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LESTAURTINIB

MIDOSTAURIN

AXITINIB

Tyrosine- TIE-2

Serine/threonine- 2Mitogen-activated protein kinase kinase kinase kinase 5 Serine/threonine-protein kinase MST2 NERATINIB SPS1/STE20-related protein kinase YSK4 SORAFENIB Dual specificity -activated protein kinase kinase 5 Proto- tyrosine-protein kinase MER Platelet-derivedTANDUTINIB beta Epithelial discoidin domain-containing receptor 1 NINTEDANIB Mixed lineage kinase 7 Macrophage colonyTyrosine-protein stimulating kinasefactor receptorreceptor UFOTyrosine-protein kinase BLK Tyrosine-protein kinase LCK NILOTINIB Serine/threonine-protein kinase 10 NT-3 growth factor receptor DiscoidinMitogen-activated domain-containing protein receptor kinase 2 kinase kinase kinase 3 Tyrosine-protein kinase ABL Nerve growth factor receptor Trk-A FORETINIBEphrin type-B receptor 6 Adaptor-associated kinaseQUIZARTINIB Ephrin type-AEphrin receptor type-B receptor5 2 Mitogen-activated proteinTyrosine-protein kinase kinase kinaseTyrosine-protein kinase JAK3 kinase 2 kinase receptor FLT3 Fibroblast growth factorSerine/threonine-protein receptor 1 kinase Aurora-B Ephrin type-A receptor 8 Serine/threonine-proteinDual specificty protein kinase kinase PLK4Mitogen-activated CLK1 protein kinase kinase kinase 12 Misshapen-like kinase 1Cyclin-dependent kinase-like 2 Platelet-derivedLINIFANIB growth factor receptorEphrin alpha type-A receptor 4 c-Jun N-terminal kinaseALISERTIB 3 Serine/threonine-protein kinase SIK1 PONATINIB Dual specificity protein kinaseStem TTK cell growthHomeodomain-interacting factor receptorTyrosine-proteinTyrosine proteinkinase kinase non-receptorkinase TYK2 4 protein 2 Maternal embryonic leucine zipper kinase Tyrosine-protein kinase ABL2NUAK family SNF1-like kinase 2 -1 receptor-associatedSerine/threonine-proteinVascular kinase endothelial 1 Neurotrophic kinasegrowth Aurora-A factortyrosine receptor kinase receptor2 type 2 Ephrin type-B receptor 3 Serine/threonine-protein kinaseTyrosine-protein SRPK1 kinaseMitogen-activated YES protein kinase kinase kinase kinase 1 Tyrosine-proteinGILTERITINIB kinase receptorBcr/AblTyrosine-protein RETfusion protein kinase TXK Non-receptor tyrosine-protein kinase TNK1 Mitogen-activated protein kinase kinase kinase 4 ILORASERTIBALECTINIBCABOZANTINIBTRAF2-OSI-930 and NCK-interacting kinase Fibroblast growth factorMAPSerine/threonine-protein receptor kinase p383 alpha AFATINIB kinase MST1 Tyrosine-protein kinaseMitogen-activated ITK/TSK protein kinase kinase kinaseSerine/threonine-protein 2 kinase 25 HepatocyteProto-oncogene growthENTOSPLETINIB factor receptor tyrosine-proteinCell division kinase protein ROS kinase 8 G protein-coupledBone morphogeneticSerine/threonine-protein receptor protein kinase receptor 4 Casein type-2 kinase kinase MST4 II alpha (prime) c-Jun N-terminal kinaseDual specificity 1 proteinDual kinase specificity CLK3 mitogen-activatedReceptorCasein protein kinase tyrosine-proteinkinase I epsilon kinase 2 kinase erbB-3 ALK tyrosineSerine/threonine-protein kinase receptor kinase RAF MAP kinaseHomeodomain-interacting signal-integrating kinase 2 protein kinaseTyrosine-protein 2 kinase SYKBRIVANIB DASATINIB Tyrosine-protein kinase Lyn Receptor protein-tyrosine kinaseSerine/threonine-protein erbB-4 kinase pknB DACTOLISIBReceptor protein-tyrosineBMP-2-inducible kinase erbB-2 protein kinase Dual specificity mitogen-activatedTRAMETINIBSerine/threonine-protein protein kinase kinase kinase 1 MRCKTyrosine-protein beta Receptor-interactingkinase Srms serine/threonine-protein kinase 1 Tyrosine-protein kinaseTyrosine-proteinFibroblast FRK growthVascular kinase factor FGR endothelialVascular receptor growthendothelial 2 factor growth receptor factor 3 receptor 1 Myosin light chainBone kinase morphogenetic protein receptor type-1B Cyclin-dependent kinase 7 c-Jun N-terminal kinase 2 VascularCOBIMETINIB Serine/threonine-proteinendothelial growth factor kinase receptorSerine/threonine-protein 16 kinase 32B Serine/threonine-proteinProtein kinase kinase N2 Chk1 EphrinSerine/threonine-proteinInterferon-induced- type-A receptor double-stranded 6 kinase TAO3 RNA-activated protein kinase ALVOCIDIB Serine/threonine-proteinSerine/threonine-protein kinase SRPK3 kinase RIO1 RibosomalTyrosine-protein protein S6 kinase kinaseIBRUTINIB alpha 3SRC TIVOZANIB Tyrosine-proteinActivin kinase receptor FES type-1 Serine/threonine-protein kinase RIO3 SIROLIMUS SEMAXANIB Dual-specificityFEDRATINIB tyrosine-phosphorylationLIM domain regulated kinase 1 kinase 1A Tyrosine-protein kinase receptor Tie-1 TRABECTEDIN Mitogen-activated protein kinase kinase kinase 3 Macrophage-stimulatingTyrosine-protein protein receptor kinase BTK Serine/threonine-proteinMammalianFocal adhesion target kinase of kinaseRapamycin GAK 1 (mTORC1)myosinInsulin light receptor-relatedchain kinaseEphrin 2 proteintype-B receptor 4 Dual specificity proteinCDK3/cyclin kinase CLK4 ELeucine-rich repeat serine/threonine-protein kinase 2 Calcium-dependent proteinActivin kinase receptor 1 type-2B Serine/threonine-proteinSerine/threonine-protein kinase ULK2Serine/threonine-protein kinase PCTAIRE-1Tyrosine-protein kinase kinase NEK2 JAK2 Tyrosine-protein kinase BMX Cyclin-dependentOMIPALISIB kinase 4/cyclin D1 Myosin IIIA CaM-kinase kinase beta Serine/threonine-protein kinaseU4/U6 PAK small Tankyrase-24 nuclear ribonucleoproteinMitogen-activatedTyrosine-protein Prp4 proteinCitronkinase Rho-interactingkinaseCTK kinase kinase kinase 13 Dual specificityMAP/ tyrosine--regulated affinity-regulating kinase kinase 2 1B cGMP-dependent protein kinaseSerine/threonine-protein 1 betaSerine/threonine-protein kinaseAMP-activated kinaseRho-associated PIM2 Aurora-C Cyclin-dependentproteinCyclin-dependent protein kinase- kinase alpha-1 kinase1kinaseCaM subunit 2 1/cyclin kinase B1I gamma Serine/threonine-proteinSerine/threonine-protein kinase kinase 24 PCTAIRE-3 cAMP-dependent protein kinase alpha-catalytic subunit Serine/threonine-protein kinase 17B Eukaryotic translation initiation factor 2-alpha kinase 4 Serine/threonine-proteinCasein kinase kinase Sgk1 Dual-specificityII Casein kinase tyrosine-phosphorylation I alphaTGF-beta receptor regulated type II kinaseSerine/threonine-protein 3 Dual specificity mitogen-activatedCasein kinase kinase PFTAIRE-1 I isoformprotein kinasealpha-like kinase 3 Ribosomal proteinSerine/threonine-proteinCaM S6 kinase kinase alpha II gamma 5 kinase 17ACyclin-dependentDANUSERTIBEpidermal growth kinase factor 9 receptor Hormonally up-regulated neu tumor-associated kinase Casein kinase I gamma 1 Receptor-typeProtein tyrosine-proteindelta homologSerine/threonine-protein 1 kinaseMitogen-activated FLT3 Interleukin-1 protein kinase kinase PRP4 receptor-associated kinasehomolog kinase 10 kinase 3 gammaTyrosine-protein subunitCyclin-dependent 2 Cyclin-dependent kinaseGCaM protein-coupled kinaseCSK kinase II alpha5 kinase receptor 7/ cyclin kinaseMAP H kinase 5 p38 Myosin light chain kinase- smooth muscle Inhibitor of nuclear factor kappa B kinase betaCyclin-dependent subunit kinaseEukaryotic 2/cyclinSerine/threonine-proteinDual A translationspecificity mitogen-activatedinitation factorkinaseEphrin WNK2 protein type-A kinase receptor kinase; 3 MEK1/2Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha Serine/threonine-proteinInhibitor kinase of nuclear RIPK2 factorG protein-coupled kappa B kinase receptor epsilonMyelin kinase subunit 6MASITINIB factor 1 Myotonin-protein kinase MAP kinase p38 gamma Testis-specificSerine/threonine-proteinDual-specificity serine/threonine-proteinProgrammed tyrosine-phosphorylation cell kinase death proteinEEF2Kkinase 42 regulated kinase 2 Cyclin-dependent kinase 4 Casein kinase I isoform gamma-3PD-0325901 CaM kinaseProtein I delta kinaseCyclin-dependent C alpha kinase 5/CDK5 activatorSerine/threonine-protein 1 kinase 36 Tyrosine-protein kinaseAMP-activated JAK1 INGENOL protein MEBUTATE kinase (AMPK)Cyclin-dependentcAMP-dependent alpha-1/beta-1/gamma-1 proteinkinase 13kinase (PKA) Chaperone activity of bc1 complex-like- mitochondrial Protein kinaseProtein C thetaProtein kinase kinase C delta C gamma Ephrin type-A receptorTyrosine-protein 2 kinase TEC Mitogen-activated protein kinase 4 CaM kinase I alphaSerine/threonine-proteinInhibitor of nuclear kinase factor PRKX kappa B kinase alpha subunit Mitogen-activated protein kinase kinase kinase 9 zeta Muscle- skeletal receptorProtein protein C (PKC) kinase alpha-1Serine/threonine-protein chain kinase PFTAIRE-2 Glycogen synthaseMAP kinase-3 kinase betap38 deltaTyrosine-proteinPhosphorylase kinaseDeath-associated FERkinase gamma protein subunit kinase 1 3 Receptor-interacting serine/threonine-protein kinase 4 Serine/threonine-proteinInsulin-like growth kinaseGlycogen factorTBK1 synthase I receptorMAP kinase-3 kinase-interactingProteinCaM alpha kinase kinaseULK3 II C serine/threonine-proteinkinasebeta kinase MNK1 Serine/threonine-protein kinase TNNI3K Serine/threonine-protein kinase PAK7 LINSITINIB MAP/microtubule affinity-regulating kinase 4 DualSerine/threonine-protein specificity protein kinase kinase CLK2 PIM1 Eukaryotic translationAnkyrin repeat initiation and factor protein 2-alpha kinase kinase domain-containing 1 protein 1 MAP Tyrosine-proteinkinase p38 beta kinase receptorInsulin TYRO3INSULIN receptor HUMAN Serine/threonine-protein kinase PAK 2 Serine/threonine-protein kinase Nek1 3-phosphoinositide dependent proteinProtein kinase-1 tyrosineSerine/threonine-protein kinase 2 beta kinase PAK 1 KW-2449 CaM-kinase kinase alpha Casein kinaseSerine/threonine-protein I PI3-kinase p110-alpha kinase NEK9 Mitogen-activatedsubunitNUAK family SNF1-like proteinEphrin kinase kinase type-AUncharacterized 1 kinase receptor kinase 1 11aarF domain-containing protein kinase 4 Rho-associated proteinTestis-specific kinase 2 serine/threonine-proteinSerine/threonine-protein kinase 1 kinase 11 Serine/threonine-protein kinase PLK3 Serine/threonine-protein kinase AKT2 Homeodomain-interacting protein kinase 1 Homeodomain-interactingMitogen-activated protein protein kinaseLeukocyte kinase3 Serine/threonine-protein kinasetyrosine kinase kinase 7 receptor kinase MRCK-A CaM kinaseRibosomal II delta protein S6 kinase alpha 2 Serine/threonine-protein kinase 38-like Serine/threonine-protein kinase tousled-like 1 MAP kinase-activatedSerine/threonine-protein protein kinase 2 kinase TAO1 Serine/threonine-protein kinase DCLK2 Protein kinase C iota Serine/threonine-proteinMitogen-activated protein kinase kinase RIO2 kinase kinaseCyclin-dependent 15 kinase-like 5 MAP kinase-activatedSerine/threonine-protein protein kinase 5kinase c-TAK1Serine/threonine-proteinSELICICLIB Tyrosine-Protein kinaseand threonine-specifickinase NEK6 C nu cdc2-inhibitorySerine/threonine-proteinSerine/threonine-protein kinase kinase TAO2 kinase ULK3 Activin receptor type-2A Serine/threonine-protein kinase PAK6 Mitogen-activated protein kinase kinaseBone kinase morphogenetic 1 protein receptor type-1A Serine/threonine-protein kinaseTASELISIB SBK1 Transient receptor potential cation channel subfamily M member 6 Protein kinaseCasein C Serine/threonine-proteinkinasemu I gammaRibosomal 2 proteinkinase S6PAK kinase 3 alpha 4 Fibroblast growth factor receptor 4 Phosphatidylinositol-4-phosphateRibosomal protein GALUNISERTIBS6 kinase 1 3-kinase C2 domain-containing beta polypeptide Serine/threonine protein kinasecGMP-dependent NLK protein kinase 2 Serine/threonine-protein kinaseSerine/threonine-protein AKT Casein kinase kinase II DCLK1alpha Mitogen-activated proteinPeripheral kinase kinaseplasma kinase membrane kinaseSerine/threonine-protein protein 4 CASK kinase LATS1 ActivinG protein-coupled receptor type-1BDual receptor specificity kinaseSTE20/SPS1-related testis-specific 7 protein proline-alanine-rich kinaseSerine/threonine-protein 1 proteinSerine/threonine-protein kinase kinase kinase ULK1 Serine/threonine-protein kinase Nek11 Serine/threonine-protein kinase SIK2 Death-associated protein kinaseCasein 2 kinaseTyrosine-protein I delta kinase ZAP-70 Mitogen-activated protein kinase 7 Serine/threonine-proteinEphrinSerine/threonine-protein kinase type-A AKT3 receptor 7 kinase tousled-like 2 SUNITINIBcAMP-dependent protein kinase beta-1 catalytic subunit Tyrosine-protein kinase HCK Serine/threonine-protein kinase Nek5 LIM domain kinase 2 Serine/threonine-proteinInterleukin-1 receptor-associated kinaseCell D2 division kinase control 4 proteinSerine/threonine-protein 2 homolog kinase MRCK gamma CaM kinase IISerine/threonine-protein beta kinase Nek4 Serine/threonine-protein kinase NIM1 Ribosomal protein S6Tyrosine-protein kinase alpha 6 kinase BRKProtein kinase C epsilonSerine/threonine-protein kinase MARK1Phosphatidylinositol-5-phosphate 4-kinase type-2 beta CaMEphrin kinase type-B IVSerine/threonine-protein receptor 1 kinaseWee1-like DCLK3 protein kinase 2 Mitogen-activated protein kinase kinase kinase 5 PI3-kinase p110-betaSerine/threonine-protein subunitSerine/threonine-protein kinase 32Akinase 32C Myosin-IIIB Cyclin-dependent kinase-like 1 Myosin light chain kinase family member 4 VATALANIB BR serine/threonine-proteinMitogen-activatedSerine/threonine-protein protein kinase kinaseSerine/threonine-protein 1 15kinase VRK2 kinase 33 Serine/threonine-protein kinase PIM3 Serine/threonine-proteinSerine/threonine-protein kinase PLK2 kinase MAK Serine/threonine-protein kinase receptor R3 Serine/threonine-protein kinase PCTAIRE-2 Dual specificity mitogen-activated protein kinase kinase 4 Serine/threonine-protein PI3-kinasekinaseSerine/threonine-protein Chk2 p110-delta subunit kinaseDual specificity38 mitogen-activatedSerine/threonine-protein protein kinase kinase 7 kinase LATS2 Ribosomal proteinSerine/threonine-protein S6 kinase alpha 1Serine/threonine--/endoribonuclease IRE1Rhodopsin kinase AMP-activatedPITSLRE protein serine/threonine-protein kinase- alpha-2Serine/threonine-protein subunit kinase CDC2L1 kinase ICK PI3-kinase p110-gamma subunit Microtubule-associated serine/threonine-protein kinase 1 PutativeSNF-related uncharacterized serine/threonine-protein serine/threonine-protein kinase kinaseSerine/threonine-protein SgK110 kinase SIK3 Phosphatidylinositol-4-phosphate 3-kinaseMitogen-activated C2 domain-containing protein subunit kinase gamma kinase kinase 6 Dual specificity mitogen-activatedTGF-beta protein receptorDual kinase serine/threoninetype kinase I 6 and tyrosine protein kinase Protein kinase C eta Mitogen-activated protein kinase 6 SELUMETINIB Phosphatidylinositol-4-phosphateSerine/threonine-protein 5-kinase kinase type-1 Nek3 gamma Serine/threonine-protein kinaseDeath-associated NEK7BR serine/threonine-protein protein kinaseCyclin-dependent 1 kinase 2 kinase 3 PITSLRE serine/threonine-protein kinase CDC2L2 Serine/threonine-protein kinase OSR1 PI4-kinase beta subunit BOSUTINIB CellMAP division kinase cycle ERK1 2-like protein kinase 6 Serine/threonine-protein kinase SRPK2 Serine/threonine-proteinPhosphatidylinositol-5-phosphate kinase Sgk3 4-kinase type-2 gamma

Serine/threonine-proteinCyclin-dependent kinase 35 kinase-like 3

CEDIRANIB

VANDETANIB

ENZASTAURIN GEFITINIB