<<

Panic, G. et al. PLOS Neglected Tropical Diseases 9, PRESENT REPORT e0003962 (2015). % Degeneracy Cpds shared with 1,323 set d (SRF) after 72 h Categorization Active Inactive M after 72 h current report 4.54 100

Acriflavinium Hydrochloride 3.61 100 1 1

Amodiaquine Dihydrochloride 3.15 81.82

Aprepitant 2.60 100

Atorvastatin 3.13 76.92 1 1

Benzalkonium Chloride 3.27 100 1 1

Benzyl Benzoate 3.34 83.33 1 1

Beta-naphthol 3.05 100

Bromhexine 2.58 100

Bromocriptine Mesylate 3.23 61.9

Butylated Hydroxyanisole 3.07 100

Chlormidazole 2.88 62.5 2.50 100 1 1

Clioquinol 3.38 100

Cloxyquin 2.54 100

Compactin, 3.51 100

Cyclandelate 2.47 100

Danazol 2.96 58.82

Desipramine 2.46 100

Dichlorophene, 2.66 100 1 1

Dicyclomine 3.11 100

Digoxin 2.55 100

Disulfiram 2.75 100 1 1

Docetaxel 2.76 92.31

Ebselen 2.78 100

Erythromycin Propionate 4.08 100

Exemestane 2.94 100

Fenbendazole 2.86 100

Fenofibrate 2.78 55.56

Formoterol 2.53 100 hexetidine 3.00 100 1 1

Isobutamben 4.67 100

Ivermectin 3.10 100 d M ≥ 2.47 and 2.51 72.73 % Naphthalenesulfonate 3.59 72 degeneracy >50 2.91 100

Mitotane 3.10 100

Mitoxantrone 4.67 75

Naftopidil Dihydrochloride, 7.29 70.83 nifuroxazide 2.63 100 1 1

Ouabain 3.14 71.43 2.72 100 1 1

Pitavastatin Calcium 4.97 78.26 primaquine 3.25 91.67 1 1

Proflavine Hemisulfate 2.47 100

Promazine 2.52 100 1 1

Propofol 3.08 100

Pyrvinium Pamoate 2.67 100 1 1

Rapamycin 3.64 68.18 2.64 60 1 1

Rimantadine 2.51 100

Salinomycin, Sodium 2.51 100 1 1

Sanguinarine Chloride, Sanguinarine Sulfate 3.45 100 1 1 2.77 100 1 1

Simvastatin 2.49 100 1 1 suloctidil 2.98 100 1 1

Sunitinib Malate 2.85 100 3.32 100 1 1

Thonzonium 2.90 69.57

Tilorone 2.93 100

Tioconazole 2.48 100

Triclosan 2.63 100 2.60 100 1 1

Triflupromazine Hydrochloride 2.50 100 1 1

Tromethamine 2.52 100

Todralazine Hydrochloride 2.64 66.67

Vilazodone Hydrochloride 2.71 88.89 22 sub- total

Yohimbine 3.54 61.54 17 active 5 inactive 77% agreement 2,6-di-t-butyl-4-methylphenol, Butylated 3.51 4.35 Hydroxytoluene 2-methoxyestradiol 2.83 13.33

2-thiouracil 3.33 3.7 3-methyl-1-phenyl-2-pyrazolin-5-one (mci-186), 3.16 5.56 Edaravone 2.63 17.39

Adenosine Phosphate 3.21 19.05

Adiphenine Hydrochloride 3.03 16

Alfacalcidol 2.59 1.72

Alprenolol Hydrochloride, 3.11 6.06

Altrenogest 3.43 21.05

Amantadine 2.84 15.38 1 1

Aminohydroxybutyric Acid 4.14 5.13

Aminopterin 3.26 0 1 1

Amorolfine 2.52 8.57

Amphotericin B 4.71 6.98 1 1

Aniracetam 2.54 3.57

Antazoline 3.06 22.73

Arecoline Hydrobromide 2.50 2.17 1 1

Artenimol 3.60 6.67

Ascorbic Acid 4.33 0 Atazanavir 3.22 6.25

Azaperone 3.86 0

Azlocillin 4.15 0

Balsalazide 2.56 3.85

Barnidipine 4.12 10

Beclomethasone 4.46 17.78

Benztropine 3.29 10

Benzydamine Hydrochloride 3.91 37.5

Bergapten 3.14 18.18

Betahistine 2.90 10.53

Betaine 2.86 0

Bifonazole 2.76 22.5

Biperiden 2.84 5.45

Bismuth Subsalicylate 3.68 0

Buflomedil, Hydrochloride 4.19 10

Cabergoline 5.23 15.62

Capecitabine 2.47 0

Captopril 3.02 11.11

Carbetapentane Citrate 2.47 7.41

Carmofur 3.78 45.71

Cefotaxime 4.78 8.89

Cefuroxime 3.04 0

Celecoxib 2.66 28

Chenodiol 2.48 19.23

Chloramphenicol 2.71 0 Chloramphenicol Hemisuccinate, 2.64 3.85 Chloramphenicol Sodium Succinate Acetate 2.49 5.56 1 1

Chloropyramine Hydrochloride 2.89 39.29

Chlorpyrifos 2.65 5

Chlortetracycline 2.90 10.53

Chlorzoxazone 2.52 3.7

Cilnidipine 4.50 25

Cilostazol 2.64 7.14

Cinnarazine 2.63 23.53 1 1

Cinromide 2.67 6.9

Ciprofibrate 2.66 2.38

Cisapride 2.85 10.71

Clobetasol Propionate 2.57 13.16

Clonazepam 4.74 0 1 1

Clonidine 2.79 4.55

Clopidogrel 2.61 11.9

Cloxacillin 2.54 9.09 colchicine 3.04 5.26 1 1

Colforsin 3.95 3.12

Cyclopentolate Hydrochloride 4.95 12 1 1 3.49 28.57

Cysteamine Hydrochloride 2.79 12.5

Dantrolene 2.97 2.63

Dasatinib 2.67 0

Daunorubicin 4.22 25

Decoquinate 2.54 2.38

Deflazacort 2.47 3.57

Delavirdine Mesylate 4.04 15.38

Deracoxib 2.70 2.44

Desoxycorticosterone Acetate 2.57 4.17 , Dexbrompheniramine 3.21 10.2 Maleate 3.34 0

Dextromethorphan Hydrobromide 4.71 32.43

Desvenlafaxine Succinate 2.47 2.7

Diaveridine 2.89 4.65

Diazoxide 4.47 11.76

Dibucaine 3.55 8 1 1

Diflorasone Diacetate 3.16 0 Methanesulfonate, 4.25 34.78 Dihydroergotamine Mesylate 5.69 22.22

Diltiazem Hydrochloride 4.51 8.7

Diminazene Aceturate 5.17 14.29

Diphenidol 2.53 13.64

Doxazosin 3.45 14.29

Doxepin 3.33 20.51

Doxepin Hydrochloride 3.81 20 1 1

Drofenine Hydrochloride 2.67 40.54

Efaroxan, Hydrochloride 2.76 13.95

Eprobemide 3.63 3.7

Ergonovine 3.23 26.67

Ergonovine Maleate 4.90 19.35

Ergotamine 2.49 0 1 1

Erythrosine Sodium 3.94 9.09 1 1

Estradiol Cypionate 2.61 16

Ethinylestradiol 2.79 13.51 1 1

Ethynodiol Diacetate 2.82 4.26

Etomidate 2.83 6.25

Etoricoxib 2.70 8.82

Famprofazone 2.75 32.26

Fenoldopam Mesylate 2.91 0

Finasteride 3.08 10.53

Flopropione 3.29 0 3.23 26.32 1 1

Flutamide 6.72 5.26

Fulvestrant 3.26 11.11 3.01 13.64

Granisetron 3.30 5.26

Guanfacine Hydrochloride 3.60 2.27

Halcinonide 3.13 3.33

Hydroquinidine 2.80 28.57

Hydroxyamphetamine Hydrobromide 2.99 21.05

Hydroxychloroquine Sulfate 2.52 4.26

Hydroxyzine 3.07 0

Ibandronate Sodium 2.58 0

Idoxuridine 2.49 0

Imatinib, Mesylate 3.23 43.48

Imipenem 3.18 0 iodipamide 2.63 10 1 1

Ipriflavone 6.26 11.76

Itopride, Hydrochloride 2.49 20 d M ≥ 2.47 (% degeneracy 3.04 11.11 <50)

Ketanserin Tartrate 2.57 4.17

Ketoprofen 3.81 17.24

Labetalol 2.50 13.33

Lansoprazole 2.50 0

Levobunolol 2.58 6.67

Levocarnitine 3.72 15.38

Levocetirizine Dihydrochloride 2.64 7.41 4.64 47.83 1 1

Lomustine 7.24 2.13

Lorazepam 3.51 4.44

Loxoprofen 3.12 2.7

L- 2.59 8.57

Mannitol 2.66 31.58

Melatonin 3.27 15.38

Melengestrol Acetate 3.32 31.03

Mesoridazine Besylate 2.47 2.22

Metaxalone 2.98 4

Methiothepin Mesylate, Maleate 3.09 44.83 1 1

Methyltestosterone 3.14 14.29

Methysergide Maleate 3.48 13.64

Mexeneone 2.85 16.22

Minoxidil 3.39 4.76

Mirtazapine 3.09 15.15

Moclobemide 4.74 6.67

Moexipril Hydrochloride 2.47 8.7

Morantel Citrate 2.51 0

Moroxydine Hydrochloride 4.07 3.7

Nanofin 2.51 0

Nefopam 4.07 2.38 7.76 7.69 2.63 6.9 1 1

Nicergoline 3.27 35.29

Nifedipine 2.50 4.17 1 1

Nithiamide 2.93 8.33

Nitrazepam 3.29 7.14

Nitrofurantoin 2.71 0

Norethindrone 2.47 11.43

Norethynodrel 3.51 13.04

Norgestimate 2.98 27.59

Nylidrin 2.96 9.68

Olmesartan 4.54 0

Olmesartan Medoxomil 2.53 10.71

Ondansetron 3.62 10.71

Ornidazole 3.71 3.85

Orphenadrine 2.78 15.79

Oxiconazole 2.60 18.92

Oxymetholone 2.92 6

Panthenol 2.49 12.5

Pentetrazole, 2.79 11.11

Pergolide 6.20 15 1 1

Perindopril Erbumine 3.39 10 1 1

Phenacetin 2.86 2.56

Phenylpropanolamine 3.58 0

Phthalylsulfathiazole 2.57 4.17

Pidolic Acid 2.89 2.7

Pidotimod 2.64 6.67

Piperacillin Sodium 2.54 2.63

Piperidolate Hydrochloride 3.22 2.94

Pirenperone 3.31 8.33

Pralidoxime Iodide, Pralidoxime Chloride 2.63 2.94

Pramipexole 5.40 9.52

Pizotyline Malate 2.77 12.5

Prasterone 2.85 7.69

Prednicarbate 3.68 6.06

Pregnenolone Succinate 2.72 10

Pridinol 3.29 26.09

Protirelin 2.88 14.29

Proxyphylline 2.95 10

Pyrilamine 3.70 3.7

Pyronaridine Tetraphosphate 3.13 4.88 1 1

Quinidine 2.71 18.52

Quinine Sulfate 2.69 3.85 1 1

Reboxetine Mesylate 2.84 12.5 1 1

Remacemide Hydrochloride 2.65 22.73 Rifampin 2.95 22.22

Ritonavir 2.55 26.32

Salmeterol 3.14 39.29

Saquinavir 3.61 11.11

Sarafloxacin Hydrochloride 2.92 6.52

Sibutramine 2.49 28.57

Solifenacin Succinate 3.66 8.33

Spiperone Hydrochloride, 2.57 21.62

Spironolactone 4.26 14.29

Stanozolol 2.48 22.22

Streptomycin Sulfate 2.55 6.45

Sulpiride 2.50 3.7 1 1

Taurine 3.25 5.56

Tazobactam 2.81 13.33

Telithromycin 2.48 0 tenylidone 2.61 22.22 1 1

Tepoxalin 2.58 5.88

Terconazole 2.92 7.69

Testosterone Propionate 2.49 40.62

Tetracaine 3.19 17.86

Thiamphenicol 2.52 2.7

Tolnaftate 3.01 24.14

Tolterodine 2.55 2.38

Toltrazuril 3.15 20

Topiramate 2.52 16.67

Topotecan, Topotecan Hydrochloride 2.64 5.88

Tramadol Hydrochloride 3.12 3.7 1 1

Triamcinolone Diacetate 2.57 3.45

Trihexyphenidyl 2.61 12.24

Trimetozine 2.47 2.78

Tripelennamine 2.98 14.29

Triprolidine Hydrochloride 3.39 46.15

Tropicamide 2.74 12.5

Tryptophan 2.89 16.67

Tulobuterol, Hydrochloride 2.53 7.14

Tyrothricin 2.80 0

Uk 14,304 2.79 2.33

Urea 2.66 6.67

Valganciclovir Hydrochloride 2.47 12.12

Valproic Acid Sodium, Sodium 3.29 7.69

Vardenafil Hydrochloride, Citrate 3.70 18.75

Vatalanib Dihydrochloride 5.29 21.43

Vidarabine 3.10 30

Vinblastine Sulfate 2.92 47.62 1 1

Vincristine 2.67 20.83 Vorinostat 2.90 17.14

Xylazine Hydrochloride, 3.09 15.38 1 1

Xylometazoline 4.88 23.08

Yohimbine Hydrochloride 3.17 17.24 30 sub-total

Zafirlukast 2.83 14.63 14 active 16 inactive 47% agreement

(-)-, Levomenthol 2.06 100

Acrisorcin 2.25 100

Afalanine 1.70 100

Alexidine Hydrochloride 2.11 100 1 1

Algestone Acetophenide 2.18 100

Allylisothiocyanate 2.00 100

Amitriptyline 2.38 91.3 1 1 2.05 100 1 1

Amlodipine Besylate 1.87 100 amscarine 1.66 100

Amsulosin 2.16 100 1.83 100 1 1

Astemizole 1.73 100

Benfluorex Hydrochloride 2.32 100

Benzethonium Chloride 2.09 100

Benzyl 1.91 100

Bepridil Hydrochloride 1.55 100 benzoxiquine 2.44 100 1 1

Bithionol 2.32 100 1 1

Bitoscanate 2.16 100

Bleomycin (bleomycin B2 Shown) 2.36 53.57

Bornyl Acetate 2.30 100

Bortezomib 1.73 100

Bronopol 1.99 100 1 1 broxaldine 1.75 100 1 1

Broxyquinoline 2.22 100

Butylparaben 1.73 100

Carvedilol, Phosphate 2.02 93.33 2.28 100 1 1

Cerivastatin, Cerivastatin Na 2.00 100

Chlorhexidine, Chlorhexidine Dihydrochloride 2.32 100

Chlorpromazine Hydrochloride, 2.02 100 1 1

Chlorprothixene Hydrochloride 1.91 100 1 1

Clemizole Hydrochloride 2.09 100

Clofibrate 2.39 100 clofoctol 1.82 100 1 1 clomiphene 2.17 100 1 1

Clomipramine 1.50 100 1 1

Cloperastine Hydrochloride 1.95 100 Clorgyline Hydrochloride, 1.84 100 Hydrochloride 2.25 100 1 1

Cyclobenzaprine 2.09 100 1 1 cyclosporine 1.62 100 1 1

Dactinomycin 2.06 100 1 1

Diazinon, Dimpylate 2.12 90.91

Dienestrol 1.93 100 digitoxin 2.39 100 1 1

Dihydroergotamine 2.33 100

Dioxybenzone 2.27 100

Dolasetron 2.31 100

Duloxetine Hydrochloride 2.02 94.44

Emetine, Emetine Dihydrochloride 1.84 100

Enoxolone 1.82 100 1.82 100 1 1

Exalamide 2.25 100

Ezetimibe 1.99 88.89

Fendiline Hydrochloride 2.42 100 1 1

Fenretinide 2.18 100

Floxuridine 1.92 88

Flufenamic Acid 1.90 100 % degeneracy Hydrochloride, Fluoxetine 1.95 100 1 1 >50 (d M <2.47) fluphenazine 1.86 100 1 1 fluvastatin 2.32 82.61 1 1

Gefitinib 2.38 100

Haloprogin 2.05 100

Homidium Bromide 1.96 100 1 1

Homoharringtonie 1.82 100 hycanthone 1.83 100 1 1

Idarubicin, Idarubicin Hydrochloride 1.85 100

Lapatinib Di-p Toluenesulfonate 2.18 100

Maprotiline 1.65 100 1.56 100 1 1 menadione 2.46 100 1 1

Mepiroxol 2.16 100

Mestranol 1.99 100

Metergoline 1.92 100

Methylbenzethonium Chloride 2.27 100 1 1

Methylene Blue 1.71 100 1 1

Mianserin 1.84 100 1 1

Monensin Sodium (monensin A Is Shown) 0.00 100 1 1

Miltefosine 1.94 100 1 1 2.31 100 1 1

Nelfinavir 1.97 100

Nitazoxanide 1.93 100 2.23 100 1 1 Nitroxoline 2.27 100

Miltefosine 2.44 100

Nortriptyline 2.03 100 1 1 oltipraz 2.35 100 1 1 2.18 100 1 1 oxethazaine 1.89 100 1 1

Paroxetine 2.16 100 1.53 100 1 1

Phenoxybenzamine 2.21 100

Pimethixene Maleate 2.23 100 2.25 100 1 1

Piperacetazine 1.77 100

Piroctone Olamine 2.21 100 1 1 2.27 77.78 1 1 1.89 100 1 1

Propafenone 1.93 100 Quinacrine Dihydrochloride, Quinacrine 2.36 100 1 1 Hydrochloride Raloxifene 1.71 100

Rosuvastatin, Rosuvastatin Calcium 2.18 100

Sertaconazole 1.90 85

Skf-525a Hydrochloride, Hydrochloride 1.90 85

Sodium Tetradecyl Sulfate 2.42 100

Sorafenib P-toluensulfonate 1.91 100 sulbentine 1.74 100 1 1

Sulfamerazine 1.61 100 tamoxifen 2.45 100 1 1

Tannic Acid 2.30 100 1.94 100 1 1

Thiothixene 2.43 100

Tolfenamic Acid 1.69 100

Tolonium Chloride 2.22 100 1 1 1.91 100 1 1

Tranylcypromine 1.62 100

Trimeprazine Tartrate 1.72 100

Trimipramine 2.22 100 50 sub-total

Troglitazone 1.28 100 37 active 13 in active 74% agreement (-)-, N-methyl, N-methyl (-)ephedrine 1.65 5.41 [1r,2s] 3-acetamidophenol 1.25 0

4-aminopyridine 2.15 9.68

Acarbose 0.00 33.33

Aceclidine Hydrochloride, 1.51 3.45

Aceclofenac 2.40 0

Acedapsone 1.73 7.69

Acedoben 1.74 7.69

Aceglutamide 1.86 2.86 Acesulfame Potassium 1.41 15

Acetaminosalol 1.85 8.82

Acetazolamide 1.89 0

Acetohexamide 2.14 0

Acetriazoic Acid 1.30 4.88

Acetylcysteine 1.39 0

Acetyl-l-leucine 1.35 5.13

Acexamic Acid 2.02 5.13

Acipimox 1.51 5.88

Actarit 1.60 0

Acyclovir 1.25 14.71

Adenine 1.74 2.5

Adipic Acid, Hexanedioic Acid 2.22 9.09

Adrenaline Bitartrate, Epinephrine Bitartrate 2.46 0

Adrenolone Hydrochloride 2.35 2.78

Aklomide 1.79 4

Alaproclate Hydrochloride, 1.81 4.76

Alclometazone Dipropionate 1.82 11.54

Alendronate Sodium 2.07 6.9 1 1

Aliskiren Hemifumarate 1.77 5.41

Allopurinol 2.46 0

Allylthiourea 1.50 0

Alpha-tochopherol 2.36 0

Alpha-tochopheryl Acetate 1.68 11.11

Alprazolam 1.81 10.64

Alprostadil 1.83 6.25

Alrestatin 1.84 25

Althiazide 1.53 3.23

Altretamine 2.03 2.7

Alverine Citrate 1.80 16.67

Ambroxol Hydrochloride 1.27 13.16

Amcinonide 1.49 4

Amifostine 1.51 0 1 1

Amikacin Sulfate 1.95 0

Aminohippuric Acid 2.11 0

Aminolevulinic Acid Hydrochloride 2.38 2.56

Aminopentamide Sulfate 1.48 0

Aminophylline, Theophylline 2.06 7.14

Aminopyrine 2.08 6.98

Aminosalicylic Acid 1.79 4.17

Aminothiazole 2.16 6.98

Amisulpride 1.94 3.7

Amlexanox 1.07 4.44

Amoxicillin 2.30 0

Amp 1.97 6.67 Ampicillin Sodium 1.71 8.11

Ampiroxicam 2.24 7.5

Amprolium 1.64 7.14

Amylene Hydrate 1.89 6.67

Anagrelide Hydrochloride 1.47 2.33

Ancitabine Hydrochloride 1.77 12.5

Anethole 0.99 8.89

Anisodamine Hydrobromide 2.46 0

Antipyrine 1.96 18.18

Apomorphine Hydrochloride 2.30 3.33

Apramycin Sulfate 1.91 6.9

Argatroban 1.47 5.41

Armodafinil 2.21 2.78

Artemether 1.31 7.41 1 1

Artemisinin 1.79 6.67 1 1

Artesunate 1.88 4.76

Ascorbyl Palmitate 2.14 46.67

Aspartame 1.53 8.33

Atracurium Besylate 1.75 11.11 1 1

Atropine 1.66 5

Atropine Oxide 1.70 6.82

Avobenzone 1.68 2.56

Azathioprine 1.49 8.57 1 1

Azelaic Acid 2.09 5.26 azelastine 2.42 4.76 1 1

Azilsartan Kamedoxomil 1.61 10.53

Aztreonam 1.33 2.22

Bacampicillin Hydrochloride 2.37 9.3

Bacitracin 1.46 3.85

Barbital 1.30 2.86

Beclamide 1.50 7.5

Beclomethasone Dipropionate 1.59 10

Benfotiamine 1.95 5.56

Benserazide 2.01 9.52

Benurestat 1.44 4.76

Benzocaine 1.48 9.68

Benzoclidine 1.37 3.33

Benzoic Acid 1.54 19.35

Benzoyl Peroxide 1.56 8.57

Benzoylpas 1.80 0

Benzthiazide 1.70 6.45 1 1

Benzyl 1.64 6.45

Berberine Chloride 2.36 7.69

Beta-carotene 1.66 0

Beta-escin 1.92 4.55 Beta- 1.70 11.11 1.75 19.35 1 1

Betamethasone Acetate 1.70 8

Betamethasone Sodium Phosphate 1.57 2.44

Betamipron 2.19 3.33

Betaxalol Hydrochloride 1.85 10.71

Bexarotene 1.36 4.65

Bezafibrate 1.50 6.67

Biotin 2.27 2.86

Bopindolol 2.41 4.17

Bretylium Tosylate 1.82 0

Bromfenac 2.17 6.82

Bromopride 1.48 3.12

Bucetin 1.32 7.69

Bucladesine 2.32 10.34

Budesonide 1.74 6.45

Bufexamac 1.69 10.42

Bumetanide 1.60 10

Bupivacaine Hydrochloride 1.86 15.15

Butacaine 1.65 0

Butamben 1.96 6.25

Butenafine 2.07 0

Caffeine 1.87 17.24

Calcifediol 2.39 0

Calcipotriene 2.14 16

Calcitriol 2.43 10

Camylofine Dihydrochloride 2.18 9.76

Candesartan 1.94 0

Canrenoic Acid, Potassium Salt 1.50 8.7

Capobenic Acid 1.99 14.29

Capreomycin Sulfate 1.33 2.94

Capsaicin 1.68 6.52

Carbachol 1.70 0

Carbamazepine 1.89 0

Carbenicillin Disodium 1.55 8.89

Carbimazole 1.81 8.57

Carbinoxamine 1.38 9.09

Carboplatin 1.90 12.2

Carisoprodol 1.47 7.14 Carnitine Hydrochloride, Carnitine (dl) 1.44 2.94 Hydrochloride Carsalam 1.97 0

Carteolol Hydrochloride 1.95 3.12

Carzenide 1.78 9.52

Casanthranol [cascaroside A Shown] 2.15 7.5

Cefadroxil 1.51 11.36 Cefalonium 1.86 0

Cefamandole Nafate 2.16 22.73 cefdinir 2.05 3.23 1 1

Cefepime 1.41 9.09

Cefixime 2.40 0

Cefmenoxime Hydrochloride 1.47 18.18

Cefonicid Sodium 1.50 0

Cefotaxime Sodium 1.74 3.45

Cefpodoxime Proxetil 1.35 5.13

Cefsulodin Sodium 1.90 0

Ceftazidime 1.34 2.94

Ceftibuten 1.57 9.09

Ceftriaxone Sodium Trihydrate 2.34 0

Cephalexin 2.03 0

Cephalothin Sodium 1.73 11.11

Cephradine 1.21 12.82

Chiniofon 1.26 2.27

Chloralose 1.51 3.12

Chlorambucil 1.81 8.57

Chloramine-t 1.54 1.89

Chloramphenicol Palmitate 2.01 12.9

Chlorazanil Hydrochloride 1.86 13.89

Chlorcyclizine Hydrochloride 1.79 10.53

Chlorpheniramine 2.41 3.57

Chlorpropamide 1.66 5.13 chlorproxithene 2.02 0

Chlorquinaldol 1.57 0 Chlortetracycline, Chlortetracycline 1.37 0 Hydrochloride Chlorthalidone 2.10 4

Cholecalciferol 1.66 13.33

Cholesterol 1.92 7.69

Cholic Acid 1.56 12.77

Choline Chloride 2.02 13.16

Chromocarb 1.61 8.57

Cianidanol 1.56 7.14

Cilastatin 1.16 2.94

Cinalukast 1.56 6.12

Cinoctramide 2.04 3.45

Cinoxacin 1.54 2.63

Ciprofloxacin 1.57 3.12

Citicoline 1.71 2.86

Citiolone 1.42 13.33

Citric Acid 2.20 5.66

Cladribine 2.08 0

Clarithromycin 2.15 18.75 , Clemastine Fumarate 1.97 20

Clenbuterol 2.09 7.14

Clidinium Bromide 2.08 0

Clindamycin Hydrochloride 1.52 3.57

Clindamycin Palmitate Hydrochloride 2.13 0

Clodronic Acid 1.57 14.29

Clofarabine 1.23 6.25

Clofibric Acid 1.43 0

Colistimethate Sodium 1.31 12.9

Cortisone 2.14 5.26

Cotinine 2.05 15.79

Coumarin 1.97 5.41

Coumophos 1.96 25

Creatinine 2.02 15.79

Crotamiton 1.42 3.03

Cyanocobalamin 2.13 9.68

Cyclamic Acid 1.28 6.67

Cyclizine 1.71 0

Cyromazine 1.94 5.56

Cytarabine 2.06 14.29

Dabigatran Etexilate Mesylate 1.76 2.86

Dapsone 2.25 33.33

D- 1.79 17.86

D-, Cycloserine (d) 1.81 6.25 1 1

Deet, Diethyltoluamide 1.98 2.7

Deferiprone 1.41 0

Deferoxamine 1.86 4.08

Dehydroacetic Acid 1.21 2.78

Dehydrocholic Acid 1.78 7.89

Demeclocycline Hydrochloride 1.63 0

Denatonium Benzoate 1.26 12.5

Dequalinium Chloride 2.39 14.71

Deslanoside 1.76 0

Desoximetasone 1.83 3.03

Dexamethasone 2.41 8

Dexamethasone Acetate 1.90 8.11

Dexamethasone Phosphate 1.62 5.88

Dexamethasone Sodium Phosphate 1.82 3.33

Dexchlorpheniramine 1.51 17.39

Dexketoprofen 1.38 2.63

Dexlansoprazole 1.94 5

Dexpanthenol 2.44 2.13

Dexpropranolol Hydrochloride 1.95 17.07

Diacerin 1.44 2.27

Diacetamate 1.77 6.06 Diatrizoic Acid 1.31 5.26

Diazepam 0.00 0

Dibekacin 1.77 17.14 1 1

Dibenzothiophene 1.42 5.56

Dibutyl Phthalate 1.89 6.06

Dichlorisone Acetate 1.54 3.57

Diclofenac 1.89 5.56

Dicloxacillin Sodium 1.77 13.04

Dicumarol 1.88 10

Didanosine 1.72 5.88

Diethylcarbamazine 1.26 10.26 1 1

Diethylstilbestrol 1.89 8

Difloxacin Hydrochloride 1.61 2.78

Diflunisal 1.88 11.54

Dihydrostreptomycin Sulfate 2.18 29.17

Diloxanide Furoate 1.76 5.41

Dimenhydrinate 2.37 11.11

Dimesna 2.15 9.68

Dimethadione 1.82 5.88

Dinitolmide 1.85 4.76

Dinoprostone 2.27 6.25

Diphenylpyraline Hydrochloride 2.27 7.69

Dipyridamole 2.47 29.17

Dipyrocetyl 2.28 3.23

Disopyramide 1.22 0

Dixanthogen 1.14 0

D-lactitol Monohydrate 1.71 2.44

D-limonene 2.18 0

Dobutamine 1.56 9.09

Doconexent 1.59 16.22

Dopamine Hydrochloride 2.01 4.35

Dorzolamide??hcl 1.44 5.88

Doxorubicin 2.20 0

Doxycycline 1.34 7.69

Doxylamine Succinate 1.56 7.14

Droperidol 2.39 0

Dyclonine Hydrochloride 1.75 7.69

Dyphylline 1.88 3.85

Edoxudine 2.02 8.16

Edrophonium Chloride 2.05 5 1 1

Efloxate 2.06 18.75

Ellagic Acid 1.86 7.5

Emtricitabine 1.49 5.26

Enilconazole 1.48 3.12

Enoxacin 1.63 3.57 Enrofloxacin 1.15 0

Entacapone 1.11 2.04

Eplerenore 1.34 2.94

Equilin 1.70 28.12

Erdosteine 1.39 0

Ergocalciferol 2.00 0

Erlotinib 1.60 3.23

Erythritol 1.66 0

Erythromycin 2.12 0

Esmolol, Hydrochloride 1.09 6.25

Estradiol 1.41 7.5

Estradiol Benzoate 2.06 0

Estriol 1.22 20.83

Estropipate 1.62 6.25

Ethamivan 1.45 3.45

Ethaverine Hydrochloride 2.33 21.62

Ethenzamide 1.60 4.17

Ethosuximide 1.80 5.56

Ethoxzolamide 1.64 0

Ethyl 1.21 5.71

Etidronate Disodium 1.57 2.86

Etodolac 1.40 5.56

Etretinate 1.62 11.11

Famciclovir 1.66 8.11 1 1

Fasudil Hydrochloride 1.78 3.45

Felbamate 1.16 9.43

Felbinac 1.50 8.33

Fenaclon 2.03 5.77

Fenamisal, Phenyl Aminosalicylate 2.25 36.67

Fenbufen 1.24 5.13

Fenoprofen 1.45 0

Fenoterol Hydrobromide 1.54 6.67

Fenspiride Hydrochloride 2.12 10

Fexofenadine 2.13 5.41

Firocoxib 2.30 7.69

Florfenicol 1.95 0

Fluconazole 1.40 4.55

Flumazenil 2.03 15.38

Flumequine 2.35 9.52

Flunisolide 2.40 3.12

Fluorescein 2.43 17.78

Fluorometholone 1.77 3.03

Flurandrenolide 1.74 2.33

Flurofamide 1.36 2.94

Fluroxene 1.31 2.44 Folic Acid 1.89 10.34

Fomepizole Hydrochloride, Fomepizole 1.82 11.9

Formestane 2.22 17.31

Foscarnet Sodium 2.19 0

Fosfosal 2.25 11.76

Fosinopril 2.32 23.81

Ftaxilide 2.04 5.26

Fumaric Acid 1.56 0

Furaltadone 1.91 12.12

Gaba, Gamma-aminobutyric Acid 1.77 5

Gabapentin 1.44 3.03

Gadoteridol 1.10 5.13

Gallic Acid 1.70 18.18

Gatifloxacin 2.29 2.27

Gemcitabine 1.78 0

Gemifloxacin Mesylate 1.75 2.33

Glibenclamide, Glyburide 1.77 0

Gliclazide 2.26 18.18

Gluconolactone 2.42 5

Glutathione 2.22 0

Guaiacol 1.86 11.11

Guanabenz 2.31 16.28

Guanadrel Sulfate 1.54 4.76

Heptaminol Hydrochloride 1.89 6.67 Dichloride, Hexamethonium 2.07 4.17 Bromide 2.24 8.82

Hydrastine (1r, 9s) 2.04 4.17

Hydrastinine Hydrochloride 1.81 0

Hydrocortisone 1.78 5.41

Hydrocortisone Butyrate 2.28 3.57

Hydrocortisone Valerate 1.70 3.12

Hydroxyprogesterone 1.30 16

Hymecromone 2.05 17.39

Hyoscyamine 1.85 2.08

Ibudilast 2.09 0

Idazoxan Hydrochloride 1.97 12.9

Idramantone 1.29 7.69

Iloprost 1.69 3.33

Imexon 1.84 13.16

Imiquimod 2.24 10.53

Indinavir 1.68 0

Inosine 1.27 11.54

Iodixanol 1.53 7.14

Iohexol 2.19 3.03

Iopanic Acid 2.13 7.14 Ioxilan 2.37 2.94

Irbesartan 2.09 0

Irinotecan, Irinotecan Hydrochloride (trihydrate) 2.33 0

Irsogladine Maleate 1.88 10.81

Isoetharine Mesylate 1.72 9.68

Isoleucine (l) 1.97 8.11

Isosorbide Dinitrate 1.90 4.17

Isotretinoin 1.97 6.06

Isovaleramide 1.18 9.09

Isoxicam 1.98 2.94 No significant 2.16 5.88 activity (d M 1.27 0 <2.47 and % degenercy <50) Ketorolac Tromethamine 1.23 5.56

Khellin 1.16 5.56

Lacitol 1.86 3.45

Lactose Monohydrate 2.05 12.5

L-alpha-methyl Dopa, 1.77 0

Lamivudine 1.68 0

Lamotrigine 2.14 2.63

Leuprolide 1.58 12.12

Levalbuterol Hydrochloride 1.48 11.43

Levetiracetam 1.20 7.69

Levobunolol Hydrochloride 1.01 5.71

Levobupivacaine 2.31 7.89

Levocabastine hcl 1.37 3.33

Levocarnitine Propionate Hydrochloride 2.05 11.11

Levodopa 1.36 4.88

Levofloxacin 2.16 4.17

Levosulpiride 1.62 7.14

Linagliptin 1.22 2.63

Lincomycin 1.81 9.09

Liothyronine 1.66 6.45

Lipoamide 1.69 5.56

Lisinopril 1.88 4.88

Lobeline 2.18 7.69

Lobendazole 1.76 0

Lonidamine 1.62 13.33

Loperamide 2.32 46.67 1 1

Loratadine 1.71 16.67

Lorglumide Sodium 1.97 16.13

Losartan, Potassium 1.87 2.94

Loxapine Succinate 1.57 0

Lufenuron 2.07 26.92

Lumiracoxib 2.17 5

Mafenide Hydrochloride 2.36 1.75 1.87 5.71

Mebeverine 2.07 9.09

Meclofenamic Acid 1.57 3.03

Meclofenoxate 1.74 9.38

Mecysteine Hydrochloride 1.95 3.12

Medroxyprogesterone Acetate 2.40 6.67

Medrysone 2.15 4.35

Mefenamic Acid 1.74 9.52

Megestrol Acetate 2.10 11.9

Meglumine 1.34 2.08

Meglutol 1.85 9.68

Meloxicam 1.77 6.45

Meparfylon 1.29 0 mepartricin 1.59 5.88 1 1

Mephenesin 1.38 2.22

Mephentermine Sulfate 2.03 3.45

Meprylcaine Hydrochloride 1.80 13.64

Meropenem 1.43 0

Mesalamine 1.65 9.09

Mesna 1.73 3.03

Meta-cresyl Acetate 1.55 22.86

Metampicillin Sodium 1.60 3.33

Metaproterenol 1.70 3.03

Metaraminol 1.31 0

Metaraminol Bitartrate 2.31 0 metformin 1.40 3.03 1 1

Methapyrilene 1.71 2.86

Methazolamide 1.76 8.33 1 1

Methocarbamol 1.74 4.76

Methoprene (s) 2.33 2.22

Methotrexate 1.95 4.26 1 1

Methotrexate(+/-) 1.54 0

Methoxamine 2.02 7.69

Methscopolamine Bromide 1.36 3.85

Methsuximide 1.65 2.44

Methylphenidate Hydrochloride 1.53 2.86 1 1

Methylprednisolone 1.71 12

Meticrane 1.22 14.29

Metolazone 1.84 3.23

Metronidazole 2.05 7.14

Mexiletine 1.63 2.17

Midodrine 2.26 0

Miglitol 1.88 0

Miglustat 1.86 5.56

Minocycline Hydrochloride 1.92 4 2.12 1.85

Mitomycin C, Mitomycin 1.89 5.71

Modaline Sulfate 2.07 10.71 montelukast 1.59 0 1 1

Montelukast Sodium 2.39 7.89

Moxalactam Disodium 2.09 4

Moxifloxacin Hydrochloride 2.07 4

Moxisylyte Hydrochoride 1.55 4.65

Mycophenolic Acid 2.28 9.09 1 1

N-acetylneuramic Acid, Aceneuramic Acid 1.73 4.55

Nadide 2.25 0

Nadifloxacin 1.38 3.03

Nafcillin Sodium 2.35 6.25

Nalbuphine 1.88 16.22

Naloxone 1.61 3.57

Naloxone Hydrochloride 1.71 10.26

Naltrexone Hydrochloride 1.93 8.82

Naproxen 1.54 7.41

Naproxol 1.35 4.35

Nateglinide 1.29 0

Nebivolol Hydrochloride 1.48 8.11

Nefazodone 2.27 25.71 1 1

Nefiracetam 1.20 9.09

Nelarabin 1.49 3.03

Neostigmine Bromide 2.42 2.94 1 1

Netilmicin Sulfate 1.46 9.43

Niacin 1.81 11.9

Niacinamide 2.45 5.71

Nicopholine 1.61 7.32

Nicotinyl Alcohol Tartrate 2.15 4.76

Nifenazone 1.94 11.43

Niflumic Acid 1.76 2.22

Nikethamide 1.66 3.57

Nilutamide 1.77 2.33

Nimesulide 2.30 12.12

Nimodipine 1.68 11.11 1 1

Nimustine 1.60 9.38

Nisoldipine 1.93 4.65 1 1

Nitrendipine 1.78 2.5 1 1

Nizatidine 1.38 13.79 1 1

Norepinephrine 2.00 0

Norfloxacin 1.79 3.03

Norgestrel, 1.48 12.12

Noscapine Hydrochloride 2.16 3.03

Novobiocin Sodium 2.36 2.63 1.51 4.55

Octodrine 1.55 8.7

Octreotide 1.91 6.45

Olanzapine 1.33 8.33

Oleandomycin Phosphate 2.04 7.69

Olopatadine Hcl 2.36 8.7

Omega-3-acid (epa Shown) 1.87 7.41

O-phospho-l-, Dexfosfoserine 1.41 0

Orbifloxacin 1.63 9.09 Aketoglutarate, Ornithine 1.67 0 Hydrochloride Orotic Acid 1.54 4

Oseltamivir 1.74 4.76

Oxaliplatin 1.59 10.71

Oxcarbazepine, Trileptal 2.03 0

Oxedrine 1.44 6.9

Oxelaidin Citrate 2.00 17.39

Oxiglutatione Disodium Salt 1.42 3.23

Oxiniacic Acid 1.56 12.9

Oxolamine Citrate 1.70 15.91

Oxolinic Acid 2.09 5.88

Oxybendazole, 2.27 2.7

Oxybenzone 2.32 16.67

Oxyphenbutazone 1.40 24.32

Oxyphencyclimine Hydrochloride 2.17 9.3

Oxyphenonium Bromide 1.66 8.11

Paliperidone 2.12 6.67

Pancuronium Bromide 1.78 3.85

Pantethine 1.67 0

Pantoprazole, Pantoprazole Sodium Salt 1.12 0

Pantothenic Acid 1.59 11.11

Paromomycin Sulfate 2.03 3.64

Paroxypropione 1.73 7.69

Pasiniazid 2.03 0

Pefloxacine Mesylate 1.65 0

Pempidine Tartrate 1.47 6.06

Penciclovir 1.36 10

Penicillamine 1.66 4.88

Penicillin V Potassium 2.24 4.35 Pentetic Acid, Diethylenetriaminepentaacetic 1.40 2.86 Acid Pentoxifylline 1.61 7.89

Phenacemide 1.11 12.24

Phenethicillin Potassium 2.12 3.23

Phenobarbital 1.38 6.67

Phenothrin 2.13 14.89

Phensuccimide 2.38 2.7 2.40 7.14

Phenylbutazone 1.42 8.33

Phthalylsulfacetamide 1.57 7.14

Picolamine 1.87 0

Piconol 1.44 8.11

Pilocarpine 1.75 5.88

Pindolol 1.81 2.78

Pioglitazone 2.47 0

Pipamperone 1.61 3.45

Pipemidic Acid 1.56 6.25

Piperacillin 1.62 8.11

Piperonyl Butoxide 2.23 3.45

Pipobroman 1.70 2.7

Piracetam 1.61 0

Piromidic Acid 2.00 2.44

Piroxicam 2.45 3.33 podofilox 2.11 0 1 1

Polymyxin B1 1.71 10.34

Pranoprofen 2.08 4.17

Pravastatin 2.20 15.79

Pravastatin Sodium 1.95 5.26

Prednisolone 2.33 2.94

Prednisolone Acetate 1.72 0

Prednisolone Sodium Phosphate 1.53 2.08

Prednisone 2.36 6.06

Prilocaine 2.10 11.11

Probenecid 2.31 8

Probucol 1.45 0

Procainamide, Pronestyl 1.68 0 1 1

Procaine, Novocain 2.12 0 1 1

Procaterol Hcl Hemihydrate 2.16 7.69

Procodazole 1.95 0

Procyclidine 2.46 19.05

Proglumide 1.65 5.13

Proguanil; Chlorguanide Hydrochloride 2.21 4.35 1 1

Pronetalol Hydrochloride 1.78 8.16

Propoxur 2.18 5.88

Propoxycaine Hydrochloride 1.50 8.57

Propoxyphene 1.74 2.63

Propranolol 2.10 3.57 Hydrochloride, Protryptyline 2.31 27.27 Hydrochloride 2.38 7.5

Pyrantel Pamoate, Pamoate 2.25 0

Pyrazinamide 2.01 0

Pyridostigmine Bromide 2.08 8.16 1 1 Pyridoxine 1.40 8.57

Pyrimethamine 2.26 13.51

Pyrithyldione 2.44 15.79

Quetiapine 1.76 5.71

Quinapril 1.59 15.62

Quinine 2.02 2.7

Quipazine Dimaleate, Maleate 0.00 42.86

R(-)- 2.29 0

Racecadotril 1.54 3.7

Racepinephrine 1.30 2.63

Ramelteon 1.20 2.38

Ranitidine 1.49 7.14

Ranolazine, Dihydrochloride 1.63 5.88

Rebamipide 1.34 2.63

Resorcinol Monoacetate 2.25 0

Retinyl Acetate 2.26 13.79

Retinyl Palmitate 2.02 9.38 riboflavin 2.14 0 1 1

Ribostamycin Sulfate 1.24 2.13

Rifabutin 2.02 18.75

Rifapentine 1.48 10.34

Rifaximin 1.72 3.7

Riluzole 2.24 39.53

Rimantadine Hydrochloride 2.41 0

Risedronate Sodium 1.25 3.7

Risperidone 1.31 0

Rivastigmine Tartrate 1.65 7.69 1 1

Rizatriptan Benzoate 2.29 6.82

Rofecoxib 1.88 3.7

Rolipram 1.90 0

Rolitetracycline 1.11 3.23

Ropinirole Hydrochloride 1.93 9.68

Ropivacaine, Hydrochloride 1.98 8.33

Rosiglitazone, Rosiglitazone Maleate 2.23 7.69

Roxithromycin 1.40 6.52

Rubitecan 1.31 0

Rufloxacin Hydrochloride 2.09 8.82

S-(-)-, Carbidopa 1.89 6.67 1 1

Salicin 1.51 6.06

Salicyl Alcohol 1.84 7.5

Salicylamide 1.52 4

Salicylanilide 1.87 21.43

Salicylic Acid 2.08 12.5

Salsalate 1.91 5.56

Scopolamine 1.66 10.71 Secnidazole 1.46 7.69

Selegiline 1.90 0

Selenomethionine 2.29 4.65

Semustine 2.10 6.06

Sennoside A 1.35 4.65

Sirolimus 1.45 25

Sisomicin Sulfate 2.36 0 Sodium Dehydrocholate, Dehydrocholate 1.81 15.79 Sodium Sodium Gluconate 1.76 5.88

Sodium Monofluorophosphate 1.72 0

Sodium Nitroprusside 1.84 0

Sodium Phenylacetate 1.52 3.03

Sorbitol 1.49 0

Spaglumic Acid 1.87 3.03

Sparteine Sulfate 1.53 20.69

Spectinomycin 2.34 8.7

Spiramycin 1.87 18.75

Streptozosin 1.74 14.29

Succimer 1.80 0

Succinylcholine Chloride 1.63 2.78

Succinylsulfathiazole 1.52 2.44

Sulfabenzamide 2.14 0

Sulfacarbamide 1.91 0

Sulfacetamide 1.79 3.85

Sulfachlorpyridazine 1.87 6.06

Sulfadimethoxine 1.92 6.25

Sulfadoxine 1.43 0

Sulfaguanidine 1.51 14.29

Sulfameter 1.99 3.85

Sulfamethazine 1.39 11.11

Sulfamethoxazole 1.82 2.94

Sulfamethoxypyridazine 2.18 17.24

Sulfamonomethoxine 1.78 0

Sulfanilamide 2.21 2.86

Sulfaphenazole 1.74 0

Sulfapyridine 1.93 6.06

Sulfasalazine 1.39 12.5

Sulfathiazole 1.98 28.57

Sulfinpyrazone 2.01 6.67

Sulfisoxazole 1.98 11.11

Sulfisoxazole Acetyl 2.09 5.13

Sulindac 1.44 5.88

Suxibuzone 1.55 0

Symclosene 1.82 20

Tacrolimus 2.01 23.53 Taxol, 2.46 21.74 1 1 Dihydrochloride, Telenzepine 2.03 0 Hydrochloride Temozolomide 1.98 11.9

Tenatoprazole 2.25 0

Teniposide 2.19 4

Tenoxicam 1.47 9.68

Terazosin 2.40 0

Terbutaline 1.92 3.03 1 1

Tetracycline 2.13 6.25

Tetrahydrozoline 1.81 3.12

Tetroquinone 1.36 7.27

Thalidomide 2.28 0

Theobromine 1.39 6.67

Thiamazole 1.76 12.5

Thiamine 1.58 5.13

Thioctic Acid 1.93 9.68

Thiotepa 1.59 3.12

Thioxolone, Tioxolone 1.43 5.88

Thip Hydrochloride, Hydrochloride 1.30 6.9

Thymol 1.92 12.5

Thyroxine, 2.36 0

Tiapride 2.14 4.76

Ticlopidine 2.03 28.57

Timolol 1.37 0

Timolol Maleate 1.68 0

Timonacic 1.60 6.67

Tinidazole 2.17 6.45 1 1

Tiopronin 1.13 3.03

Tiotropium Br 1.82 0

Tiratricol 2.36 10.34

Tizanidine Hydrochloride 1.91 13.33

Tobramycin 1.55 5.41

Tolazamide 1.77 7.69

Tolazoline, Priscoline 1.49 12.5

Tolbutamide 1.45 15.62

Tolcapone 1.44 3.57

Tolmetin Sodium 1.17 10.71

Tramadol 2.35 18.92

Tranexamic Acid 1.82 17.65

Trazodone 1.11 4.08

Triacetin 1.34 2.63

Triamcinolone 1.94 7.14

Triamcinolone Acetonide 1.88 0

Trichlormethiazide 2.44 9.68 1 1

Trientine Hydrochloride 2.19 13.04 Trifluridine 1.78 5

Trimebutine Maleate 1.33 10.26

Trimetazidine 2.45 0

Trimethadione 2.29 4.35

Trimethobenzamide Hydrochloride 1.98 3.03

Trioxsalen 2.06 11.76

Triptorelin 2.08 3.23

Troclosene Potassium 1.75 7.14

Tropisetron 1.90 7.69

Troxerutin 2.02 9.68

Tuaminoheptane Sulfate 2.26 12.5

Tylosin Tartrate 1.70 2.38

Tyloxapol 1.44 11.11

Tyrosine 1.37 6.45

Uracil 1.55 9.68

Valacyclovir, Valaciclovir Hydrochloride 1.66 3.23

Valdecoxib 2.15 3.57

Valsartan 1.58 5.88

Vancomycin 1.61 7.14

Vancomycin Hydrochloride 2.29 11.43

Vecuronium Bromide 1.20 0

Venlafaxine, Hydrochloride 2.06 2.38 1 1

Vincamine 1.54 14.81

Vinorelbine 1.69 5.56

Viomycin Sulfate 1.80 6.9

Zaprinast 1.66 3.45

Zidovudine [azt] 1.66 0

Zoledronic Acid 1.98 14.81 42 sub-total

Zolmitriptan 1.33 2.63 13 active 29 inactive 69% agreement , Zolpidem Tartrate 1.97 3.85 (between inactives) 2.15 5.26 144 81 63

Concordance (for actives and inactives) between the two data sets is 67%