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Orally Active Compound Library (96-Well)

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Orally Active Compound Library (96-Well) • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com Orally Active Compound Library (96-well) Product Details: Catalog Number: CS-L061 Formulation: A collection of 2244 orally active compounds supplied as pre-dissolved Solutions or Solid Container: 96- or 384-well Plate with Peelable Foil Seal; 96-well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode Storage: -80°C Shipping: Blue ice Packaging: Inert gas Plate layout: CS-L061-1 1 2 3 4 5 6 7 8 9 10 11 12 a Empty Vonoprazan Mivebresib AZD0156 BAY-876 Tomivosertib PQR620 NPS-2143 R547 PAP-1 Delpazolid Empty Varenicline b Empty Varenicline (Hydrochlorid Varenicline A-205804 CI-1044 KW-8232 GSK583 Quiflapon MRK-016 Diroximel Empty e) (Tartrate) fumarate SHP099 c Empty A 922500 SHP099 (hydrochlorid Nevanimibe Pactimibe Pactimibe GNF-6231 MLi-2 KDM5-IN-1 PACMA 31 Empty e) hydrochloride (sulfate) Rilmenidine d Empty Cadazolid Treprostinil GSK3179106 Esaxerenone (hemifumarat Rilmenidine Fisogatinib BP-1-102 Avadomide Aprepitant Empty e) (phosphate) Cl-amidine AZD5153 (6- e Empty Maropitant Abscisic acid (hydrochlorid BGG463 WNK463 Ticagrelor Axitinib Hydroxy-2- CGS 15943 Pipamperone Empty e) naphthoic Setogepram Teglarinad f Empty Y-27632 GSK2193874 Lanabecestat CXD101 Ritlecitinib YL0919 PCC0208009 (sodium salt) (chloride) Futibatinib Empty TAK-659 g Empty NCB-0846 GS-444217 (hydrochlorid Navitoclax ABX464 Zibotentan Simurosertib (R)- CEP-40783 MK-8617 Empty e) Simurosertib Choline JNJ- h Empty CCT251236 (bitartrate) Sarcosine Brensocatib AS-605240 PF-06840003 EED226 Filibuvir 39758979 Vorapaxar Empty Plate layout: CS-L061-2 1 2 3 4 5 6 7 8 9 10 11 12 S1p receptor Cyclo(his-pro) Coenzyme a Empty Asenapine Silodosin agonist 1 Vadadustat Iberdomide FK614 PF-01247324 (TFA) Q9 Ralfinamide Empty GKT136901 b Empty (±)- Zanubrutinib Emodepside Fenobam GZD856 GKT136901 (hydrochlorid MRX-2843 Linrodostat Avapritinib Empty Zanubrutinib (formic) e) Elimusertib Nilotinib c Empty GDC-0077 JNJ- Elimusertib (hydrochlorid Roblitinib Darovasertib Bosutinib Gefapixant Nilotinib (monohydroc Empty 64619178 e) hloride Tecalcet NPS-2143 ZM223 d Empty MSC2530818 Olaparib Ilaprazole (Hydrochlorid (hydrochlorid GSK2982772 TM5441 Ziritaxestat NE 52-QQ57 (hydrochlorid Empty e) e) e) Dasatinib e Empty RG7800 RG7800 MLN8054 CP671305 Dasatinib (hydrochlorid Anle138b BMS-309403 BMS-309403 ASP7663 Empty hydrochloride e) (sodium) Ruboxistaurin CB-1158 f Empty Linsitinib DS-1040 BMS-816336 Prostaglandin (hydrochlorid CPI-444 (dihydrochlori Navarixin AZD4635 Rucaparib Empty (Tosylate) E2 e) de) (Camsylate) Sorafenib SSTR5 g Empty Sorafenib SB756050 (Tosylate) RG3039 antagonist 1 OSI-930 Cediranib Apimostinel Amuvatinib SR 57227A Empty Masitinib h Empty NS13001 Pazopanib Masitinib (mesylate) BIIB021 Everolimus Rapamycin Vorinostat Ixabepilone Panobinostat Empty Plate layout: CS-L061-3 1 2 3 4 5 6 7 8 9 10 11 12 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com NVP- a Empty Belinostat Bortezomib Saracatinib Telaprevir Boceprevir Danoprevir Simeprevir ADW742 PD0325901 Sunitinib Empty Edoxaban Dabigatran b Empty Vandetanib Afatinib Afatinib BMS-536924 Edoxaban Edoxaban (tosylate Betrixaban Dabigatran etexilate Empty (dimaleate) (tosylate) monohydrate) etexilate (mesylate) MK-3207 c Empty Linagliptin Saxagliptin Narlaprevir TC-G-1008 MK-3207 Gusacitinib (Hydrochlorid LY3200882 Repotrectinib CLP290 Empty e) d Empty E7046 Fananserin SB 243213 SB-200646A ROCK-IN-2 Doramapimod Falnidamol Desidustat RSVA405 TC ASK 10 Empty Regorafenib Fasudil e Empty Toceranib ML218 Toceranib Regorafenib (monohydrate BMS-690514 L-006235 Proglumide Stiripentol (Hydrochlorid Empty (phosphate) ) (sodium) e) Raltegravir MK-2206 IPN60090 Samuraciclib f Empty Raclopride Sotrastaurin Raltegravir (potassium (dihydrochlori IPN60090 (dihydrochlori PTC-028 ROC-325 (hydrochlorid Empty salt) de) de) e) Samuraciclib g Empty (trihydrochlori Seclidemstat Ensartinib Sutezolid Linezolid Emricasan ACY-957 Losmapimod IDH-305 Cintirorgon Empty de) hydrochloride Fedratinib h Empty Vorasidenib Pamiparib QC6352 Pamapimod Talmapimod Theliatinib Pocapavir Ki20227 Fedratinib (hydrochlorid Empty e hydrate) Plate layout: CS-L061-4 1 2 3 4 5 6 7 8 9 10 11 12 Dapagliflozin Empty AZD-8055 OSI-027 HPGDS Vismodegib Balapiravir Capsaicin Capsaicin Dapagliflozin ((2S)-1,2- Canagliflozin Empty a inhibitor 1 (purity>99%) propanediol, Daclatasvir b Empty Ixazomib Ixazomib Delanzomib TAK-715 (dihydrochlori Daclatasvir LY2811376 Fasiglifam Cobicistat Lexibulin Empty citrate de) Secoisolaricir Pomaglumeta c Empty esinol d methionil (Z)-Orantinib Darapladib GSK1904529 Telatinib GSK-626616 ARRY-380 Tegobuvir Ketanserin Empty diglucoside (hydrochlorid A (analog ) Sarpogrelate Y-27632 d Empty Ketanserin (hydrochlorid SRX246 Ponesimod Nevirapine Delavirdine Efavirenz Rilpivirine Flurbiprofen (dihydrochlori Empty (tartrate) e) (mesylate) de) Valproic acid Alagebrium Rucaparib e Empty Valproic acid (sodium salt) 5-Azacytidine RO-28-1675 GSK356278 Zamicastat Liarozole chloride Dazoxiben (phosphate) Empty Niraparib f Empty Rucaparib Niraparib (hydrochlorid Niraparib T0901317 SB-705498 Arimoclomol Rentiapril Neticonazole Palosuran Empty e) (tosylate) (maleate) Palosuran Epertinib g Empty (hydrochlorid Voclosporin Furprofen SY-640 Ningetinib Ningetinib PF-03463275 Selamectin PQR530 (hydrochlorid Empty e) Tosylate e) Asimadoline h Empty Tetrahydrobio (hydrochlorid AX-024 AX-024 SC-26196 PD-166793 Abrocitinib E6130 AS1269574 SIB-1553A Empty pterin e) hydrochloride Plate layout: CS-L061-5 1 2 3 4 5 6 7 8 9 10 11 12 Ganaplacide a Empty L 152804 PAT-505 Ximelagatran Cilomilast Ritanserin Hyaluronidas GNE-6776 Mirogabalin Ferric maltol (hydrochlorid Empty e besylate e) Facinicline Almorexant CP-100356 b Empty CCT 137690 Almorexant (hydrochlorid (hydrochlorid GNE-493 Pemetrexed Pemetrexed (R)- PF-06471553 (hydrochlorid Empty e) e) (disodium) Bicalutamide e) Foliglurax c Empty GW 501516 Emedastine Talazoparib Pretomanid Delamanid Loxoribine URB-597 L-368,899 GNE-781 (monohydroc Empty tosylate hydrochloride hloride) Seltorexant d Empty Clotrimazole Istradefylline Preladenant Rosiptor Seltorexant (hydrochlorid Tucidinostat Vorolanib Balovaptan Baloxavir Empty e) marboxil Parsaclisib e Empty Mavacamten Praliciguat Tulrampator Atabecestat Elenbecestat Enarodustat Firibastat Fulacimstat Lazertinib (hydrochlorid Empty e) Lanraplenib Danegaptide f Empty Ralaniten Cilofexor Edicotinib Lanraplenib (succinate) Nidufexor Pemigatinib Soticlestat Hydrochloride Ziresovir Empty g Empty GW2580 Rezivertinib Tolebrutinib Camicinal S 18986 VER-82576 AZD1390 IRAK4-IN-7 RG7112 Alisertib Empty Trametinib h Empty MK-0752 Lenvatinib Lenvatinib Pomalidomid MGCD-265 Tozadenant Ibrutinib Trametinib (DMSO NDT 9513727 Empty (mesylate) e analog solvate) Plate layout: CS-L061-6 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com 1 2 3 4 5 6 7 8 9 10 11 12 Eplivanserin LM11A-31 a Empty (±)-CPSI- AS601245 A-770041 (hemifumarat (dihydrochlori Rivastigmine TC-G 1005 Risperidone PF-02413873 SNT-207707 Empty 1306 e) de) (tartrate) Alendronate b Empty SNT-207858 CVT-12012 NS11394 Fingolimod SB 239063 SD 0006 Asenapine (sodium Sitaxsentan JNJ- Empty (free base) (maleate) hydrate) (sodium) 38877618 Nintedanib c Empty AZD7325 esylate GLPG1837 PF-05180999 Finerenone E-7386 MK-8353 EBI-2511 AZD7594 BAY-677 Empty (Rac)- d Empty BAY-678 GDC-0927 INCB-057643 LSZ-102 RGX-104 RGX-104 NMDAR NAcM-OPT Tafenoquine BAY-1316957 Empty (free Acid) antagonist 1 (Succinate) 3,4'- e Empty FT113 TAS0728 Calcium Pinaverium Tyk2-IN-5 CWHM-1008 DMX-5804 Dihydroxyflav BI-749327 GSK2983559 Empty dobesilate bromide one GDC-0575 f Empty Unesbulin PF-06869206 ABBV-744 eCF506 PRN1008 GDC-0575 dihydrochlorid ARQ 531 VIT-2763 O-304 Empty e H3B-6545 g Empty ACP-105 S-23 T025 TAS6417 AZ32 Ripretinib Menaquinone H3B-6545 (hydrochlorid CF53 Empty -7 e) Retagliptin PF-06700841 h Empty H3B-5942 UCB9608 SMN-C3 CG-806 (phosphate) Retagliptin PF-06747711 (P-Tosylate) SMS2-IN-2 ACT-709478 Empty Plate layout: CS-L061-7 1 2 3 4 5 6 7 8 9 10 11 12 Almonertinib 5- a Empty PXS-4728A Almonertinib (hydrochlorid TVB-2640 TL02-59 Mito-TEMPO DT-061 (1S,2S,3R)- Methyltetrahy Anserine Empty e) DT-061 drofolic acid PLX5622 Se- b Empty Sphingomyeli trans-AUCB BI-671800 (hemifumarat VTP50469 (S)-PF- Olutasidenib Methylseleno LY3295668 Sotorasib Empty n e) 06873600 cysteine PXS-5153A c Empty (monohydroc Salcaprozate Ly93 FGFR1/DDR2 DLK-IN-1 N,N'-Diacetyl- ONO-7475 SHP394 VU6012962 GB1107 Empty hloride) (sodium) inhibitor 1 L-cystine Pyridoxal d Empty MRTX-1257 LY2940094 Rineterkib LY2452473 Benproperine Eslicarbazepi MA-0204 isonicotinoyl JNJ- G5-7 Empty (phosphate) ne hydrazone 63576253 Propiverine e Empty Glumetinib BIBB 515 (hydrochlorid URB937 BRD0705 BRD5648 Purfalcamine Dabuzalgron UTL-5g AZD7507 Empty e) S55746 f Empty Deucravacitini S55746 (hydrochlorid USP25/28 MJN110 Ibrolipim UNC569 THPP-1 ABX-1431 RG7834 Empty b e) inhibitor AZ1 DDD107498 Enclomiphen g Empty (succinate) Eprosartan Danicopan Org-12962 AS-041164 e (citrate) AZD1940 SX-682 S18-000003 Ensifentrine Empty Fingolimod Erlotinib PF-06446846 Pazopanib BMS-599626 h Empty Trofosfamide AZD9567 (hydrochlorid Afizagabar (Hydrochlorid PFE-360 (hydrochlorid (Hydrochlorid (Hydrochlorid MW-150
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