WO 2019/038250 Al 28 February 2019 (28.02.2019) W P O PCT
(12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (10) International Publication Number (43) International Publication Date WO 2019/038250 Al 28 February 2019 (28.02.2019) W P O PCT (51) International Patent Classification: C07F5/02 (2006.01) A61P 35/00 (2006.01) A61K 31/69 (2006.01) (21) International Application Number: PCT/EP20 18/072485 (22) International Filing Date: 2 1 August 2018 (21.08.2018) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 17187636.0 24 August 2017 (24.08.2017) EP (71) Applicant: MERCK PATENT GMBH [DE/DE] ; Frank¬ furter Strasse 250, 64293 Darmstadt (DE). (72) Inventors: KLEIN, Markus; Lindenweg 35, 64291 DARMSTADT (DE). SCHADT, Oliver; Forststrasse 4, 635 17 RODENBACH (DE). ESDAR, Christina; Am Bre- itwiesenberg 2, 64287 DARMSTADT (DE). (81) Designated States (unless otherwise indicated, for every kind of national protection available) : AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
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