Aads. See Aminoacetonitrile Derivatives
363 Index a anaerobic NADH-fumarate reductase AADs. See aminoacetonitrile derivatives system 275 (AADs) anthelmintic discovery ABZ-nitazoxanide 266 medicinal chemistry approaches ABZ-sulfone 260, 265, 266 CODP 242–245 ABZ-sulfoxide 260, 265, 266, 272 intervet multicyclics 235, 238 Acid fast bacilli (AFB) 329, 330 VAChT inhibitors 238, 240, 241 acoziborole 129, 130 new molecules, from patent literature acute fascioliasis 294 232–235 adult flukes 295, 300 anti-bacterial approach 169, 171 adult worms 164, 166, 170–172, 175, antibacterial therapy vs. host directed 180, 190–192, 194–198, 200, 201, therapy 354 206, 207, 254, 290, 293–296, 304 antibody-based therapeutics 67–69 African animal trypanosomiasis (AAT) anticancer drugs 194 118, 119 anti-microbial properties 271 albendazole 2, 3, 9, 169, 171, 227–229, metallo-organic ruthenium 257, 272, 275, 303 complexes 271 Alpha-1-acid glycoprotein (AGP) proteasome inhibitor 271, 273 203, 212 anti-foodborne trematode drugs 304, α-difluoromethylornithine 265 311 17-α-ethynylestradiol 298 anti-fungal agent 260 Alpinia nigra 307, 311 anti-fungal compound amphotericin B Alveolar echinococcosis (AE) 253 desoxycholate (cAMB) 267 benzimidazole treatments 257, anti-infective agents 259–261 anti-echinococcal activities 267 clinical presentation 255, 257 anti-malarial drugs 268 Aminoacetonitrile derivatives (AADs) extracellular protozoan parasites 233, 234, 238 267 patents 233 intracellular protozoan parasites amino-acetonitrile linker 234 267 amino-malononitrile linker 234 anti-infective thiazolide 260 amino ozonids 267 anti-malarial compounds 267 amino-pyrazole 147, 148 anti-malarial drugs 268 amphotericin B 2, 3, 7, 140, 143, 144, antimalarials dihydroartemisinin 267 148, 260, 267, 272, 275 anti-metacestodal activity 271 Neglected Tropical Diseases: Drug Discovery and Development, First Edition.
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