, is the 6-maleimidocaproyl Monoamine Oxidase (MAO) *Available package size: 5,10,50,100mg hydrazone derivative prodrug of the anthracycline antibiotic doxorubicin (DOXO-EMCH) with antineoplastic activity. A10828 SB 743921 A10078 Aniracetam *Available package size: 10,25,50,100mg A11050 Arry-520 CI-994 is a histone deacetylase (HDAC) inhibitor and induces histone A10818 Safinamide Mesylate (FCE28073) A11170 AZ 3146 A12409 Epirubicin hyperacetylation in living cells. A11722 Rasagiline mesylate *Available package size: 10,50,100mg

A12556 Resminostat

AZ 3146 is a potent and selective monopolar spindle 1 (Mps1) kinase inhibitor (IC50 = 35 nM). It interferes with chromosome alignment and overrides spindle assembly checkpoint and also Inhibits the Rasagiline is an irreversible inhibitor of monoamine oxidase used as recruitment of Mad1, Mad2 and centromere protein E (CENP-E) to a monotherapy in early Parkinson's disease or as an adjunct therapy kinetochores. in more advanced cases. Epirubicin is a cell-permeable antitumor antibiotic. A stereoisomer *Available package size: 5,10,50,100mg of Doxorubicin that exhibits reduced cardiotoxicity. Epirubicin’s *Available package size: 50,100mg antitumor actions are mediated by targeting and inhibiting Topo II A11976 Monastrol Resminostat, also known as RAS2410, is a potent inhibitor of histone A11777 SL251188 (topoisomerase II). deacetylase (HDAC) classes I and II. It binds to and inhibits HDACs *Available package size: 10,25,50,100mg leading to an accumulation of highly acetylated histones. A11885 Moclobemide DNA, RNA and Protein Synthesis *Available package size: 10,25,50,100mg A13294 Safinamide A12890 Thiostrepton A13353 Bifemelane hydrochloride A10036 Cycloheximide (Actidione) A12722 Scriptaid A10152 Bleomycin sulfate CYP17 A12745 Apicidin A10182 Carboplatin Factor Xa A11044 TAK-700 (Orteronel) A12911 BRD9757 A10221 Cisplatin A10082 Apixaban (BMS-562247-01) A11138 TOK-001 (Galeterone) A13218 RGFP966 A10224 Clafen (Cyclophosphamide) A10228 Clofarabine Sir2-like Family Deacetylases (sirtuins) A10281 Dacarbazine A10346 Oxaliplatin (Eloxatin) A10377 EX 527 A10392 Floxuridine A10466 Ifosfamide Apixaban is an anticoagulant for the prevention of venous A10532 Lincomycin hydrochloride (U-10149A) TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor. thromboembolism and venous thromboembolic events. A10568 Mercaptopurine *Available package size: 5,10,50,100mg *Available package size: 5,10,50,100mg A10597 Mizoribine A10632 Nelarabine (Arranon)

A11409 Cyproterone acetate A11084 Anacetrapib (MK-0859) A13004 INCB024360 A13515 TAK-700 (salt) Ferroptosis

A12916 Ferrostatin-1 (ethyl ester) Phospholipases A13247 Ferrostatin-1 (Fer-1) A13822 Erastin A10206 Chlorpromazine hydrochloride A10548 LY315920 (Varespladib) INCB024360 is an orally available hydroxyamidine and inhibitor of indoleamine 2,3-dioxygenase (IDO1), with potential immunomodulating and antineoplastic activities. Anacetrapib (MK-0859) is a CETP inhibitor being developed to treat *Available package size: 5,10,25,50mg hypercholesterolemia (elevated cholesterol levels) and prevent cardiovascular disease. *Available package size: 5,10,50,100mg A11213 JTT-705 (Dalcetrapib) PI3K / Akt / mTOR LY315920 (Varespladib) is an inhibitor of the IIa, V, and X isoforms of A11397 Evacetrapib (LY2484595) secretory phospholipase A2 (sPLA2). *Available package size: 5,10,50,100mg DNA Methyltransferases Akt A13460 Deguelin Lipid Metabolism A10105 Azacitidine(Vidaza) A10003 MK-2206 dihydrochloride PI3-Kinase (PI3K) A10292 Decitabine A10094 AT7867 A11230 PF 429242 A12744 SGI-110 A10088 AS-605240 A10112 AZD6482 HMG-CoA Reductase A10133 BEZ235 (NVP-BEZ235) A10172 CAL-101 (GS-1101) A10737 Pitavastatin calcium (Livalo) A10421 GDC-0941 A10438 GSK1059615 A10463 IC-87114 PF 429242 is a reversible, competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease. AT7867 is a novel and potent inhibitor of both AKT and the downstream kinase p70 S6 kinase (p70S6K) and also of protein *Available package size: 10,25,50,100mg kinase A. A11242 Torcetrapib (CP-529414) *Available package size: 10,25,50,100mg A12318 SC-26196 A10453 Honokiol Pitavastatin Calcium is a competitive inhibitor of the enzyme HMGCR A10709 Perifosine (NSC-639966) (HMG-CoA reductase) results in a reduction in LDL cholesterol FAAH synthesis. A11024 PF-04691502 A11049 URB597 *Available package size: 10,25,50,100mg A11030 GSK690693 IC-87114 was the first isoform-selective PI3K inhibitor: p110M-NM- A11031 CCT128930 4(IC50 = 0.13 M-BM-5M) vs. p110M-NM-1(IC50 = 200 M-BM-5M), A11800 Atorvastatin calcium A11032 PHT-427 p110M-NM-2(IC50 = 16 M-BM-5M) and p110M-NM-3(IC50 = 61 M-BM-5M). A11877 Lovastatin (Mevacor) A11033 Triciribine phosphate (NSC-280594) *Available package size: 5,10,25,100mg A11912 Pravastatin sodium A11034 A-674563 A10547 LY294002 A13709 Mevastatin A11246 GDC-0068 A10693 Palomid 529 (P529) URB597 is a relatively selective inhibitor of the enzyme fatty acid A13743 Atorvastatin A11286 AKT inhibitor VIII (AKTI-1/2) amide hydrolase (FAAH). A11287 A-443654 *Available package size: 5,25,50,100mg Neuronal Metabolism A11759 AZD5363 A12420 JNJ 1661010 A12877 KP372-1 A12404 ONO 2506 A13210 Triciribine

Palomid 529 is a dual TORC1/2 inhibitor of the PI3K/Akt/ mTOR pathway having broad activity in angiogenesis and cellular proliferation ONO 2506 inhibits S100B synthesis in activated cultured astrocytes. *Available package size: 10,50,100,200mg JNJ 1661010 is a selective and reversible inhibitor of fatty acid amide *Available package size: 10,25,50,100mg hydrolase (FAAH) (IC50 = 12nM). A10727 PIK-293 *Available package size: 10,25,50,100mg IDO A10728 PIK-294 CETP Triciribine, also known as API-2, suppresses the phosphorylation level and kinase activity of Akt. *Available package size: 10,25,50,100mg

A11151 3-Methyladenine A11784 GSK2636771 A10746 PP242 A11161 Wortmannin A11956 TG 100713 A11162 NVP-BGT226 A12422 IPI-145 A11169 CH5132799 A11196 CAY10505 A11197 AS-604850

PIK-294 is a PI3 Kinase inhibitor that is 20- to 60-fold more potent than the parent compound, PIK-293. It is one of the most potent IPI-145, also known as INK-1197, is an orally bioavailable, highly selective and potent small molecule inhibitor of the delta and PP242 is a potent and selective mTOR inhibitor in both mTORC1 and mTORC2. *Available package size: 5,10,50,100mg gamma isoforms of phosphoinositide-3 kinase (PI3K) with potential p110δ-selective inhibitors that has been reported. immunomodulating and antineoplastic activities. *Available package size: 5,10,50,100mg A10729 PIK-75 AS-604850 inhibited MCP-1-mediated monocyte chemotaxis with *Available package size: 5,10,25,50mg A10782 Rapamycin (Sirolimus) A10730 PIK-90 an IC50 value of 21 µM and reduced RANTES-induced peritoneal neutrophil recruitment in a murine model of leukocyte chemotaxis A12480 VS-5584 A10906 Temsirolimus (Torisel) A10731 PIK-93 with an ED50 value of 42.4 mg/kg. A12704 SF1126 A10989 WYE-354 A10765 Quercetin dihydrate (Sophoretin) *Available package size: 5,10,50,100mg A12831 GDC-0032 A10766 Quercetin (Sophoretin) A11198 D-106669 A12935 PF-04979064 A10922 TG100-115 A11202 A66 A11207 PP121

WYE-354 is a potent cell-permeable inhibitor of mTOR (IC50 = 4.3 PF-04979064 is a highly potent and orally bioavailable PI3K/mTOR nM) which blocks signaling through both mTOR complex 1 (mTORC1) dual inhibitor. respectively). TG100-115 inhibits PI3K γ and -δ(IC50 values of 83 and 235 nM, *Available package size: 2,5,10mg nM) and other kinases. *Available package size: 5,10,25,100mg PP121 is a dual inhibitor of receptor tyrosine kinases (RTKs) (IC50 < and mTORC2. It is a much weaker inhibitor of PI3K α (IC50 = 1026 *Available package size: 5,10,25,50mg A10923 TGX-221 A13021 HS-173 A11038 WYE-125132 (WYE-132) 0.02 μM for Abl, Src, VEGFR-2 and PDGFR) and PI 3-K family kinases A13224 KU 0060648 A10995 XL147 *Available package size: 10,25,50,100mg (IC50 < 0.06 μM for p110α, DNA-PK and mTOR). A11056 OSI-027 A10997 XL765 A13879 CNX-1351 A11261 PX-866 A11079 PKI-587 A11014 ZSTK474 mTOR A11187 WYE-687 A11188 WAY-600 A10114 AZD8055 A11303 AZD2014

PX-866 is a small-molecule wortmannin analogue inhibitor of the ZSTK474 is an ATP-competitive inhibitor of class I alpha, gamma, and delta isoforms of phosphoinositide 3-kinase (PI3K) phosphatidylinositol 3 kinase isoforms. AZD2014 is an orally bioavailable inhibitor of the mammalian target with potential antineoplastic activity. AZD8055 is a potent, selective, and orally bioavailable ATP- *Available package size: 10,25,50,100mg of rapamycin (mTOR) with potential antineoplastic activity. mTOR *Available package size: 5,10,25,50mg competitive mTOR kinase inhibitor with an IC50 of 0.8 nM. A11016 BKM120 (NVP-BKM120) kinase inhibitor. A11328 BYL719 *Available package size: 10,25,50,100mg A11023 GDC-0980 (RG7422) *Available package size: 5,10,25,50mg A10295 Deforolimus (Ridaforolimus) A11035 GSK2126458 A11443 GDC-0349 A10374 Everolimus (RAD001) A11064 YM201636 A11461 INK 128 A10505 KU-0063794 A11089 PKI-402 A11098 NU-7441 (KU-57788) A11099 AS-252424

BLY719 is an orally bioavailable phosph-atidylinositol 3-kinase (PI3K) inhibitor with potential antineoplastic activity. *Available package size: 5,10,25,50mg

A11363 CZC24832 INK 128 is a TORC1/2 inhibitor, is also an orally bioavailable inhibitor KU-0063794 is a selective inhibitor of mammalian target of of raptor-mTOR (TOR complex 1 or TORC1) and rictor-mTOR (TOR A11511 NVP-BAG956 rapamycin (mTOR) (IC50 ~10 nM for mTORC1 and mTORC2 AS-252424 is a potent inhibitor of PI3K with selectivity for the γ complex 2 or TORC2) with potential antineoplastic activity. values of 30, 940, 20,000, and 20,000 nM respectively. A11766 BAY 80-6946 respectively). isoform. It inhibits human recombinant PI3Kγ, α, β, and δ with IC50 *Available package size: 5,10,25,50mg *Available package size: 5,10,50,100mg *Available package size: 5,25,50,100mg

A11586 Torin 2 A11558 SU-5402 A10963 Vandetanib (ZD6474) DNA-dependent protein kinase (DNA-PK) A11752 Lapatinib (free base) A10967 Vatalanib (PTK787) 2HCl

A10726 PI-103 A11948 AP26113 A10996 XL184 free base (Cabozantinib) A11949 AG-17 A11263 BMS-690514 A12448 Butein A11396 E-7050 (Golvatinib) A12650 PKC 412 A11407 Apatinib (YN968D1) A12867 CGP-52411 A11496 Motesanib (AMG706) Torin 2 is a potent and selective mTOR inhibitor (IC50 = 2.1 nM). A12868 ARRY-543 A11557 SU14813 Displays 800-fold cellular selectivity for mTOR over PI3K (cellular A13588 Tyrphostin AG 183 A11772 CP-547632 EC50 values are 0.25 and 200 nM for mTOR and PI3K respectively). A13681 AZD-9291 A11954 ZM 323881 hydrochloride *Available package size: 10,25,50,100mg PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of phosphatidylinositol 3-kinase (PI3K) family members with selectivity A13718 Icotinib Hydrochloride A11955 ZM 306416 hydrochloride A11587 Torin 1 A13755 CNX-2006 A11978 Delphinidin chloride A11950 Zotarolimus *Available package size: 5,10,25,50mg A13825 Icotinib A12027 (-)-Catechin gallate toward DNA-PK, PI3K (p110α), and mTOR. A12395 XL388 A11098 NU-7441 (KU-57788) A12437 SU 5416 (Semaxinib) A11778 Compound 401 FGFR A13234 SKLB1002 PDK1 A12752 NU7026 A13377 SAR131675 A10703 PD173074 A13465 SKLB610 A10681 OSU-03012 A11075 AZD4547 A13966 TPT-260 (Dihydrochloride) A11148 BX-795 Ribosomal S6 protein kinases (RSK) A11159 BGJ398 (NVP-BGJ398) A11149 BX-912 A11244 LY 2874455 Type 1 insulin-like growth factor receptor (IGF- A11160 SL 0101-1 1R) A11423 FMK PDGFR A11755 PF 4708671 A10440 GSK1904529A A12452 BI-D1870 A10504 KRN 633 A10658 NVP-ADW742 BX-795 is a potent PDK1 inhibitor that blocks PDK1/Akt signaling in A10880 Sunitinib Malate tumor cells and inhibits the anchorage-dependent growth of a variety A11021 NVP-AEW541 of tumor cell lines in culture or induced apoptosis. A10903 Telatinib (BAY 57-9352) *Available package size: 10,25,50,100mg A11052 Crenolanib (CP-868596) A11350 CP-673451 A11511 NVP-BAG956 A11581 Toceranib (PHA 291639, SU 11654) A12767 GSK 2334470 A11753 MK-2461 A13484 PS 48 A11978 Delphinidin chloride

VEGFR NVP-AEW541 is a selective IGF-1R kinase inhibitor that inhibits A10025 Linifanib (ABT-869) the autophosphorylation activity of IGF-1R (IC50 = 0.086 uM) and Receptor Tyrosine Kinases prevents IGF-1-mediated survival and proliferation of MCF-7 cells A10049 Albendazole (IC50 = 0.16 and 1.64 uM, respectively). A10101 Tivozanib (AV-951) A10702 PD153035 (HCl salt) *Available package size: 2,5,10,25mg EGFR/HER2 A10103 Axitinib A10706 Pelitinib (EKB-569) A10137 Bibf1120 (Vargatef) A11053 OSI-906 A10043 AEE788 A10990 WZ3146 A10162 Brivanib alaninate (BMS-582664) A10047 AG-490 A10991 WZ4002 A10185 Cediranib (AZD2171) A10053 Tyrphostin AG 879 A10992 WZ8040 A10204 Chloroxine A10062 AST-6 A11022 AG-1478 (Tyrphostin AG-1478) A10248 CYC116 A10116 AZD8931 A11027 Arry-380 A10254 Brivanib (BMS-540215) A10141 BIBW2992 (Afatinib) A11028 AV-412 A10259 Imatinib (Gleevec) A10210 Chrysophanic acid (Chrysophanol) A11051 PF299804 OSI-906 is a potential first-in-class selective small molecule, dual A10340 E7080 (Lenvatinib) kinase inhibitor of both insulin-like growth factor-1 receptor (IGF-1R) A10211 Canertinib (CI-1033) A11057 XL647 A10495 Kaempferol and insulin receptor (IR). A10242 CP-724714 A11155 AST-1306 *Available package size: 5,10,50,100mg A10502 Ki8751 A10362 Erlotinib Hydrochloride A11158 ARRY334543 A10504 KRN 633 A11054 BMS-536924 A10422 Gefitinib (Iressa) A11209 BMS 599626 (AC480) A10608 Motesanib Diphosphate (AMG-706) A11059 BMS-754807 A10514 Lapatinib Ditosylate A11236 TAK-285 A10699 Pazopanib Hydrochloride (GW786034) A11400 AG-1024 (Tyrphostin) A10612 Mubritinib (TAK 165) A11263 BMS-690514 A10893 Taxifolin A11951 PQ 401 A10638 Neratinib (HKI-272) A11334 BIBX 1382 A10953 TSU-68 (SU6668) A12195 Picropodophyllin A10678 OSI-420 A11407 Apatinib (YN968D1) A13069 XL-228

A10154 BMS-794833 AP24534 (Ponatinib) is a potent multi-kinase and pan-BCR-ABL FLT3 (FMS-like tyrosine kinase 3) A10493 JNJ-38877605 inhibitor. *Available package size: 10,25,50,100mg A10027 AC220 (Quizartinib) A10587 MGCD-265 A10119 Bafetinib (INNO-406) A10408 FTY720 (Fingolimod) A10468 Imatinib Mesylate A10644 Nilotinib (AMN-107)

TAE684 is a inhibitor of ALK and also a potent inhibitor of LRRK2 MGCD265 is a multitargeted tyrosine kinase inhibitor that binds to kinase activity (IC(50) of 7.8nM against wild-type LRRK2, 6.1nM AC220 (Quizartinib) is a uniquely potent and selective FLT3 inhibitor and inhibits the phosphorylation of several RTKs, including the c-Met against the G2019S mutant). with IC50 of 0.56 ± 0.3 nM and >10 mM for MC4-11 and A375, *Available package size: 5,10,50,100mg respectively. and MST1R. receptor (HGFR); the Tek/Tie-2 receptor; VEGFR types 1, 2, and 3; A10712 PF-2341066 (Crizotinib) *Available package size: 5,10,50,200mg *Available package size: 5,10,50,100mg A10198 Dovitinib Dilactic acid A10826 SB 431542 Nilotinib is a Bcr-Abl inhibitor with IC50 less than 30 nM. A10610 MP470 (MP-470) A10352 ENMD-2076 A11083 GW788388 *Available package size: 25,50,100,200mg A10711 PF-04217903 A11134 CH5424802 A10988 WP1130 ( Degrasyn ) A10713 PHA-665752 A11175 GSK1838705A A11200 DCC-2036 (Rebastinib) A10839 SGX-523 A11205 LDN193189 A11439 GNF 2 A10869 SU11274 A10998 Foretinib (GSK1363089, XL880) A11055 AMG-458 ENMD-2076 is a novel, orally-active antimitotic and antiangiogenic molecule inhibits Aurora A as well as tyrosine kinases that drive A11087 ARQ 197 tumor vascularization, including VEGFR2 (KDR), PDGFR and the FGF receptors. *Available package size: 5,10,50,100mg LDN193189 is a highly potent small molecule BMP inhibitor that inhibits BMP type I receptors ALK2 (IC50: 5 nM), ALK3 (IC50: 30 A10508 KW-2449 A10887 Tandutinib (MLN518) phosphorylation. GNF 2 is a Bcr-abl inhibitor that inhibits proliferation and induces nM) and ALK6 (TGFβ1/BMP signaling) and subsequent SMAD apoptosis in Bcr-abl-expressing cells. A11411 Dovitinib (TKI-258) *Available package size: 2,5,25,50mg *Available package size: 10,25,50mg A11773 ASP3026 ARQ-197 is a selective inhibitor of the c-Met receptor tyrosine kinase. A11948 AP26113 A13120 PD173955 *Available package size: 10,50,100,200mg A13065 AZD3463 A13237 GNF-5 A11132 INCB28060 A13238 LDK-378 FAK

Dovitinib is a small-molecule multitargeted receptor tyrosine kinase A11142 PF 431396 inhibitor, which inhibits Ba/F3 cells transformed to IL3 independence by ZNF198-FGFR1 or BCR-FGFR1 with IC50 values of 150 nM and 90 A11192 PF-562271 nM, respectively. *Available package size: 10,25,50,100mg

A12427 TCS 359 INCB28060, a novel inhibitor of c-MET kinase. INCB28060 exhibits picomolar enzymatic potency and is highly specific for c-MET with LDK378 is a highly selective, orally bioavailable and ATP-competitive A13454 SB1317 (TG-02) more than 10,000-fold selectivity over a large panel of human small molecule inhibitor of ALK (Anaplastic Lymphoma Kinase), a kinases. This inhibitor potently blocks c-MET phosphorylation and receptor tyrosine kinase considered to be an important lung cancer activation of its key downstream effectors in c-MET-dependent tumor drug target. c-MET cell lines. *Available package size: 5,10,25,50mg *Available package size: 5,10,25,50mg A10063 AMG 208 PF-562271 is an orally bioavailable small molecule and ATP- A11150 NVP-BVU972 A13744 CEP-28122 competitive focal adhesion kinase (FAK) inhibitor with potential A10153 BMS-777607 A11257 EMD-1214063 antineoplastic and antiangiogenic activities. A11396 E-7050 (Golvatinib) BCR-ABL *Available package size: 5,10,50,100mg ALK A10080 AP24534 (Ponatinib) A11235 PF 573228 A11929 PF-04554878

A10662 TAE684 A12580 PF-00562271 SRC BMS-777607 is a MET tyrosine kinase inhibitor that binds to c-Met protein, or HGFR, preventing binding of HGF and disrupting the MET signaling pathway. *Available package size: 5,10,50,100mg

A10108 Saracatinib (AZD0530) Masitinib (AB1010) is a protein tyrosine kinase inhibitor. AMG-Tie2-1 is a highly potent, non-selective inhibitor of Tie-2 (IC50 *Available package size: 10,25,50,100mg <1 nM). Axl *Available package size: 5,10,25,50mg A10679 OSI-930 A10153 BMS-777607 A11518 Pazopanib(GW-786034) Bone Morphogenetic Proteins (BMP) A10996 XL184 free base (Cabozantinib) A13741 R428 Spleen tyrosine kinase (Syk) A10959 UK-383367 Saracatinib (AZD0530) is a highly selective, orally available, dual- A10161 Bosutinib (SKI-606) Tyrosine kinase specific Src/Abl kinase inhibitor with IC50 of 2.7 and 30 nM for c-Src and Abl kinase, respectively. A11472 Ki 20227 *Available package size: 10,25,100,200mg A13587 AG-1288 A10290 Dasatinib (BMS-354825) A13589 AG 957 A11020 PCI-32765

UK-383367 is a potent and selective inhibitor of BMP-1. Bosutinib (SKI-606) is a tyrosine kinase inhibitor undergoing *Available package size: 10,25,50,100mg research for use in the treatment of cancer. A12820 DMH-1 *Available package size: 10,50,100,200mg A12821 LDN-212854 A10769 R406 Tyrphostin AG 957 is a potent tyrosine kinase inhibitor. Selectively Bruton's tyrosine kinase blocks the tyrosine kinase activity of human p210bcr-abl (Ki = 750 PCI-32765 is an orally bioavailable small-molecule inhibitor of A11020 PCI-32765 Bruton's tyrosine kinase (BTK) with potential antineoplastic activity. *Available package size: 5,10,25,50mg nM) over p140c-abl (Ki = 10 μM). *Available package size: 5,10,25,100mg A11348 CGI1746 A12706 GDC-0834 A11177 KX2-391 R406 is an orally available spleen tyrosine kinase inhibitor with an A13202 AVL-292 Trk Receptors A12214 KX1-004 IC50 of 41 nM. A12417 MLR 1023 A13730 GNF 5837 *Available package size: 2,5,10,25mg A12723 PP2 A10770 R406 (freebase) A12724 PP1 A10771 R935788 A11320 BAY 61-3606 AVL-292 is a highly selective, covalent Btk inhibitor. A11926 R788 (Fostamatinib) *Available package size: 5,10,25,50mg A11952 P505-15 A13233 CNX-774 GNF-5837 is a potent, selective, and orally bioavailable pan-TRK A12162 Piceatannol inhibitor that inhibited tumor growth in a mouse xenograft model A12731 PRT062607 HCL derived from RIE cells expressing both TRKA and NGF. A13884 GS-9973 *Available package size: 10,25,50,100mg

PP2 is a selective inhibitor of Src-family tyrosine kinases. Inhibits CNX-774 is a potent Btk inhibitor (IC50 < 1 nM). p56lck and p59fynT (IC50 values are 4 and 5 nM respectively). Displays > 10000-fold selectivity over ZAP-70 and JAK2. Moderately *Available package size: 5,10,25,50mg

*Available package size: 10,25,50,100mg inhibits CSK (IC50 = 0.73 μM). A13232 1-NA-PP1 GS-9973 is an oral inhibitor of spleen tyrosine kinase (Syk), with A13290 A-419259 potential antineoplastic activity. NF-kB/IkB A13573 PP1 Analog II, 1NM-PP1 *Available package size: 10,25,50,100mg Deferasirox is a rationally-designed oral iron chelator. Its main use is A13821 CGP77675 NF-kB to reduce chronic iron overload in patients who are receiving long- Tie-2 term blood transfusions for conditions such as beta-thalassemia and c-Kit A10293 Deferasirox other chronic anemias. A10932 Tie2 kinase inhibitor *Available package size: 5,10,25,50mg A10250 Regorafenib (BAY 73-4506) A13456 AMG-Tie2-1 A11318 BMS 345541 A10558 Masitinib (AB1010) A11338 Bay 65-1942 HCl A11339 Bay 65-1942 A11821 Bindarit A12669 Teglarinad chloride

A12748 QNZ A10535 Lomustine (CeeNU) A11579 TPCA-1 A12746 SC-514 TGF-β / Smad

A11010 Zoledronic Acid TGF-β / Smad Inhibitors A11060 CX-4945 (Silmitasertib)

A10827 SB 525334 A11554 Sotrastaurin (AEB071) QNZ inhibits the activation of the transcription factor NF-κB and has *Available package size: 5,10,25,50mg been used to investigate NF-κB signaling.

Cytokines includingSC-514 is JNK, an orally p38, MK2 active, and ATP-competitive ERK. IKKβ inhibitor (IC50 = 3 - 12 μM) that displays > 10-fold selectivity over 28 other kinases *Available package size: 10,25,50,100mg A10881 Suplatast tosilate A12548 VGX-1027 A12836 IKK-16 A12837 IMD 0354 A13108 PHA 408 IKK SB525334 is a selective inhibitor of transforming growth factor-β expressionreceptor I in(ALK5, kidney TGF-βRI) cells. (IC50 = 14.3 nM). Inhibits TGF-β1- Sotrastaurin is a protein kinase C inhibitor for the prevention of induced smad2/3 nuclear localization and TGF-βRI-induced mRNA transplant rejection and treatment of psoriasis. *Available package size: 5,10,50,100mg *Available package size: 5,10,25,50mg A11017 LY2157299 JAK / Stat A11133 LY2109761 A12399 Ruboxistaurin (LY333531) A11157 SB-505124 A12419 Go 6976 A13094 alpha-Amyloid Precursor Protein Modulator A12808 CEP33779 JAK A13197 GF 109203X A13082 PF-03394197 (oclacitinib) A10095 AT9283 A13162 GLPG0634 Protein Kinase A A10104 AZ-960 A13454 SB1317 (TG-02) A10110 AZD1480 A13457 JAK Inhibitor I A11935 H 89 dihydrochloride A14049 WHI-P 154 type I receptor (ALK5), ALK4 and ALK7 (IC50 values are 47 and 129 nMSB-505124 for ALK5 is and a selective ALK4 respectively). inhibitor of transforming growth factor-β Stat *Available package size: 5,25,50,100mg

A10244 Cryptotanshinone A11405 Astragaloside A AZD1480 is a novel potent small JAK2 inhibitor with an IC50 of 0.26 A10395 Fludarabine Phosphate (Fludara) A11762 RepSox (SJN 2511) H 89 dihydrochloride is a cell-permeable, selective, reversible, ATP- nM. competitive and potent inhibitor of protein kinase. A10396 Fludarabine (Fludara) A12358 A 83-01 *Available package size: 5,10,50,200mg *Available package size: 10,,25,50,100mg A10817 S3I-201 (NSC 74859) A12924 ITD-1 A10241 CP-690550 (Tofacitinib citrate) A10263 Cyt387 Protein Kinase C (PKC) Protein kinase D (PKD)

A10196 Chelerythrine Chloride A12416 CID 2011756 A10356 LY317615 (Enzastaurin) A12423 kb NB 142-70 A13804 CID 755673 S3I-201 (NSC 74859) is a novel inhibitor of Stat3 that inhibits Stat3, Stat3 complex formation and Stat3-DNA binding activity in vitro (IC50 = 86 ± 33 µM) and Stat3-dependent transcriptional activities. CYT387 is an inhibitor of Janus kinases JAK1 and JAK2, acting as an *Available package size: 5,10,50,100mg ATP competitor with IC50 values of 11 and 18 nM, respectively. *Available package size: 10,25,50,200mg Proteases A10546 LY2784544 Pim Kinase A11041 INCB018424 (Ruxolitinib) A10838 SGI-1776 (free base) Caspase Proteasome A11082 TG-101348 A11945 SMI-4a A11180 TG101209 A10984 VX-765 A10085 Artemether (SM-224) A11967 TCS PIM-1 4a A11193 NVP-BSK805 A11090 PAC-1 A10160 Bortezomib (Velcade) A12896 CX-6258 A11241 BMS-911543 A11944 Apoptosis Activator 2 A10284 Danoprevir (RG7227) A11329 Baricitinib (LY3009104) A12373 Z-VAD-FMK A10320 Disulfiram A11795 WP1066 A13070 LY573636 (Tasisulam) A10600 MLN2238 A12394 XL019

A10602 MLN9708 BIIB021 is an oral fully synthetic Hsp90 inhibitor that selectively and HIV Protease potently inhibits the molecular chaperone Hsp90 thereby inhibiting the proper assembly of multiple oncogenic proteins involved in tumor A10096 Atazanavir sulfate (BMS-232632-05) growth and survival. *Available package size: 5,10,50,100mg A10097 Atazanavir A10512 Lamivudine A10178 Capsaicin A10537 Lopinavir (ABT-378) MLN9708 is a proteasome inhibitor, which inhibits the activity of the A10343 Elesclomol proteasome, blocking the targeted proteolysis normally performed by VX-222 is a small molecule non-nucleoside inhibitor of HCV NS5B A10659 AUY922 (NVP-AUY922) the proteasome. polymerase that is being investigated for the treatment of hepatitis C *Available package size: 5,10,50,100mg virus infection. *Available package size: 5,10,50,100mg A10617 Nafamostat mesylate A11043 MG-132 A11295 Asunaprevir (BMS-650032)

Lopinavir is an inhibitor of the HIV protease. *Available package size: 10,100,200mg

A10799 Ritonavir AUY922 (NVP-AUY922) is highly potent and oral inhibitor of Hsp90 MG-132 is a potent cell-permeable inhibitor of proteasome (IC50 = with IC50=21 nM in Hsp90 FP binding assay and inhibits proliferation of various human cancer cell lines in vitro, with GI50 average 9 nM. *Available package size: 10,25,50,100mg *Available package size: 5,10,25,100mg 100 nM) and calpain (IC50 = 1.2 μM). A11145 CEP-18770 A10660 NVP-BEP800 A11025 Geldanamycin A11062 AT13387 Asunaprevir is an inhibitor of the viral enzyme serine protease NS3. *Available package size: 5,10,25,50mg A11074 PF-04929113 (SNX-5422) A11332 Boceprevir (SCH-503034) Ritonavir inhibits the HIV viral proteinase enzyme which prevents A11130 PU-H71 cleavage of the gag-pol polyprotein, resulting in noninfectious, A11131 MPC-3100 immature viral particles. A11189 SNX-2112 *Available package size: 10,25,50,100mg A11195 KW-2478 A11378 Saquinavir CEP-18770 is a novel orally active proteasome inhibitor with a favorable tumor selectivity profile for the treatment of MM and other A11853 Darunavir Ethanolate (Prezista) malignancies responsive to proteasome inhibition. A11871 Indinavir sulfate *Available package size: 5,10,50,100mg A11985 Amprenavir A11278 PR-171 (Carfilzomib) Boceprevir is a protease inhibitor used as a treatment for hepatitis C genotype 1. *Available package size: 5,10,25,50mg

A11335 Balapiravir (R1626) KW-2478 is an agent that targets the human heat-shock protein 90 A11336 BMS-790052 2HCl (Hsp90) with potential antineoplastic activity. *Available package size: 5,10,50,100mg A11343 Ciluprevir (BILN 2061) Amprenavir is an human immunodeficiency virus (HIV) protease A11519 PSI-6130 inhibitor with IC50 of 14.6 ± 12.5 ng/ml for wild-type HIV isolates A11251 XL-888 A11529 PSI-7977 *Available package size: 5,10,25,50mg PR-171 (Carfilzomib) is a tetrapeptide epoxyketone and a selective A11269 IPI-504 (Retaspimycin hydrochloride) proteasome inhibitor. It is an analog of epoxomicin. A11530 PSI-6206 A12583 Fosamprenavir A11272 IPI-493 *Available package size: 5,10,25,50mg A11583 Tegobuvir (GS-9190) A13156 GSK2838232A A11522 Pralatrexate A12357 BMS-790052 A12003 (-)-Gallocatechin A12374 VCH-916 Heat Shock Proteins (HSP) A12768 Lactacystin A13105 Setrobuvir (ANA-598) A12933 P 22077 A13118 Celgosivir A10010 17-AAG (KOS953) A13711 Gliotoxin A13155 Ledipasvir (GS 5885) A10011 17-DMAG HCl (Alvespimycin) A14048 PSI A10143 BIIB021

IPI-493 is a potent and orally bioavailable HSP90 inhibitor with Ki of HCV Protease 21 nM. *Available package size: 1,2,5,10mg A10159 BMS-790052 A10902 Telaprevir (VX-950)

A10980 VX-222 Ledipasvir is an inhibitor of the hepatitis C virus HCV NS5A protein. *Available package size: 5,10,25,50mg

A11768 Radicicol Linagliptin is a DPP-4 inhibitor, an enzyme that degrades the incretin hormones glucagon-like peptide-1 (GLP-1) and glucose-dependent MMP Cathepsin A12388 MKT 077 insulinotropic polypeptide (GIP). A12648 CUDC-305 (DEBIO-0932 ) *Available package size: 5,10,50,100mg A12826 Marimastat A12020 Balicatib A12850 HSP-990 A12848 4-epi-Chlortetracycline Hydrochloride A13256 CA-074 A12528 Vildagliptin A13351 VER 155008 A13072 NSC 405020 A13817 VER-50589 A13311 Alogliptin Benzoate A13312 Trelagliptin Succinate (SYR-472) Aminopeptidase Thrombin Epigenetics A10208 CHR2797 (Tosedostat) A10138 BIBR 953 (Dabigatran, Pradaxa) Bromodomain A12948 UNC1215 Integrase A13068 CPI-203 A11440 GSK 525762A (I-BET-762) A13163 Bromosporine A10042 Fluorouracil (Adrucil) A11783 GSK 1210151A (I-BET151) A13165 I-CBP112 A10156 BMS-707035 A13227 SGC-CBP30 A10347 Elvitegravir (GS-9137) A13717 UNC 669 BIBR 953 (Dabigatran, Pradaxa) has shown antithrombotic efficacy A13749 MS436 in animal models of thrombosis, with a rapid onset of action and predictable pharmacodynamic response. A13890 OTX015 *Available package size: 5,10,50,100mg A14015 GSK2801 A11325 BCX 1470 methanesulfonate Histone demethylases GSK1210151A is a novel selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4. A12918 GSK J1 *Available package size: 5,10,25,50mg

Elvitegravir (GS-9137) is a potent inhibitor of the strand-transfer A12545 PFI-1 step of integration mediated by human immunodeficiency virus type A12729 (+)-JQ1 1 (HIV-1) integrase. BCX 1470 blocks the esterolytic and hemolytic activities of the *Available package size: 10,50,100mg complement enzymes Cls and factor D in vitro. *Available package size: 5,10,25,50mg A10775 Raltegravir (MK-0518) A11331 BCX 1470 A11517 Otamixaban (FXV 673)

GSK J1 is a potent and selective inhibitor of the H3K27 histone Angiotensin-Converting Enzyme (ACE) demethylases JMJD3 and UTX. *Available package size: 10,25,50,100mg A10670 Olmesartan (RNH6270, CS-088) Raltegravir (MK-0518) targets integrase, an HIV enzyme that A10710 Perindopril Erbumine (Aceon) A13246 OG-L002 integrates the viral genetic material into human chromosomes, a A11317 Moxonidine critical step in the pathogenesis of HIV. A13358 Tranylcypromine hydrochloride A11615 Olmesartan medoxomil *Available package size: 5,10,50,100mg (+)-JQ1 is a potent, high affinity, selective BET bromodomain A11738 Captopril inhibitor. A11068 S/GSK1349572 A11748 Fosinopril sodium *Available package size: 5,10,25,50mg A11135 MK-2048 A11867 Imidapril (Tanatril) A11876 Lisinopril (Zestril) Dipeptidyl Peptidase IV (DPP-4) A12769 Zofenopril calcium Stem Cells A10430 Glimepiride Matrix Metalloprotease A10848 Sitagliptin phosphate monohydrate A11109 Saxagliptin (BMS-477118) A11345 CTS-1027 Stem Cell Proliferation Stem Cell Differentiation A11224 Linagliptin (BI-1356) A12985 Batimastat (BB-94) A12922 ID 8 A12926 Kartogenin Other Proteases

A11764 Camostat mesylate A12928 MI 2

CHIR-98014 is a very potent, selective, cell-permeable reversible A12737 IWR-1-endo inhibitor of GSK-3. A12816 LGK-974 *Available package size: 5,10,50,100mg GSK-3 / Wnt / Hedgehog A11143 SB-705498 A11223 TWS119 A10249 Cyclopamine γ-Secretase A10258 GDC-0449 (Vismodegib) A11048 LY2940680 A10157 BMS-708163 LGK974 is a highly potent, selective and orally bioavailable Porcupine A10288 DAPT (GSI-IX) inhibitor (Wnt signaling antagonist) with an IC50 <1 nM in the Wnt signaling reporter assay and Porcupine binding assay. *Available package size: 5,10,25,50mg

A12951 Wnt-C59 TWS119 is a 4,6 disubstituted pyrrolopyrimidine that potently GDC-0449 (Vismodegib) is a more potent novel and specific synthetic A13978 IWP-L6 oral hedgehog pathway inhibitor with an IC50 of 3 nM. *Available package size: 5,10,25,50mg inhibits GSK3β with an IC50 value of 30 nM.1 At 400 nM. *Available package size: 25,50,200mg A11592 Tideglusib A11351 TAK-441 β-catenin A11941 TDZD-8 DAPT (GSI-IX) is an inhibitor of γ-secretase that causes a reduction in A11442 GANT 58 Aβ40 and Aβ42 levels in human primary neuronal cultures with IC50 *Available package size: 5,10,50,100mg A12418 HhAntag A12737 IWR-1-endo values of 115 and 200 nM for total Aβ and Aβ42 respectively. A12920 Hh-Ag1.5 A13795 FH535 A10802 RO4929097 A13095 SANT-1 A10836 Semagacestat (LY450139) A13252 GANT61 A11174 YO-01027 GSK-3 TDZD-8 protects the brain against I/R injury by inhibiting GSK-3beta activity. A10199 CHIR-99021 *Available package size: 5,10,25,50mg

A12741 LY2090314 A12819 AZD1080 GANT61 is an inhibitor for GLI1 as well as GLI2-induced transcription, A13060 AZD2858 A13728 AR-A 014418 other pathways, such as TNF and glucocorticoid receptor gene inhibits hedgehog with IC50 of 5 μM, displays selectivity over agent. transactivation. YO-01027 is a dipeptidic γ-secretase inhibitor, an antiAlzheimer *Available package size: 5,10,25,50mg *Available package size: 10,25,50,100mg Smoothened

A11176 LY-411575 A11480 Purmorphamine Wnt A12774 LDE225 Diphosphate CHIR99021 is an aminopyrimidine derivative that inhibits GSK3α and *Available package size: 2,5,25,100mg A10994 XAV 939 GSK3β with IC50 values of 10 and 6.7 nM, respectively. A10471 Indirubin A10825 SB 216763 A11061 SB 415286

LY-411575 is a selective, cell permeable, small molecule gamma secretase inhibitor. *Available package size: 5,10,50,100mg TNKS1 and TNKS2 respectively). LDE225 is an orally bioavailable small-molecule Smoothened (Smo) XAV 939 is a TNKS inhibitor (IC50 values are 0.011 and 0.004 μM for antagonist with potential antineoplastic activity. *Available package size: 10,25,50,100mg A11194 MK-0752 *Available package size: 5,10,25,50mg SB 415286 is a potent and selective cell-permeable, ATP-competitive A11337 BMS 433796 A12362 KY02111 A12775 PF-5274857 A11393 E 2012 A12707 IWP-2 A13204 BMS-833923 (XL-139) inhibitor of GSK3α with an IC50 value of 78 nM (similar potency for A11776 LY2811376 *Available package size: 10,25,50,100mg GSK3β) and a Ki value of 31 nM. A12433 Flurizan A11085 CHIR-98014 A12444 BMS 299897 A13815 FLI-06

IWP-2 is an inactivator of Porcn function and inhibitor of Wnt BMS-833923 (or XL-139) is an orally bioavailable small-molecule Hedgehog production, and blocks beta-catenin accumulation. Wnt/b-catenin SMO (Smoothened) inhibitor with potential antineoplastic activity. ('canonical') pathway maintains transcriptional programs that enable *Available package size: 5,10,25,50mg stem cells to remain multipotent. *Available package size: 5,10,25,100mg A13881 PF-04449913

A13372 CHC P-gp Transporters Neurotransmitter Transporters A11584 Tariquidar (XR9576) A12004 Cynarin A10222 Citalopram Hydrobromide Rostafuroxin (PST-2238) is an ouabain-inhibitor counteracting A12363 Selamectin ATPase specific forms of hypertension. A10319 Dipyridamole *Available package size: 5,10,25,50mg A11919 Reboxetine mesylate CRM1 A10086 Artemisinin A11960 LY 2183240 A10213 Ciclopirox A13647 (-)-Blebbistcitin A13099 UCPH 101 A12582 KPT-330 A12975 KPT185 Multidrug Transporters AMPA receptor A10549 LY335979 A12349 Ampalex (CX-516) A11080 PSC-833 A12424 LY404187 Ciclopirox is currently being investigated as an alternative treatment A12324 Elacridar to ketoconazole for seborrhoeic dermatitis as it suppresses growth A12425 LY450108 of the yeast Malassezia furfur.It acts by inhibiting the membrane A13109 NBQX KPT185 is a selective CRM1 inhibitor. KPT-185 significantly inhibits transfer system by interrupting the Na+ K+ ATPase. leukemia cell proliferation with IC50 ranging from 100 nM to 500 A13882 DNQX *Available package size: 10,25,50,100mg nM, and induces cell-cycle arrest and apoptosis of AML cell lines and A14010 IEM 1754 Dihydrobromide primary AML blasts. A10669 Oligomycin A *Available package size: 10,25,50,100mg A10672 Omeprazole Elacridar is a prototypical BCRP inhibitor which inhibits the Bcrp1- A11156 Brefeldin A mediated transport. A11408 PF 3716556 *Available package size: 5,10,25,50mg A11696 Pantoprazole (Protonix) Sodium-dependent Glucose Cotransporter Ion Channels

(SGLT) CK-1827452 is a selective cardiac specific myosin activator. A10155 EGT1442 Calcium Channels *Available package size: 5,10,50,100mg A10285 Dapagliflozin (BMS512148) Pantoprazole is a proton pump inhibitor drug that inhibits gastric A10068 Amlodipine A11219 Azelnidipine acid secretion. A10069 Amlodipine besylate (Norvasc) A11314 AMG 073 (Cinacalcet) *Available package size: 100,500mg A10215 Cilnidipine A11729 Lacidipine A11933 KB-R7943 mesylate A10219 AMG-073 HCl (Cinacalcet HCl) A11730 Benidipine hydrochloride A11961 Bafilomycin A1 A11731 Nilvadipine (ARC029) A12022 Bufalin A11746 Clevidipine A12023 Resibufogenin Dapagliflozin inhibits subtype 2 of the sodium-glucose transport A12684 Pinaverium Bromide proteins (SGLT2), which is responsible for at least 90% of the glucose A13989 BAPTA tetrapotassium reabsorption in the kidney. AMG-073 HCl (Cinacalcet HCl) represents a new class of compounds *Available package size: 5,10,50,100mg A14023 BAPTA/AM for the treatment of hyperparathyroidism known as calcimimetics, A11100 Canagliflozin which reduce parathyroid hormone (PTH) synthesis and secretion by A12440 Empagliflozin increasing the sensitivity of the parathyroid calcium-sensing receptor (CaR) to extracellular calcium. A12680 LX-4211 *Available package size: 10,50,100mg A12690 Tofogliflozin Bufalin is a cardiotonic steroid originally isolated from the Chinese A10309 Diethylstilbestrol toad venom. A10311 Diltiazem HCl BAPTA/AM, an intracellular calcium chelator, induces delayed *Available package size: 10,25,50,100mg Monocarboxylate transporters (MCT) A10487 Isradipine necrosis by lipoxygenase-mediated free radicals in mouse cortical cultures. A12024 Bufotalin A11293 AR-C155858 A10553 Manidipine (Manyper) *Available package size: 25,50,100mg A12032 Cinobufagin A10554 Manidipine dihydrochloride A12726 Dynasore A10643 Nifedipine Ligand-gated Ion Channels A12755 Ouabain A10645 Nimodipine A13283 Rostafuroxin (PST-2238) A10921 Tetrandrine (Fanchinine) A10006 (-)-Huperzine A A11140 NPS-2143 (SB-262470) A10414 Gabapentin Hydrochloride A11206 CK-1827452 (Omecamtiv mecarbil) A10444 GYKI-52466 dihydrochloride A10490 Ivermectin AR-C155858 is a potent inhibitor of monocarboxylate transporters A10748 Prasugrel (Effient) MCT1 and MCT2 that binds to an intracellular site involving A10966 Varenicline transmembrane helices 7-10. *Available package size: 5,10,25mg A11107 GW791343 HCl

A11233 PNU 282987 A10986 VX-809 A12932 Optovin Potassium Channels A12519 VX-661 A13278 HC-030031 A13000 PPQ-102 A13333 Flufenamic acid A10433 Glyburide A13511 IOWH032 A13560 Icilin A10593 Minoxidil (U-10858) A13723 CFTR-Inhibitor-II A10629 Nateglinide (Starlix) PNU 282987 is a drug that acts as a potent and selective agonist for NMDA Receptors A10641 Nicorandil *Available package size: 10,25,50,100mg A10783 Repaglinide Transient Receptor Potential Channels A13729 MDL 29951 the α7 subtype of neural nicotinic acetylcholine receptors. A11290 A-867744 A11239 TAK-438 A12353 A 967079 A11701 Ondansetron (Zofran) A11708 Memantine hydrochloride A11862 Felbamate MDL-29951 is a novel glycine antagonist of NMDA receptor activation A11873 Lamotrigine (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo. A11947 TCN 201 *Available package size: 5,10,25,50mg A12426 SDZ 220-581 A 967079 is a selective TRPA1 channel blocker (IC50 values are 67 TAK-438 is a novel potassium-competitive acid blocker. A12681 Methyllycaconitine citrate and 289 nM at human and rat TRPA1 receptors respectively). *Available package size: 2,5,10,25mg A12751 NMDA *Available package size: 10,25,50,100mg A11521 PAP-1 (5-(4-Phenoxybutoxy)psoralen) A13784 Bretazenil Sodium Channels AMPK / Insulin Receptor A10064 Amiloride hydrochloride PAP-1 is a selective inhibitor of Kv1.3, voltage-gated potassium A10510 Lacosamide A11970 BML-275 channel. PAP-1 (EC50=2 nM) potently inhibits human T effector AMPK A10530 Lidocaine (Alphacaine) memory cell proliferation and delayed hypersensitivity. A10721 Phenytoin (Lepitoin) *Available package size: 5,10,25,50mg A10028 Acadesine (Aicar,NSC 105823) A10722 Phenytoin sodium (Dilantin) A10717 Phenformin hydrochloride A11884 Mitiglinide calcium A10795 Riluzole (Rilutek) A11071 A-769662 A11922 Retigabine (Ezogabine) A11102 PF-04971729 A11934 NS 309 A11234 A 803467 A12783 TRAM-34 A12857 E-4031 dihydrochloride

BML-275 is a cell-permeable pyrazolopyrimidine compound shown to be an AMP-activated protein kinase (AMPK) and fatty acid synthase Chloride Channels A-769662 is a new activator of AMP-activated protein kinase (AMPK). inhibitor. *Available package size: 5,10,50,100mg A 803467 is a selective blocker of NaV1.8 channels (IC50 values are A10985 VX-770 (Ivacaftor) *Available package size: 5,10,50mg 8, 2450, 6740, 7340 and 7380 nM for hNaV1.8, hNaV1.3, hNaV1.7, A13339 Talniflumate hNaV1.5 and hNaV1.2 channels respectively). *Available package size: 10,25,50,100mg Cystic Fibrosis Transmembrane Regulator A11602 Vinpocetine (CFTR) ATM / ATR A11715 Proparacaine HCl A10758 PTC124 (Ataluren) A11605 VE-821 A11728 Amiloride hydrochloride dihydrate ATM A13191 CGK 733 A11750 Ibutilide fumarate A13205 AZ-20 A13760 QX 314 chloride A10506 KU-55933 ATR PTC124 also known as Ataluren is CFTR-G542X nonsense allele inhibitor. A13289 VE-822 *Available package size: 10,25,50,100mg A10985 VX-770 (Ivacaftor)

KU-55933 is an ATM inhibitor by suppressing cell proliferation and induces apoptosis by blocking Akt in cancer cells with overactivated QX 314 chloride is a membrane impermeable quaternary derivative Akt. VE-822 is an potent ATR inhibitor. of lidocaine, a voltage-activated Na+ channel blocker. *Available package size: 5,10,50,100mg *Available package size: 5,10,25,50mg *Available package size: 50,100,250mg A13328 ETP-46464 VX-770 (Ivacaftor) is known as a CFTR potentiator. A10507 KU-60019 *Available package size: 5,10,50,100mg A11086 CP-466722

A10061 Amfebutamone (Bupropion) Acetylcholine Muscarinic Receptors A10067 Amisulpride 7-TM Receptors A10032 Acetylcysteine A10125 Benserazide hydrochloride (Serazide) A10098 Atropine A10236 Clozapine A10329 Domperidone A13766 SDZ 205-557 HCl A10147 Biperiden hydrochloride A10331 Dopamine hydrochloride 5-HT Receptors A13767 Tropanserin A10180 Bethanechol chloride A10446 Haloperidol (Haldol) A13833 RU 24969 hemisuccinate A10386 Fesoterodine fumarate (Toviaz) A10017 5-hydroxytryptophan (5-HTP) A10416 Galanthamine hydrobromide A10747 Pramipexole 2HCl monohyrate A10048 Agomelatine Adrenergic Receptors A10417 Gallamine triethiodide A10956 U 95666E A10091 Asenapine maleate A10476 Ipratropium bromide A11118 Rotigotine hydrochloride A10231 Clomipramine hydrochloride A10052 Alfuzosin HCl A10480 Irsogladine A11119 Thioridazine hydrochloride A10287 Dapoxetine hydrochloride A10149 Bisoprolol fumarate A10579 Methscopolamine bromide A11341 B-HT 920 2HCl A10437 Granisetron Hydrochloride A10232 Clonidine hydrochloride A10635 Neostigmine bromide (Prostigmin) A11553 Rotigotine A10497 Ketanserin (Vulketan Gel) A10296 Dehydroepiandrosterone A10684 Oxybutynin A11559 SB-277011 A10588 Mianserin hydrochloride A10298 Detomidine hydrochloride A10803 Rocuronium bromide A11720 Fenoldopam A10607 Mosapride citrate A10325 Dobutamine hydrochloride A10808 SVT-40776 (Tarafenacin) A11824 Blonanserin A10624 Naratriptan A10334 Doxazosin mesylate A10937 Tolterodine tartrate (Detrol LA) A11915 Ropinirole A10667 Olanzapine (LY170053) A10484 Isoprenaline HCl A11166 5-hydroxymethyl tolterodine A11916 Ropinirole HCl A10674 Ondansetron HCl (GR 38032F) A10555 Maprotiline hydrochloride A11203 PNU-120596 A11937 GBR-12935 dihydrochloride A10691 Paliperidone A10618 Naftopidil (Flivas) A11215 Solifenacin succinate A11998 Rotundine A10759 Puerarin (Kakonein) A10619 Naftopidil Dihydrochloride A11706 Tropicamide A12415 BP897 A10797 Risperidone (Risperdal) A10630 Nebivolol HCl A11712 Orphenadrine citrate A12536 Pramipexole dihydrochloride A10931 Tianeptine sodium A10686 Oxymetazoline hydrochloride A11719 Rivastigmine tartrate A12991 GR 103691 A11106 LY310762 A10719 Phenoxybenzamine hydrochloride A11975 Methoctramine hydrate A13087 Naxagolide A11116 Vilazodone A10794 Rilmenidine A11987 Darifenacin A13694 L-741626 A11165 RS-127445 A10819 Salbutamol sulfate (Albuterol) A13071 Arecoline A13844 Cabergoline A11178 BRL-15572 A10882 Synephrine (Oxedrine) A11182 WAY-100635 A11229 Metroprolol succinate Histamine Receptors Opioid Receptors A11666 Phenylephrine hydrochloride A11208 BMY 7378 A10350 Enalapril maleate A11668 DL-Adrenaline A10117 Azelastine hydrochloride (Allergodil) A11226 Tropisetron (ICS 205930) A10561 MCOPPB trihydrochloride A11713 Metoprolol tartrate A10195 Cetirizine Dihydrochloride A11310 Alosetron A11072 ADL5859 HCl A11721 Betaxolol A10205 Chlorpheniramine maleate A11418 Eletriptan hydrobromide A11076 JTC-801 A11732 Formoterol hemifumarate A10218 Cimetidine A11702 Mirtazapine A11210 BRL 52537 hydrochloride A11733 Betaxolol hydrochloride A10226 Clemastine fumarate A11703 Trazodone hydrochloride A11322 BAN ORL 24 A11734 Phentolamine mesilate A10538 Loratadine A11704 Urapidil hydrochloride A11718 Trimebutine A11740 Terazosin hydrochloride A10671 Olopatadine hydrochloride A11705 Duloxetine A13843 Nalmefene hydrochloride A11717 Duloxetine HCl A11788 Salmeterol A11117 Ciproxifan maleate A11222 Rupatadine A11743 Tegaserod maleate A11807 Adrenalone HCl GABA Receptors A11771 Prucalopride A11843 Carvedilol A11340 Bepotastine Besilate A11868 Ivabradine HCl (Procoralan) A11360 Ciproxifan A11799 Almotriptan malate (Axert) A10121 Baicalin A11905 Procaterol HCl A11699 Brompheniramine A11801 Aripiprazole (Abilify) A10397 Flumazenil A11914 Prazosin HCl A11709 Cyproheptadine hydrochloride A11925 SB269970 HCl A10412 Furosemide A11923 ARN-509 A11724 Mizolastine A12378 Lorcaserin A10413 Gabapentin A12657 Tamsulosin A11859 Fexofenadine HCl A12521 Lu AE58054 A10754 Primidone (Mysoline) A12795 Arformoterol tartrate A11921 Roxatidine acetate hydrochloride A12598 lorcaserin hydrochloride (APD-356) A10849 SKF 89976A hydrochloride A12844 Formoterol A12356 Rupatadine Fumarate A12602 Vortioxetine hydrobromide A12590 (+)-Bicuculline A13080 Tetrahydrozoline Hydrochloride A12661 Bilastine A13075 Eletriptan A12689 Phenazepam A13225 ICI 118,551 hydrochloride A12713 JNJ7777120 A13092 NAD 299 hydrochloride (Robalzotan) A13696 2-Hydroxysaclofen A13406 Bisoprolol A12845 Bepotastine A13267 PRX-08066 A13726 AWD 131-138 A13293 Tandospirone A13413 Medetomidine hydrochloride A13086 Metiamide A13757 PU 02 A13419 Octopamine hydrochloride Purinergic (P2Y) Receptors A13762 N-Desmethylclozapine A13422 Pindolol Dopamine Receptors A13738 Nebivolol

A10233 Clopidogrel (Plavix) A10556 Maraviroc (UK-427857) A11238 Ticagrelor (AZD6140) A10971 Vicriviroc Malate Adenosine Receptors Leukotriene receptor A11486 MRS 2578 A11097 SRT3109 A10040 Adenosine A11607 MK-0679 (Verlukast) A11104 INCB 3284 dimesylate A10066 Aminophylline A11908 Pranlukast (ONO 1078) A11127 MK-0812 Metabotropic glutamate receptors (mGluR) A10339 Dyphylline A13090 LY 255283 A11315 AMD 070 A10544 LY2140023 (LY404039) A11451 Istradefylline (KW-6002) A11555 SCH-527123 A11126 BINA A11560 SYN-115 Orexin Receptors A11577 SRT3190 A11181 ADX-47273 A11619 CGS 21680 hydrochloride A11953 AMD 3465 Hexahydrobromide A11500 MK-4305 (Suvorexant) A11754 VU 0357121 A12695 SCH 442416 A12383 Reparixin A12651 SB-649868 A11968 CTEP A12846 Tamsulosin hydrochloride A12588 WZ811 A12786 SB 334867 A12467 VU 0361737 A13745 CVT 6883 A12596 MSX-122 A13439 TCS 1102 A12589 MPEP hydrochloride A13074 AMD3100 (Plerixafor) A12664 VU 0364439 Cannabinoid Receptors Somatostatin Receptors A12705 PHCCC G Protein A11253 GW842166X A12782 Octreotide A13123 LY 379268 A11513 Org 27569 A13236 MPEP HCl A11228 QS 11 A11547 Rimonabant (SR141716) A13758 SIB 1757 NK1 Receptors A11373 CCG-63802 A11780 JWH 133 A13759 SIB 1893 A12912 CASIN A11932 WIN 55,212-2 mesylate A13103 GW679769 (Casopitant) A13886 EHT 1864 A11938 BML-190 A13104 Ibodutant (MEN 15596) Angiotensin Receptors A11939 MDA 19 A11942 CP 945598 hydrochloride A10891 Tasosartan Platelet-Activating Factor (PAF) Receptors Protease-Activated Receptors (PAR) A12849 AB-FUBINACA A10905 Telmisartan A13495 ML 161 A10429 Ginkgolide B A12914 AM251 A11121 Eprosartan A11739 Ginkgolide A A11775 Azilsartan (TAK-536) Neurotensin Receptors A13747 Eprosartan mesylate Endothelin Receptors A11770 SR 48692 Melatonin Receptors A11006 Zibotentan (ZD4054) A11091 Bosentan A10564 Melatonin A11291 Ambrisentan (BSF 208075) Endocrinology / Hormones A11564 Sitaxsentan sodium (TBC-11251) Peptide Receptors A10598 MK 3207 hydrochloride P2X Receptor Pregnane X Receptors A11255 MK-0974 (Telcagepant) A11107 GW791343 HCl A10791 Rifampin A11567 SB-408124 A11316 A 740003 A11700 Meclizine dihydrochloride A11594 Tolvaptan A11473 KN-62 A11909 Pregnenolone A11820 Prostaglandin E1 (PGE1) A11690 Ticlopidine hydrochloride A11979 YIL 781 TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist. A11972 NF 279 A12158 BIIE 0246 Estrogen Receptors *Available package size: 5,10,50,100mg A12412 A-317491 sodium salt hydrate A12350 Ozarelix A10230 Clomifene citrate A11665 Bazedoxifene acetate A12351 Desmopressin LPA Receptor A10308 Dienogest A11667 Ethisterone A12646 Melanotan II A10336 Drospirenone A11965 GW9508 A12790 Parathyroid Hormone 1-34, Human A10501 Ki16425 A10375 Evista (Raloxifene Hydrochloride) A12083 Liquiritigenin A12860 THIQ A11966 Ki16198 A10410 Fulvestrant (Faslodex) A13299 XCT 790 A13102 BMS-927711 A10439 GSK1292263 A13740 Zearalenone Prostanoid Receptors A10451 Hexestrol Smoothened Receptors A10550 LY500307 A10688 Ozagrel(OKY-046) Progesterone Receptors A10591 Mifepristone (Mifeprex) A10520 LDE225 (NVP-LDE225) A11483 Laropiprant (MK0524) A10336 Drospirenone A11018 TAK-875 A11742 Ozagrel hydrochloride A10529 Levonorgestrel Chemokine Receptors (CCR5) A13498 Cloprostenol (sodium salt) A10885 Tamoxifen Citrate A13751 BAY-u 3405

A12166 Mogroside II A2 Renin-angiotensin-aldosterone system (RAAS) A12652 T0901317 Vitamin D Receptors

A10123 Benazepril hydrochloride A12865 Cerpegin A11413 Ercalcidiol A10175 Candesartan (Atacand) Aromatase GnRH receptor MDV3100 is androgen-receptor inhibitor. Highly recommended inhibitor in AR research. A10075 Anastrozole A12375 NBI-42902 *Available package size: 5,10,25,50mg A10378 Exemestane A12376 SR 144528 A10523 Letrozole A12396 AZD3514 A12805 BMS564929 A13398 Bopindolol malonate

Candesartan is an angiotensin receptor blocker (also called an A13407 Clenbuterol hydrochloride angiotensin-II receptor antagonist or an AIIRA). *Available package size: 5,10,50,100mg PPAR A10176 Candesartan cilexetil (Atacand) A10424 Gemfibrozil (Lopid) SR 144528 displays a Ki value of 0.6 nM for rat spleen and human A10351 Enalaprilat dihydrate recombinant CB2 receptors and a Ki value of 400 nM for rat brain and A10807 Rosiglitazone (BRL-49653) Letrozole is an Aromatase inhibitor. CGS 20267 is a new non-steroidal human recombinant CB1 receptors. A10810 Rosuvastatin calcium (Crestor) compound which potently inhibits aromatase in vitro (IC50 of 11.5 *Available package size: 5,10,25,50mg A11122 Rosuvastatin *Available package size: 10,50,100mg A11123 Aliskiren hemifumarate nM) and in vivo (ED50 of 1–3 μg/kg p.o.) A12613 Abarelix Acetate A11184 Clinofibrate A10563 Megestrol Acetate A12840 Degarelix acetate A11616 Aliskiren (CGP 60536) A11088 Fadrozole A12862 Ganirelix A11736 Quinapril hydrochloride Rosiglitazone works as an insulin sensitizer, by binding to the PPAR A11745 Moexipril hydrochloride receptors in fat cells and making the cells more responsive to insulin. Retinoic Acid Receptors GPR A11747 Cilazapril monohydrate *Available package size: 25,50,100,200mg A11749 Temocapril A11792 AM 580 A13186 AZD1981 A10809 Rosiglitazone maleate A13201 PD 123319 ditrifluoroacetate A11793 CD 437 A11137 Cetaben A12430 Palovarotene A11437 GW 501516 A13113 Talarozole A11727 Ciprofibrate A11981 Troglitazone A11982 GW 7647 Glucocorticoid receptors A11983 L-165,041 A10457 Hydrocortisone(Cortisol) AZD1981, as a potent antagonist in a disease relevant cell system, A11984 GW 9662 inhibits DK-PGD2-induced CD11b expression in human eosinophils A11860 Fluticasone propionate PD 123319 ditrifluoroacetate is a potent, selective, non-peptide with IC50 of 10 nM. angiotensin AT2 receptor antagonist. IC50 values are 34 and 210 nM A12360 pirinixic acid (WY 14643) *Available package size: 5,10,25mg in rat adrenal tissue and brain respectively. A12391 GSK-3787 *Available package size: 10,25,50,100mg A12392 GSK 0660 A12413 GW6471 Androgen Receptors A10008 (R)-Bicalutamide Liver X receptors (LXRs) Transferases A10009 17 alpha-propionate A10076 Andarine (GTX-007) A11141 GW4064 Glucocorticoid receptors A10142 Bicalutamide (Casodex) A11186 WAY-362450 A10253 Ostarine (MK-2866) A11204 GW3965 HCl A11199 A 922500

Etomoxir is an inhibitor of carnitine palmitoyltransferase A (CPT1), which is required for the oxidation of long-chain acyl CoA esters. Also a strong inhibitor of mitochondrial CPT1 and a candidate as an anti- diabetic drug. Ostarine is an androgen receptor modulator (SARM). A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor *Available package size: 5,10,25,50mg (IC50 values are 7 and 24 nM at human and mouse DGAT-1 *Available package size: 5,10,50,200mg GW3965 HCl is a selective and orally active liver X receptor (LXR) full respectively). agonist. A10562 MDV3100 *Available package size: 5,10,50,100mg *Available package size: 5,10,50,100mg Phosphorylases A11415 Etomoxir A11173 CP-91149

EPZ005687 is a potent inhibitor of EZH2 (K(i) of 24 nM). Methyltransferases *Available package size: 5,10,25,50mg A11763 BIX 01294 A12712 EPZ-6438 Ubiquitin A12735 EPZ-5676 A13209 IU1 activating enzyme E1 A13277 P005091

A13254 PYR-41

BIX 01294 is a G9a-like protein and G9a histone lysine methyltransferase inhibitor. *Available package size: 10,25,50,100mg EPZ-5676 is a small molecule inhibitor of histone methyltransferase with potential antineoplastic activity. A13110 Opicapone (BIA 9-1067) P005091 is a selective inhibitor of ubiquitin-specific protease (USP) 7 *Available package size: 5,10,25,50mg (IC50 = 4.2 uM). *Available package size: 10,25,50mg Protein Prenyltransferases A12812 Chaetocin PYR-41 is a cell-permeable, irreversible ubiquitin-activating enzyme A12941 SGC 0946 A12368 FTI 277 *Available package size: 10,25,50,100mg (E1) inhibitor (IC50 < 10 μM). p97 A14020 LB42708 A12377 NMS-873 E3 ubiquitin ligase FPTase A13253 SMER-3 A12328 Lonafarnib (SCH66336)

SGC 0946 is a potent DOT1L methyltransferase inhibitor that blocks DUB H3K79 methylation in A431 cells and MCF10A cells. A12715 LDN-57444 *Available package size: 5,10,25,50mg A13190 PR-619 NMS-873 is a potent and specific small molecule allosteric inhibitor A12983 EPZ004777 of the ATPase VCP/p97 (IC50 ~0.03 uM), identified by a high- A13114 GSK343 throughput screening. A13194 UNC0646 *Available package size: 5,10,25,50mg A13200 UNC0321 A12736 DBeq Lonafarnib (SCH 66336) is a selectively FPTase inhibitor for A13690 UNC 0638 H-ras, K-ras-4B and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM, respectively. *Available package size: 5,10,25,50mg PR-619 is a cell-permeable, reversible, and broad-spectrum inhibitor Histone Methyltransferase of the deubiquitinylating enzymes (DUBs). *Available package size: 5,10,25,50mg A11377 DZNep

UNC 0638 is a selective inhibitor of G9a and GLP histone lysine methyltransferases. Others *Available package size: 10,25,50mg A10035 Acitretin Histone Acetyltransferases Other inhibitors A10038 Adapalene A10005 (-)-Epigallocatechin gallate A10044 Aesculin (Esculin) A12814 Garcinol A10013 3-Indolebutyric acid A10051 Alfacalcidol 3 Deazaneplanocin A (DZNep) is a cyclopentenyl analog of A12815 C646 A10014 4-Demethylepipodophyllotoxin A10054 Alizarin 3-deazaadenosine, originally synthesized as an inhibitor of A13378 NU 9056 A10055 Allopurinol S-adenosyl-L-homocysteine hydrolase. A10015 4-Methylumbelliferone (4-MU) A10056 Allopurinol sodium *Available package size: 1,2,5,10mg DNA Methyltransferases A10016 5-Aminolevulinic acid hydrochloride A10018 7-Aminocephalosporanic acid A10057 Aloe-emodin A12439 EPZ005687 A12785 Lomeguatrib A10023 ABT-492 A10058 Aloin (Barbaloin) A10029 Acarbose A10059 Altretamine A10031 Acetanilide A10065 Aminocaproic acid (Amicar) A10033 Acipimox A10070 Ammonium Glycyrrhizinate (AMGZ) A10034 Acitazanolast A10072 Amorolfine Hydrochloride

A10073 Amphotericin B A10245 Crystal violet A10427 Gentamycin sulfate (Gentacycol) A10616 Myricitrin (Myricitrine) A10074 Amygdalin A10247 Curcumol A10428 Gestodene A10621 Nanchangmycin A10077 Andrographolide A10252 Dihydromyricetin (Ampeloptin) A10432 L-Glutamine A10626 Naringin (Naringoside) A10083 Aprepitant (MK-0869) A10260 Cyclosporin A A10434 Glycyrrhizic acid A10627 Naringin Dihydrochalcone A10084 Arbutin (Uva, p-Arbutin) A10261 Bryostatin 1 A10435 Gossypol A10628 Natamycin (Pimaricin) A10087 Artesunate A10262 Cyclovirobuxin D (Bebuxine) A10436 Gramine A10633 Neohesperidin A10099 Azomycin (2-Nitroimidazole) A10265 Cytarabine A10443 Guaifenesin (Guaiphenesin) A10634 Neohesperidin dihydrochalcone A10106 Azalomycin-B A10266 Cytisine (Baphitoxine, Sophorine) A10445 Gynostemma Extract A10636 Nepafenac A10107 Azathioprine A10282 Daidzein A10447 Hematoxylin (Hydroxybrazilin) A10651 Nobiletin (Hexamethoxyflavone) A10118 Aztreonam (Azactam, Cayston) A10283 Daidzin A10450 Hesperidin A10652 Norfloxacin (Norxacin) A10124 Bendamustine HCl (SDX-105) A10289 Daptomycin A10454 Hordenine A10656 Phenprocoumon A10126 Berberine Hydrochloride A10291 D-Cycloserine A10455 Hydralazine hydrochloride A10663 NXY-059 (Cerovive) A10127 Bergenin (Cuscutin) A10294 Deflazacort A10456 Hydrochlorothiazide A10666 Ofloxacin (DL8280) A10128 Beta Carotene A10297 Desonide A10458 Hydroxocobalamin (Vitamin B12a) A10668 Oleanolic Acid (Caryophyllin) A10129 Betamethasone A10299 Dexamethasone A10459 Hydroxyurea A10675 Oridonin (Isodonol) A10130 Betamethasone dipropionate A10300 Dexrazoxane Hydrochloride A10460 Hyodeoxycholic acid A10676 Orlistat A10131 Betamethasone valerate A10302 D-glutamine A10467 Iloperidone A10677 Orotic acid (6-Carboxyuracil) A10136 Biapenem A10305 Diclofensine A10469 Imiquimod (Aldara) A10680 Osthole A10139 BIBR-1048 (Dabigatran etexilate) A10306 Didanosine A10470 Indapamide (Lozol) A10682 Oxacillin sodium monohydrate A10144 Bilobalide A10307 Dienestrol A10472 Indocyanine green A10685 Oxymatrine (Matrine N-oxide) A10145 Bimatoprost (Lumigan) A10310 Dihydroartemisinin A10473 Indole-3-carbinol A10687 Oxytetracycline (Terramycin)

A10146 Biochanin A (4-Methylgenistein) A10313 Dimesna (BNP7787) A10481 Isoconazole nitrate A10690 Paeonol (Peonol) A10165 BTZ043 (BTZ038, BTZ044) A10314 Dioscin (Collettiside III) A10482 Isoliquiritigenin A10692 Palmatine chloride A10166 Budesonide A10315 Diosgenin A10489 Itraconazole (Sporanox) A10694 Pamidronate Disodium A10167 Bumetanide A10316 Diosmetin A10503 Kinetin A10698 Parthenolide ((-)-Parthenolide) A10168 Bupivacaine hydrochloride A10317 Diosmin A10509 L(+)-Rhamnose Monohydrate A10708 Pentagastrin A10169 Busulfan (Myleran, Busulfex) A10318 Diphenhydramine hcl A10515 Lappaconite Hydrobromide A10723 Phloretin (Dihydronaringenin) A10170 Butylscopolamine BR A10321 Divalproex sodium A10517 L-Ascorbyl 6-palmitate A10724 Phlorizin (Phloridzin) A10171 Caffeic acid A10322 DL-Carnitine hydrochloride A10521 Leflunomide A10725 Vanoxerine 2HCl (GBR-12909) A10173 Calcitriol (Rocaltrol) A10323 D-Mannitol A10524 Leucovorin Calcium A10732 Pimecrolimus A10181 Carbidopa A10327 Docosanol A10531 Limonin A10734 Piperine (1-Piperoylpiperidine) A10186 Cefaclor A10328 Dofetilide A10533 Linezolid (PNU-100766) A10738 Pizotifen malate A10187 Cefdinir A10332 Doripenem Hydrate A10539 Loteprednol Etabonate A10741 Polydatin (Piceid) A10189 Cefoselis sulfate A10333 Dorzolamide HCL A10540 Lubiprostone A10744 Posaconazole A10190 Cefprozil hydrate (Cefzil) A10335 Doxercalciferol A10543 LY2886721 A10750 Praziquantel (Biltricide) A10191 Ceftiofur hydrochloride A10341 Ecdysone A10551 Magnolol A10752 Prednisone (Adasone) A10192 Celastrol A10342 Econazole nitrate A10552 Malotilate A10753 Prilocaine A10197 Chenodeoxycholic acid A10348 Emodin A10557 Marbofloxacin A10758 PTC124 (Ataluren) A10201 Chlormezanone (Trancopal) A10353 Glycyrrhetinic acid (Enoxolone) A10565 Meloxicam (Mobic) A10767 Quetiapine fumarate A10202 Chlorogenic acid A10361 Ergosterol A10567 Meprednisone (Betapar) A10772 Racecadotril (Acetorphan) A10203 Chlorothiazide A10376 Evodiamine (Isoevodiamine) A10569 Meropenem A10777 Ramelteon (TAK-375) A10207 Chlorprothixene A10379 Ezetimibe (Zetia) A10572 Mestranol A10786 Rhein (Monorhein) A10209 Chrysin A10388 Fisetin (Fustel) A10573 Metformin hydrochloride A10787 Rheochrysidin (Physcione) A10214 Cidofovir (Vistide) A10389 FK-506 A10574 Methacycline HCl (Physiomycine) A10790 Rifabutin A10220 Cinchonidine A10394 Flucytosine A10575 Methazolastone A10792 Rifapentine (Priftin) A10225 Clarithromycin A10406 Formononetin (Formononetol) A10581 Methyl Hesperidin A10793 Rifaximin (Xifaxan) A10227 Clindamycin hydrochloride A10407 Tegafur A10584 Metolazone A10796 Risedronate sodium A10229 Clofibrate A10409 Fudosteine A10594 Mitotane A10814 Rutaecarpine (Rutecarpine) A10235 Cloxacillin sodium A10411 Fumalic acid (Ferulic acid) A10595 Mitoxantrone A10815 Rutin (Rutoside) A10237 Coenzyme Q10 (CoQ10) A10415 Gadodiamide (Omniscan) A10605 Morin hydrate A10820 Salicin (Salicoside, Salicine) A10239 Cortisone acetate A10418 Gastrodin (Gastrodine) A10613 Mycophenolate mofetil (CellCept) A10821 Salidroside (Rhodioloside) A10243 Crotamiton A10423 Gemcitabine HCl (Gemzar) A10614 Mycophenolic acid A10822 Salinomycin (Procoxacin) A10426 Genistin (Genistoside) A10615 Myricetin (Cannabiscetin) A10831 Sclareol

A10832 Sclareolide (Norambreinolide) A11260 MLN4924 A11664 Telithromycin (Ketek) A11878 Iopromide A10837 Sesamin (Fagarol) A11265 Odanacatib (MK-0822) A11669 L-Thyroxine A11894 Nadifloxacin A10840 Shikimic acid (Shikimate) A11283 P005672 HCl A11670 Noradrenaline bitartrate monohydrate A11904 Paroxetine HCl A10842 Silibinin (Silybin) A11284 Cefozopran A11671 Inulin A11910 Pyridoxine HCl A10844 Silymarin (Silybin B) A11294 Anguizole A11672 ATP (Adenosine-Triphosphate) A11911 Pidotimod A10846 Sinomenine (Cucoline) A11297 Adoprazine (SLV313) A11674 Epalrestat A11936 ML 7 hydrochloride A10854 Sodium orthovanadate A11298 Adarotene (ST1926) A11675 Risedronic acid (Actonel) A11946 OC 000459 A10857 Sophocarpine A11299 Avibactam A11676 Alibendol A11958 Moxalactam Sodium A10861 Spectinomycin HCl A11300 ASC-J9 A11677 Genipin A11959 GW2580 A10864 Staurosporine A11301 Avosentan (SPP301) A11678 Miglitol (Glyset) A11963 Y320 A10866 STF-62247 A11302 Armodafinil A11679 NAD+ A11973 Necrostatin-1 A10867 Stigmasterol (Stigmasterin) A11312 Azaphen (Pipofezine) A11680 Pioglitazone (Actos) A11974 GW 4869 A10868 Streptozotocin (Zanosar) A11319 BMS-509744 A11681 Strontium ranelate (Protelos) A11989 Apocynin (Acetovanillone) A10888 Tangeretin (Tangeritin) A11323 Bardoxolone methyl (RTA 402) A11683 Cyclocytidine A11991 Schisandrin B A10889 Tanshinone I A11324 Bardoxolone (CDDO) A11684 Etidronate (Didronel) A12000 Guanosine A10890 Tanshinone IIA (Tanshinone B) A11330 Besifloxacin HCl A11685 Pamidronic acid A12026 Carnosic Acid A10892 Taurine A11342 Calcipotriol monohydrate A11687 Prednisolone acetate (Omnipred) A12159 Ezatiostat A10894 Tazarotene A11346 Calcipotriol A11688 Fluocinonide(Vanos) A12161 Catharanthine sulfate A10910 Tenoxicam A11359 CB 300919 A11689 Fenoprofen calcium A12163 Fenretinide A10912 Terbinafine hydrochloride (Lamisil) A11362 Calcitetrol A11691 Mometasone furoate A12258 HPGDS inhibitor 1 A10913 Plerixafor 8HCl (DB06809) A11364 Caspofungin Acetate A11698 Aspartame A12323 Efaproxiral A10918 Indacaterol A11367 Calcifediol A11707 Idebenone A12325 Indisulam (E7070) A10920 Tetrahydropapaverine hydrochloride A11401 PA-824 A11710 Pramiracetam A12345 Anamorelin HCl A10925 Theobromine (3,7-Dimethylxanthine) A11404 Chondroitin sulfate A11711 Carisoprodol A12346 Anamorelin A10933 Tigecycline A11406 LY2608204 A11714 Lafutidine A12347 cis-(Z)-Flupentixol dihydrochloride A10942 Tranilast (SB 252218) A11420 Fagomine A11716 Adiphenine HCl A12355 Nipradilol A10952 Troxerutin A11435 GSK-923295 A11723 Naltrexone HCl A12361 Pristinamycin A10961 Ursolic acid (Malol) A11495 MK 0893 A11725 Edaravone (MCI-186) A12364 Nalbuphine Hydrochloride A10964 Vanillylacetone A11497 MK-2894 A11726 Heparin sodium A12365 CHIR-090 A10986 VX-809 A11499 MLN4924 (HCL Salt) A11735 Geniposide A12369 Stiripentol A10993 Xanthone (Genicide) A11542 Rilpivirine (R 278474, TMC 278) A11737 Buflomedil HCl A12370 ANX-510 A11003 Yohimbine hydrochloride (Antagonil) A11561 Salmefamol A11741 Moxonidine HCl A12380 Quarfloxin (CX-3543) A11015 A11585 TMC353121 A11744 Mecarbinate A12389 Benperidol A11069 Fosaprepitant dimeglumine A11591 Tedizolid (TR-701) A11751 Probucol β-Sitosterol A12400 MifaMurtide A11070 AG-L-59687 A11593 Tonabersat (SB-220453) A11756 MK-0517 (Fosaprepitant) A12406 Apaziquone A11093 Nitisinone A11613 Zanamivir A11757 GSK126 A12407 TMPA A11094 Bexarotene (LGD1069) A11614 Zaurategrast (CDP323) A11761 Merck SIP Agonist A12428 WF 11899A A11095 URB754 A11632 Cephalomannine A11769 Loxiglumide (CR1505) A12432 ALPHA-ERGOCRYPTINE A11096 UR-144 A11641 Pranoprofen A11774 Argatroban A12441 Halofuginone A11103 BAPTA A11645 Ganciclovir A11781 PF 670462 A12479 Siramesine Hydrochloride A11110 Folinic acid calcium salt (Leucovorin) A11648 Sulbactam A11783 GSK 1210151A (I-BET151) A12547 Lithocholic acid A11111 Rasagiline A11652 Clindamycin palmitate HCl A11787 Aminopterin A12568 Tirasemtiv A11113 Pneumocandin B0 A11653 Oseltamivir phosphate (Tamiflu) A11802 Atracurium besylate A12569 Ametantrone A11124 Peramivir A11654 Oxibendazole A11805 Amidopyrine A12579 Nalfurafine hydrochloride A11128 Laquinimod (ABR-215062) A11655 Tioconazole A11806 Azacyclonol A12581 P7C3-A20 A11136 INCB8761 (PF-4136309) A11656 Flubendazole (Flutelmium) A11808 Articaine HCl A12592 Ascomycin A11139 Retapamulin (SB-275833) A11657 Tolnaftate A11809 Altrenogest A12634 MBX-2982 A11185 Ribitol (Adonitol) A11658 Balofloxacin A11829 Butenafine HCl A12654 Ombrabulin A11201 BMS-806 (BMS 378806) A11659 Sarafloxacin hydrochloride A11831 Cabazitaxel A12658 Verteporfin A11214 Lurasidone (SM13496) A11660 Prulifloxacin (Pruvel) A11840 ENOblock (AP-III-a4) A12660 Carebastine A11216 Entecavir A11661 Rimantadine (Flumadine) A11852 Fenticonazole nitrate A12666 AZ 23 A11227 Chaetominine A11662 Isepamicin A11870 Ibandronate sodium A12668 Pemetrexed disodium A11232 Troxacitabine (SGX-145) A11663 Arbidol HCl A11874 Levosimendan A12673 Pyronaridine Tetraphosphate

A12676 Salubrinal A13007 TTNPB A13360 ML 171 A14050 WW298 A12686 Eltrombopag A13032 AT 56 A13369 5-BrdU A14051 WK23 A12687 JNJ-28312141 A13036 Siramesine A13370 BCH A14052 YH249 A12691 Palifosfamide A13046 N6022 A13404 FABP4 Inhibitor A14070 TAPI-1 A12696 Vancomycin A13073 Clemizole A13410 Imipramine Hydrochloride A14071 NVP-AAM077 Tetrasodium Hydrate A12698 Telavancin A13084 Arbidol A13411 Isotetrandrine A14072 STF 118804 A12727 AMG517 A13085 LODENOSINE A13455 GSK369796 A12747 JZL184 A13088 Trimipramine A13475 SF1670 Carbonic Anhydrase A12753 RC-3095 A13089 ent Naxagolide Hydrochloride A13516 Coluracetam A10303 Diclofenamide A12754 Tirapazamine A13091 Nimorazole A13520 Isatoribine monohydrate A11673 Tioxolone A12756 Cyclamic Acid A13096 Panipenem A13530 Flumatinib mesylate A11765 Brinzolamide A12771 Acolbifene (EM 652, SCH57068) A13097 Ioversol A13570 ML314 A12773 Bleomycin hydrochloride A13098 Tipiracil A13642 Etofenamate A12780 Freselestat A13100 Triphendiol (NV-196) A13663 Nifuratel Cholinesterase

A12781 Ibutamoren mesylate (MK-677) A13101 ME-143 A13667 Geranylgeranylacetone A10330 Donepezil hydrochloride A12784 Embramine A13106 GSK221149A (Retosiban) A13668 Levomefolate Calcium A13079 Donepezil A12793 Vofopitant (GR 205171) A13111 R1530 A13692 PTZ-343 A13584 A-3 Hydrochloride A12797 Miglustat hydrochloride A13112 GGTI-2418 A13693 Gemcitabine elaidate A12799 Prochloraz manganese A13117 NSC348884 A13708 Atovaquone Casein Kinase 2 A12801 Sapacitabine (CYC682) A13119 Balamapimod (MKI-833) A13716 AR-231453 A12802 Ibutamoren (MK-677) A13122 Amsilarotene (TAC-101) A13719 Treprostinil A10344 Ellagic acid A12803 Cardiolipin A13124 SNT-207707 A13725 10058-F4 A12806 Ravuconazole A13134 CP-640186 A13732 TGR5-Receptor-Agonist Soluble guanylyl cyclase (sGC) A12807 Ceftobiprole medocaril A13150 XEN445 A13733 NSI-189 A11549 Riociguat (BAY 63-2521) A12818 Doripenem A13157 TEMPOL A13734 ZLN005 A12402 YC-1 A12832 Vorapaxar (SCH 530348) A13167 AMG-47a A13739 SCH 54292 A12835 MK7622 A13187 RI-1 A13742 TC-DAPK6 A12838 NQDI 1 A13188 SRPIN340 A13746 FAI Reagents

A12843 Cangrelor (AR-C69931) A13195 UNC0631 A13748 GNE-7915 A11980 TPEN A12847 a-Apo-oxytetracycline A13207 Pirodavir A13756 Cambendazole A12852 D2PM hydrochloride A13215 (Glp1)-Apelin-13 A13764 ST 101(ZSET1446) Integrin Receptors A12859 GKA50 A13230 TP808 A13768 AdipoRon A12861 Mirabegron A13235 NVP-231 A13783 Tirofiban Hydrochloride Hydrate A12371 Cilengitide trifluoroacetate A12863 Lomifyllin A13242 Quinacrine 2HCl A13807 BMS303141 A12372 Cilengitide A12864 Delamanid A13243 Apramycin Sulfate A13814 Atglistatin A12787 Firategrast (SB 683699) A12873 Tafenoquine A13248 MGL-3196 A13819 TG 100801 A12876 Pyrintegrin A13251 GS-9620 A13820 TG 100572 Toll-like Receptors A12878 SNT-207858 A13261 Nolatrexed Dihydrochloride A13826 PTC-209 A12683 Toll-Like Receptor 7 Ligand II A12879 Tepoxalin A13268 Ansamitocin P-3 A13828 APY29 A12841 VTX-2337 A12887 4-Epi Minocycline A13269 Caspofungin A13830 (S)-Reticuline A12895 Thiamet G A13270 Micafungin A13831 PX 12 Beta-secretase (BACE) A12899 PluriSln 1 A13271 Fidaxomicin A13832 RPI-1 A12905 AR7 A13276 KN-93 A13835 PF-06687859 A12825 AZD3839 A12906 BAF312 A13279 Flurazepam dihydrochloride A13876 C7280948 A13249 AZD5423 A12908 Bioymifi A13281 Pyrroloquinoline quinone A13883 CGP 57380 A12909 JNJ-40411813 A13292 Arzoxifene HCl A13887 TP-434 LRRK2 A12910 Lupulone A13296 SP-420 A13983 ATB 346 A12798 GSK2578215A A12913 Cilliobrevin D A13297 Deferitrin (GT-56-252) A13990 Fosfluconazole A12919 HG-10-102-01 A12931 OAC1 A13300 Palosuran A14018 Chlorin E6 A13448 CZC-25146 A12934 P7C3 A13310 MK-3102 A14033 NHS-Biotin A13969 GNE0877 A12945 StemRegenin 1 (SR1) A13324 BAY57-1293 A14035 Biotin Hydrazide A12954 Monomethyl auristatin E A13331 laxogenin A14040 Biotin-X-NHS MELK A12990 Lobucavir A13354 Harmane A14041 BMPS

A12851 OTSSP167 alpha-Amyloid Precursor Protein Modulator------30 AS 602801 (Bentamapimod)------6 ALPHA-ERGOCRYPTINE------52 AS-252424------21 A Altrenogest------52 AS-604850------21 Altretamine------48 AS-605240------20 β-lactamase Alvimopan (ADL 8-2698)------15 AS703026------5 A 740003------43 AM 580------46 Asaraldehyde (Asaronaldehyde)------15 A12384 Clavulanic acid A 803467------39 AM251------44 ASC-J9------51 A 83-01------30 Ambrisentan (BSF 208075)------43 Ascomycin------52 A 922500------46 AMD 070------43 Asenapine maleate------41 A 967079------40 AMD 3465 Hexahydrobromide------43 Asiatic acid------6 Gluconeogenesis A-3 Hydrochloride------54 AMD3100 (Plerixafor)------43 Asiaticoside------6 A-317491 sodium salt hydrate------43 Ametantrone------52 ASP3026------26 A10419 Gatifloxacin A-419259------27 Amfebutamone (Bupropion)------42 Aspartame------52 A-443654------20 AMG 073 (Cinacalcet)------38 AST-1306------3,23 A66------21 AMG 208------25 AST-6------2,23 A-674563------20 AMG 900------9 Astragaloside A------30 Cholinesterases A-769662------40 AMG-073 HCl (Cinacalcet HCl)------38 Asunaprevir (BMS-650032)------31 A-867744------39 AMG-458------25 AT 56------53 A-966492------9 A13079 Donepezil AMG-47a------53 AT101------1 a-Apo-oxytetracycline------53 AMG517------53 AT13387------32 Abacavir------12,13 AMG-Tie2-1 ------27 AT-406------2 Abacavir sulfate------12,13 Amidopyrine------52 AT7519------8 Aldose Reductase Abarelix Acetate------46 Amiloride hydrochloride------39 AT7519 HCl------8 AB-FUBINACA------44 Amiloride hydrochloride dihydrate------39 AT7867------20 A13083 Tolrestat Abiraterone (CB-7598)------13 Aminocaproic acid (Amicar)------48 AT9283------29 Abiraterone Acetate (CB7630)------13 Aminophylline------44 AT9283 ------9 ABT------13 Aminopterin------52 Atazanavir------32 ABT-199------1 Amisulpride------42 Atazanavir sulfate (BMS-232632-05)------32 Nitric Oxide Signaling ABT-263 (Navitoclax)------1 Amlodipine------38 ATB 346------54 ABT333------18 Amlodipine besylate (Norvasc)------38 ATB-337------15 A13359 Diphenyleneiodonium chloride ABT-492------48 Ammonium Glycyrrhizinate (AMGZ)------48 Atglistatin------54 ABT-737------1 Amonafide (AS1413)------11 Atorvastatin------19 ABT-751------11 Amorolfine Hydrochloride------48 Atorvastatin calcium------19 ABT-888 (Veliparib)------9 Ampalex (CX-516)------38 Atovaquone------54 Adenylyl Cyclase AC220 (Quizartinib)------25 Amphotericin B------49 ATP (Adenosine-Triphosphate)------52 Acadesine (Aicar,NSC 105823)------40 Amprenavir------32 Atracurium besylate------52 A12917 Forskolin Acarbose------48 Amrubicin------11 Atropine ------42 Acemetacin (Emflex)------15 Amsacrine------12 Aurora A Inhibitor I------9 A13586 NKY 80 Acetaminophen------15 Amsilarotene (TAC-101)------53 AUY922 (NVP-AUY922)------32 Acetanilide------48 Amygdalin------49 AV-412------3,23 Acetylcysteine------42 AN2728 ------14 Avanafil------14 Aciclovir (Acyclovir)------5 Anacetrapib (MK-0859)------19 Avasimibe (CI-1011)------13 IDH1 Acipimox ------48 Anamorelin ------52 Avibactam------51 Acitazanolast------48 Anamorelin HCl------52 AVL-292------28 A12923 IDH-C227 Acitretin------48 Anastrozole------46 Avosentan (SPP301)------51 Acolbifene (EM 652, SCH57068)------53 Andarine (GTX-007)------45 AWD 131-138------42 Actinomycin D------12 Andrographolide------49 Axitinib------4,24 ACY-1215 (Rocilinostat)------17 Anguizole------51 AZ 23------52 LSD1 inhibitor Adapalene ------48 Aniracetam------17 AZ 3146------18 Adarotene (ST1926)------51 Ansamitocin P-3------53 AZ-20------40 A12927 LSD1-C76 Adefovir dipivoxil------12 ANX-510------52 AZ628------7 Adenine sulfate------18 AP24534 (Ponatinib)------26 AZ-960------29 Adenosine------44 AP26113------3,24 Azacitidine(Vidaza)------19 Adiphenine HCl------52 AP26113 ------26 Azacyclonol------52 Casein Kinase 1 AdipoRon ------54 Apatinib (YN968D1)------3,24 Azalomycin-B------49 ADL5859 HCl------42 Apatinib (YN968D1) ------24 Azaphen (Pipofezine)------51 A13574 LH 846 Adoprazine (SLV313)------51 Apaziquone------52 Azathioprine------49 Adrenalone HCl------41 Apicidin------17 AZD1080------36 A13949 D4476 Adriamycin------11 Apigenin------13 AZD1152-HQPA (Barasertib)------9 ADX-47273------43 Apixaban (BMS-562247-01)------17 AZD1480------29 AEE788------2,23 Apocynin (Acetovanillone)------52 AZD1981------46 Lipoxygenase Aesculin (Esculin)------48 Apoptosis Activator 2------1,30 AZD2014------22 AG 957------28 Apramycin Sulfate------53 AZD-2461------10 AG-014699 (Rucaparib)------9 Apremilast (CC 10004)------14 AZD2858------36 A13346 MK 886 AG-1024 (Tyrphostin)------24 Aprepitant (MK-0869)------49 AZD3463------26 AG-1288------28 APY29------54 AZD3514------45 AG14361 ------10 AR-231453------54 AZD3839------54 Sigma-1 receptor AG-1478 (Tyrphostin AG-1478) ------3,23 AR-42 (HDAC-42)------17 AZD4547------3,24 AG-17------3,24 AR7------53 AZD5363------20 AG-490------2,23 AR-A 014418------36 AZD5423------54 A12504 S1RA AGI-5198 (IDH-C35)------15 Arbidol------53 AZD5438------8 AGI-6780------15 Arbidol HCl------51 AZD6244 (Selumetinib) ------5 AG-L-59687------51 Arbutin (Uva, p-Arbutin)------49 AZD6482------20 Agomelatine------41 AR-C155858------37 AZD7762------7 AK-7 ------17 Arctigenin------6 AZD8055------22 AKT inhibitor VIII (AKTI-1/2)------20 Arecoline------42 AZD8330 ------5 Albendazole------4,24 Arformoterol tartrate------41 AZD8931------2,23 Alendronate sodium hydrate------12 Argatroban------52 AZD-9291------3,24 Alfacalcidol------48 Aripiprazole (Abilify)------41 Azelastine hydrochloride (Allergodil)------42 Alfuzosin HCl------41 Armodafinil------51 Azelnidipine------38 Alibendol------52 ARN-509------41 Azilsartan (TAK-536)------43 Aliskiren (CGP 60536)------45 ARQ 197------25 Azithromycin (Zithromax)------18 Aliskiren hemifumarate------45 ARRY334543------3,23 Azomycin (2-Nitroimidazole)------49 Alizarin------48 Arry-380------3,23 Aztreonam (Azactam, Cayston)------49 Allopurinol------48 Arry-520------18 Allopurinol sodium------48 ARRY-543------3,24 Almotriptan malate (Axert)------41 Artemether (SM-224)------30 Aloe-emodin------48 Artemisinin------37 Alogliptin Benzoate------33 Artesunate------49 B Aloin (Barbaloin)------48 Articaine HCl------52 Alosetron------41 Arzoxifene HCl------53

BAF312------53 BML-190------44 Candesartan cilexetil (Atacand)------45 Cilengitide trifluoroacetate------54 CZC-25146 ------54 Dorzolamide HCL------49 Bafetinib (INNO-406)------26 BML-275------40 Canertinib (CI-1033)------2,23 Cilliobrevin D------53 Dovitinib (TKI-258)------25 Baicalein------13 BML-277------8 Cangrelor (AR-C69931)------53 Cilnidipine------38 Dovitinib Dilactic acid------25 Baicalin------42 BMN673------10 Capecitabine (Xeloda)------16 Cilomilast (SB-207499)------14 Doxazosin mesylate------41 Balamapimod (MKI-833)------53 BMPS------54 Capsaicin------32 Cilostazol------14 Doxercalciferol------49 Balapiravir (R1626)------31 BMS 299897------35 Captopril------33 Ciluprevir (BILN 2061)------31 D Drospirenone------44 Balicatib------34 BMS 345541------28 Carbamazepine------16 Cimetidine------42 Drospirenone ------44 Balofloxacin------51 BMS 433796------35 Carbidopa------49 Cinchonidine------49 Droxinostat------16 D-106669------21 BAM 7------1 BMS 599626 (AC480)------3,23 Carboplatin------18 Cinobufagin------37 Duloxetine------41 D2PM hydrochloride------53 BAN ORL 24------42 BMS-265246------8 Cardiolipin------53 Ciprofibrate------45 Duloxetine HCl------41 D4476 ------55 BAPTA------51 BMS303141------54 Carebastine------52 Ciproxifan------42 Dutasteride (Avodart)------5 Dabrafenib (GSK2118436A)------7 BAPTA tetrapotassium------38 BMS-509744------51 Carisoprodol------52 Ciproxifan maleate------42 Dynasore------37 Dacarbazine------18 BAPTA/AM------38 BMS-536924------24 Carmofur------16 cis-(Z)-Flupentixol dihydrochloride------52 Dyphylline------44 Daidzein------49 Bardoxolone (CDDO)------51 BMS564929 ------45 Carnosic Acid------52 Cisplatin------18 Daidzin------49 Bardoxolone methyl (RTA 402)------51 BMS-690514------3,23 Carvedilol------41 Citalopram Hydrobromide------38 Danoprevir (RG7227)------30 Baricitinib (LY3009104)------29 BMS-690514 ------24 CASIN------43 CK-1827452 (Omecamtiv mecarbil)------38 Danusertib (PHA-739358)------9 Batimastat (BB-94)------33 BMS-707035------33 Caspofungin------53 CK-636------12 Dapagliflozin (BMS512148)------37 E BAY 1000394------8 BMS-708163------35 Caspofungin Acetate------51 Cladribine------16 Daphnetin------16 Bay 11-7821------1 BMS-740808------18 Catharanthine sulfate------52 Clafen (Cyclophosphamide)------18 Dapivirine------13 Bay 60-7550------14 BMS-754807 ------24 CAY10505------21 Clarithromycin------49 E 2012------35 Dapoxetine hydrochloride------41 BAY 61-3606------27 BMS-777607------25 CB 300919------51 Clavulanic acid ------55 E-4031 dihydrochloride------39 DAPT (GSI-IX)------35 Bay 65-1942------28 BMS-777607 ------28 CC-401------6 Clemastine fumarate------42 E-7050 (Golvatinib)------4,24,25 Daptomycin------49 Bay 65-1942 HCl------28 BMS-790052------31,31 CCG-63802------43 Clemizole------53 E7080 (Lenvatinib)------4,24 Darifenacin------42 BAY 80-6946------21 BMS-790052 2HCl------31 CCT128930------20 Clenbuterol hydrochloride------45 Ecdysone------49 Darunavir Ethanolate (Prezista)------32 BAY 87-2243------5 BMS-794833------25 CCT129202------9 Clevidipine------38 Econazole nitrate------49 Dasatinib (BMS-354825)------27 BAY57-1293------53 BMS-806 (BMS 378806)------51 CCT137690------9 Clindamycin hydrochloride------49 Edaravone (MCI-186)------52 DBeq------48 BAY-u 3405------43 BMS-833923 (XL-139)------36 CCT239065------18 Clindamycin palmitate HCl------51 Efaproxiral------52 DCC-2036 (Rebastinib)------26 Bazedoxifene acetate------44 BMS-863233 (XL-413)------8 CCT241533------9 Clinofibrate------45 EGT1442------37 D-Cycloserine------49 BCH------54 BMS-911543------29 CCT241533 ------7 Clofarabine------18 EHop-016------11 Decitabine------16 BCX 1470------33 BMS-927711------43 CD 437------46 Clofibrate------49 EHT 1864 ------43 Decitabine ------19 BCX 1470 methanesulfonate------33 BMY 7378------41 Cediranib (AZD2171)------4,24 Clomifene citrate------44 Elacridar------37 Deferasirox------28 Belinostat (PXD101)------16 Boceprevir (SCH-503034)------31 Cefaclor------49 Clomipramine hydrochloride------41 Elesclomol------32 Deferitrin (GT-56-252)------53 Benazepril hydrochloride------45 Bopindolol malonate------45 Cefdinir------49 Clonidine hydrochloride------41 Eletriptan------41 Deflazacort------49 Bendamustine HCl (SDX-105)------49 Bortezomib (Velcade)------30 Cefditoren pivoxil------5 Clopidogrel (Plavix)------43 Eletriptan hydrobromide------41 Deforolimus (Ridaforolimus)------22 Benidipine hydrochloride------38 Bosentan------43 Cefoselis sulfate------49 Cloprostenol (sodium salt)------43 Ellagic acid------54 Degarelix acetate------46 Benperidol------52 Bosutinib (SKI-606)------27 Cefozopran------51 Clotrimazole------13 Eltrombopag------53 Deguelin------20 Benserazide hydrochloride (Serazide)------42 BP897------42 Cefprozil hydrate (Cefzil)------49 Cloxacillin sodium------49 Elvitegravir (GS-9137)------33 Dehydroepiandrosterone------41 Bepotastine------42 BRAF inhibitor------7 Ceftiofur hydrochloride------49 Clozapine------42 Embramine------53 Delamanid------53 Bepotastine Besilate------42 BRD9757------17 Ceftobiprole medocaril------53 CNX-1351------22 EMD-1214063------25 Delavirdine mesylate------12 Berberine Hydrochloride------49 Brefeldin A------37 Celastrol------49 CNX-2006------3,24 Emodin------49 Delphinidin chloride------3,24 Bergenin (Cuscutin)------49 Brequinar------15 Celecoxib------15 CNX-774------28 Empagliflozin------37 Delphinidin chloride ------24 Besifloxacin HCl------51 Bretazenil------39 Celgosivir------31 Cobicistat(GS-9350)------13 Emtricitabine------12 Deltarasin-HCl------14 Beta Carotene------49 Brinzolamide------54 CEP-18770------31 Coenzyme Q10 (CoQ10)------49 Enalapril maleate------42 Desmopressin------43 Beta-Lapachone------11 Brivanib (BMS-540215)------4,24 CEP-28122------26 Colchicine------11 Enalaprilat dihydrate------45 Desonide------49 Betamethasone------49 Brivanib alaninate (BMS-582664)------4,24 CEP33779------29 Coluracetam------54 ENMD-2076------25 Detomidine hydrochloride------41 Betamethasone dipropionate------49 BRL 52537 hydrochloride------42 Cephalomannine------51 Combretastatin A4------5 ENOblock (AP-III-a4)------52 Dexamethasone------49 Betamethasone valerate ------49 BRL-15572------41 Cerpegin------46 Compound 401------23 ent Naxagolide Hydrochloride------53 Dexrazoxane Hydrochloride------49 Betaxolol------41 Bromfenac sodium------16 Cerubidine------11 Cortisone acetate------49 Entecavir------51 D-glutamine------49 Betaxolol hydrochloride------41 Bromosporine------34 Cetaben------45 Costunolide------12 Epalrestat------52 Diazepinomicin------7 Bethanechol chloride------42 Brompheniramine------42 Cetirizine Dihydrochloride------42 CP 945598 hydrochloride------44 Epirubicin------18 Diclofenac sodium------15 Betrixaban------18 Bryostatin 1------49 Cevipabulin (TTI-237)------12 CP-466722------40 Epirubicin Hydrochloride------11 Diclofenamide------54 Betulinic acid------12 BS-181 HCl------8 CFTR-Inhibitor-II------40 CP-547632------4,24 Epothilone A------12 Diclofensine------49 Bexarotene (LGD1069)------51 BSI-201 (Iniparib)------10 CGI1746------28 CP-640186 ------53 Epothilone B (EPO906)------12 Didanosine------49 BEZ235 (NVP-BEZ235) ------20 BTZ043 (BTZ038, BTZ044)------49 CGK 733------40 CP-673451------3,24 Epothilone D------12 Dienestrol------49 BGJ398 (NVP-BGJ398)------3,24 Budesonide------49 CGP 3466B maleate------15 CP-690550 (Tofacitinib citrate)------29 Eprosartan------43 Dienogest------44 B-HT 920 2HCl------42 Bufalin------37 CGP 57380------54 CP-724714------2,23 Eprosartan mesylate------43 Diethylstilbestrol------38 BI 2536------10 Buflomedil HCl------52 CGP-52411------3,24 CP-91149------46 EPZ004777------47 Dihydroartemisinin------49 BI6727 (Volasertib)------10 Bufotalin------37 CGP60474------8 CPI-203------34 EPZ005687------47 Dihydromyricetin (Ampeloptin)------49 Biapenem------49 Bumetanide------49 CGP77675------27 CPI-613------15 EPZ-5676------47 Diltiazem HCl------38 Bibf1120 (Vargatef)------4,24 Bupivacaine hydrochloride------49 CGS 21680 hydrochloride------44 Crenolanib (CP-868596)------3,24 EPZ-6438------47 Dimebon dihydrochloride------14 BIBR 1532------12 Busulfan (Myleran, Busulfex)------49 CH5132799------21 Crotamiton------49 Erastin------20 Dimesna (BNP7787)------49 BIBR 953 (Dabigatran, Pradaxa)------33 Butein------3,24 CH5424802------26 Cryptotanshinone------29 Ercalcidiol------46 Dinaciclib (SCH 727965)------8 BIBR-1048 (Dabigatran etexilate)------49 Butenafine HCl------52 Chaetocin------47 Crystal violet------49 Ergosterol------49 Dioscin (Collettiside III)------49 BIBW2992 (Afatinib)------2,23 Butylscopolamine BR ------49 Chaetominine------51 CTEP------43 Eribulin Mesylate------12 Diosgenin------49 BIBX 1382 ------3,23 BX-795------23 CHC------38 CTS-1027------33 Erlotinib Hydrochloride ------2,23 Diosmetin------49 Bicalutamide (Casodex)------45 BX-912------23 Chelerythrine Chloride------30 CUDC-101------16 Ethisterone------44 Diosmin------49 BI-D1870------23 BYL719------21 Chenodeoxycholic acid------49 CUDC-305 (DEBIO-0932 )------33 Etidronate (Didronel)------52 Diphenhydramine hcl------49 Bifemelane hydrochloride------17 CHIR-090 ------52 CUDC-907------17 Etofenamate------54 Diphenyleneiodonium chloride------55 BIIB021------32 CHIR-124------7 Curcumol------49 Etomoxir------46 Dipyridamole------38 BIIE 0246------43 CHIR-98014------36 CVT 6883------44 Etoposide (VP-16)------11 Disulfiram------30 Bilastine------42 CHIR-99021------36 CW069------12 ETP-46464------40 Divalproex sodium------49 Bilobalide------49 Chloramphenicol------13 CX-4945 (Silmitasertib)------30 Evacetrapib (LY2484595)------19 C DL-Adrenaline------41 Bimatoprost (Lumigan)------49 Chlorin E6------54 CX-5461------18 Everolimus (RAD001)------22 DL-Carnitine hydrochloride------49 BINA------43 Chlormezanone (Trancopal)------49 CX-6258------29 Evista (Raloxifene Hydrochloride)------44 C646------47 D-Mannitol------49 Bindarit ------28 Chlorogenic acid------49 CYC116------4,24 Evodiamine (Isoevodiamine)------49 C7280948------54 DMH-1------28 Biochanin A (4-Methylgenistein)------49 Chlorothiazide------49 CYC116 ------9 EX 527------17 CA-074------34 DMOG------15 Biotin Hydrazide------54 Chloroxine------4,24 Cyclamic Acid------53 Exatecan mesylate------11 Cabazitaxel------52 DMXAA (ASA404)------4 Biotin-X-NHS------54 Chlorpheniramine maleate------42 Cyclocytidine------52 Exemestane------46 Cabergoline------42 DNQX------38 Bioymifi------53 Chlorpromazine hydrochloride------19 Cycloheximide (Actidione)------18 Ezatiostat------52 Caffeic acid------49 Dobutamine hydrochloride------41 Biperiden hydrochloride------42 Chlorprothixene------49 Cyclopamine------35 Ezetimibe (Zetia) ------49 CAL-101 (GS-1101)------20 Docetaxel (Taxotere)------12 Birinapant (TL32711)------2 Chondroitin sulfate------51 Cyclophosphamide monohydrate------2 Calcifediol------51 Docosanol------49 Bisoprolol------41 CHR2797 (Tosedostat)------33 Cyclosporin A------49 Calcipotriol ------51 Dofetilide------49 Bisoprolol fumarate------41 Chrysin------49 Cyclovirobuxin D (Bebuxine)------49 Calcipotriol monohydrate------51 Domperidone------42 BIX 01294------47 Chrysophanic acid (Chrysophanol)------2,23 Cynarin ------38 Calcitetrol------51 Donepezil------54 BIX 02189 ------5 CI994 (Tacedinaline)------17 Cyproheptadine hydrochloride ------42 F Calcitriol (Rocaltrol)------49 Donepezil ------55 BIX02188------5 Ciclopirox------37 Cyproterone acetate------19 Cambendazole------54 Donepezil hydrochloride------54 BKM120 (NVP-BKM120)------21 CID 2011756------30 Cyt387------29 FABP4 Inhibitor------54 Camostat mesylate------33 Dopamine hydrochloride------42 Bleomycin hydrochloride------53 CID 755673------30 CYT997------11 Fadrozole------46 Camptothecin------11 Doramapimod (BIRB-796)------6 Bleomycin sulfate------18 Cidofovir (Vistide)------49 Cytarabine------49 Fagomine------51 Canagliflozin------37 Doripenem------53 Blonanserin------42 Cilazapril monohydrate------45 Cytisine (Baphitoxine, Sophorine)------49 FAI ------54 Candesartan (Atacand)------45 Doripenem Hydrate------49 BM-1074------1 Cilengitide------54 CZC24832------21 Fasudil HCl (HA-1077)------10

Adooq Bioscience Email: [email protected] Phone: 1-866-930-6790 Fax: 1-866-333-9607 Adooq Bioscience Email: [email protected] Phone: 1-866-930-6790 Fax: 1-866-333-9607 Alphabetical Product Index Alphabetical Product Index

Febuxostat (TEI-6720)------15 Geldanamycin------32 H 89 dihydrochloride------30 IOX 2------5 LY2603618 (IC-83)------7,9 Felbamate------39 Gemcitabine elaidate------54 HA-1077 dihydrochloride------11 IPI-145------22 LY2608204------51 Fenoldopam------42 Gemcitabine HCl (Gemzar)------49 HA14-1------1 IPI-493------32 L LY2784544------29 Fenoprofen calcium------52 Gemfibrozil (Lopid)------45 Halofuginone------52 IPI-504 (Retaspimycin hydrochloride)------32 LY2811376------35 Fenretinide ------52 Genipin------52 Haloperidol (Haldol)------42 Ipratropium bromide------42 LY2835219------8 Fenticonazole nitrate------52 Geniposide------52 Harmane------53 Irbesartan (Avapro)------11 L(+)-Rhamnose Monohydrate------50 LY2886721------50 Ferrostatin-1 (ethyl ester)------20 Genistin (Genistoside)------49 HC-030031------40 Irinotecan------11 L-165,041------45 LY294002------20 Ferrostatin-1 (Fer-1)------20 Gentamycin sulfate (Gentacycol)------50 Hematoxylin (Hydroxybrazilin)------50 Irinotecan HCl Trihydrate (Campto)------11 L-741626------42 LY2940680------35 Fesoterodine fumarate (Toviaz)------42 GENZ-644282------12 Heparin sodium------52 Irsogladine------42 L-779450------7 LY310762------41 Fexofenadine HCl------42 Geranylgeranylacetone------54 Hesperadin------9 Isatoribine monohydrate------54 Lacidipine------38 LY315920 (Varespladib)------19 FG-4592------5 Gestodene------50 Hesperetin------14 Isepamicin------51 Lacosamide------39 LY317615 (Enzastaurin)------30 FH535------36 GF 109203X------30 Hesperidin------50 Isoconazole nitrate------50 Lactacystin------31 LY335979------37 Fidaxomicin------53 GGTI-2418------53 Hexestrol------44 Isoliquiritigenin------50 Lafutidine------52 LY404187------38 Finasteride------5 Gimeracil------15 HG-10-102-01------54 Isoprenaline HCl------41 Lamivudine------32 LY-411575------35 Firategrast (SB 683699)------54 Ginkgolide A------43 Hh-Ag1.5------35 Isotetrandrine------54 Lamotrigine------39 LY450108------38 Fisetin (Fustel)------49 Ginkgolide B------43 HhAntag------35 Isotretinoin------14 Lapatinib (free base)------3,24 LY500307------44 FK 3311------16 GKA50------53 HIF-C2------5 Ispinesib (SB-715992)------18 Lapatinib Ditosylate------2,23 LY573636 (Tasisulam)------1,30 FK-506------49 Glimepiride------33 HMN-214------10 Isradipine------38 Lappaconite Hydrobromide------50 FK866------2 Gliotoxin------31 Honokiol------5 ISRIB (trans-isomer)------2 LAQ824 (NVP-LAQ824)------16 Flavopiridol (Alvocidib)------8 GLPG0634 ------29 Honokiol ------20 Istradefylline (KW-6002)------44 Laquinimod (ABR-215062)------51 Flavopiridol HCl------8 Glyburide------39 Hordenine------50 ITD-1------30 Laropiprant (MK0524)------43 FLI-06------35 Glycyrrhetinic acid (Enoxolone)------49 HPGDS inhibitor 1------52 ITF2357 (Givinostat)------16 L-Ascorbyl 6-palmitate------50 M Floxuridine------18 Glycyrrhizic acid------50 HQL-79------12 Itraconazole (Sporanox)------50 laxogenin------53 Flubendazole (Flutelmium)------51 GNE0877------54 HS-173------22 IU1------48 LB42708------47 Magnolol------50 Flucytosine------49 GNE-7915------54 HSP-990------33 Ivabradine HCl (Procoralan)------41 LBH589 (Panobinostat)------16 Malotilate------50 Fludarabine (Fludara)------29 GNF 2------26 Hydralazine hydrochloride------50 Ivermectin------38 LCL-161------2 Manidipine (Manyper)------38 Fludarabine (Fludara) ------16 GNF 5837------28 Hydrochlorothiazide------50 IWP-2------36 LDE225 (NVP-LDE225)------43 Manidipine dihydrochloride------38 Fludarabine Phosphate (Fludara)------29 GNF-5------26 Hydrocortisone(Cortisol)------46 IWP-L6------36 LDE225 Diphosphate ------36 Maprotiline hydrochloride------41 Fludarabine Phosphate (Fludara) ------16 Go 6976------30 Hydroxocobalamin (Vitamin B12a)------50 IWR-1-endo------36 LDK-378------26 Maraviroc (UK-427857)------43 Flufenamic acid------40 Gossypol------50 Hydroxyflutamide------13 Ixabepilone------12 LDN193189------26 Marbofloxacin------50 Flumatinib mesylate------54 GR 103691------42 Hydroxyurea------50 LDN-212854------28 Marimastat------34 Flumazenil------42 Gramine------50 Hyodeoxycholic acid------50 LDN-57444------48 Masitinib (AB1010)------27 Flumequine------11 Granisetron Hydrochloride------41 Hypothemycin------2 Ledipasvir (GS 5885)------31 MBX-2982------52 Flunixin meglumine------15 GS-9620------53 LEE011------8 MC1568------16 Fluocinonide(Vanos)------52 GS-9973------27 Leflunomide------50 MCOPPB trihydrochloride------42 Fluorouracil (Adrucil)------33 GSK 0660------45 J Lenalidomide (CC-5013)------1 MDA 19------44 Flupirtine maleate------16 GSK 1210151A (I-BET151)------34,52 Lersivirine (UK-453061)------13 MDL 29951------40 Flurazepam dihydrochloride------53 GSK 2334470------23 I Letaxaban (TAK-442)------18 JAK Inhibitor I------29 MDM2 Inhibitor------2 Flurizan------35 GSK 269962------11 Letrozole------46 JK 184------15 ME-143------53 Fluticasone propionate------46 GSK 525762A (I-BET-762)------34 Ibandronate sodium------52 Leucovorin Calcium------50 JNJ 1661010------19 Mecarbinate------52 FM19G11------5 GSK J1------34 Ibodutant (MEN 15596)------44 Levomefolate Calcium------54 JNJ 26854165------1 Meclizine dihydrochloride------44 FMK------23 GSK1059615------20 Ibudilast (KC-404)------14 Levonorgestrel------44 JNJ-26481585------16 Medetomidine hydrochloride------41 Folinic acid calcium salt (Leucovorin)------51 GSK1070916------9 Ibuprofen (Advil)------15 Levosimendan------52 JNJ-28312141------53 Megestrol Acetate------46 Foretinib (GSK1363089, XL880)------25 GSK1120212 (JTP-74057, Trametinib)------5 Ibuprofen Lysine (NeoProfen)------15 LGK-974------36 JNJ-38877605 ------25 MEK162 (ARRY-438162) ------6 Formononetin (Formononetol)------49 GSK126------52 Ibutamoren (MK-677)------53 L-Glutamine------50 JNJ-40411813------53 Melanotan II------43 Formoterol------41 GSK1292263------44 Ibutamoren mesylate (MK-677)------53 LGX 818------7 JNJ-7706621------8 Melatonin------43 Formoterol hemifumarate------41 GSK1838705A------26 Ibutilide fumarate------39 LH 846------55 JNJ7777120------42 Meloxicam (Mobic)------50 Forskolin------55 GSK1904529A------24 IC-87114------20 Licofelone------15 JNK-IN-8------6 Memantine hydrochloride------39 Fosamprenavir------32 GSK2126458------21 Icariin------14 Lidocaine (Alphacaine)------39 JTC-801------42 Mephenytoin------14 Fosaprepitant dimeglumine------51 GSK221149A (Retosiban)------53 I-CBP112------34 Limonin------50 JTT-705 (Dalcetrapib)------19 Meprednisone (Betapar)------50 Fosbretabulin disodium (CA4P)------12 GSK256066------14 ICI 118,551 hydrochloride------41 Linagliptin (BI-1356)------33 JW 55------10 Mercaptopurine------18 Fosfluconazole------54 GSK2578215A------54 Icilin------40 Lincomycin hydrochloride (U-10149A) ------18 JWH 133------44 Merck SIP Agonist------52 Fosinopril sodium------33 GSK2606414 ------2 Icotinib------3,24 Linezolid (PNU-100766)------50 JZL184------53 Meropenem------50 Freselestat------53 GSK2636771------22 Icotinib Hydrochloride------3,24 Linifanib (ABT-869)------3,24 Mestranol------50 FTI 277------47 GSK2656157------2 ID 8------34 Liquiritigenin------44 Metformin hydrochloride------50 FTY720 (Fingolimod)------26 GSK2801------34 Idarubicin HCl------11 Lisinopril (Zestril)------33 Methacycline HCl (Physiomycine)------50 Fudosteine------49 GSK2838232A------32 Idebenone------52 Lithocholic acid------52 Methazolastone------50 Fulvestrant (Faslodex)------44 GSK343------47 IDH-C227 ------55 K Lobucavir------53 Methoctramine hydrate------42 Fumalic acid (Ferulic acid)------49 GSK369796------54 IEM 1754 Dihydrobromide------38 LODENOSINE------53 Methotrexate (Abitrexate)------15 Furosemide------42 GSK-3787------45 Ifosfamide------18 Kaempferol------4,24 Lomeguatrib------47 Methoxsalen (Oxsoralen)------13 GSK429286A------10 Iguratimod (T 614)------15 Kartogenin------34 Lomifyllin------53 Methoxyresorufin------14 GSK461364------10 IKK-16------29 kb NB 142-70------30 Lomustine (CeeNU)------29 Methscopolamine bromide------42 GSK690693------20 Iloperidone------50 KB-R7943 mesylate------37 Lonafarnib (SCH66336)------47 Methyl Hesperidin------50 GSK-923295------51 Imatinib (Gleevec)------4,24 Kenpaullone------8 Lopinavir (ABT-378)------32 Methyllycaconitine citrate------39 G Guaifenesin (Guaiphenesin)------50 Imatinib Mesylate------26 Ketanserin (Vulketan Gel)------41 Loratadine------42 Methylprednisolone------2 Guanosine------52 IMD 0354------29 Ketoconazole------13 Lorcaserin------41 Metiamide ------42 Gabapentin------42 GW 4869------52 Imidapril (Tanatril)------33 Ki 20227------28 lorcaserin hydrochloride (APD-356)------41 Metolazone------50 Gabapentin Hydrochloride------38 GW 501516------45 Imipramine Hydrochloride------54 Ki16198------43 Lornoxicam (Xefo)------15 Metoprolol tartrate------41 Gadodiamide (Omniscan)------49 GW 5074------7 Imiquimod (Aldara)------50 Ki16425------43 Loteprednol Etabonate------50 Metroprolol succinate------41 Galanthamine hydrobromide------42 GW 7647------45 Inauhzin------17 Ki8751------4,24 Lovastatin (Mevacor)------19 Metyrapone------15 Gallamine triethiodide------42 GW 9662------45 INCB 3284 dimesylate------43 Kinetin------50 Loxiglumide (CR1505)------52 Mevastatin------19 Gambogic acid------2 GW2580------52 INCB018424 (Ruxolitinib)------29 KN-62------43 LSD1-C76 ------55 MG-132------31 Ganciclovir------51 GW3965 HCl------45 INCB024360------20 KN-93------53 L-Thyroxine------52 MGCD0103 (Mocetinostat)------16 Ganirelix------46 GW4064------45 INCB28060------25 Kobe0065------6 Lu AE58054------41 MGCD-265 ------25 GANT 58------35 GW6471------45 INCB8761 (PF-4136309)------51 Kobe2602------7 Lubiprostone------50 MGL-3196------53 GANT61------35 GW679769 (Casopitant)------44 Indacaterol------51 KP372-1------20 Luliconazole------13 MI 2 ------33 Garcinol------47 GW788388------26 Indapamide (Lozol)------50 KPT185------38 Lupulone------53 Mianserin hydrochloride------41 Gastrodin (Gastrodine)------49 GW791343 HCl------38,43 Indinavir sulfate------32 KPT-330 ------38 Lurasidone (SM13496)------51 Micafungin------53 Gatifloxacin ------55 GW842166X------44 Indirubin------36 KRN 633------3,24 Luteolin------14 MifaMurtide------52 GBR-12935 dihydrochloride------42 GW843682X------10 Indisulam (E7070)------52 KU 0060648------22 LX 1606------15 Mifepristone (Mifeprex)------44 GDC-0032------22 GW9508------44 Indocyanine green------50 KU-0063794------22 LX 1606 Hippurate------14 Miglitol (Glyset)------52 GDC-0068------20 GYKI-52466 dihydrochloride------38 Indole-3-carbinol------50 KU-55933------40 LX-4211------37 Miglustat hydrochloride------53 GDC-0349------22 Gynostemma Extract------50 Indomethacin (Indocid, Indocin)------15 KU-60019------40 LY 2183240------38 Milrinone (Primacor)------14 GDC-0449 (Vismodegib)------35 INH1------13 KW-2449------25 LY 255283------44 Minoxidil (U-10858)------39 GDC-0834------28 INK 128------22 KW-2478------32 LY 2874455------3,24 Mirabegron------53 GDC-0879------6 INNO-206 (Aldoxorubicin)------18 KX1-004 ------27 LY 379268------43 Mirtazapine------41 GDC-0941------20 INO-1001 ------10 KX2-391------27 LY2090314------36 Mitiglinide calcium------39 GDC-0973------6 Inulin------52 KY02111------36 LY2109761------30 Mitotane------50 GDC-0980 (RG7422) ------21 H Iopromide------52 LY2140023 (LY404039)------43 Mitoxantrone------50 GDC0994 ------6 Ioversol------53 LY2157299------30 Mitoxantrone Hydrochloride------11 Gefitinib (Iressa)------2,23 IOWH032------40 LY2228820------6

Mizolastine------42 NBI-42902------46 Ondansetron HCl (GR 38032F)------41 PF 477736------7 PPQ-102------40 Rapamycin (Sirolimus)------22 Mizoribine------18 NBQX------38 ONO 2506------19 PF 4981517------13 PQ 401------24 Rasagiline------51 MK 0893------51 N-Desmethylclozapine------41 Opicapone (BIA 9-1067)------47 PF 573228------26 PR-171 (Carfilzomib)------31 Rasagiline mesylate------17 MK 3207 hydrochloride------43 Nebivolol ------41 Optovin------40 PF 670462------52 PR-619------48 Ravuconazole------53 MK 886 ------55 Nebivolol HCl------41 Org 27569------44 PF-00562271------26 Pralatrexate------31 Razaxaban------18 MK-0517 (Fosaprepitant)------52 Necrostatin-1------1,52 Oridonin (Isodonol)------50 PF-03394197 (oclacitinib)------29 Pramipexole 2HCl monohyrate------42 RC-3095------53 MK-0679 (Verlukast)------44 Nefiracetam (Translon)------5 Orlistat------50 PF-03814735------9 Pramipexole dihydrochloride------42 Reboxetine mesylate------38 MK-0752------35 Nelarabine (Arranon)------18 Orotic acid (6-Carboxyuracil)------50 PF-04217903 ------25 Pramiracetam------52 Refametinib (RDEA-119, BAY 86-9766)------6 MK-0812------43 Neohesperidin------50 Orphenadrine citrate------42 PF-04447943------14 Pranlukast (ONO 1078)------44 Regorafenib (BAY 73-4506)------27 MK-0974 (Telcagepant)------43 Neohesperidin dihydrochalcone ------50 Oseltamivir phosphate (Tamiflu)------51 PF-04449913------36 Pranoprofen------51 Repaglinide------39 MK-1439------13 Neostigmine bromide (Prostigmin)------42 OSI-027------22 PF-04554878------26 Prasugrel (Effient)------38 Reparixin------43 MK-1775------7 Nepafenac------50 OSI-420 ------2,23 PF-04691502------20 Pravadoline (WIN 48098)------15 RepSox (SJN 2511)------30 MK-2048------33 Nepicastat (free base) (SYN-117)------14 OSI-906------24 PF-04880594------7 Pravastatin sodium------19 Resibufogenin------37 MK-2206 dihydrochloride------20 Nepicastat hydrochloride------15 OSI-930------27 PF-04929113 (SNX-5422)------32 Praziquantel (Biltricide)------50 Resminostat ------17 MK-2461------3,24 Neratinib (HKI-272)------2,23 Ostarine (MK-2866) ------45 PF-04971729------39 Prazosin HCl------41 Resveratrol------17 MK-2894------51 Nevirapine (Viramune)------12 Osthole------50 PF-04979064------22 Prednisolone acetate (Omnipred)------52 Retapamulin (SB-275833)------51 MK-3102------53 NF 279------43 OSU-03012------23 PF-06687859------54 Prednisone (Adasone)------50 Retigabine (Ezogabine)------39 MK-4305 (Suvorexant)------44 NHS-Biotin------54 Otamixaban (FXV 673)------33 PF-2341066 (Crizotinib)------26 Pregnenolone------44 Reversine------9 MK-4827------10 Nicorandil------39 OTSSP167 ------55 PF-2545920------14 Prilocaine------50 RGFP966------17 MK-5108 (VX-689)------9 Nifedipine------38 OTX015------34 PF299804------3,23 PRIMA-1------1 Rhein (Monorhein)------50 MK7622------53 Nifuratel------54 Ouabain------37 PF-3758309------2 Primidone (Mysoline)------42 Rheochrysidin (Physcione)------50 MK-8245------15 Nilotinib (AMN-107)------26 Oxacillin sodium monohydrate ------50 PF-3845------15 Pristinamycin------52 RI-1------53 MK-8745------9 Nilvadipine (ARC029)------38 Oxaliplatin (Eloxatin)------18 PF-5274857 ------36 Probucol------52 Ribitol (Adonitol)------51 MKT 077------33 Nimesulide------15 Oxibendazole------51 PF-562271------26 Procaterol HCl------41 Rifabutin------50 ML 161------44 Nimodipine------38 Oxybutynin------42 PFI-1------34 Prochloraz manganese------53 Rifampin------44 ML 171------54 Nimorazole------53 Oxymatrine (Matrine N-oxide)------50 PH-797804------6 Proparacaine HCl------39 Rifapentine (Priftin)------50 ML 7 hydrochloride------52 Nipradilol------52 Oxymetazoline hydrochloride------41 PHA 408------29 Prostaglandin E1 (PGE1)------43 Rifaximin (Xifaxan)------50 ML-3043------6 Nitisinone------51 Oxytetracycline (Terramycin)------50 PHA-665752------25 PRT062607 HCL------27 Rilmenidine------41 ML314------54 NKY 80------55 Ozagrel hydrochloride------43 PHA-680632------9 Prucalopride------41 Rilpivirine (R 278474, TMC 278)------51 MLN 0905------10 NMDA------39 Ozagrel(OKY-046)------43 PHA-767491------8 Prulifloxacin (Pruvel)------51 Riluzole (Rilutek)------39 MLN2238------30 NMS-873------48 Ozarelix------43 PHA-793887------8 PRX-08066------41 Rimantadine (Flumadine)------51 MLN2480 (BIIB-024)------7 Nobiletin (Hexamethoxyflavone)------50 PHA-848125 (Milciclib)------8 PS 48------23 Rimonabant (SR141716)------44 MLN4924------51 Nocodazole------12 PHCCC------43 PSC-833------37 Riociguat (BAY 63-2521)------54 MLN4924 (HCL Salt)------51 Nolatrexed Dihydrochloride------53 Phenacetin------15 PSI------31 Risedronate sodium------50 MLN8054------9 Noradrenaline bitartrate monohydrate------52 P Phenazepam------42 PSI-6130------31 Risedronic acid (Actonel)------52 MLN8237 (Alisertib)------9 Norfloxacin (Norxacin)------50 Phenformin hydrochloride------40 PSI-6206------31 Risperidone (Risperdal)------41 MLN9708------31 NPI-2358 (Plinabulin)------5 P 22077------31 Phenoxybenzamine hydrochloride------41 PSI-7977------31 RITA (NSC 652287)------1 MLR 1023------27 NPS-2143 (SB-262470)------38 P005091------48 Phenprocoumon------50 PTC124 (Ataluren)------50 Ritonavir------32 Moclobemide------17 NQDI 1------53 P005672 HCl ------51 Phentolamine mesilate------41 PTC124 (Ataluren) ------39 Rivaroxaban (Xarelto)------18 Moexipril hydrochloride------45 NS 309------39 P276-00------8 Phenylbutazone------15 PTC-209------54 Rivaroxaban Diol------18 Mogroside II A2------46 NS-398------15 P505-15------27 Phenylephrine hydrochloride------41 PTZ-343------54 Rivastigmine tartrate------42 Mometasone furoate------52 NSC 131463 (DAMPA)------15 P7C3 ------53 Phenytoin (Lepitoin)------39 PU 02------41 RKI-1447------11 Monastrol------18 NSC 23766------11 P7C3-A20------52 Phenytoin sodium (Dilantin)------39 Puerarin (Kakonein)------41 Ro 61-8048------15 Monomethyl auristatin E------53 NSC 319726------1 PA-824------51 Phloretin (Dihydronaringenin)------50 PU-H71------32 Ro 90-7501------14 Morin hydrate------50 NSC 405020------34 PAC-1------1,30 Phlorizin (Phloridzin)------50 Purmorphamine------36 RO3280------10 Mosapride citrate------41 NSC-207895 (XI-006)------2,18 Paclitaxel (Taxol)------12 PHT-427------20 Purvalanol B------8 RO4927350------5 Motesanib (AMG706)------4,24 NSC348884------53 Paeonol (Peonol)------50 PI-103------23 PX 12------54 RO4929097------35 Motesanib Diphosphate (AMG-706)------4,24 NSI-189------54 Palifosfamide------53 Piceatannol ------27 PX-866------21 RO4987655------6 Moxalactam Sodium------52 NU 6102------8 Paliperidone------41 Picropodophyllin------24 PYR-41------48 RO5126766------6 Moxifloxacin HCl------11 NU 9056------47 Palmatine chloride------50 Pidotimod------52 Pyridoxine HCl------52 Rocuronium bromide------42 Moxonidine------33 NU7026------23 Palomid 529 (P529)------20 Pifithrin-alpha------1 Pyrintegrin------53 Rofecoxib (Vioxx)------15 Moxonidine HCl------52 NU-7441 (KU-57788)------21,23 Palosuran------53 Pifithrin-beta------1 Pyronaridine Tetraphosphate------52 Roflumilast------14 MP470 (MP-470)------25 Nutlin 3a------2 Palovarotene------46 Pifithrin-u------1 Pyroxamide (NSC 696085)------16 Rolipram------14 MPC-3100------32 Nutlin 3b------2 Pamidronate Disodium------50 PIK-293------20 Pyrroloquinoline quinone------53 Romidepsin (FK228 ,Depsipeptide)------17 MPEP HCl ------43 Nutlin-3------2 Pamidronic acid------52 PIK-294------20 Ropinirole------42 MPEP hydrochloride------43 NVP-231------53 Panipenem------53 PIK-75------21 Ropinirole HCl------42 MRS 2578------43 NVP-AAM077 Tetrasodium Hydrate ------54 Pantoprazole (Protonix)------37 PIK-90------21 Roscovitine (Seliciclib)------8 MS-275 (Entinostat)------16 NVP-ADW742------24 PAP-1 (5-(4-Phenoxybutoxy)psoralen)------39 PIK-93------21 Rosiglitazone (BRL-49653)------45 MS436 ------34 NVP-AEW541------24 Parathyroid Hormone 1-34, Human------43 Pimecrolimus------50 Q Rosiglitazone maleate------45 MSX-122------43 NVP-BAG956------21,23 Parecoxib------16 Pimobendan (Vetmedin)------14 Rostafuroxin (PST-2238)------37 Mubritinib (TAK 165)------2,23 NVP-BEP800------32 Paroxetine HCl------52 Pinaverium Bromide------38 QNZ------1,29 Rosuvastatin------45 Mycophenolate mofetil (CellCept)------50 NVP-BGT226------21 Parthenolide ((-)-Parthenolide)------50 Pindolol------41 QS 11------43 Rosuvastatin calcium (Crestor)------45 Mycophenolic acid------50 NVP-BHG712------6 Pazopanib Hydrochloride (GW786034)------4,24 Pioglitazone (Actos)------52 Quarfloxin (CX-3543)------52 Rotigotine------42 Myricetin (Cannabiscetin)------50 NVP-BSK805------29 Pazopanib(GW-786034)------27 Piperine (1-Piperoylpiperidine)------50 Quercetin (Sophoretin)------21 Rotigotine hydrochloride------42 Myricitrin (Myricitrine)------50 NVP-BVU972------25 PCI-24781------16 Pirarubicin------11 Quercetin dihydrate (Sophoretin)------21 Rotundine------42 NXY-059 (Cerovive)------50 PCI-32765------27 pirinixic acid (WY 14643)------45 Quetiapine fumarate------50 Roxatidine acetate hydrochloride------42 PCI-32765 ------28 Pirodavir------53 Quinacrine 2HCl------53 RPI-1------54 PCI-34051------17 Piroxicam (Feldene)------15 Quinapril hydrochloride------45 RS-127445------41 N PD 0332991 HCl------8 Pitavastatin calcium (Livalo)------19 QX 314 chloride------39 RU 24969 hemisuccinate------41 O PD 123319 ditrifluoroacetate------45 Pizotifen malate------50 Ruboxistaurin (LY333531)------30 PD 169316------6 PJ 34 hydrochloride------10 Rupatadine------42 N6022 ------53 PD0325901------5 PKC 412------3,24 Rupatadine Fumarate------42 NAD 299 hydrochloride (Robalzotan)------41 OAC1------53 PD153035 (HCl salt)------2,23 PKI-402------21 Rutaecarpine (Rutecarpine)------50 NAD+------52 Obatoclax mesylate (GX15-070)------1 PD173074------3,24 PKI-587------22 R Rutin (Rutoside)------50 Nadifloxacin------52 OC 000459------52 PD173955------26 Plerixafor 8HCl (DB06809)------51 Nafamostat mesylate------31 Octopamine hydrochloride------41 Pluripotin (SC-1)------2 PD184352 (CI-1040) ------5 R1530------53 Naftopidil (Flivas)------41 Octreotide------44 PluriSln 1------53 PD318088 ------5 R406------27 Naftopidil Dihydrochloride------41 Odanacatib (MK-0822)------51 PLX4032 (Vemurafenib)------6 PD98059------5 R406 (freebase)------27 Nalbuphine Hydrochloride------52 Ofloxacin (DL8280)------50 PLX-4720------6 S Pefloxacin mesylate------11 R428------28 Nalfurafine hydrochloride------52 OG-L002------34 Pneumocandin B0------51 Pelitinib (EKB-569)------2,23 R547------8 Nalmefene hydrochloride------42 Olanzapine (LY170053)------41 PNU 282987------39 Pemetrexed (Alimta)------15 R788 (Fostamatinib)------27 S/GSK1349572------33 Naltrexone HCl------52 Olaparib (AZD2281)------10 PNU-120596------42 Pemetrexed disodium------52 R935788 ------27 S1RA ------55 Nanchangmycin------50 Oleanolic Acid (Caryophyllin)------50 Podophyllotoxin------11,12 Pentagastrin------50 Racecadotril (Acetorphan)------50 S3I-201 (NSC 74859)------29 Naproxen sodium------15 Oligomycin A------37 Polydatin (Piceid)------50 Peramivir------51 Radicicol------33 Sabutoclax------1 Naratriptan------41 Olmesartan (RNH6270, CS-088)------33 Pomalidomide (CC-4047)------1 Perifosine (NSC-639966)------20 RAF265 (CHIR-265)------7 Safinamide------17 Naringenin------13 Olmesartan medoxomil------33 Posaconazole------50 Perindopril Erbumine (Aceon)------33 Raf265 derivative------7 Safinamide Mesylate (FCE28073)------17 Naringin (Naringoside)------50 Olopatadine hydrochloride------42 PP1------27 PF 3716556------37 Raltegravir (MK-0518)------33 Salbutamol sulfate (Albuterol)------41 Naringin Dihydrochalcone------50 Ombrabulin------52 PP1 Analog II, 1NM-PP1------27 PF 429242------19 Raltitrexed (Tomudex)------12 Salicin (Salicoside, Salicine)------50 Natamycin (Pimaricin)------50 Omeprazole------37 PP121------21 PF 431396 ------26 Ramelteon (TAK-375)------50 Salidroside (Rhodioloside)------50 Nateglinide (Starlix)------39 ON-01910------10 PP2------27 PF 4708671------23 Ranolazine------15 Salinomycin (Procoxacin)------50 Naxagolide------42 Ondansetron (Zofran)------39 PP242------22

Salmefamol------51 SRT3109------43 Tenoxicam------51 WZ3146------3,23 4-Epi Minocycline------53 Salmeterol------41 SRT3190------43 Tepoxalin------53 WZ4002------3,23 4-epi-Chlortetracycline Hydrochloride------34 Salubrinal------53 ST 101(ZSET1446)------54 Terazosin hydrochloride------41 U WZ8040------3,23 4-Methylumbelliferone (4-MU) ------48 SANT-1------35 Staurosporine------51 Terbinafine hydrochloride (Lamisil)------51 WZ811------43 5-Aminolevulinic acid hydrochloride------48 Sapacitabine (CYC682)------53 StemRegenin 1 (SR1)------53 Tetrahydropapaverine hydrochloride------51 5-BrdU------54 Saquinavir------32 STF 118804------54 Tetrahydrozoline Hydrochloride------41 U 95666E------42 5-hydroxymethyl tolterodine------42 SAR131675------4,24 STF-62247------51 Tetrandrine (Fanchinine)------38 U0126-EtOH------5 5-hydroxytryptophan (5-HTP)------41 Saracatinib (AZD0530)------27 Stigmasterol (Stigmasterin)------51 TG 100572------54 UCPH 101------38 7-Aminocephalosporanic acid------48 Sarafloxacin hydrochloride------51 Stiripentol------52 TG 100713------22 UK-383367------28 X Saxagliptin (BMS-477118)------33 Streptozotocin (Zanosar)------51 TG 100801------54 UNC 0638------47 SB 202190------6 Strontium ranelate (Protelos)------52 TG003------8 UNC 669------34 Xanthone (Genicide)------51 SB 203580------6 SU 5416 (Semaxinib)------4,24 TG100-115------21 UNC0321------47 XAV 939------35 SB 216763------36 SU11274------25 TG101209------29 UNC0631------53 XCT 790------44 SB 239063------6 SU14813------4,24 TG-101348------29 UNC0646------47 XEN445 ------53 SB 334867------44 SU-5402------3,24 TGR5-Receptor-Agonist------54 UNC1215------34 XL019------29 SB 415286 ------36 Sulbactam------51 TGX-221------21 UPF 1069------10 XL147------21 SB 431542------26 Sulindac (Clinoril) ------15 TH-302------13 UR-144------51 XL184 free base (Cabozantinib)------4,24,28 SB 525334------30 Sunitinib Malate------3,24 Theobromine (3,7-Dimethylxanthine)------51 Urapidil hydrochloride------41 XL-228------24 SB 743921------18 Suplatast tosilate------29 Thiamet G------53 URB597------19 XL388------23 SB1317 (TG-02) ------8,25,29 SVT-40776 (Tarafenacin)------42 Thiazovivin------10 URB754------51 XL647------3,23 SB269970 HCl------41 SYN-115------44 Thioridazine hydrochloride------42 Ursolic acid (Malol)------51 XL765------21 SB-277011------42 Synephrine (Oxedrine)------41 Thiostrepton------18 XL-888------32 SB-408124------43 THIQ------43 SB-505124------30 Tianeptine sodium------41 SB590885------7 Ticagrelor (AZD6140)------43 V SB-649868------44 Ticlopidine hydrochloride------43 Y SB-705498------36 Tideglusib------36 SB939------16 T Tie2 kinase inhibitor------27 Valdecoxib------16 Vancomycin------53 Y-27632 dihydrochloride------10 SC-26196------19 Tigecycline------51 Y320------52 SC-514------29 T0901317------46 Tioconazole------51 Vandetanib (ZD6474)------4,24 T-705 (Favipiravir)------12 Vanillylacetone------51 Y-33075------11 SCH 442416------44 Tioxolone------54 YC-1------54 SCH 54292------54 TAE684------25 Tipifarnib (Zarnestra)------2 Vanoxerine 2HCl (GBR-12909)------50 Tafenoquine------53 Vardenafil------14 YH249------54 SCH 900776 (MK-8776)------7 Tipiracil ------53 YIL 781------43 SCH-527123------43 TAK-285------3,23 Tirapazamine------53 Varenicline------38 TAK-438------39 Vatalanib (PTK787) 2HCl------24 YM155------1 SCH772984------6 Tirasemtiv------52 YM201636------21 SCH900776------7 TAK-441------35 Tirofiban Hydrochloride Hydrate------54 Vatalanib (PTK787) 2HCl Base ------4 TAK-632------7 VCH-916------31 YO-01027------35 Schisandrin B------52 Tivozanib (AV-951)------4,24 Yohimbine hydrochloride (Antagonil)------51 Sclareol------50 TAK-700 (Orteronel)------13 TMC353121------51 VE-821------40 Sclareolide (Norambreinolide)------51 TAK-700 (Orteronel) ------18 TMPA------52 VE-822------40 Scriptaid------17 TAK-700 (salt)------19 TMS------13 VER 155008------33 SDZ 205-557 HCl------41 TAK-715------6 Toceranib (PHA 291639, SU 11654)------3,24 VER-50589------33 SDZ 220-581------39 TAK-733------5 Tofogliflozin------37 Verteporfin------52 Z Selamectin------38 TAK-875------44 TOK-001 (Galeterone)------13 VGX-1027------29 Semagacestat (LY450139)------35 TAK-901------9 TOK-001 (Galeterone) ------18 Vicriviroc Malate------43 Sesamin (Fagarol)------51 TAK-960------10 Tolfenamic acid------15 Vilazodone------41 Zanamivir------51 Setrobuvir (ANA-598)------31 Talarozole------46 Toll-Like Receptor 7 Ligand II------54 Vildagliptin------33 Zardaverine------14 SF1126------22 Talmapimod (SCIO-469)------6 Tolnaftate------51 Vinblastine------12 Zaurategrast (CDP323)------51 SF1670------54 Talniflumate------39 Tolrestat ------55 Vincristine sulfate------12 ZCL-278------8 SGC 0946------47 TAME------12 Tolterodine tartrate (Detrol LA)------42 Vinflunine Tartrate------12 Zearalenone------44 SGC-CBP30------34 Tamoxifen Citrate------44 Tolvaptan------43 Vinorelbine (Navelbine)------6 Zibotentan (ZD4054)------43 SGI-110------19 Tamsulosin------41 Tonabersat (SB-220453)------51 Vinpocetine------39 ZLN005------54 SGI-1776 (free base)------29 Tamsulosin hydrochloride------44 Topotecan HCl (Hycamtin)------11 Vofopitant (GR 205171)------53 ZM 306416 hydrochloride------4,24 SGX-523 ------25 Tandospirone------41 Torcetrapib (CP-529414)------19 Vorapaxar (SCH 530348)------53 ZM 323881 hydrochloride------4,24 Shikimic acid (Shikimate)------51 Tandutinib (MLN518)------25 Torin 1------23 Voriconazole (Vfend)------13 ZM 336372------7 SIB 1757------43 Tangeretin (Tangeritin)------51 Torin 2------23 Vorinostat (SAHA)------17 ZM-447439------9 SIB 1893------43 Tanshinone I------51 TP-434------54 Vortioxetine hydrobromide------41 Zofenopril calcium------33 Silibinin (Silybin)------51 Tanshinone IIA (Tanshinone B)------51 TP808------53 VRT752271 ------6 Zoledronic Acid------30 Silymarin (Silybin B)------51 TAPI-1------54 TPCA-1------29 VS-5584 ------22 Zotarolimus------23 Sinomenine (Cucoline)------51 Tariquidar (XR9576)------38 TPEN ------54 VTX-2337------54 ZSTK474------21 Siramesine------53 Tasosartan------43 TPT-260 (Dihydrochloride)------4,24 VU 0357121------43 Z-VAD-FMK------1,30 Siramesine Hydrochloride------52 Taurine------51 TRAM-34------39 VU 0361737------43 Sitagliptin phosphate monohydrate ------33 Taxifolin ------4,24 Tranilast (SB 252218)------51 VU 0364439------43 Sitaxsentan sodium (TBC-11251)------43 Tazarotene------51 Tranylcypromine hydrochloride------34 VX-222------31 Skepinone-L ------6 TC-DAPK6------54 Trazodone hydrochloride------41 VX-661------40 VX-680 (MK-0457, Tozasertib)------9 Others SKF 89976A hydrochloride------42 TCN 201------39 Trelagliptin Succinate (SYR-472)------33 SKLB1002------4,24 TCS 1102------44 Treprostinil------54 VX-702------6 SKLB610------4,24 TCS 359------25 Trichostatin-A (TSA)------16 VX-745------6 ------51 SL 0101-1------23 TCS ERK 11e (VX-11e)------6 Triciribine------20 VX-765------1,30 (-)-Blebbistcitin------37 SL251188------17 TCS JNK 5a------6 Triciribine phosphate (NSC-280594)------20 VX-770 (Ivacaftor)------39 (-)-Catechinβ-Sitosterol gallate------4,24 SMER-3------48 TCS PIM-1 4a------29 Trimebutine------42 VX-809------40,51 (-)-Epigallocatechin gallate------48 SMI-4a------29 TDZD-8 ------36 Trimetrexate------15 (-)-Gallocatechin------31 SN 38------11 Tedizolid (TR-701)------51 Trimipramine------53 (-)-Huperzine A------38 SNS-032 (BMS-387032)------8 Tegafur------49 Triphendiol (NV-196)------53 (+)-Bicuculline------42 SNS-314------9 Tegaserod maleate------41 Troglitazone------45 W (+)-JQ1------34 SNT-207707------53 Teglarinad chloride------28 Tropanserin------41 (Glp1)-Apelin-13 ------53 Tegobuvir (GS-9190)------31 (R)-Bicalutamide------45 SNT-207858------53 Tropicamide------42 WAY-100635------41 Telaprevir (VX-950)------31 (S)-(+)-Flurbiprofen------15 SNX-2112------32 Tropisetron (ICS 205930)------41 WAY-362450------45 Telatinib (BAY 57-9352)------3,24 (S)-10-Hydroxycamptothecin------11 Sodium Danshensu------13 Troxacitabine (SGX-145)------51 WAY-600------22 Telavancin------53 (S)-Reticuline------54 Sodium orthovanadate------51 Troxerutin------51 WF 11899A------52 Telithromycin (Ketek)------52 10058-F4------54 Solifenacin succinate------42 TSU-68 (SU6668)------4,24 WHI-P 154------29 Telmisartan------43 1400W Dihydrochloride------12 Sophocarpine------51 TTNPB------53 WIN 55,212-2 mesylate------44 Temocapril------45 17 alpha-propionate------45 Sorafenib (Nexavar)------6 Tubacin------17 WK23------54 TEMPOL------53 17-AAG (KOS953)------32 Sotrastaurin (AEB071)------30 Tubastatin A HCl------17 Wnt-C59------36 Temsirolimus (Torisel)------22 17-DMAG HCl (Alvespimycin)------32 SP-420------53 TW-37 ------1 Wortmannin------21 Tenofovir (Viread)------12 1-NA-PP1------27 SP600125------6 TWS119------36 WP1066------29 Tenofovir (Viread) ------12 2-Hydroxysaclofen------42 Spectinomycin HCl------51 Tyrphostin AG 183------3,24 WP1130 ( Degrasyn )------26 Tenofovir Disoproxil Fumarate------10 2-Methoxyestradiol------5 SR 144528------46 Tyrphostin AG 879------2,23 WW298------54 Tenofovir Disoproxil Fumarate ------13 3-Cyano-7-ethoxycoumarin------13 SR 3677 dihydrochloride------11 WYE-125132 (WYE-132)------22 Tenovin-1------1 3-Indolebutyric acid------48 SR 48692------44 WYE-354------22 Tenovin-3------1 3-Methyladenine------21 SRPIN340------53 WYE-687------22 SRT1720------17 Tenovin-6------1 4-Demethylepipodophyllotoxin------48

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