Functional Group Table of Contents-1

Functional Group Table of Contents-1

Acids and Derivatives 1 Aromatic Carboxylic Acid Derivatives, 1 Azinyloxy, and Phenoxy-Diaryl-Carboxylic Acid Derivatives, Their Preparation and Use as Mixed ETA/ETB Endothelin Receptor Antagonists, 6 Cinnamic Acid Derivatives, 10 Compounds Derived from Benzoic Acid Esters, Composition Containing Said Compounds and Use Thereof, 15 1,2-Diarylmethylene Derivatives, Their Methods of Preparation, and Their Uses in Therapeutics, 17 Geranic Acid Derivatives, 21 Halogenated Cinnamic Acids and Esters Thereof, Processes for the Preparation Thereof and Halogenated Aryldiazonium Salts, 23 Halogenation Catalyst, 25 Method for Producing Alkoxy Malonic Acid Nitriles, 27 Phosphonosuccinic Acid Derivatives, Processes for Their Preparation and Medicaments Containing These Compounds, 29 Preparation of Cyclohexane Carboxylate Derivatives, 32 Water Soluble Fullerenes with Antiviral Activity, 38 Alcohols 42 Butyne Diol Derivatives, 42 1,2-Dithin Anti-infective Agents, 47 Oligiocycloalkanoid Compounds and Methods of Use, 50 Polymers with Controlled Physical State and Bioerodibility, 55 4-Quinolinemethanol Derivatives as Purine Receptor Antagonists, 57 Synthesis of 5-Decenyl Acetate and Other Pheromone Components, 60 Aldols 63 Stereospecific Synthesis of Aldols, 63 Aldehydes 65 Process for Selective Catalytic Oxidation of Olefins to Aldehydes, Ketones With Cleavage of C=C Bonds, 65 Alkenes 68 Carbonyl Containing Compounds, 68 Alkynes 70 Diaryl-enynes, 70 DNA-Cleaving Anti-Tumor Agents, 74 Amides 78 Adamantane Derivatives, 78 o-Anisamide Derivatives, 81 Benzamide Analogues Useful as PARP (ADP-Ribosyltransferase, ADPRT) DNA Repair Enzyme Inhibitors, 84

Carboxamide Compositions, Methods, and Compositions for Inhibiting PARP Activity, 88 Heterocyclic Amides, 91 Phosphoramide Compounds 96 Amines 99 Aminophenyl Ketones Derivatives and a Method for the Preparation Thereof, 99 Arylamine Synthesis, 103 Fungicidal Spirocyclic Amines, 106 Method for Producing Propargylamine Compounds, 110 One Pot Process for the Preparation of 1-[2-Methylamino-(4-Methoxy- phenyl)-Ethyl]Cyclohexanol, 113 Organic Electroluminescence Device and Phenylenediamine Derivative, 115 Process for Preparing N-Substituted Hydroxylamines and Salts Thereof, 120 Sodium Channel Modulators, 122 Substituted 2-Aminoalkyl 1,4-Diaminobenzene Compounds and Oxidation Dye Precursor Containing the Same, 125 Aminoacids 127 Aminoindanes, 127 Aminopropylphosphinic, 130 Cyclic Aminoacids and Derivatives Thereof Useful as Pharmaceutical Agents, 132 Isocyanoalkyl, Carbonic Acid Derivatives, Their Conversion into Secondary Amidoalkyl Carbonic Acid Derivatives by Isocyanide Multicomponent Reactions, as well as these Secondary Amidoalkyl Carbonic Acid, 135 Spirodiamino Acid Scaffold for Combinatorial Synthesis, 138 Anthracenones 142 10-Substituted 1,8-Dihydroxy-9(10H) Anthracenone Pharmaceuticals, 142 Aza and Diaza Bi- and Tricyclics 146 Bi- and Tri-cyclic Aza Compounds and Their Uses, 146 Certain Tricyclic Substituted Diazabicyclo[3.2.1]octane Derivatives, 151 Dopamine Transporter Imaging Agent, 154 N-Alkyl and N-Acyl Derivatives of 3,7-Diazabicyclo-[3.3.1]Nonanes and Selected Salts Thereof as Multiclass Antirrhythmic Agents, 157 Process for the Manufacture of Tropenol, 160 Aza Benzazolium Salts 163 Aza-Benzazolium Containing Cyanine Dyes, 163 Aza-Dihydroquinoxaline 166 8-Aza, 6-Aza and 6,8-Diazo-1,4-dihydroquinoxaline-2,3-diones and the Use Thereof as Antagonists for the Glycine/NMDA Receptor, 166 Aza-Indolyls 169 Aza-Indolyl Derivatives for Treating Obesity, 169 Aza-Oxindoles 172 Substitued Aza-Oxindole Derivatives, 172 Azides 175 Stereoselective Ring Opening Reactions, 175

Aziridines/Diazirines 180 Diazirine Derivatives of Aromatic Heterocyclic Compounds, 180 Preparation of N-arylmethyl Aziridine Derivatives 1,4,7,10- Tetraazacyclo- Dodecane Derivatives Obtained Therefrom and N-Arylethyl- ethanolamine Sulfonate Esters as Intermediates, 183 Process for Producing Aziridine Compounds, 186 Benzodiazopines 188 Benzodiazepines, 188 Benzoxazoles 192 Benzoxazoles, 192 Benzopyrans 197 Benzopyran Derivatives, 197 Benzothiophenes 201 Pentacyclic Compounds, Intermediates, Processes, Compositions, and Methods, 201 Benzotriazoles 206 Method of Synthesizing t-Amido-Substituted 2-(2-Hydroxyphenyl) benzotriazole Compounds in a One-Step Process, 206 Carbamates/Ureas 209 Herbicidal Sulfonylureas, Their Preparation and Use, 209 Process for the Preparation of Aminocarbonyl Derivatives of Geneseroline Having Selective Brain Anticholinesterase Activity, 212 Catalysis 215 Highly Reactive Form of Copper and Reagents Thereof, 215 Lewis Acid Catalyst Composition, 218 Cumulenes 221 Aromatic Allene Compounds of the Formula (CH2=CH-O)n-R-(A)m in Which R is an Aromatic Group and Preparation Thereof, 221 Preparation of Unsaturated Ketones, 224 (S)-4-Amino-Hepta-5,6-Dienoic Acid and Intermediates Thereof, 227 Cycloanhydrins 230 Method for the Stereoselective Production of Substituted Cyclohexyl- anhydrins, 230 Cyclodextrane/dextrane 233 Conjugation of Biomolecules Using Diels-Adler Cycloaddition, 233 Nohr-McDonald Elimination Reaction, 237 Cyclopentadiene 233 Cyclopentadienyl Derivatives and Process for Their Preparation, 233 Cyclopropanes 240 Aryl Phenylcyclopropyl Sulfide Derivatives and Their Use as Cell Adhesion Inhibiting Anti-inflammatory and Immune Suppressive Agents, 240 Cyclic Compounds Having a Cycloalkylene Chain 246 2-Hydroxymethylcyclopropylidene-methylpurines and -Pyrimidines as AntiViral Agents, 251 Process of Producing Cyclopropanecarboxylate Compounds, 256

Process for the Preparation of Methylenecyclopropane, 258 Synthesis of Cyclopropaneacetylene by a One Pot Process, 260 Dentrimers 262 Dentrimeric Fullerene Derivatives, Process for Their Preparation, and Use as Neurprotectants, 262 Starburst Conjugates, 265 Enamines 269 Use of Enamines as Light Protection Agents, 269 Enaminones 272 Phenyl-Substituted Cyclic Enaminones, 272 Ethers 276 Diaryl Ether Condensation Reactions, 276 Preparation and Use of Ionic Liquids in Microwave-Assisted Chemical Transformations, 279 Wurster’s Crown Ligands, 281 Formazan 283 Formazan Metal Complexes, 283 Furazancarboxylic Acid 286 Hydroxymethylfurazancarboxylic Acid Derivatives, 286 Furanones 289 Furanone Derivatives, 289 Guanidines 291 Cyclic Guanidine Derivatives and Their Use as Pesticides, 291 Guanines 294 Substituted O6-Benzyl-8-Aza-Guanines, 294 Hydrazine 297 Diacylhydrazine Derivatives, 297 Method for Synthesizing Hydrazodicarbonamide, 300 Imidazole 302 Method for Preparing Cycloheptimidazoles, 302 Substituted Imidazole Compounds, 305 Imidazolidine 309 Cis-Imidazolines, 309 Spiroimidazolidine Derivatives, Their Preparation, Their use and Pharmaceutical Preparations Formed Therefrom, 312 Imidazolone 317 Fungicidal 2-Imidazolin-5-ones and Imidazoline-5-thiones, 317 Imidazoltriazionones 320 2-Phenyl Substituted Imidazotriazinones as Phosphodiesterase Inhibitors, 320 Imide Derivatives 324 Photocleavable Agents and Conjugates for the Detection and Isolation of Biomolecules, 324 Process for the Preparation of Alkyl 4[2-(Phthalimido)ethoxy]- acetoacetate, 329

Iminocarboxylic acid methyl amides 331 Preparation of α-Methoxyiminocarboxylic Acid Methylamides and Intermediates Therefore, 331 Indoles 335 Process for the Preparation of Indole Derivatives and Intermediates of the Process, 335 Synthetic Compounds for Treatment of Inflammation, 340 Tetrahydro-β-Carbolines, 342 Indoline 346 Amination Process, 346 Isocoumarins 349 Process for Preparing Isocoumarins, 349 Isoxazolines 353 Method for Producing Isoxazoline-3-yl-acyl Benzene, 353 Ketones 357 Acetoacetic Acid Derivatives, Process for Their Preparation and Their Use, 357 Methods for Making Substituted Phenylketoenols, 360 Process for Preparing 3-Hydroxymethyl-4-(Aryl or Heterocyclic)- Cyclopentanones, 363 Process for Preparing Trifluoromethyl Ketones, 368 Process for the Preparation of High Purity Alkyladamanantyl Esters, 370 Lactams 372 Anticonvulsant and Anxiolytic Lactam and Thiolactam Derivatives, 372 β-Lactams as Antiproliferative Agents, 375 β-Lactam-like Chaperone Inhibitors, 379 N-Thiolated β-Lactam Antibiotics, 382 Process for Preparing Beta Lactam Compound, 386 6-(Spirocyclopropyl)-Penicillanic Acid-4,4-Dioxides, 389 Lactones 392 Benzylidene-γ-Butryolactones, Process for Their Preparation and Their Use as UV Absorbers, 392 Ring-Opened Azlactone Inititators for Nitroxide-Mediated Polymerization, 395 Macocyclic Rings 398 β-Diketone Compounds, β-Diketone Compounds Coordinated to Metal, Method of Organic Synthesis with These, and Catalyst, 398 1,4-Dioxacylcycloalkane-2-one and 1,4-Dioxacylcycloalkene-2-one, 402 Synthesis of Macrocyclic Tetraamido-N Ligands, 405 The Preparation of Giant Ring Compounds, 408 Morpholines 411 Lewis Acid-Catalyzed Claisen Rearrangements in the Preparation of Chiral Products, 411 Naphthopyans 413 Indeno-fused Photochromic Naphthopyrans, 413

Naphthyridines 418 4-Hydroxy-1,8-Naphthyridine-3-Carboxamides as Antiviral Agents, 418 Nitro Derivatives 422 Geminal-Dinitro-1,5-Diazocine Derivatives, 422 Methods of Preparing Salts of Dinitromethane, 428 Vicarious Nucleophilic Substitution Using 4-Amino-1,2,4- Triazole, Hydroxylamine or O-Alkylhydroxylamine to Prepare 1,3-Diamino- 2,4,6-Trinitrobenzene or 1,3,5-Triamine-2,4,6-Trinitrobenzene, 430 Nitrones 432 Furan Nitrone Compounds, 432 Organometallics 435 Aryl Borates, 435 Boric Ester Synthesis, 438 Method for Producing Monoaryloxy-ansa-Metallocenes, 440 Process for Preparing Bisallylboranes and Non-aromatic Boronic Acids, 443 Synthetic Molecules That Specifically React with Target Sequences, 445 Orthocarbonates, -esters, and derivatives 449 Spiroorthocarbonates Containing Epoxy Groups, 449 Substituted Sprioalkylamino and Alkoxy Heterocyclics, Processes for Their Preparation, and Their Use as Pesticides and Fungicides, 452 Synthesis of Spiro Ortho Esters, Spiro Ortho Carbonates, and Intermediates, 455 Oxadiazines 458 Oxadiazine Derivative, 458 1,3,4-Oxadiazine Derivatives and Their Use as Pesticides, 461 Oxathiolanes 464 Antiviral Activity and Resolution of 2-Hydroxylmethyl-5- (5-fluorocytosin-1-yl)-1,3-Oxathiolane, 464 Substituted 1,3-Oxathiolanes with Antiviral Properties, 468 Oxazines 472 Photochromic Oxazine Compounds and Methods for Their Manufacture, 472 Oxazolidinones 475 Process to Prepare Cyclic-Sulfur Fluorine Containing Oxazolidinones, 475 Oxetanes 480 Fluorinated Oxetane Derivatives and Production Process Thereof, 480 Process for the Production of 3-Alkyl-3-Hydroxymethyloxetanes, 482 Oxetanones 484 Oxetanone Derivatives, 484 Oximes 486 O-Acyloxime Photoinitiators, 486 Oxime Derivatives and Their Use Thereof as Latent Acids, 489 Oxirane 491 Diels-Adler Adducts of Epoxybutene and Epoxybutene Derivatives, 491 Process for the Preparation of an Oxirane, Aziridine or Cyclopropane, 493

Phenols 496 Calixarene Derivatives, 496 Dimeric Arylisoquinoline Alkaloids and Synthesis Method Thereof , 500 Process for Preparing Procyanidin (4-6 or 4-8) Oligomers and Their Derivatives, 504 Piperidine 508 N-acyl Cyclic Amine Derivatives, 508 Opiate Compounds, Methods of Making and Methods of Use, 511 Process for Production of Piperidine Derivatives, 515 Spiropiperidine Derivatives, 519 Piperizines 523 Piperazine Derivatives, 523 Porphyrins 525 1,3-Dipolar Cycloadditions to Polypyrrolic Macrocycles, 525 Pyrans 527 Synthesis of 3,6-Dialkyl-5,6-Dihydro-4-Hydroxy-Pyran-2-One, 527 Pyrazoles 530 Parasiticidal Compounds, 530 Spiropyrazole Compounds, 534 Pyridine 537 Process for Preparing Tribromomethylsulfonylpyridine, 537 3-Pyridinyl Compounds, 539 Pyridone and tetrahydropyridone 542 Pyridone Derivatives, Their Preparation and Their Use as Synthesis Intermediates, 542 Solid Phase Synthesis of Heterocycles, 546 Pyrimidines 549 N-Heterocyclic Derivatives as NOS Inhibitors, 549 Pyrrols 552 7-Azabicyclo[2.2.1]Heptane and Heptene Derivatives as Cholinergic Receptor Ligands, 552 Colormetric Sensor Compositions and Methods, 555 Quinones 558 Compositions and Methods for Treating Viral Infections, 558 Quinone Compound, Liquid Crystal Composition, and Guest-Host-Type Liquid Crystal Cell Employing the Same, 562 Polycyclic Aryl and Heteroaryl Substituted 1,4-Quinones Useful for Selective Inhibition of the Coagulation Cascade, 565 Synthesis of Coenzyme Q10, Ubiquinone, 570 Radiolabelled Reagents 574 Radioligands and Their Use for Identifying Potassium Channel Modulators, 574 Synthesis of 2H- and 13C-Substituted Dithanes, 578 Tritioacetylating Reagents and Processes for Preparation Thereof, 580 Saccharides 582 2-Saccharinylmethyl Heterocyclic Carboxylates Useful as Proteolytic, 582

Sugars 587 Heavily Fluorinated Sugar Analogues, 587 Preparation of Thioarabinofuranosyl Compounds and Use Thereof, 591 Process for the Alkaline Oxidative Degradation of Reducing Sugars, 596 Sugar Derivatives of Hydromorphorine, Dihydromorphorine and Dihydroisomorphorine Compositions Thereof and Uses for Treating or Preventing Pain, 599 Sulfonamides 602 Thioaryl Sulfonamide Hydroxamic Acid Compounds, 602 Sulfones 607 α-Amino-β-Sulfonyl Hydroxamic Acid Compounds, 607 Nitromethylthiobenzene Derivatives as Inhibitors of Aldose Reductase, 610 Process for the Preparation of Ethanesulfonyl-piperidine Derivatives, 614 α,β-Unsaturated Sulfones for Treating Proliferative Disorders, 618 Sulfonylimides 621 Sulfonylimide Compounds, 621 Tetrabenazine 623 Iodine Derivatives of Tetrabenazine, 623 Tetracyclines 626 7-Substituted Fused Ring Tetracycline Compounds, 626 Tetrahydrobenzoquinoxaline Diones 629 Pyrrolyl Tetrahydrobenzoquinoxaline Diones, Their Preparation and Use As Glutamate Receptor Antagonist, 629 Tetrahydrobenzothiepines 633 Method for the Preparation of Tetrahydrobenzothiepines, 633 Tetrahydroisoquinolines 638 Pictet-Spengler Reaction for the Synthesis of Tetrahydroisoquinolines and Related Heterocyclic Compounds, 638 Tetrahydroquinolines 640 Dimeric Compounds, 640 Tetrazoles 643 Tetrazolyl-Phenyl Actamide Glucokinase Activators, 643 Thiazoles 648 Oxazolo, Thiazolo and Selenazolo [4,5-c]-Quinolin-4-Amines and Analogues Thereof, 648 Tri-Aryl-Substituted-Ethane PDE4 Inhibitors, 651 Thiophenes 656 3,4-Diaryl Thiopenes and Analogs Thereof Having Use as Antiinflammatory Agents, 656 Oligiothiophenes and Synthesis Thereof, 660 Polyaryl Antitumor Agents, 663 Triazines 666 Aryloxy- and Arylthiosubstituted Pyrimidines and Triazines and Derivatives Thereof, 666 Method of Alkylating Triazine Derivatives, 670

Triazoles 673 One Step Synthesis of 1,2,3-Triazole Carboxylic Acids, 673 Triazolyl-Tetrazinyl-Aminotriazine Compounds Useful in Pyrotechnic Compositions and Process Thereof, 676 Trioxolanes 679 Spiro and Dispiro 1,2,4-Trioxolane Anti-malarials, 679

Product Utility Table of Contents-2

Additives t-Amido-Substituted 2-(2-Hydroxyphenyl)benzotriazole Compounds Ultraviolet Light Absorbing Coating Additives, 206 Aromatic Allene Compounds as Chemical Intermediates and Paint Components, 221 Colorant Stabilizer from Ultra Violet Light Using β-Cyclodextrin Inclusion Complexs, 269 Method for Synthesizing the Blowing Agent Hydrazodicarbonamide, 300 Oxime Derivatives as Photoresist Latent Acid for Acid-Curable Resins, 489 Resin and Fire-Retardant Materials Using Triazine Derivatives, 670 Sun Screen Additive Using Halogenated Cinnamic Acids and Esters Thereof, 23 Analytical Agents Analytical and Diagnostic Reagents Useful as Immunogens, 324 Aza-Benzazolium Containing Cyanine Dyes Fluorescencing Molecular Probes, 163 Biological Imaging Agent Using N-Arylmethyl Aziridine 1,4,7,10- Tetraazacyclododecane Derivatives, 183 Calaxarene Derivatives for Use as Chelating Agents for Actinide and Lanthanide Metal Cations, 496 DNA Labeling Agents Using Synthetic Molecules That Specifically React with Target Sequences, 445 Dopamine Transporter Imaging Agent Useful as Early Diagnosis Agents for Neurodegenerative Disorders, 154 New Analytic Reagents for Detection of Fluoride, Chloride, and Phosphate Anions Using Colormetric Sensor Compositions and Methods, 555 Photocleavable Agents and Conjugates for Use as Biological Tagging Agent for Nucleic Acids, 324 Catalysts and Methods Acetyl Chlorination Catalyst, 25 Arylamine Synthesis Method Using Tris(dibenzylideneacetone)dipalladium, 103 Chiral Morpholine Derivatives, 411 Diels-Alder Epoxybutene Adducts, 491 Epoxide Preparation Using Insitu Diazo Intermediates, 493 High Yielding Alkylation Method Using Ionic Solvents, 279 High Yielding Method for Preparing Adamanantyl Methacrylates, 370 High Yielding Method for Preparing Isocoumarin Derivatives, 349 Highly Reactive Form of Copper and Reagents Thereof, 215 Improved Method for Preparing N-Substituted Hydroxylamines and Derivatives, 120 Improved Method for Preparing 1,2,3-Triazole Carboxylic Acid Derivatives, 679 Improved Method for Preparing Tribromomethylsulfonylpyridine, 537 Improved Method for Preparing Ubiquinone, 570

Lewis Acid Catalyst Using Ytterbium Tris(trisperfluorooctanesulfonyl)- methide, 218 Method for Preparing Aminopropargyl and Derivatives, 110 Method for Producing Monoaryloxy-ansa-Metallocenes for Use as Olefin Polymerization Catalyst, 440 Method for the Stereoselective Production of Substituted Cyclohexylanhydrins Using (R)- or (S)-Oxynitrilase, 230 Olefin Oxidizing Reagent for the Selective Catalytic Oxidation of Olefins to Aldehydes, Ketones With Cleavage of C=C Bonds, 63 Reagent for Aromatic Ether Coupling Using Cesium carbonate and Di(copper triflate).benzene 279 Synthesis of Macrocyclic β-Diketone Rings, 398 Synthesis of Macrocyclic Tetraamido-N-Ligands for Oxidizing Complexes, 405 Synthetic Method for Preparing Indolines, 346 Vicarious Nucleophilic Substitution Using 4-Amino-1,2,4- Triazole, Hydroxylamine or O-Alkylhydroxylamine to Prepare 1,3-Diamino-2,4,6- Trinitrobenzene or 1,3,5-Triamine-2,4,6-Trinitrobenzene, 430 Zirconium or Titanium Catalysis Ligands for α-Olefin Polymerisation, 240 Chemical Intermediates Acetoacetic Acid Derivatives, Process for Their Preparation, and Their Use Perfume and Fragrance Intermediates, 357 Arylboron Derivatives, 435 Automotive Lubricant Intermediate, 68 Boric Acid Intermediates, 438 Cumulene Ketones Intermediates, 224 Halodiazirine and Cyclopropane Derivatives, 180 Indole Derivatives and Intermediates Chemical Preecursor in the Treatment of Hyperlipoproteinaemia and Arteriosclerosis, 335 Intermediate for Anti-hypertensive and Anti-ischaemic Drugs, 329 Intermediate in Commerical Prepartion of HIV Chemokine CCR-5 Receptor Antagonists, 363 Isocyanoalkyl, Carbonic Acid Derivatives as Amino Acid Precursors, 135 Method for Producing Alkoxy Malonic Acid Dinitriles Anesthetic Intermediate, 27 One Pot Process for the Preparation of the Anti-depressant Intermediate, 1-[2- Methylamino-(4-Methoxyphenyl)-Ethyl]Cyclohexanol, 113 Preparation of Cyclopropanecarboxylate Compounds as Pyrethroid Precursors, 256 Process for Preparing Bisallylboranes and Non-aromatic Boronic Acids, 443 Process for Preparing Trifluoromethyl Ketones as Pesticide Precursors, 368 Process for Producing Aziridine Compounds as Amino Acid and β-Lactam Antibiotic Intermediates, 186 Spirodiamino Acid Scaffold Template for the Preparation of Synthetic Receptor and Enzyme Intermediates, 138 Starburst Agricultural and Pharmaceutical Intermediate, 265 Stereoselective Azide Ring Opening Reactions, 175

Stereospecific Routes to Polypropinates and Chiral 2-Substituted-1,3 Diols, 65 Synthesis of Cyclopropaneacetylene by a One Pot Process Precursor for the Preparation of HIV Reverse Transcriptase, 260 Synthesis of 3,6-Dialkyl-5,6-Dihydro-4-Hydroxy-Pyran-2-One as a Tetrahydrolipstatin Intermediate, 484 Cosmetics 2-Aminoalkyl 1,4-Diaminobenzene Compounds as Hair Coloring Agent Precursors, 125 Fragrance and Perfume Component from Geranic Acid Derivatives, 21 Fragrances and Perfumes from 1,4-Dioxacylcycloalkane-2-one and 1,4- Dioxacylcycloalkene-2-one, 402 Photochromic Oxazine Compounds Used in Sunlight-Induced Darkening Sunglasses, 472 Photosensitive Opthalmic Plastic Lenses Using Indeno-fused Photochromic Naphthopyrans, 413 Benzylidene-γ-Butryolactones as a Sunscreen Component in Cosmetics, 392 Dyes Organic Dyes Bases on Formazan Metal Complexes, 283 Electronic Electroluminescence Device for Reducing Voltage Using Phenylenediamine Derivatives, 115 Lithium Batteries Containing Sulfonylimide Compounds as Electrolyte, 621 Energetic Materials Geminal-Dinitro-1,5-Diazocine Derivatives, 422 Methods of Preparing Salts of Dinitromethane, 428 Triazolyl-Tetrazinyl-Aminotriazine Compounds Useful in Pyrotechnic Compositions and Process Thereof, 676 Free Radical Agents Furan Nitrones as Spin Radical Trapping Agents, 432 Tetrahydroisoquinolines as Free Radical Trapping Agents and Precursors, 643 Fungicides Agricultural Fungicides Based on 2-Imidazolin-5-ones and Imidazoline-5- thiones, 317 Antifungal Agents Based on 1,2-Dithin Ester Derivatives, 47 Antifungal Agents Derived from Spirocyclic Amines, 106 Preparation of α-Methoxyiminocarboxylic Acid Methylamides for Use as Fungicides, 331 Herbicides Herbicidal Agents Containing Sulfonylureas, 209 Herbicides Derived from Aminophenyl Ketones Derivatives, 99 Method for Producing Isoxazoline-3-yl-acyl Benzene for Use as an Herbicide, 353 Liquid Crystals Liquid Crystal Cells for Electrode Substrates Prepared from a Quinone Compound and Liquid Crystal, 562 Wurster’s Crown Ligands as Liquid Crystal Displays, 281

Parasiticide 4-Ethynylpyrazole Derivatives Useful as Parasiticides, 530 Pesticides Animal Pesticides Based on Cyclic Guanidine Derivatives 291 Insect Pheromones Prepared from 5-Decenyl Acetate, 60 Oxadiazine Derivatives Useful as Pesticides, 458 1,3,4-Oxadiazine Derivatives and Their Use as Pesticides, 461 Pesticides Prepared from Substituted Phenylketoenols, 360 Phenyl-Substituted Cyclic Enaminones Useful as Pesticides and Herbicides, 272 Substituted Sprioalkylamino and Alkoxy Heterocyclics, Processes for Their Preparation, and Use as Pesticides and Fungicides, 452 Pharmaceuticals Analgesics Spiropyrazole Compounds as Opioid Receptor Ligands, 534 Sugar Derivatives of Hydromorphorine, Dihydromorphorine and Dihydroisomorphorine, 599 Treatment of Neuropathic Pain Using Amino Di(benzylether) Derivatives, 122 Analgesic Antagonists Piperidine Derivatives as Opioid Analgesic Antagonists, 511 Antibacterial Agents Cyclic-Sulfur Fluorine Containing Oxazolidinones as Antibacterial Agents, 475 β-Lactam-like Chaperone Inhibitors, 379 Antibiotics N-Thiolated β-Lactam Antibiotics, 382 Process for Preparing β-Lactam Compounds, 386 6-(Spirocyclopropyl)-Penicillanic Acid-4,4-Dioxides, 389 7-Substituted Fused Ring Tetracycline Compounds, 626 Anticonvulsant Anticonvulsant and Anxiolytic Lactam and Thiolactam Derivatives, 389 Anticoagulants Polycyclic Aryl and Heteroaryl Substituted 1,4-Quinones Useful for Selective Inhibition of the Coagulation Cascade, 565 Pyridone Derivatives as Anticoagulants and Antithrombotic Agents, 542 Anticycotoxicity Agent Substitued Aza-Oxindole Derivatives for Use in Reducing Epithelial Cytotoxicity Induced During Chemotherapy, 172 Anti-inflammatory Agents Anti-inflammatory and Analgesic Agents Based on 1,2-Diarylmethylene Derivatives, 17 Aryl Phenylcyclopropyl Sulfide Derivatives and Their Use as Cell Adhesion Inhibiting Anti-inflammatory and Immune Suppressive Agents, 243 Benzodiazepines as Cell Adhesion Modulators for Regulating Inflammatory and Immune Responses, 188 N-Heterocyclic Derivatives as Nitric Oxide Synthase Inhibitors, 549 10-Substituted 1,8-Dihydroxy-9(10H) Anthracenone Pharmaceuticals, 142

Substituted Imidazole Compounds as CSBP/p38 Kinase Inhibitor, 305 Treatment of Immune or Inflammatory Disorders with Cinnamic Acid Derivatives, 10 Anti-Malarials Spiro and Di-spiro Adamantane 1,2,4-Trioxolane Antimalarials, 679 Anti-neoplastic Agents Animal Anti-neoplastic Agents Based on Phosphoramide Compounds, 96 Antiproliferation Agents Based on Oxazolo, Thiazolo and Selenazolo [4,5-c]- Quinolin-4-Amines and Analogues Thereof, 648 Benzamide Analogues Useful as DNA Repair Enzyme Inhibitors, 84 Cis-Imidazolines as Antiproliferation Agents, 309 DNA-Cleaving Anti-Tumor Agents, 74 Heavily Fluorinated Sugar Analogues, 587 β-Lactams as Antiproliferative Agents, 375 Poly(2-thienyl) Containing AntiTumor Agents, 663 Preparation of Thioarabinofuranosyl Compounds and Use Thereof, 591 Process for Preparing Procyanidin (4-6 or 4-8) Oligomers and Their Derivatives, 505 Substituted O6-Benzyl-8-Aza-Guanines, 294 Therapeutic Photosensitizing Agents Prepared from1,3-Dipolar Cycloadditions to Polypyrrolic Macrocycles, 525 α,β-Unsaturated Sulfones for Treating Proliferative Disorders, 618 Arthritis 3,4-Diaryl Thiopenes and Analogs Thereof Having Use as Anti-inflammatory Agents in the Treatment of Arthriris, 656 Spiroimidazolidine Derivatives, Their Preparation, Their use and Pharmaceutical Preparations Formed Therefrom in the Treatment of Rheumatoid Arthritis or Allergic Disorders, 312 Cardiovascular Disorders Adamantane Derivatives for Treatment of Cardiovascular Disorders, 78 Azinyloxy, and Phenoxy-Diaryl-Carboxylic Acid Derivatives, Their Preparation and Use as Mixed ETA/ETB Endothelin Receptor Antagonists, 6 Benzopyran Derivatives as α1-Adrenergic Receptor Inhibitors, 197 Diacylhydrazine Derivatives as Integrin Inhibitors, 297 N-Alkyl and N-Acyl Derivatives of 3,7-Diazabicyclo-[3.3.1]Nonanes and Selected Salts Thereof as Multiclass Antirrhythmic Agents, 157 2-Phenyl Substituted Imidazotriazinones as Phosphodiesterase Inhibitors, 320 Central Nervous Disorders Piperazine Derivatives for Treatment of Central Nervous Disorders, 523 2-Saccharinylmethyl Heterocyclic Carboxylates Useful as Proteolytic Enzyme Inhibitors and Compositions and Method of Use Thereof, 582 Dermatology Aromatic Carboxylic Acid Derivatives for Treatment of Photodamaged Skin, 1

Compounds Derived from Benzoic Acid Esters, Composition Containing Said Compounds and Use Thereof in the Treatment of Alopecia, 15 Diabetes Nitromethylthiobenzene Derivatives as Inhibitors of Aldose Reductase for Treatment of Diabetic Peripheral and Autonomous Complications, 610 Tetrazolyl-Phenyl Actamide Glucokinase Activators for Treatment for Type II Diabetes Disorder, 643 Drug Delivery Oligiocycloalkanoid Compounds and Methods of Use as Drug Delivering Agents, 50 Polymers with Controlled Physical State and Bioerodibility, 55 The Preparation of Giant Ring Compounds for Use as Macrocyclic Lipids in Drug Delivery Systems, 408 Gastrointestinal Disorders Aminopropylphosphinic Acids and Derivatives for Treatment of Upper Gastrointestinal Tract Disorders, 130 Aza-Indolyl Derivatives for Treating Obesity, 169 Hormonal Pentacyclic Compounds, Intermediates, Processes, Compositions, and Methods for Treatment of Post-Menopausal Syndrome, 201 Hypertension Butyne Diol Derivatives as Endothelin Receptor Antagonists, 42 Method for Preparing Cycloheptimidazoles for Treatment of Hypertension Metabolic Disorders o-Anisamide Derivatives for Treatment of Metabolic Diseases, 81 Phosphonosuccinic Acid Derivatives, Processes for Their Preparation, and Medicaments Containing These Compounds in Treatment of Calcium Metabolic Disorders, 29 Metalloprotease Enzyme Disorders α-Amino-β-Sulfonyl Hydroxamic Acid Compounds for Use as Matrix Metalloprotease Inhibitors, 607 Thioaryl Sulfonamide Hydroxamic Acid Compounds for Use as Metalloproteinases, 602 Muscle Relaxants Muscle Relaxants Derived from Hydroxymethylfurazancarboxylic Acid Derivatives, 286 Neurological Aminoindanes for Treatment of Chronic Neurodegenerative Diseases, 127 8-Aza, 6-Aza and 6,8-Diazo-1,4-dihydroquinoxaline-2,3-diones and the Use Thereof as Antagonists for the Glycine/NMDA Receptor, 166 Carboxamide Compositions, Methods, and Compositions for Inhibiting PARP Activity, 88 Cyclic Aminoacids and Derivatives Thereof Useful as Pharmaceutical Agents for Treatment of Neuropathological Diseases, 132

Dentrimeric Fullerene Derivatives, Process for Their Preparation, and Use as Neurprotectants, 262 Diaryl-enynes as Glycine Uptake Inhibitors, 70 Furanone Derivatives for Treatment of Neurodegenerative Disorders, 289 Process for the Preparation of Aminocarbonyl Derivatives of Geneseroline Having Selective Brain Anticholinesterase Activity, 212 Process for the Preparation of Ethanesulfonyl-piperidine Derivatives, 614 3-Pyridinyl Compounds for Treatment of Parkinson's Disease, 539 Pyrrolyl Tetrahydrobenzoquinoxaline Diones, Their Preparation and Use As Glutamate Receptor Antagonist, 629 Tetrahydroquinolines Dimeric Compounds for Treatment of Alzheimer’s Disease, 640 Psychiatric Aryloxy- and Arylthiosubstituted Pyrimidines and Triazines and Derivatives Thereof for Treatment of Psychiatric Disorders and Neurological Diseases, 666 7-Azabicyclo[2.2.1]Heptane and Heptene Derivatives as Cholinergic Receptor Ligands, 552 Bi- and Tri-cyclic Aza Compounds and Their Uses Neurotransmitter Re-uptake Inhibitors, 146 Certain Tricyclic Substituted Diazabicyclo[3.2.1]octane Derivatives for Treatment of Schizophrenia, 151 (S)-4-Amino-Hepta-5,6-Dienoic Acid and Intermediates Thereof as Irreversible GABA-T Inhibitor, 227 Tetrahydro-β-Carbolines for Treatment of Eating and Sexual Disorders, 343 Respiratory Diseases Benzoxazoles as Phosphodiesterases (PDEs) Inhibitor for Treating Asthma, 192 Heterocyclic Amides as Human Neutrophil Elastase Inhibitors, 89 N-Acyl Cyclic Amine Derivatives for Treatment of Respiratory, Urinary and Digestive Diseases, 508 Process for Preparing Piperidine Derivatives for Use as Non-sedating Anti- Histamine, 515 Spiropiperidine Derivatives for Use as Inhibitor for Respiratory Tract Contractions, 519 Tri-Aryl-Substituted-Ethane PDE4 Inhibitors as Anti-asthmatic and Anti- inflammatory Precursors, 651 Serum Cholesterol Lowering Agents Method for the Preparation of Tetrahydrobenzothiepines as Ileal Bile Acid Transporter for Lowering Blood Serum Cholesterol, 638 Oxetanone Derivatives as Lipase Inhibitors for Lowering Cholesterol, 484 Sleep Disorders Cyclic Compounds Having a Cycloalkylene Chain for Preventing and Treatment of Melatoninergic Disorders, 246

Virucides Antiviral Activity and Resolution of 2-Hydroxylmethyl-5-(5-fluorocytosin-1- yl)-1,3-Oxathiolane for Treatment of HIV, 464 Compositions and Methods for Treatment of HIV-1 and HIV-2 Using Desmethylhypericin and Derivatives , 558 Dimeric Arylisoquinoline Alkaloids and Synthesis Method Thereof as Antiviral Agents in the Treatment of HIV, 500 2-Hydroxymethylcyclopropylidene-methylpurines and -Pyrimidines as AntiViral Agents, 251 4-Hydroxy-1,8-Naphthyridine-3-Carboxamides as Antiviral Agents Treatment of Herpes Simplex Viruses Using 4-Hydroxy-1,8-Naphthyridine-3- Carboxamides, 418 Substituted 1,3-Oxathiolanes with as HIV Replication Inhibitor, 468 Water Soluble Fullerenes with Antiviral Activity, 38 Polymer Initiators Azlactone Polymerization Initiators, 395 Photopolymerization Agents using O-Acyloximes, 486 Photopolymerization Agents using Spiroorthocarbonate, 449 Prepolymers Fluoropolymer Precursor, 480 Polymer Precursor for Polymeric Drug Delivery Devices, 455 Polythiophene Precursor, 660 Production and Industrial Preparations Alkaline Oxidative Degradation of Reducing Sugars, 596 3-Ethyl-3-hydroxylmethyloxetane Preparation, 482 Methylene-cyclopropane Scale Up, 258 Preparation of Cyclohexane Carboxylate Derivatives for Use as Neuraminidase Inhibitors, 32 Tropenol Production, 160 Radiolabelled Reagents Iodine Derivatives of the Monoamine Uptake Inhibitor Tetrabenazine and Radiolabeled 125I-Derivatives, 623 125I-Radioligands for Identifying Potassium Channel Modulators, 575 Synthesis of 2H- and 13C-Substituted Dithanes, 579 The Use of Tritium Gas in Preparing Tritioacetylating Reagents, 580