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Membrane Transporter/Ion Channel Compound Library (96-well)

Product Details:

Catalog Number: CS-L011

Formulation: A collection of 849 Membrane Transporter/ related compounds supplied as pre-dissolved Solutions or Solid

Container: 96- or 384-well Plate with Peelable Foil Seal; 96-well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode

Storage: -80°C

Shipping: Blue ice

Packaging: Inert gas

Plate layout: CS-L011-1

1 2 3 4 5 6 7 8 9 10 11 12

SKF-96365 a Empty (hydrochlorid Vonoprazan BAY-876 Ko 143 JNJ- PAP-1 Varenicline (Hydrochlorid HC-067047 Empty e) 17203212 e)

SKF89976A ML133 DMCM b Empty Varenicline (hydrochlorid (hydrochlorid Naminidil MCHR1 (hydrochlorid MRK-016 Nigericin (S)- Linaprazan Empty (Tartrate) e) e) antagonist 2 e) (sodium salt) ML753286

LY2365109 D-α- c Empty (hydrochlorid ZL006 IC87201 A-804598 Hydroxyglutar BAPTA-AM Abscisic acid CaCCinh-A01 T16Ainh-A01 U93631 Empty e) ic acid

Norverapamil (-)- Pirmenol d Empty D-AP5 GSK2193874 AM-2099 (hydrochlorid (methobromid gamma-DGG (hydrochlorid Kynurenic Quinolinic D- Empty e) e) e) acid acid

Isoguvacine 7- 7- (RS)-AMPA Diphenylenei 5′- e Empty Guvacine (hydrochlorid Chlorokynure Chlorokynure (monohydrate YM-58483 odonium diphosphorib FG 7142 NPPB Empty hydrochloride e) nic acid nic acid ) chloride ose (sodium)

8-Bromo- 4- f Empty Y-26763 MK-8998 Org-26576 DHBP ZD7288 cGMP PF-01247324 ICA-069673 Acetamidobut Empty (dibromide) (sodium) anoic acid

Vanilpyruvic JNJ- Polyoxyethyle g Empty L-DABA acid 47965567 GAL-021 NS-638 CDN1163 Pico145 ne stearate TRPC6-IN-1 Empty

CP-409092 EIPA h Empty Gefapixant (hydrochlorid Ilaprazole AMG9810 EIPA (hydrochlorid ML213 Fasentin ASP7663 PSB-12062 Empty e) e)

Plate layout: CS-L011-2

1 2 3 4 5 6 7 8 9 10 11 12

Gaboxadol GYKI 53655 a Empty CM-4620 NS13001 THIP (hydrochlorid CLP290 (hydrochlorid SCH28080 ML218 Empty e) e)

Fasudil b Empty MRS1845 trans-Ned 19 Eact Talniflumate DCPIB (Hydrochlorid Ro15-4513 (S)- CGP52432 Empty hydrochloride e) SNAP5114

SSD114 Dapagliflozin c Empty (hydrochlorid TTA-Q6 ML335 NecroX-5 ML402 Capsaicinoid Dapagliflozin ((2S)-1,2- Empty e) propanediol,

ABT-418 Tariquidar d Empty Canagliflozin (hydrochlorid PF 04531083 Piromelatine Tariquidar (methanesulf Ketanserin Ketanserin Empty e) onate, (tartrate)

Eniporide Nelonemdaz e Empty BNC210 Bay K 8644 Endovion Zamicastat hydrochloride SB-705498 AMG 517 HMR 1556 Nelonemdaz (potassium) Empty

Caroverine (2S)-6- f Empty (hydrochlorid PF-03463275 Prenylnaringe Selamectin Azosemide (hydrochlorid SKA-121 LE135 Kynurenic Empty e) nin mesylate e) acid (sodium)

WAY-213613 α-Cyano-4- Desformylflus Aminooxyacet g Empty DL-TBOA (hydrochlorid AS1269574 UBP310 hydroxycinna SN 6 trabromine SIB-1553A SEN12333 ic acid Empty e) mic acid hydrochloride (hemihydrochl

Facinicline CP-100356 h Empty ABT-107 (hydrochlorid (dihydrochlori (Rac)- Pivagabine AM-0902 (hydrochlorid WS-12 Empty besylate e) de) Lanicemine e)

Plate layout: CS-L011-3

1 2 3 4 5 6 7 8 9 10 11 12

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

XE 991 a Empty ML-SA1 A-967079 Pyr3 QX-314 P-1075 dihydrochlorid Flindokalner VU591 VU591 NS5806 Empty (chloride) e hydrochloride

AZ10606120 b Empty DMP-543 BMS-191011 PD-118057 BL-1249 (dihydrochlori Broflanilide Fluxametamid LY3130481 Lavendustin NSC 15364 Empty de) e B

(R)- c Empty Dotinurad Tulrampator Licogliflozin Posenacaftor Posenacaftor CX516 LY450108 S 18986 Empty (sodium) (sodium)

NS8593 d Empty (hydrochlorid VU0463271 ZSET1446 NS19504 ML 297 CIM0216 BX430 MK6-83 Empty e)

(Rac)- e Empty NS11394 A-803467 AZD7325 GSK1702934 GLPG1837 JT010 Synta66 NMDAR Pinaverium Empty A antagonist 1

JNJ- PSEM 89S TRPM8 IK1 inhibitor f Empty Gboxin SKA-31 PTI-428 61432059 BI-749327 PF-06869206 (TFA) HC-070 antagonist 2 PA-6 Empty

L- L- L- Taurolithochol RO2959 g Empty AMG 333 ACT-709478 ONO- Palmitoylcarni Palmitoylcarni Palmitoylcarni ic acid Etiocholanolo (monohydroc Azumolene Empty 8590580 tine tine (chloride) tine (TFA) (sodium salt) ne hloride)

TRPV4 Propiverine h Empty GDC-0276 (-)-(S)-B- PF-06305591 PF-06305591 GT 949 -1 DS16570511 (hydrochlorid Metaflumizon Lotilaner Empty 973B (dihydrate) (free base) e) e

Plate layout: CS-L011-4

1 2 3 4 5 6 7 8 9 10 11 12 N-(p- Empty AUT1 VU041 amylcinnamo Tifenazoxide Cav 2.2 Bifenazate GLPG2451 Afizagabar ML67-33 GSK205 Empty a yl) Anthranilic blocker 1

GSK369796 b Empty Dihydrochlori PF-06372865 (hydrochlorid A-867744 CCMI NS 1738 PNU-120596 CGP 36742 (Rac)-MEM (hydrochlorid Empty de e) 1003 e)

VU0134992 c Empty ABT-239 ASP2905 AC1903 ICA-27243 BAY-8002 SB-366791 (hydrochlorid Aurintricarbox TRPM4-IN-1 Empty e) ylic acid

PEAQX d Empty ML418 Rostafuroxin (tetrasodium Oxatomide ISX-9 ML277 ML365 ORM-10962 KGA-2727 VU0071063 Empty hydrate)

(Rac)-ABT- Naspm e Empty 202 BI 01383298 NS-1619 GV-58 (hydrochlorid CFM-2 Pyr6 CX546 Naspm (trihydrochlori Empty (dihydrochlori e de)

Nicardipine f Empty GSK-7975A DSP-2230 PEPA (hydrochlorid GSK-5498A CFTR (sodium PNU-282987 Empty e) corrector 2 hemiheptahy

Sigma-1 D- g Empty Tubocurarine GS967 Quisqualic Nav1.1 Mirogabalin R(+)-IAA-94 VU0810464 LDN-212320 AZD3965 Empty antagonist 3 (chloride acid activator 1

5-(N,N- h Empty YHO-13177 YHO-13351 Raxatrigine Hexamethyle Optovin PF-04856264 BNC375 ORM-10103 WEHI-9625 Empty (free base) hydrochloride ne)-

Plate layout: CS-L011-5

1 2 3 4 5 6 7 8 9 10 11 12

ML204 Dibutyryl- a Empty PF 05089771 EN6 BPAM344 Clomethiazol ML204 (hydrochlorid NMDA-IN-1 cGMP Empty (tartrate) e e) (sodium)

SDZ 220-581 b Empty SDZ 220-581 (hydrochlorid BAY-1797 Isotachysterol NS 11021 DS-1971a TPC2-A1-N TPC2-A1-P AR-C155858 Empty e) 3 hemioxalate

GABAA Zatebradine c Empty Lumacaftor KN-62 Vinpocetine nAChR GFB-8438 receptor Lu AE98134 Tofogliflozin (hydrochlorid Zatebradine Empty agonist 1 agent 1 (hydrate) e)

Ethacizine (R)- (S)-Verapamil A2764 d Empty Ionomycin Indophagolin ML-SI1 (hydrochlorid TRAM-34 (hydrochlorid (hydrochlorid OR-1896 (dihydrochlori Urolithin C Empty (calcium) e) e) e) de)

BzATP AMPA e Empty Cisatracurium P2X3 H3B-120 SUVN-911 (triethylammo receptor Sepimostat MDR-652 Encequidar Encequidar Empty (besylate) antagonist 34 nium salt) modulator-2 (mesylate)

5- (S)-UFR2709 f Empty Hydroxydeca Lansoprazole (R)- SR33805 Methionine Oleandrin COR659 (hydrochlorid (E/Z)- Ebselen Empty noate Lansoprazole e) Sivopixant

Vernakalant g Empty A2793 Spinosad A 839977 Nav1.7 Ro 25-6981 PPQ-102 (Hydrochlorid (hydrochlorid Levcromakali Empty inhibitor (Maleate) e) e) m

Gallopamil GTS-21 h Empty Verapamil (hydrochlorid Levosimenda (dihydrochlori L-655708 NP118809 AF-353 (dihydrochlori Empty e) n monohydrate de) de)

Plate layout: CS-L011-6 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

1 2 3 4 5 6 7 8 9 10 11 12

L-Glutamic a Empty Rosiglitazone L- (hydrochlorid Levamlodipin Monepantel Radiprodil Ipragliflozin Remogliflozin Empty (maleate) acid (monosodium e) e besylate etabonate

Chembridge- b Empty HC-030031 5861528 CNQX DNQX NBQX Fanapanel hydrate (maleate) Empty

(-)-Dizocilpine (S)-(-)-Bay-K- (R)-(+)-Bay- Glibenclamid Lesinurad Vonoprazan c Empty (maleate) MDL 105519 8644 K-8644 e Lesinurad (sodium) (Fumarate) Vigabatrin Empagliflozin Empty

Ertugliflozin GW791343 A 438079 d Empty KB-R7943 NS309 Tezacaftor Ertugliflozin L- (dihydrochlori A 438079 (hydrochlorid SEA0400 Empty (mesylate) hydrochloride pyroglutamic de) e)

Mibefradil A-317491 LY 303511 e Empty Sotagliflozin S0859 E-4031 (dihydrochlori APD668 A-317491 (sodium salt GW9508 (hydrochlorid Empty de) hydrate) e)

SAR7334 Istaroxime Carboxyamid f Empty SAR7334 (hydrochlorid QNZ46 NS6180 (hydrochlorid CGP37157 NBI-98782 BTB06584 Tenapanor otriazole Empty e) e) (Orotate)

D-3263 g Empty Carboxyamid (hydrochlorid MDL-29951 Minodronic Transcrocetin (hydrochlorid Etifoxine Oligomycin A CFTR(inh)- Empty otriazole e) enacarbil acid ate disodium e) 172

(S)-(-)-5- Eleclazine h Empty VU 0240551 SN 2 Fluorowillardii (R)-Funapide (Trifluoroacet Verinurad (hydrochlorid Valbenazine Empty ne ate) e)

Plate layout: CS-L011-7

1 2 3 4 5 6 7 8 9 10 11 12

Bepridil a Empty ICA-121431 RPR-260243 NS1643 Mavatrep (hydrochlorid JNJ 303 Afoxolaner Dofequidar Acamprosate Empty e hydrate) (Maleate) (fumarate) (calcium)

Ranolazine b Empty (R)- Atazanavir Rosiglitazone (-)-Huperzine (dihydrochlori (dihydrochlori Empty () A (calcium) de) de) (acetate)

Mefloquine Pantoprazole Meclofenoxat c Empty (hydrochlorid Omberaceta Rosuvastatin Pantoprazole (sodium Coluracetam e Empty e) m (Calcium) (sodium) hydrate) (hydrochlorid

Radafaxine BI-9627 d Empty (hydrochlorid Bexagliflozin Tegoprazan Mizagliflozin PCI 29732 BI-9627 (hydrochlorid KCC2 blocker GlyH-101 Empty e) e) 1

Azimilide Endoxifen (Z- e Empty IOWH-032 (Dihydrochlori RQ- SYM2206 L-701324 CIQ isomer STF-31 PF-4840154 Adjudin Empty de) 00203078 hydrochloride

SSR180711 AZD9056 SCH-23390 f Empty Rimeporide WZB117 Nav1.7-IN-2 Pyr10 (hydrochlorid (hydrochlorid (hydrochlorid GSK1016790 Empty e) e) e) A

BPO-27 g Empty Branaplam NSC23925 Lemildipine Cariporide ABT-639 KS176 GSK2798745 (racemate) (dicitrate) Empty

CRAC CRAC 1- h Empty DAA-1106 XEN907 BCTC KM11060 RN-1734 RN-1747 intermediate intermediate Aminocyclobu Cycloleucine Empty 1 2 tanecarboxyli

Plate layout: CS-L011-8

1 2 3 4 5 6 7 8 9 10 11 12

Transcrocetin Elacridar a Empty Clofilium Ca2+ channel (-)-Aspartic meglumine Senicapoc A-740003 NNC 55-0396 Elacridar (hydrochlorid Cinepazide Empty tosylate agonist 1 acid salt e) (Maleate)

Dronedarone Galanthamine Gabapentin Verapamil Diphenidol b Empty (-)- (Hydrochlorid (hydrobromid Gabapentin (hydrochlorid (hydrochlorid (hydrochlorid Trimethadion (hydrochlorid Empty e) e) e) e) e) e e)

Vigabatrin c Empty Deslanoside Baclofen D- (hydrochlorid Etomidate (hydrochlorid Etiracetam Empty e) e)

Omeprazole Oxcarbazepin Vecuronium d Empty Omeprazole (sodium) e (bromide) Furosemide (sodium) Empty

L-Ascorbic e Empty L-Ascorbic acid (sodium Lidocaine (hydrochlorid Riluzole Empty acid salt) e) hydrochloride

Carbamazepi Methocarbam Oxybutynin f Empty ne Indapamide ol Oxybutynin (chloride) (chloride) Empty

Amiloride Amiloride g Empty (hydrochlorid hydrochloride Atracurium Amlodipine Amlodipine Cromolyn Empty e) dihydrate (besylate) (maleate) (besylate) (sodium)

Flunarizine Adiphenine h Empty Chlormezano A (dihydrochlori (hydrochlorid (hydrochlorid Empty ne de) (citrate) e) (fumarate) e)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Plate layout: CS-L011-9

1 2 3 4 5 6 7 8 9 10 11 12

Propafenone a Empty Pancuronium (hydrochlorid Phenytoin Mepivacaine (hydrochlorid Empty (dibromide) e) (sodium) e)

Amitriptyline Dibucaine Ropivacaine b Empty (hydrochlorid Probenecid (hydrochlorid Dibucaine (hydrochlorid Ropivacaine (hydrochlorid (hydrochlorid Ropivacaine Empty e) (Octahydrate) e hydrate) e) e e) (mesylate)

(+)- c Empty Hexamethoni Decamethoni Tetrabenazin Tetrabenazin Tetrabenazin (hydrochlorid Empty um (Bromide) um (Bromide) Pyrithione e e (Racemate) e e)

Levobupivaca Tiagabine Dihydroergoto d Empty ine Rabeprazole Lubiprostone (hydrochlorid Eslicarbazepi dihydrochlorid xine Nitenpyram Empty (hydrochlorid (sodium) e) ne acetate e (mesylate)

Lobeline e Empty Acetamiprid Bifenthrin Dinotefuran Proflavine Meticrane Benzethoniu (hydrochlorid (hydrochlorid Metergoline Empty (hemisulfate) m chloride e) e)

N- f Empty Acetylprocain L-Cycloserine Flufenamic (hydrochlorid Thonzonium Empty amide acid e) (bromide) hydrochloride

Oxybuprocain Mecamylamin g Empty e hydrochloride e Chlorpropami Minoxidil Empty hydrochloride monohydrate (hydrochlorid de sulfate

Benidipine Procyclidine 2,2,2- h Empty Esomeprazol (hydrochlorid Domiphen Clopamide (hydrochlorid (hydrochlorid Picrotoxinin Trichloroetha (hydrochlorid Empty e e) (bromide) e) e) nol e)

Plate layout: CS-L011-10

1 2 3 4 5 6 7 8 9 10 11 12

Chloroprocain Tetraethylam a Empty (Z)-Capsaicin e Ethacrynic (+)- Mivacurium Pregnenolone monium (hydrochlorid Empty (hydrochlorid acid (dichloride) monosulfate (chloride) e)

6-Methoxy-2- b Empty β-Cyfluthrin naphthoic (hydrochlorid Tannic acid Ilaprazole Cloperastine 7ACC1 DIDS (sodium Quinine Empty acid e) (sodium) fendizoate salt)

Indole-2- γ- (±)- c Empty 7ACC2 carboxylic Canagliflozin Ginsenoside Ginsenoside Ginsenoside Aminobutyric Solamargine Praeruptorin Phloretin Empty acid (hemihydrate) Rb1 Rc Rd acid A

L- d Empty Phlorizin Monensin Caffeic acid Cytisinicline Phenylalanin Bicuculline Daurisoline Bulleyaconitin Catharanthine Empty sodium salt e e A

Thiocolchicosi Dihydrocapsa N- Sinapine e Empty Imperatorin de icin Lappaconitine Gomisin J Methylcytisine 8- (thiocyanate) Empty

Reserpine 20(S)- f Empty (hydrochlorid Ophiopogonin (-)-α-Pinene Ginsenoside Ginsenoside Ginsenoside Jujuboside A alpha- Oxypeucedan Rhoifolin Empty e) D Rf Rg3 Ro Asarone in

(20S)- g Empty Protopanaxad Shikonin Bufalin Menthol (E)- Oleic acid Sodium Chrysosplene Pulegone Empty iol Cardamonin oleate tin

Halofuginone h Empty Loureirin B Halofuginone (hydrobromid Coniferyl Allocryptopine Isosinensetin Miltirone Acevaltrate Heteroclitin D (-)-Securinine Empty e) ferulate

Plate layout: CS-L011-11

1 2 3 4 5 6 7 8 9 10 11 12

3- a Empty Songorine Kavain Deoxyaconitin Podocarpic Methyllycaco Arecaidine Diphyllin Paris saponin Glaucine Empty e acid nitine citrate VII

6,2'- b Empty Trilobatin Hypophyllant Sinapine Beta- Dihydroxyflav 6- Cirsimaritin Veratridine Cyclopiazonic Empty hin Eudesmol one Methylflavone acid

4,6-O- c Empty Hydroxy-α- 1,4-Cineole Ethylidene-α- Neriifolin Tat-NR2B9c CALP3 CALP2 (TFA) Methyl Rabeprazole (+)- Empty sanshool D-glucose (TFA) syringate Sulfide

2-Aminoethyl 1,2,4- 3,4,5- TRPM8 d Empty diphenylborin Trihydroxybe (±)- Trimethoxycin GI-530159 antagonist Decanoic acid N-Methyl-DL- Empty ate nzene Naringenin namic acid WS-3

Methyl p- Dehydronitros e Empty 1-Octanol homoveratrat OR-1855 Hydroxybenz DL-Menthol Empty Empty e aldehyde onisoldipine

f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected]