PHARMA PATENTS GRANTED DURING 2010-11 TO 2013-14 ( UP TO 31-7-2013) Application No Date of Filing Patent No Patent Grant Date Title Applicant 1074/MUM/2006 07-07-2006 239822 01-04-2010 A MODIFIED RELEASE PHARMACEUTICAL COMPOSITION PANACEA BIOTEC LIMITED OF BICALUTAMIDE 1115/MUMNP/2007 25-07-2007 238424 02-04-2010 A TRIAZOLO [4,5-d]PYRIMIDINE COMPOUND OF ASTRA ZENECA AB FORMULA (II) 3902/DELNP/2005 01-09-2005 239827 05-04-2010 A GEL FORMULATIONS ANTARES PHARMA IPL AG 359/CAL/1995 31-03-1995 239838 06-04-2010 A 1 H-SUBSTITUTED-INDOLE-3-GLYOXYLAMIDE COMPOUND AND PROCESS OF PREPARATION THEREOF

13/CAL/2000 10-01-2000 239851 06-04-2010 NOVEL BENZOTHIOPHENE COMPOUNDS, ELI LILLY AND COMPANY INTERMEDIATES, COMPOSITIONS AND METHODS THEREOF 3803/DELNP/2005 26-08-2005 239895 07-04-2010 A PHARMACEUTICAL COMPOSITION FOR TREATING OR JARROW FORMULAS, INC. PREVENTING HUMAN IMMUNODEFICIENCY VIRUS (HIV) INFECTION, MALARIA OR BOTH 3702/DELNP/2006 28-06-2006 239909 09-04-2010 FURANCARBONYLGUANIDINE DERIVATIVES, THEIR KOREA RESEARCH INSTITUTE OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS CHEMICAL TECHNOLOGY. CONTAINING THEM 1165/DELNP/2005 23-03-2005 239936 12-04-2010 A PHARMACEUTICAL FORMULATION FOR TREATMENT SHIRE LLC OF PATIENTS HAVING ATTENTION DEFICIT HYPERACTIVITY DISORDER(ADHD) 2221/DELNP/2006 24-04-2006 239954 15-04-2010 NUTRITIONAL COMPOSITION AGAINST SIDE EFECTS OF NESTEC S.A. CHEMOTHERAPY OR RADIOTHERAPY 1053/DELNP/2004 20-04-2004 239997 21-04-2010 A LYOPHILIZED PHARMACEUTICAL COMPOSITION PRODUCTS INC. 5037/DELNP/2005 03-11-2005 240018 23-04-2010 SUBSTITUTED-1-PHTHALAZINAMES AS VR-1 MERCK SHARP & DOHME LIMITED ANTAGONISTS 2695/DEL/2005 07-10-2005 240034 23-04-2010 A PROCESS TO OBTAIN A PHARMACEUTICAL PRODUCT MADAN, DR. ANIL KUMAR WITH AN ENHANCED DISSOLUTION RATE AND THE PHARMACEUTICAL PRODUCT RESULTING THEREOF

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877/MUMNP/2007 11-06-2007 240123 28-04-2010 AN OILY ISOTROPE PHARMACEUTICAL COMPOSITION SA VETOQUINOL

402/DELNP/2006 23-01-2006 240207 29-04-2010 A FLUORO SUBSTITUTED OMEGA-CARBOXYARYL BAYER HEALTHCARE LLC DIPHENYL UREA COMPOUND OR A SALT, AN ISOLATED STEREOISOMER THEREOF

365/DELNP/2005 01-02-2005 240219 29-04-2010 A COMPOUND 2-(3-AMINOARYL) AMINO-4-ARYL- AB SCIENCE THIAZOLES OF FORMULA I. 50/CAL/2001 30-01-2001 240197 29-04-2010 A VACCINE PREPARED FOR THE TREATMENT OR RICAN LIMITED PROPHYLAXIS OF HELICOBACTER PYLORI INFECTION

3435/DELNP/2004 04-11-2004 240229 30-04-2010 A 3, 17-DISUBSTITUTED MORPHINAN COMPOUND AND JENKEN BIOSCIENCES, INC PHARMACEUTICAL COMPOSITION THEREOF 1599/DELNP/2005 20-04-2005 240249 30-04-2010 AN IMIDAZOLE COMPOUND USES AS CARDIOVASCULAR PORTELA & C.A., SA. AGENTS 1516/DELNP/2005 15-04-2005 240264 30-04-2010 AN ANALOGUE OF KAHALALIDE F PHARMA MAR, S.A.U 4540/DELNP/2006 07-08-2006 240268 30-04-2010 NEW AZABICYCLIC COMPOUNDS, A PROCESS FOR THEIR LES LABORATORIES SERVIER PREPARATION AND PHARMACEUTICAL. COMPOSITIONS CONTAINING THEM 927/KOLNP/2006 13-04-2006 240314 04-05-2010 DERIVATIVES OF N-[PHENYL (PYRROLIDINE-2-YL) SANOFI-AVENTIS METHYL ] BENZAMIDE AND N-[ ( AZEPAN-2-YL ) PHENYLMETHYL ] BENZAMIDE, PREPARATION METHOD THEREOF AND APPLICATION OF SAME IN THERAPEUTICS IN/PCT/2002/01272/DEL 20-12-2002 240340 05-05-2010 A COMPOSITION USEFUL AGAINST NEURONAL DAMAGE HUNTER FLEMING LIMITED

30/DELNP/2003 10-01-2003 240341 05-05-2010 A PYRIDOPYRROLOPYRIMIDINE COMPOUND USED AS PHARMA MAR, S.A. ANTITUMOURAL AGENT 1286/DELNP/2005 31-03-2005 240358 05-05-2010 DEVELOPMENT OF NOVEL HEREBAL FORMULATION COUNCIL OF SCIENTIFIC & INDUSTRIAL USED AS AN ANTI-DIABETIC ON TRADITIONAL RESEARCH INDIGENOUS KNOWLEDGE IN/PCT/2001/01142/MUM 19-09-2001 240371 06-05-2010 ANTHELMINTIC COMPOSITIONS ASHMONT HOLDINGS LIMITED 6170/DELNP/2005 30-12-2005 240378 06-05-2010 HYDROXYPYRIDINE CGRP RECEPTOR ANTAGONISTS MERCK AND CO.INC. 4733/DELNP/2005 18-10-2005 240379 06-05-2010 PHARMACEUTICAL FORMULATION OF THE SODIUM BOEHRINGER INGELHEIM SALT OF TELMISARTAN INTERNATIONAL GMBH IN/PCT/2001/00708/DEL 08-08-2001 240383 06-05-2010 A BRANCHED CHAIN AMINO ACID-DEPENDENT WARNER-LAMBERT COMPANY AMINOTRANSFERASE INHIBITORS COMPOUND 779/MUMNP/2006 05-07-2006 240396 07-05-2010 A PHARMACEUTICAL COMPOSITION CONTAINING MERZ PHARMA GMBH & CO. KGAA MEMANTINE FOR THE TREATMENT OF MILD AND MILD- TO-MODERATE ALZHEIMER S DISEASE 1330/DEL/2004 19-07-2004 240422 10-05-2010 A HERBAL COMPOSITION FOR THE TREATMENT OF HIV PANDEY , SANTOSH KUMAR AND A PROCESS OF PREPARING THE SAME 446/KOLNP/2004 02-04-2004 240474 12-05-2010 PHARMACEUTICAL COMPOSITION COMPRISING GAMA- KALVINSH IVARS BUTYROBETAINE 5950/DELNP/2005 20-12-2005 240515 14-05-2010 HETEROARYLOXY NITROGENOUS SATURATED BANYU PHARMACEUTICAL CO.,LTD. HETEROCYCLIC DERIVATIVE 767/DELNP/2006 15-02-2006 240599 19-05-2010 , SPRAY-DRIED AMORPHOUS POWDER BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG. 1903/DELNP/2004 02-07-2004 240690 26-05-2010 COMPOSITION, SYNTHESIS, DIAGNOSTIC AND MICHAEL A. MURPHY  THERAPEUTIC APPLICATIONS OF POLYAMINES 1564/DELNP/2005 19-04-2005 240734 26-05-2010 AN IMMUNOGEN FOR PREPARATION OF THERAPEUTIC INSTITUTE OF IMMUNOLOGY, PLA VACCINES FOR TREATMENT OF HEPATITIS B AND PRODUCING METHOD THEREOF 2657/DELNP/2004 09-09-2004 240755 28-05-2010 PHARMACEUTICAL PREPARATION CONTAINING EURO-CELTIQUE S.A., OXYCODONE AND NALOXONE" 450/DELNP/2005 07-02-2005 240762 28-05-2010 A METALLOPROTEINASE INHIBITOR COMPOUND AND ASTRAZENEECA AB PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 762/DEL/2000 25-08-2000 240763 28-05-2010 AN IMPROVED MALE CONTRACEPTIVE FORMULATION SUJOY KUMAR GUHA

714/MUMNP/2006 19-06-2006 240768 31-05-2010 COMPOSITION AND METHOD FOR REDUCING THE HINDUSTAN UNILEVER LIMITED EFFECTS OF STRESS ON SKIN CONDITION 946/KOLNP/2006 17-04-2006 240787 01-06-2010 DERIVATIVES OF N-[PHENYL(ALKYLPIPERIDINE-2- SANOFI-AVENTIS YL)METHYL]BENZAMIDE 1693/DELNP/2004 15-06-2004 240817 02-06-2010 ISOTRETINOIN NANOPARTICULATE COMPOSITIONS RANBAXY LABORATORIES LIMITED 5582/DELNP/2005 01-12-2005 240818 02-06-2010 A SUBSTITUTED BENZAMIDE COMPOUND AND ASTELLAS PHARMA INC. PHARMACEUTICAL COMPOSITION THEREOF 921/DEL/1998 13-04-1998 240834 03-06-2010 A CELL STRUCTURE MEDIUM COMPOSITION FOR THE BAYER CORPORATION PRODUCTION OF RECOMBINANT FACTOR VIII 4611/DELNP/2005 10-10-2005 240846 04-06-2010 SELECTIVE SPIROCYCLIC GLUCOCORTICOID RECEPTOR MERCK SHARP & DOHME CORP., MODULATORS 640/DELNP/2005 18-02-2005 240871 07-06-2010 COMPOSITION FOR SOLUBILIZATION OF DAEHWA PHARM. CO., LTD. AND PREPARATION METHOD THEREOF IN/PCT/2002/1483/KOL 02-12-2002 240925 10-06-2010 A TOPICAL ORAL COMPOSITION THE PROCTER & GAMBLE COMPANY 2210/CAL/1998 23-12-1998 240930 10-06-2010 PRODRUGS OF ASPARTYL PROTEASE INHIBITORS INCORPORATED 1185/DEL/1999 07-09-1999 240939 10-06-2010 A SPATTER CURE COMPOUND AND A PROCESS FOR THE MADAN MOHAN BANDYOPADHYAY PREPARATION THEREOF FOR USE DURING THE WELDING PROCESS 925/KOLNP/2006 13-04-2006 240989 14-06-2010 N - HETEROCYCLYL - METHYLBENZAMIDE DERIVATIVE SANOFI-AVENTIS COMPOUNDS 3115/DELNP/2005 13-07-2005 240990 14-06-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN ASTRAZENECA AB AROMATASE INHIBITOR,A PROGESTIN AND AN OESTROGEN 461/DELNP/2005 07-02-2005 241002 14-06-2010 COMPOSITION COMPRISING THE EXTRACT OF Helixir Co., Ltd. ACTINIDIA ARGUTA AND RELATED SPECIES FOR THE PREVENTION AND TREATMENT OF ALLERGIC DISEASE AND NON-ALLERGIC INFLAMMATORY DISEASE

5320/DELNP/2005 21-11-2005 241017 15-06-2010 MACROCYCLIC QUINAZOLINE DERIVATIVES AS JANSSEN PHARMACEUTICA N.V. ANTIPROLIFERATIVES AGENTS 228/DELNP/2004 03-02-2004 241018 15-06-2010 NOVEL COMPOUNDS AS ANTI-INFLAMMATORY, 4SC AG Germany IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 250/MUM/2004 01-03-2004 241016 15-06-2010 GASTRIC RETENTION CONTROLLED DRUG DELIVERY SUN PHARMA ADVANCED RESEARCH SYSTEM COMPANY LIMITED 1910/KOLNP/2004 13-12-2004 241066 17-06-2010 COMPOUNDS AS MODULATORS OF STEROID ELI LILLY AND COMPANY HORMONE NUCLEAR RECEPTORS 1077/MUMNP/2005 03-10-2005 241110 17-06-2010 POLYMERIC OLIGONUCLEOTIDE PRODRUGS ENZON PHARMACEUTICALS, INC. 207/CAL/1998 09-02-1998 241050 17-06-2010 PEPTIDES FOR DIAGNOSING AND TREATMENT OF GERHILD WILDNER AUTOIMMUNE DISEASES IN/PCT/2003/00001/DEL 01-01-2003 241117 18-06-2010 TOPICAL LIPOSOMAL FORMULATION COMPRISING CENTRO DE INVESTIGACIÓN Y CLOBETASOL PROPIONATE ENCAPSULATED IN DESARROLLO DE MEDICAMENTOS LIPOSOMES (CIDEM) 1210/DEL/2004 30-06-2004 241119 18-06-2010 A NOVEL COBALT COMPLEX USEFUL FOR REVERSAL OF INDIAN COUNCIL OF MEDICAL DRUG RESISTANCE AND THE PREPARATION THEREOF RESEARCH

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529/MUMNP/2006 09-05-2006 241597 14-07-2010 METHOXY PHOSPHONATE NUCLEOTIDE PRODRUG , INC. 1243/MUM/2005 03-10-2005 241583 14-07-2010 A HERBAL PAIN- RELIEF COMPOSITION PHARMACON REMEDIES [BOMBAY] PVT. LTD., 1610/DELNP/2005 20-04-2005 241646 17-07-2010 A BIOADHESIVE PHARMACEUTICAL COMPOSITION COLUMBIA LABORATORIES (BERMUDA) COMPRISING AN IONIC TREATING AGENT AND AN IONIC LIMITED POLYMER POLYCARBOPHIL IN/PCT/1999/00001/DEL 07-12-1999 241656 19-07-2010 PYRIMIDINONE COMPOUNDS AND PROCESS FOR BORYUNG PHARMACEUTICAL CO. LTD., PREPARING THE SAME 215/DELNP/2006 12-01-2006 241658 19-07-2010 INFANT OR FOLLOW-ON FORMULA NESTEC S.A. 1649/DELNP/2006 27-03-2006 241659 19-07-2010 A COMBINATION COMPRISING CANDESARTAN OR A ASTRAZENECA UK LIMITED. PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 3409/DELNP/2005 01-08-2005 241660 19-07-2010 PHARMACEUTICAL LIQUID FORMULATION ARAKIS LTD 1960/DELNP/2004 08-07-2004 241677 20-07-2010 A PHARMACEUTICAL COMPOSITION COMPRISING A NERVIANO MEDICAL SCIENCES S.R.L. PHARMACEUTICALLY ACCEPTABLE CARRIER OR EXCIPIENT AND, AS ACTIVE INGREDIENT, AN ACRYLOYL DISTAMYCIN DERIVATIVE 2258/DELNP/2006 24-04-2006 241685 20-07-2010 A COMPOSITION LI, GUOQIAO 769/DELNP/2006 15-02-2006 241721 22-07-2010 ANTIMICROBIAL COMPOSITIONS CONTAINING THE TRUSTEES OF COLUMBIA SYNERGISTIC COMBINATIONS OF QUATERNARY UNIVERSITY IN THE CITY OF NEW YORK AMMONIUM COMPOUNDS AND ESSENTIAL OILS AND/OR CONSTITUENTS THEREOF 1415/MUMNP/2005 20-12-2005 241735 22-07-2010 AN ISOLATED ANTIBODY BAYER SCHERING PHARMA AKTIENGESELLSCHAFT IN/PCT/2002/00588/DEL 10-06-2002 241773 24-07-2010 PYRROLO[2,3-d] PYRIMIDINE COMPOUNDS PFIZER PRODUCTS INC. 2090/DEL/1998 20-07-1998 241782 24-07-2010 A PHARMACEUTICAL COMPOSITION COMPRISING 5-[4- SMITHKLINE BEECHAM P.L.C [2(N-METHYL-N-(2-PYRIDYL)AMINO] ETHOXY]BENZYL]THIAZOLIDINE-2,4-DIONE 128/DELNP/2004 19-01-2004 241823 27-07-2010 A PROLONGED RELEASE MUCOADHESIVE TABLET BIOALLIANCE PHARMA 2226/DEL/2004 08-11-2004 241827 27-07-2010 A COMPOSITION FOR ENHANCING BIOAVAILABILITY OF COUNCIL OF SCIENTIFIC AND DRUGS/NUTRACEUTICALS. INDUSTRIAL RESEARCH 708/CHENP/2004 05-04-2004 241838 28-07-2010 AN ANGIOTENSIN PEPTIDE MOIETY-CARRIER CYTOS BIOTECHNOLOGY AG CONJUGATE. 462/KOLNP/2005 18-03-2005 241844 28-07-2010 9, 10-DEHYDRO-DESOXY-EPOTHILONE COMPOUNDS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH 5943/DELNP/2005 20-12-2005 241905 30-07-2010 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP., 2868/CHENP/2004 16-12-2004 241952 02-08-2010 A COMPOSITION FOR ENHANCING IMMUNE RESPONSE CYTOS BIOTECHNOLOGY AG

1683/MUMNP/2007 15-10-2007 241989 04-08-2010 TABLET- TYPE CONTROLLED-RELEASE PREPARATION HENNIG ARZNEIMITTEL GMBH & CO. CONTAINING CINNARIZINE AND DIMENHYDRINATE FOR KG COMBATING VERTIGO 1278/DELNP/2005 31-03-2005 241999 05-08-2010 SUBSTITUTED CARBAMIC ACID QUINOLIN-6-YL ESTERS COUNCIL OF SCIENTIFIC & INDUSTRIAL AS ACETYLCHOLINESTERASE INHIBITORS RESEARCH 3331/DELNP/2006 09-06-2006 242015 06-08-2010 A 2-QUINOLINONE OR 2-QUINOXALINONE COMPOUND JANSSEN PHARMACEUTICA N.V.

5565/DELNP/2006 25-09-2006 242021 06-08-2010 THE COMPOUNDS 2-[(2-FLUORO-6- PFIZER INC METHOXZYPHENOXY)(3-FLUOROPHENYL) METHYL]MORPHOLINE AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF 1182/DELNP/2005 24-03-2005 242025 06-08-2010 AN OCULAR TREATMENT SOLUTION FOR THE JIN JUN ZHANG TREATMENT OR PREVENTION OF POSTERIOR CAPSULAR OPACIFICATION 2630/DELNP/2004 08-09-2004 242026 06-08-2010 A QUINAZOLINE DERIVATIVE ASTRAZENECA AB 471/CHENP/2006 06-02-2006 242036 06-08-2010 METHODS AND COMPOSITIONS FOR CANCER THERAPY HENRY FORD HEALTH SYSTEM USING NOVEL ADENOVIRUS 53/DEL/2004 12-01-2004 242024 06-08-2010 A PHARMACEUTICAL PREPARATION FOR THE EURO-CELTIQUE S.A., PREVENTION OR THE TREATMENT OF INFECTIONS IN THE INTERIOR OF THE HUMAN OR ANIMAL BODY

4759/DELNP/2005 19-10-2005 242056 09-08-2010 PHARMACEUTICAL COMPOSITION FOR A MERCK SHARP & DOHME CORP., ATHEROSCLEROSIS,DYSLIPIDEMIAS AND RELATED CONDITIONS 1265/DELNP/2006 08-03-2006 242095 11-08-2010 AN ORAL COMPOSITION OF ITRACONAZOLE HAVING HANMI PHARM.CO. LTD. IMPROVED ITRACONAZOLE BIOAVAILABILITY

413/MUM/2003 25-04-2003 242111 11-08-2010 CRYSTALLINE CLOPIDOGREL BESYLATE AND PROCESS CADILA HEALTHCARE LIMITED FOR PREPARATION THEREOF 489/DEL/2001 16-04-2001 242113 11-08-2010 A RUMEN BYPASS COMPOSITION CONTAINING A JUBILANT ORGANOSYS LIMITED BIOACTIVE SUBSTANCE 2472/DELNP/2005 08-06-2005 242134 16-08-2010 THE COMPOUND (-) TENATOPRAZOLE, OR (-)-5- SIDEM PHARMA SA METHOXY -2[[(4-METHOXY-3,5-DIMETHYL-2- PYRIDYL)METHYL]SULFINYL]IMIDAZO-[4,5-B]PYRIDINE

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991/DEL/2003 12-08-2003 242180 18-08-2010 A COMPOSITION USEFUL FOR THE TREATMENT OF COUNCIL OF SCIENTIFIC AND LEISHMANIASIS INDUSTRIAL RESEARCH 3296/DELNP/2006 08-06-2006 242247 19-08-2010 AMINOBENZIMIDAZOLES AND BENZIMIDAZOLES AS TIBOTEC PHARMACEUTICALS LTD. INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION 1855/KOLNP/2006 04-07-2006 242344 24-08-2010 INHIBITOR OF PROTEIN MODIFICATION PRODUCTS TOKAI UNIVERSITY EDUCATIONAL FORMATION SYSTEM 1702/KOLNP/2006 20-06-2006 242347 24-08-2010 NOVEL COMBINATION OF ANTICHOLINERGIC AND beta MEDA PHARMA GMBH & CO. KG MIMETICS FOR THE TREATMENT OF RESPIRATORY DISEASES 4232/KOLNP/2007 05-11-2007 242351 24-08-2010 COMPOUND USEFUL AS AMPA RECEPTOR ELI LILLY AND COMPANY POTENTIATORS 3811/KOLNP/2007 08-10-2007 242352 24-08-2010 PHARMACEUTICAL COMPOSITION AND METHOD USING TOYAMA CHEMICAL CO., LTD. ANTIFUNGAL AGENT IN COMBINATION 2071/KOLNP/2006 24-07-2006 242354 24-08-2010 PHARMACEUTICAL COMPOSITION FOR PROMOTING OTSUKA PHARMACEUTICAL ANGIOGENESIS. CO. LTD 4484/KOLNP/2007 21-11-2007 242367 24-08-2010 A PHARMACEUTICAL COMPOSITION ADVANCED SCIENTIFIC DEVELOPMENTS

135/DEL/2003 18-02-2003 242387 25-08-2010 HERBAL HEALTH PROTECTIVE AND PROMOTIVE COUNCIL OF SCIENTIFIC AND NUTRACEUTICAL FORMULATION FOR DIABETICS AND INDUSTRIAL RESEARCH PROCESS FOR PREPARING THE SAME 327/DEL/2000 28-03-2000 242390 25-08-2010 NOVEL α-HYDROXY-9, 12-TRICOSDIENOIC ACID COUNCIL OF SCIENTIFIC AND USEFUL AS THERAPEUTIC AGENT INDUSTRIAL RESEARCH 3140/DELNP/2006 01-06-2006 242466 27-08-2010 MORPHOLINYL CONTAINING BENZIMIDAZOLES AS TIBOTEC PHARMACEUTICALS LTD. INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION 6010/DELNP/2005 22-12-2005 242467 27-08-2010 A COMPOSITION FOR THE BETTER TREATMENT OF INDENA S.P.A. RHEUMATOID ARTHRITIS 403/CHENP/2004 27-02-2004 242497 30-08-2010 PHARMACEUTICAL COMPOSITION COMPRISING NOVARTIS AG LUMIRACOXIB 2991/DELNP/2005 05-07-2005 242504 30-08-2010 A COMPOSITIONS FOR INTRANASAL DELIVERY OF ARCHIMEDES DEVELOPMENT LIMITED FENTANYL 2785/KOLNP/2006 25-09-2006 242537 31-08-2010 BENZIMIDAZOLE DERIVATIVE AND A PROCESS FOR THE TAKEDA PHARMACEUTICAL COMPANY PREPARATION THEREOF LIMITED 849/KOLNP/2007 09-03-2007 242552 01-09-2010 SULPHONAMIDE DERIVATIVES, THE PREPARATION LABORATORIOS DEL DR. ESTEVE, S.A. THEREOF AND THE APPLICATION OF SAME AS MEDICAMENTS 2628/DELNP/2006 10-05-2006 242729 07-09-2010 AN OIL-BASED FORMULATION FOR NASAL APPLICATION MATTERN UDO

2159/MUM/2006 29-12-2006 242722 07-09-2010 A COMPOSITION FOR BODY WEIGHT LOSS Dr. Kishori Ganpat Apte 3415/DELNP/2004 03-11-2004 242804 14-09-2010 MODIFIED RELEASE PHARMACEUTICAL FORMULATION ASTRAZENECA AB

258/DELNP/2005 24-01-2005 242831 15-09-2010 AN ANTI-MICROBIAL COMPOSITION THE QUIGLEY CORPORATION 1449/MUM/2005 21-11-2005 242838 15-09-2010 COMPOSITION FOR ENHANCING ANTIBACTERIAL ADVANCED ENZYME TECHNOLOGIES ACTIVITY OF ANTIBACTERIAL AGENTS LIMITED 24/DELNP/2005 04-01-2005 242889 17-09-2010 COMPOUNDS HAVING ANTI-PARASITIC,IN PARTICULAR CENTRE NATIONAL DE LA RECHERCHE ANTIMALARIAL ATIVITY AND COMPOSITIONS THEREOF SCIENTIFIQUE (CNRS)

39/DELNP/2005 05-01-2005 242893 17-09-2010 A SUSTAINED-RELEASE PHARMACEUTICAL PHARMACIA CORPORATION, COMPOSITION 2266/DELNP/2004 04-08-2004 242898 17-09-2010 A PHARMACEUTICAL COMPOSITION COMPRISING 4-(3'- ASTRAZENECA AB, CHLORO-4'-FLUOROANILINO)-7- METHOXY-6-(3- MORPHOLINOPROPOXY) QUINAZOLINE OR A PHARMACEUTICALLY-ACCEPTABLE SALT THEREOF 3455/DELNP/2004 05-11-2004 242901 17-09-2010 A COMPOUND FOR COMBATING URINARY TRACT MOUNT COOK BIOSCIENCES  DYSFUNCTION AND A FORMULATION THEREOF INC.  43/DELNP/2005 05-01-2005 242902 17-09-2010 A SUSTAINED-RELEASE PHARMACEUTICAL PHARMACIA CORPORATION COMPOSITION 5590/DELNP/2005 01-12-2005 242904 17-09-2010 3-DEMETHYL-AND 3-DEMETHYLTHIO-COLLCHICHINE INDENA S.P.A. DERIVATIVES 1613/DELNP/2003 07-10-2003 242910 18-09-2010 A PHARMACEUTICAL COMPOSITION FOR THE HF ARZNEIMITTELFORSCHUNG GMBH TREATMENT OF COGNITIVE DISTURBANCES OCCURRING AS SEQUELAE 4138/DELNP/2004 27-12-2004 242912 18-09-2010 AN ORALLY DELIVERABLE PHARMACEUTICAL PHARMACIA CORPORATION COMPOSITION 1114/DELNP/2005 21-03-2005 242928 20-09-2010 A PHARMACEUTICAL COMPOSITION FOR PREPARING A IDEC MA INC., MEDICAMENT FOR THE TREATMENT OF CHRONIC DEMYELINATING MOTOR NEUROPATHY

2015/DELNP/2006 12-04-2006 242935 20-09-2010 IMPLANTS WITH ATTACHED SILYLATED THERAPEUTIC SMART TECH LP., AGENTS 382/DELNP/2005 02-02-2005 242939 21-09-2010 A COMPOUND 1-(4-BENZOYLPIPERAZIN-1-YL)-2-(4- BRISTOL-MYERS SQUIBB COMPANY FLUORO-7-(1 H-1,2,3-TRIAZOL-1-YL)-1H-PYRROLO[2,3- YL)ETHANE-1,2-DIONE OF FORMULA (A)

416/DELNP/2005 03-02-2005 242987 23-09-2010 ANTIBODIES AND IMMUNOCONJUGATES BINDING TO BOARD OF REGENTS, THE UNIVERSITY AMINOPHOSPHOLIPIDS AND THEIR USE IN TREATING OF TEXAS SYSTEM VIRAL INFECTIONS 865/DELNP/2005 04-03-2005 243032 24-09-2010 NOVEL COMPOUND, A COMPSITION COMPRISING SUCH GALDERMA RESEARCH & NOVEL COMPOUND AND A PROCESS THEREOF" DEVELOPMENT, S.N.C.,

2728/CHENP/2006 24-07-2006 243035 24-09-2010 ANALOGS OF BENZOQUINONE-CONTAINING INFINITY DISCOVERY INC ANSAMYCINS FOR THE TREATMENT OF CANCER 1669/DELNP/2005 25-04-2005 243061 27-09-2010 A DIRECTLY TABLETABLE GASTRORESISTANT SPHEROID ETHYPHARM AND METHOD FOR PREPARING THE SAME

1310/DELNP/2005 01-04-2005 243091 27-09-2010 CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITOR NEURO3D COMPOUNDS 555/DELNP/2005 14-02-2005 243249 30-09-2010 LIQUID FORMULATIONS FOR MUCOSAL GW PAHRMA LIMITED ADMINISTRATION 3243/DELNP/2006 06-06-2006 243281 01-10-2010 N-ARYL PIPERIDINE SUBSTITUTED JANSSEN PHARMACEUTICA N.V. BIPHENYLCARBOXAMIDES AS INHIBITORS OF APOLIPOPROTE IN B 1045/KOLNP/2005 01-06-2005 243339 06-10-2010 NEW BIOREVERSIBLE ESTER PRODRUG AND ORION CORPORATION PHARMACEUTICAL COMPOSITON CONTAINING THE SAME 2241/DELNP/2003 22-12-2003 243378 08-10-2010 A DISPIRO 1,2,4,-TRIOXOLANE MEDICINES FOR MALARIA VENTURE 2219/DELNP/2005 25-05-2005 243438 18-10-2010 A COMPOSITION FOR TREATING PULMONARY TRANSAVE, INC. INFECTION IN A PATIENT 1482/DELNP/2005 13-04-2005 243445 19-10-2010 LACTOFERRIN COMPOSITIONS AGENNIX INCORPORATED IN/PCT/2002/00248/DEL 28-02-2002 243451 19-10-2010 A PHARMACEUTICAL COMPOSITION (MEDICAMENT) SCHERING AKTIENGESELLSCHAFT

1572/DELNP/2005 19-04-2005 243463 19-10-2010 A FORMULATION THAT PROVIDES COLLEGIUM PHARMACEUTICAL, INC PULSATILE RELEASE OF MILNACIPRAN IN/PCT/2001/01164/DEL 18-12-2001 243473 20-10-2010 ANESTHETIC COMPOSITION FOR INTRAVENOUS KUHNIL PHARM CO., LTD. INJECTION COMPRISING PROPOFOL 1709/DELNP/2003 20-10-2003 243499 21-10-2010 A PIPERIDINYL BENZOXAZOLONE COMPOUND OF EURO-CELTIQUE, S.A FORMULA I 267/DELNP/2005 24-01-2005 243502 21-10-2010 4-(SUBSTITUTED ARYL)-5-HYDROXYISOQUINOLINONE KYORIN PHARMACEUTICAL CO.,LTD DERIVATIVE 1680/DELNP/2003 16-10-2003 243508 21-10-2010 SPIROPYRAZOLE COMPOUNDS EXHIBITING AFFINITY EURO-CELTIQUE, S.A FOR THE OPIOID RECEPTOR-LIKE (ORLI) RECEPTOR 3854/DELNP/2004 06-12-2004 243509 21-10-2010 A BIFUNCTIONAL COMPOUND COMPRISING A PROTEIN DUOTOL AB CONJUGATED WITH AN IMMUNOMODULATING NUCLEIE ACID 2958/DELNP/2004 29-09-2004 243516 21-10-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN PFIZER INC EP4 RECEPTOR ANTAGONIST 890/DELNP/2007 02-02-2007 243571 26-10-2010 AMINOPYRIDINE COMPOUNDS AS PROTEIN KINASE PFIZER INC. INHIBITORS FOR THE TREATMENT OF CANCER

153/DEL/2004 30-01-2004 243559 26-10-2010 A NOVEL COMBINATORIAL LIBRARY OF 3 AND 30- COUNCIL OF SCIENTIFIC AND SUBSTITUTED LUP-20(29)- ENE DERIVATIVES USEFUL AS INDUSTRIAL RESEARCH ANTI-MALARIAL AGENTS IN/PCT/2002/00150/DEL 04-02-2002 243610 27-10-2010 AN AQUEOUS COMPOSITION COLGATE-PALMOLIVE COMPANY 47/DEL/2000 21-01-2000 243577 27-10-2010 A THERAPEUTIC COMPOSITION FOR PANACEA BIOTEC LIMITED TOPICAL/TRANSDERMAL USE AND A PROCESS FOR PREPARATION THEREOF 1299/DEL/1999 28-09-1999 243594 27-10-2010 CONTROLLED RELEASE COMPOSITION COMPRISING PANACEA BIOTEC LIMITED NIMESULIDE 567/CHE/2004 17-06-2004 243595 27-10-2010 NOVEL INTERMEDIATE FOR THE PRERPARATION OF ORCHID CHEMICALS & CEFOTIAM PHARMACEUTICALS LTD IN/PCT/2000/207/KOL 10-08-2000 243613 28-10-2010 A CYCLOALKENE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED 648/DELNP/2003 29-04-2003 243648 28-10-2010 A SOLID ORAL CONTROLLED-RELEASE COMPOSITION EURO-CELTIQUE S.A.

1113/DELNP/2006 02-03-2006 243668 29-10-2010 AMIDOMETHYL- SUBSTITUTED 1-(CARBOXYALKYL)- SOLVAY PHARMACEUTICALS GMBH CYCLOPENTYLCARBONYLAMINO-BENZAZEPINE-N- ACETIC ACID COMPOUNDS OF THE GENERAL FORMULA 1, ITS COMPOSITION AND PROCESS FOR PREPARING THE SAME 02196/DELNP/2003 16-12-2003 243687 29-10-2010 VITAMIN D ANALOGUES AND COMPOSITION GALDERMA RESEARCH & CONTAINING THE SAME DEVELOPMENT S.N.C 5192/DELNP/2006 11-09-2006 243714 02-11-2010 CONTROLLED-RELEASE PHARMACEUTICAL EISAI R & D MANAGEMENT CO.  COMPOSITION AND METHOD FOR PRODUCING THE LTD. SAME 1778/DELNP/2004 22-06-2004 243759 03-11-2010 QUICK RELEASE FLUDARA TABLET COMPOSITION ALCAFLEU MANAGEMENT GMBH & CO. KG, 2054/DELNP/2003 02-12-2003 243790 08-11-2010 TOPICAL APPLICATION OF THIAZOLYLAMIDES AICURIS GMBH & CO.KG 118/DELNP/2005 13-01-2005 243791 08-11-2010 MULTI-COMPONENT PHARMACEUTICAL CAPSULE FOR GLAXO GROUP LIMITED RETAINING DRUG SUBSTANCE IN/PCT/2002/01271/DEL 20-12-2002 243802 08-11-2010 A COMPOSITION USEFUL FOR PROTECTING AGAINST HUNTER-FLEMING LIMITED ACUTE OR CHRONIC NEURONAL DAMAGE 1133/DELNP/2005 22-03-2005 243822 09-11-2010 A THERAPEUTIC COMPOSITION FOR THE TREATMENT STEROGENE BIOSEPARATIONS, INC., OF CANCER 3875/DELNP/2006 05-07-2006 243848 09-11-2010 FORMULATION FOR TREATING OBESITY AND SCANDINAVIAN CLINICAL NUTRITION I ASSOCIATED METABOLIC SYNDROME SVERIGE AB  922/MUM/2006 13-06-2006 243835 09-11-2010 HERBAL COMPOSITION FOR RELIEVING PAIN FROM BABULAL BHAWARLAL JAIN JOINTS AND BONES AND METHOD THEREOF 1326/DELNP/2005 01-04-2005 243859 10-11-2010 PHARAMACEUTICAL COMPOSITION COMPRISING HANMI PHARM CO., LTD CRYSTALLINE SIBUTRAMINE METHANESUFONATE HEMIHYDRATE 253/DELNP/2005 24-01-2005 243870 10-11-2010 PYRIMIDYL SULPHONE AMIDE DERIVATIVES AS ASTRAZENECA AB CHEMOKINE RECEPTOR MODULATORS 2174/DELNP/2005 24-05-2005 243874 10-11-2010 PULVERULENT FORMULATION FOR INHALATION BOEHRINGER INGELHEIM PHARMA CONTAINING TIOTROPIUM GMBH & CO. KG 1485/DELNP/2005 13-04-2005 243878 10-11-2010 A METHOD FOR MANUFACTURING MEDICAMENT AND INSTITUT PASTEUR AND INSTITUT A MEDICAMENT THEREOF NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE IN/PCT/2002/00758/DEL 02-08-2002 243881 10-11-2010 CONDENSATION DERIVATIVES OF THICOLCHICINE AND INDENA S.P.A. BACCATIN AS ANTITUMOR AGENTS 746/DELNP/2004 23-03-2004 243912 10-11-2010 A PHARMACEUTICAL COMPOSITION FOR ORAL APOGEPHA ARZNEIMITTEL GMBH ADMINISTRATION 308/DELNP/2005 27-01-2005 243913 10-11-2010 NOVEL BENZOIMIDAZOLE DERIVATIVES USEFUL AS PFIZER PRODUCTS INC. ANTIPROLIFERATIVE AGENTS" 90/MUM/2005 28-01-2005 243858 10-11-2010 SYNERGISTIC INJECTABLE COMBINATION OF SANJEEV KHANDELWAL ANTISPASMODIC AND ANTIPYRETIC - ANALGESIC IN/PCT/2002/00438/DEL 29-04-2002 243922 11-11-2010 A SOLID ORAL CONTROLLED RELEASED COMPOSITION EURO-CELTIQUE S.A.

301/DELNP/2005 27-01-2005 243930 11-11-2010 ECHINACEA ANGUSTIFOLIA ROOT EXTRACT INDENA S.P.A COMPOSITION AND PROCESS FOR PREPARATION THEREOF 182/DELNP/2005 18-01-2005 243957 11-11-2010 A 1H-IMIDAZO[4,5-C] QUINOLINE 4-PHTHALIMIDE TEVA PHARMACEUTICAL WORKS COMPOUND OF FORMULA (II) AND PROCESS FOR PRIVATE LIMITED COMPANY PREPARING THE SAME 1268/DEL/2002 17-12-2002 243921 11-11-2010 A MEDICINAL COMPOSITION FOR TREATMENT OF SANDEEP SINGH HYPOXIA 51/DEL/2001 22-01-2001 243924 11-11-2010 THERAPEUTIC COMPOSITION CONTAINING NIMESULIDE PANACEA BIOTEC LIMITED AND PROCESS FOR THEIR PREPARATION

542/DEL/2004 22-03-2004 243944 11-11-2010 A MEDICINAL COMPOSTION USEFUL IN TREATMENT OF BANARSI LAL DUA HIV/AIDS 696/DEL/2004 12-04-2004 243949 11-11-2010 DIMMER OF PHENAZINE-1-CARBOXYLIC ACID AND TO DEPARTMENT OF BIOTECHNOLOGY, THE PROCESS OF PREPARATION THEREOF 577/DELNP/2003 16-04-2003 243972 12-11-2010 PHARMACEUTICAL COMPOSITION COMPRISING AKL TECHNOLOGIES LIMITED GINKGOLIDE AND APOCYNIN 29/DELNP/2003 08-01-2003 243999 15-11-2010 BRANCHED-CHAIN LIPOPHILIC COMPOUND, D-PHARM LTD. PHARMACEUTICAL COMPOSITION AND USES THEREOF

994/DELNP/2005 15-03-2005 244000 15-11-2010 INHALATION COMPOSITIONS WITH HIGH DRUG RATIOS NORTON HEALTHCARE LTD.

996/DELNP/2005 15-03-2005 244005 15-11-2010 INHALATION COMPOSITION NORTON HEALTHCARE LTD 816/DEL/2004 30-04-2004 244027 15-11-2010 A SYNERGISTIC HERBAL COMPOSITION FOR THE PRASAD VAIDYA BANKE TREATMENT OF ANIMAL BITE ESPECIALLY SNAKE BITE AND EARLY STAGES OF HYDROPHOBIA. 582/DEL/2003 08-04-2003 244034 15-11-2010 A HERBAL COMPOSITION AGAINST BRONCHIAL THE DIRECTOR, CENTRAL COUNCIL FOR ASTHMA AND PROCESS FOR PREPARATION THEREOF RESEARCH IN UNANI MEDICINE

1611/DELNP/2003 07-10-2003 244074 16-11-2010 A PHARMACEUTICAL COMPOSITION FOR THE HF ARZNEIMITTELFORSCHUNG GMBH TREATMENT OF DEFUNCTIONALIZATION MANIFESTATIONS OR CHRONIC PSYCHIARTIC SYMPTOMS 313/DELNP/2005 27-01-2005 244095 18-11-2010 BENZIMIDAZOL COMPOUNS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG., 998/DELNP/2006 24-02-2006 244106 18-11-2010 PIPERIDINE COMPOUNDS EURO-CELTIQUE S. A. 601/MUMNP/2005 13-06-2005 244113 18-11-2010 BENZOYLGUANIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG 796/DEL/2003 11-06-2003 244158 22-11-2010 A FORMULATION FOR DELIVERY OF BIOACTIVE AGENT NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) 1832/DELNP/2003 06-11-2003 244188 23-11-2010 QUICK-DISINTEGRATING TABLET IN THE BUCCAL CAVITY ASTELLAS PHARMA INC. AND MANUFACTURING METHOD THEREOF 460/DELNP/2005 07-02-2005 244195 23-11-2010 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING CJ CORPORATION THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME 2297/DELNP/2003 31-12-2003 244197 23-11-2010 A COMPOSITION FOR PHARMACOLOGICAL THERAPY OF HF ARZNEIMITTELFORSCHUNG GMBH DEPENDENCE 475/DEL/1997 25-02-1997 244182 23-11-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN PFIZER INC. ESTROGEN AGONIST/ANTAGONIST 5114/DELNP/2006 05-09-2006 244217 24-11-2010 A POWDERY COMPOSITION COMPRISING A STEROIDAL BAYER SCHERING PHARMA MOLECULE AND A PHARMACEUTICALLY ACCEPTABLE AKTIENGESELLSCHAFT CARRIER 2530/KOLNP/2006 04-09-2006 244233 25-11-2010 DIPEPTIDYL PEPTIDASE INHBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED 855/MUM/2007 03-05-2007 244264 26-11-2010 POTENTIZED FORMULATION OF ANALOG RAJESH SHAH

37/DEL/2004 08-01-2004 244306 30-11-2010 4-ARYL-2,6-DIMETHYL-3, 5-DICARBOETHOXY-1, 4- COUNCIL OF SCIENTIFIC AND DIHYDROPYRIDINES AND CORRESPONDING HYDROXY INDUSTRIAL RESEARCH DERIVATIVES 2439/KOLNP/2006 28-08-2006 244339 01-12-2010 A THIAZOLE DERIVATIVE TAISHO PHARMACEUTICAL CO. LTD IN/PCT/2001/01189/DEL 20-12-2001 244342 01-12-2010 OPTICALLY ACTIVE QUINOLINE CARBOXYLIC ACID EU Biotech Development Ltd. DERIVATIVES 823/CAL/1999 05-10-1999 244355 02-12-2010 A POLYPHARMACEUTICAL COMPOSITION FOR THE MR. ABDUL MUEED TREATMENT OF HYPERTENSION 1623/DELNP/2005 21-04-2005 244379 06-12-2010 SUSTAINED RELEASE COMPOSITION FOR ORAL HANMI PHARM. CO., LTD. ADMINISTRATION OF DRUGS 1434/DELNP/2005 08-04-2005 244381 06-12-2010 MICROSPHERE FOR CONTROLLED RELEASE OF TIANJIN TASLY GROUP CO., LTD. TEMOZOLOMIDE AND MEHTOD FOR PREPARATION THEREOF 225/MUMNP/2006 24-02-2006 244464 07-12-2010 STERILE PREPARATIONS OF PHOSPHOLIPIDS AND ANTI- The Board of Regents of the University INFLAMMATORY PHARMACEUTICALS AND METHODS of Texas System FOR MAKING AND USING SAME 693/MUMNP/2006 13-06-2006 244465 07-12-2010 OXAZOLIDINONE-QUINOLONE HYBRID ANTIBIOTICS MORPHOCHEM AKTIENGESELLSCHAFT FUR KOMBINATORISCHE CHEMIE.

557/MUM/2004 14-05-2004 244433 07-12-2010 A CONTROLLED RELEASE DELIVERY COMPOSITION OF CADILA HEALTHCARE LIMITED METFORMIN 7293/DELNP/2006 04-12-2006 244472 08-12-2010 PHARMACEUTICAL COMPOSITION OF CORTICOSTEROID ALMIRALL  S.A. AND ANTAAGONIST OF M3 MUSCARINIC RECEPTORS FOR USE IN THE RESPIRATORY DISORDERS 3668/DELNP/2005 18-08-2005 244474 08-12-2010 A NOVEL (E)-4-CARBOXYSTYRYL-4-CHLOROBENZYL TEMPLE UNIVERSITY - OF THE SULFONE COMPOUND COMMONWEALTH SYSTEM OF HIGHER EDUCATION 1682/MUMNP/2007 15-10-2007 244488 08-12-2010 PELLET- TYPE CONTROLLED- RELEASE PREPARATION HENNIG ARZNEIMITTEL GMBH & CO. CONTAINING CINNARIZINE AND DIMENHYDRINATE FOR KG. COMBATING VERTIGO 579/MUM/2003 06-06-2003 244479 08-12-2010 AN IMMEDIATE RELEASE FORMULATION OF CADILA HEALTHCARE LIMITED FLUVASTATIN 22/MUM/2004 09-01-2004 244489 08-12-2010 NOVEL SUBSTITUTED HYDROXAMIC ACID DERIVATIVES CADILA HEALTHCARE LIMITED

5050/DELNP/2006 01-09-2006 244519 09-12-2010 A SYNERGISTIC COMPOSITION FOR REGULATING THE GIULIANI S.P.A. TROPHISM OF FOLLICLES AND OPTIONALLY THE SKIN PRODUCTION OF SEBUM 3467/DELNP/2006 16-06-2006 244529 09-12-2010 3-CYANO-QUINOLINE COMPOUNDS AS KINASE JANSSEN PHARMACEUTICA N.V. INHIBITORS, PHARMACEUTICAL COMPOSITION THEREOF AND PROCESS FOR PREPARATION 1449/CAL/1997 05-08-1997 244524 09-12-2010 PHARMACEUTICAL COMPOSITION CONTAINING 4- MERCK PATENT GESELLSCHAFT MIT OXOBUTANOIC ACIDS RESCHRANKTER HAFTUNG 1476/DELNP/2005 13-04-2005 244563 10-12-2010 A NON-EFFERVESCENT TABLET FORMULATION FOR BAYER CONSUMER CARE AG ORAL ADMINISTRATION OF SODIUM IBUPROFEN 894/MUM/2007 10-05-2007 244558 10-12-2010 HOMEOPATHY BASED FORMULATION FOR TREATMENT RAJESH SHAH OF LICHEN PLANUS 3719/DELNP/2004 24-11-2004 244635 13-12-2010 A DUAL COMPONENT ANTIPLAQUE ORAL COLGATE-PALMOLIVE COMPANY COMPOSITION 25/CAL/1998 06-01-1998 244606 13-12-2010 PHARMACEUTICAL COMPOSITION IN THE FORM OF SONUS PHARMACEUTICALS INC EMULSION MICRO EMULSION OR MICELLAR SOLUTION FOR DELIVERY OF POORLY SOLUBLE DRUGS

198/MUM/2004 20-02-2004 244585 13-12-2010 NOVEL DRUG DELIVERY SYSTEM TORRENT PHARMACEUTICALS LTD. 838/CAL/1999 12-10-1999 244608 13-12-2010 A POLYPHARMACEUTICAL COMPOSITION FOR THE MR. ABDAL MUEED TREATMENT OF CORYZA CATARRH POLYPUS TONSILS, HEADACHE MIGRAINE APTHAE THRUSH SPRUE GLOSSITIS ITCHING AND PUSTULES 2056/MUM/2006 15-12-2006 244626 13-12-2010 STABLE DUAL RELEASE PHARMACEUTICAL TABLET IPCA LABORATORIES LIMITED COMPRISING METOPROLOL AND CHLORTHALIDONE

3536/KOLNP/2006 27-11-2006 244638 14-12-2010 HISTAMINE H3 RECEPTIOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY THERAPEUTIC USES 4710/KOLNP/2007 05-12-2007 244647 14-12-2010 A SUBSTITUTED TETRAHYDROCARBAZOLE COMPOUND ELI LILLY AND COMPANY USEFUL AS ANDROGEN RECEPTOR MODULATORS (SARM) AND PHARMACEUTICAL COMPOSITION THEREOF 5917/DELNP/2005 19-12-2005 244662 15-12-2010 A TOPICAL COMPOSITION FOR THE TREATMENT OF POLICHEM S.A ONYCHOSCHIZIA 1010/KOLNP/2006 20-04-2006 244695 15-12-2010 AQUEOUS SOLUTION PREPARATION CONTAINING SENJU PHARMACEUTICAL CO., LTD. AMINOGLYCOSIDE ANTIBIOTIC AND BROMFENAC 472/DELNP/2005 08-02-2005 244698 15-12-2010 A PHARMACEUTICAL FORMULATION IN THE FORM OF BRISTOL-MYERS SQUIBB COMPANY AN INCLUSION COMPLEX IN/PCT/2001/00453/DEL 31-05-2001 244699 15-12-2010 AN IMPROVED COMPOSITION OF A DRUG MALIREDDY S. REDDY 1012/MUM/2005 26-08-2005 244675 15-12-2010 NOVEL DRUG DELIVERY SYSTEM TORRENT PHARMACEUTICALS LIMITED

1397/DELNP/2003 01-09-2003 244724 17-12-2010 A DELAYED RELEASE ORAL SOLID COMPOSITION PENWEST PHARMACEUTICALS CO 569/DELNP/2003 16-04-2003 244734 17-12-2010 A PHARMACEUTICAL COMPOSITION COMPRISING FOURNIER LABORATORIES IRELAND PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR LIMITED (PPAR) AND COENZYME Q10. IN/PCT/2002/00622/DEL 19-06-2002 244741 17-12-2010 COMPOUNDS SPECIFIC TO ADENOSINE A1 A2 AND A3, OSI PHARMACEUTICAL INC. RECEPTORS AND USES THEREOF 3306/KOLNP/2006 10-11-2006 244780 20-12-2010 A CYCLIC AMIDE COMPOUND AND A COMPOSITION TAKEDA PHARMACEUTICAL COMPANY COMPRISING THE SAME LIMITED 301/DELNP/2003 05-03-2003 244794 20-12-2010 SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC APPLIED RESEARCH SYSTEMS ARS AND IONISABLE MOIETIES AS INHIBITOR OF PROTEIN HOLDING N.V JUNKINASES 196/DELNP/2005 19-01-2005 244809 21-12-2010 SUSTAINED RELEASE FORMULATIONS COMPRISING GLAXO GROUP LIMITED LAMOTRIGINE 680/DELNP/2005 21-02-2005 244827 21-12-2010 NUCLEOSIDE ANALOG COMPOUND ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY 6238/DELNP/2006 25-10-2006 244837 21-12-2010 4-PHENYLAMINO-QUINAZOLIN-6-YL-AMIDES AND A WARNER -LAMBERT COMPANY PHARMACEUTICAL COMPOSITION COMPRISING THE LLC  SAME 1739/DELNP/2003 23-10-2003 244886 23-12-2010 4-ANILINOQUINOLINE-3-CARBOXAMIDE OF THE ASTRA ZENECA AB FORMULA I (A) 911/MUM/2005 05-08-2005 244866 23-12-2010 TOPICAL PHARMACEUTICAL COMPOSITIONS GLENMARK PHARMACEUTICALS CONTAINING ADAPALENE AND CLINDAMYCIN LIMITED IN/PCT/2002/00340/DEL 28-03-2002 244925 27-12-2010 FORMULATION FOR MENOPAUSAL WOMEN DRUGTECH CORPORATION 812/KOLNP/2006 04-04-2006 244997 28-12-2010 MODAFINIL MODIFIED RELEASE PHARMACEUTICAL , INC COMPOSITIONS 2982/CHENP/2006 14-08-2006 245016 29-12-2010 GLP-1 ANALOGUES SOCIETE DE CONSEILS DE RECHERCHES ET D"APPLICATIONS SCIENTIFIQUES SAS

1341/CHE/2005 21-09-2005 245033 29-12-2010 DERIVATIVES OF 4,6-DISUBSTITUTED 1,2,4- TRIAZOLO- JAWAHARLAL NEHRU CENTRE FOR 1,3,4-THIADIAZOLE, A PROCESS AND USES THEREOF ADVANCED SCIENTIFIC RESEARCH

756/KOLNP/2006 29-03-2006 245052 30-12-2010 CONDENSED RING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. 984/CHENP/2005 20-05-2005 245117 03-01-2011 COMPOSTION COMPRISING A CHEMOTHERAPEUTIC M/S. THE BOARD OF TRUSTEES OF THE AGENT AND AN ENDOTHELIN B AGONIST. UNIVERSITY OF ILLINOIS

688/DELNP/2006 10-02-2006 245128 04-01-2011 A SUBSTITUTED QUINAZOLINE COMPOUND INCLUDING ARRY BIOPHARMA, INC. RESOLVED ENANTIOMERS,DIASTEREOMERS,AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF

4781/DELNP/2005 19-10-2005 245131 04-01-2011 N-[1-(3-CHLORO-1-NAPHTHALENYL)ETHYL]-2-[4-(4- GLAXO GROUP LIMITED FLUOROPHENYL)-1-METHYL-4-PIPERIDINYL]-N- METHYLACETAMIDE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, ITS COMPOSITION AND PROCESS FOR PREPARING THE SAME 1578/DELNP/2004 07-06-2004 245132 04-01-2011 NITROGEN-CONTAINING HETEROARYL DERIVATIVES BTG INTERNATIONAL LTD., 3710/DELNP/2004 24-11-2004 245171 06-01-2011 A COMPOSITIONS FOR LOWERING INTRAOCULAR , INC PRESSURE AND PROVIDING NEUROPROTECTIOIN IN A PATIENT IN NEED THEREOF 6740/DELNP/2006 14-11-2006 245187 06-01-2011 CINNAMIDE COMPOUND EISAI R&D MANAGEMENT CO., LTD 2605/DELNP/2006 09-05-2006 245196 06-01-2011 RADIOLABELED 3,7-BIS [2-(4-NITRO [3,5-3H] PHENYL) ASTRAZENECA AB ETHYL] -3,7-DIAZABICYCLO [3,3,1] NONANE

1295/DELNP/2003 14-08-2003 245212 07-01-2011 PHARMACEUTICAL COMPOSITIION CONTAINING ONE BOEHRINGER INGELHEIM PHARMA OR MORE TIOTROPIUM SALTS GMBH & CO. KG. IN/PCT/2002/00728/DEL 29-07-2002 245257 11-01-2011 SULFONAMIDE COMPOUNDS THAT MODULATE THE TEXAS BIOTECHNOLOGY CORPORATION ACTIVITY OF ENDOTHELIN 281/DELNP/2005 25-01-2005 245306 13-01-2011 A PHARMACEUTICAL COMPOSITION FOR INHIBITING HELIX BIOPHARMA CORP. GROWTH OF CANCER CELLS 709/DELNP/2005 22-02-2005 245310 13-01-2011 N-PYRID-2YL,N'-4,7-DI-HALO- MEDIVIR AB TETRAHYDROCYCLOPROPA (-C-) CHROMEN-1-YL(THIO) UREA COMPOUNDS OF THE FORMULA U 291/DELNP/2005 25-01-2005 245335 13-01-2011 A COMPOSITION COMPRISING A SYNERGISTIC RATIO OF PFIZER INC. AN ALPHA-2-DELTA LIGAND AND A PDEV INHIBITOR

344/DELNP/2005 28-01-2005 245337 13-01-2011 A 2'-C-METHYL-RIBOFURANOSYL CYTIDINE-3'-O-L- IDENIX (CAYMAN) LIMITED VALINE ESTER COMPOUND 654/DELNP/2005 18-02-2005 245339 13-01-2011 A NOVEL CYTOTOXIC LINKABLE TAXANE COMPOUND IMMUNOGEN, INC

560/DELNP/2005 14-02-2005 245340 13-01-2011 AQUEOUS PHARMACEUTICAL COMPOSITION FOR BOEHRINGER INGELHEIM PHARMA INHALATION GMBH & CO. KG 108/DELNP/2005 12-01-2005 245350 14-01-2011 1 2-CYANO-4-FLUOROPYRROLIDINE DERIVATIVE" ASTELLAS PHARMA INC. 678/MUMNP/2005 27-06-2005 245363 17-01-2011 ORALLY ADMINISTRABLE PREPARATION BAYER SCHERING PHARMA AKTIENGESELLSCHAFT 207/DELNP/2005 19-01-2005 245368 17-01-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL ACRUX DDS PTY.LTD. DELIVERY 1136/DELNP/2005 22-03-2005 245372 17-01-2011 A PHARMACEUTICAL COMPOUND AND COMPOSITION BAUSCH & LOMB INCORPORATED THEREOF 419/DELNP/2005 03-02-2005 245396 18-01-2011 A SUSTAINED RELEASE BICIFADINE COMPOSITION NASCIME LIMITED 123/DELNP/2005 13-01-2005 245400 18-01-2011 COMPOSITION FOR TOPICALLY TREATING SEBORRHEIC PARKS, L., DEAN DERMATITIS 214/DELNP/2005 19-01-2005 245401 18-01-2011 AN ORALLY CONSUMABLE FILM COMPOSITION FOR COLGATE-PALMOLIVE COMPANY DELIVERING BREATH FRESHENING AGENTS TO THE ORAL CAVITY 1029/DELNP/2005 16-03-2005 245410 18-01-2011 A PHARMACEUTICAL COMPOSITION COMPRISING A HUMAN INTERLEUKIN-11(IL-11')POLYPEPTIDE" IN/PCT/2002/01202/DEL 05-12-2002 245422 19-01-2011 PHARMACEUTICAL COMPOSITIONS CONTAINING D-PHARM LTD. PHOSPHOLIPID DERIVATIVES OF VALPROIC ACIDS" IN/PCT/2002/00852/DEL 28-08-2002 245424 19-01-2011 PYRROLOPYRIMIDONE DERIVATIVES AND PROCESS OF S.K. CHEMICALS CO., LTD. PREPARATION THEREOF 3677/DELNP/2005 19-08-2005 245428 19-01-2011 A FACTOR VIII COMPOSITION INC. 2052/DELNP/2005 13-05-2005 245431 19-01-2011 TIZANIDINE COMPOSITION TEVA PHARMACEUTICAL INDUSTRIES LTD. 1752/DELNP/2005 29-04-2005 245446 19-01-2011 A PHARMACEUTICAL COMPOSITION COMPRISING NEUROPHARMACOLOGY SERVICES,LLC. OXYTOCIN 1708/DELNP/2005 27-04-2005 245448 19-01-2011 PYRIDOPYRROLIZINE AND PYRIDOINDOLIZINE MERCK FROSST CANADA & CO. DERIVATIVES 1633/DELNP/2005 21-04-2005 245450 19-01-2011 PHENYLNAPHTHALENE COMPOUNDS AND LES LABORATOIRES SERVIER PHARMACEUTICAL COMPOSITION THEREOF 5949/DELNP/2005 20-12-2005 245452 20-01-2011 COMPOUNDS FOR TREATING OCULAR HYPERTENSION MERCK & CO.INC. AND COMPOSITIONS THEREOF 1090/DELNP/2005 21-03-2005 245455 20-01-2011 6-METHYL-2[4-(4--MORPHOLINO) ANILINO] NICOTINIC B & C BIOPHARM ACID AND METHOD FOR PREPARING THEREOF

1139/DELNP/2005 23-03-2005 245458 20-01-2011 AN INJECTABLE EMULSION FORMULATION OF A BAXTER INTERNATIONAL INC. VOLATILE ANESTHETIC 1361/DELNP/2005 05-04-2005 245460 20-01-2011 AN ASIALO-INTERFERON PHARMACEUTICAL THE GENERAL HOSPITAL CORPORATION COMPOSITION 1420/DELNP/2005 07-04-2005 245492 21-01-2011 NOVEL QUINOLYLPROPYLPIPERIDINE COMPOUNDS AND NOVEXEL PROCESS FOR PREPARATION THEREOF 2224/DELNP/2004 30-07-2004 245502 21-01-2011 CARBAMOYL SUBSTITUTED COMPOUNDS USEFUL TANABE SEIYAKU CO. LTD FORαLß2 INHIBITION OF INTEGRIN MEDIATED CELL ADHESION 99/KOLNP/2007 09-01-2007 245570 25-01-2011 OXAZOLE DERIVATIVES AS HISTAMINE H3 RECEPTOR ELI LILLY AND COMPANY AGENTS, PREPARATION AND THERAPEUTIC USES

2093/DELNP/2005 17-05-2005 245573 25-01-2011 A 3,5 SUBSTITUTED OXAZOLIDINONE COMPOUND OF ASTRAZENECA AB THE FORMULA (I) 751/DELNP/2005 24-02-2005 245578 25-01-2011 A 3-(SULFONAMIDOETHYL)-INDOLE COMPOUND AND A BOEHRINGER INGELHEIM METHOD OF MAKING FORMULA (I) PHARMACEUTICALS INC. 2090/DELNP/2005 17-05-2005 245583 25-01-2011 A CONTROLLED RELEASE TABLET CONTAINING CILAG AG TOPIRAMATE, HYDROCHLORIDE AND XANTHAN GUM 2007/DELNP/2004 13-07-2004 245611 27-01-2011 AN OSMOTIC PHARMACEUTICAL TABLET PFIZER PRODUCTS INC 2918/DELNP/2004 28-03-2004 245616 27-01-2011 AN INDAZOL COMPOUND JNK INHIBITOR EISAI R&D MANAGEMENT CO., LTD 1871/KOLNP/2007 25-05-2007 245644 28-01-2011 A COMPOUND OF FORMULA (I) AND A COMPOSITION ELI LILLY AND COMPANY USED AS ALLOSTERIC POTENTIATORS OF THE M4 MUSCARINIC RECEPTOR

1073/DELNP/2003 08-07-2003 245684 28-01-2011 A GELDANAMYCIN DERIVATIVE THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES IN/PCT/2002/01240/DEL 13-12-2002 245685 28-01-2011 A COMPOUND OF THE 3`-O-VALINYL ESTER OF 2`- IDENIX (CAYMAN) LIMITED DEOXY-[BETA]-L-CYTIDINE 3501/DELNP/2004 09-11-2004 245725 31-01-2011 A HERBAL COMPOSITION USEFUL FOR GASTRO- COUNCIL OF SCIENTIFIC & INDUSTRIAL INTESTINAL DISORDERS & PROCESS THEREOF RESEARCH. 910/CHE/2005 08-07-2005 245780 01-02-2011 NOVEL BIO-ACTIVE DERIVATIVES ORCHID CHEMICALS & PHARMACEUTICALS LTD 318/KOLNP/2007 29-01-2007 245805 02-02-2011 VAGINAL RING CONTAINING THE POPULATION COUNCIL, INC. RECEPTOR MODULATORS 1154/DEL/2001 16-11-2001 245820 02-02-2011 NOVEL DIALLYLDISULPHIDE COMPOUNDS HAVING DEPARTMENT OF SCIENCE AND ANTILIPIDEMIC AND ANTIOXIDANT ACTIVITY TECHNOLOGY 1501/MUMNP/2006 07-12-2006 245843 03-02-2011 A PHARMACEUTICAL COMPOSITION COMPRISING BOEHRINGER INGELHEIM PHARMA TIOTROPIUM AND FORMOTEROL GMBH & CO. KG. 1124/MUM/2004 20-10-2004 245846 03-02-2011 SEDATIVES LOADED INTRANASAL NASOADHESIVE AMBIKANANDAN MISRA MICROEMULSIONS FOR BRAIN TARGETED DELIVERY IN INSOMNIA 843/CHE/2006 12-05-2006 245854 03-02-2011 NOVEL THROMBOLYTIC MOLECULES AND A PROCESS BHARAT BIOTECH INTERNATIONAL THEREFOR LIMITED 2543/DELNP/2005 13-06-2005 245887 04-02-2011 A COMPOSITION FOR TREATING PERSONS SUFFERING ALCON, INC. FROM ACUTE OR CHRONIC DEGENERATIVE CONDITIONS OR DISEASES OF THE EYE

3220/DELNP/2005 20-07-2005 245920 07-02-2011 PHARMACEUTICAL COMPOSITION USEFUL AGAINST CENTRO DE INGENIERIA GENETICA Y NEOPLASIA BIOTECNOLOGIA 3029/DELNP/2005 06-07-2005 245936 07-02-2011 A LACTOFERRIN COMPOSITION FOR TREATING AGENNIX INCORPORATED BACTEREMIA OR SEPSIS 3254/DELNP/2005 22-07-2005 245943 07-02-2011 COMPOSITION FOR PREVENTIVE TREATMENT OF COLD PRONOVA MEDICAL B.V. SORES 3481/DELNP/2004 09-11-2004 245978 08-02-2011 COMPOSITION, FORMULATIONS & KIT FOR TREATMENT EPIGENESIS PHARMACEUTICALS, LLC. OF RESPIRATORY & LUNG DISEASE WITH (S) STEROID & AN ANTI- MUSCARINIC AGENT(S) 6091/DELNP/2005 27-12-2005 245986 09-02-2011 MODIFIED-RELEASE COMPOSITION BIOVAIL LABORATORIES INTERNATIONAL SRL. 2139/KOLNP/2006 28-07-2006 246005 09-02-2011 NOVEL INHIBITORS OF GLUTAMINYL CYCLASE PROBIODRUG AG 935/KOLNP/2006 13-04-2006 246008 09-02-2011 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN VERTEX PHARMACEUTICALS KINASES INCORPORATED 232/DELNP/2004 03-02-2004 246010 09-02-2011 ANTITUMORAL ANALOGUES OF ECTEINASCIDIN PHARMA MAR, SA. IN/PCT/2002/00703/DEL 16-07-2002 246021 09-02-2011 A COMPOSITION USEFUL AGAINST ASEPTIC HU, SHIQING INFLAMMMATIONS AND STUBBORN PAINS 372/DELNP/2003 12-03-2003 246112 15-02-2011 17-METHYLENE STEROIDS, PROCESS FOR THEIR SCHERING AKTIENGESELLSCHAFT PRODUCTION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THESE COMPOUNDS 5042/DELNP/2005 03-11-2005 246115 15-02-2011 HETEROARYL AMIDE DERIVATIVES AND THEIR USE AS ASTRAZENECA AB P2X7 , RECEPTOR ANTAGONISTS 1301/KOLNP/2006 17-05-2006 246121 15-02-2011 DUAL MOLECULES CONTAINING PEROXY DERIVATIVE, CENTRE NATIONAL DE LA RECHERCHE THE SYNTHESIS SCIENTIFIQUE 1125/KOLNP/2007 02-04-2007 246133 15-02-2011 HALOGENATED BENZAMIDE DERIVATIVES ROMARK LABORATORIES, L.C. 2037/DELNP/2006 13-04-2006 246159 17-02-2011 A COMPOUND OF FORMULA (I) FOR USE AS PFIZER INC. MEDICAMENT 252/MUM/2007 09-02-2007 246147 17-02-2011 A PHARMACEUTICAL COMPOSITION AND A PROCESS INDUS BIOTECH PRIVATE LIMITED THEREOF 1588/DEL/1998 10-06-1998 246186 18-02-2011 A 4 -SUBSTITUED-9-DEOXO-9A-AZA-9A- PFIZER PRODUCTS INC. HOMOERYTHROMYCIN A COMPOUND" 3827/DELNP/2004 02-12-2004 246195 21-02-2011 PHARMACEUTICAL COMPOSITION AND PROCESS OF INSIGNION HOLDINGS LIMITED PREPRATION THEREOF 828/KOLNP/2006 05-04-2006 246198 21-02-2011 2,4-DIOXO-3-QUINAZOLINYL SULFONYLUREAS PORTOLA PHARMACEUTICALS, INC. 1428/DELNP/2005 07-04-2005 246202 21-02-2011 A GLP-2 PEPTIDE AND PHARMACEUTICAL NOVA NORDISK A/S COMPOSITION THEREOF 4753/DELNP/2005 19-10-2005 246215 21-02-2011 AN ARYL AMINOTHIAZOLE COMPOUND NEUROGENETIC PHARMACEUTICALS , INC. 1594/DELNP/2004 08-06-2004 246226 22-02-2011 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS KINETEK PHARMACEUTICALS INC THERAPEUTICS 3736/DELNP/2006 29-06-2006 246229 22-02-2011 A PARENTERAL PHARMACEUTICAL COMPOSITION PFIZER PRODUCTS INC. 1241/DELNP/2005 30-03-2005 246249 22-02-2011 A COMPOUND OF FORMULA (I) OR ASTRAZENECA AB PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF 5369/DELNP/2005 23-11-2005 246279 23-02-2011 BETA-STRAND MIMETICS AND METHODS RELATING CHOONGWAE PHARMA CORPORATION THERETO 1872/KOLNP/2007 25-05-2007 246285 23-02-2011 AN AMIDE OF COMPOUND 2-DEOXY-2, 2- ELI LILLY AND COMPANY DIFLUOROCYTIDINE AND PHARMACEUTICAL COMPOSITION THEREOF 2713/DEL/2006 19-12-2006 246278 23-02-2011 PHARMACEUTICAL COMPOSITION LES LABORATOIRES SERVIER 172/DELNP/2007 08-01-2007 246305 24-02-2011 BIS(THIO-HYDRAZIDE AMIDE) SALTS FOR TREATMENT SYNTA PHARMACEUTICALS CORP OF CANCERS, PHARMACEUTICAL COMPOSITION AND METHOD OF PREPARATION THEREOF

961/CHENP/2004 05-05-2004 246323 24-02-2011 CYCLOOXYGENASE -2 INHIBITOR/HISTONE NOVARTIS AG DEACETYLASE INHIBITOR COMBINATION 402/CHENP/2004 27-02-2004 246328 24-02-2011 AN AEROSOL SUSPENSION FORMULATION FOR SCHERING CORPORATION INHALATION 7329/DELNP/2006 05-12-2006 246335 24-02-2011 A PHARMACEUTICAL COMPOSITION SUITABLE FOR USE ALMIRALL  S.A. IN THE RESPIRATORY DISORDERS COMPRISING PDE4 INHIBITORS AND ANTAGONIST OF M3 MUSCARINIC RECEPTORS IN/PCT/2002/00749/DEL 01-08-2002 246355 25-02-2011 A SYNERGISTIC PHARMACEUTICAL COMPOSITION AVENTIS PHARMA S.A. COMPRISING A COMBINATION OF CAMPTOTHECIN WITH CAPECITABINE 1748/DELNP/2003 27-10-2003 246359 25-02-2011 A NOVEL COMPOUND HAVING CORTICOTROPIN- EISAI R & D MANAGEMENT CO. LTD RELEASING FACTOR RECEPTOR ANTAGONISTIC ACTIVITY, SALTS THEREOF AND HYDRATES OF THE FOREGOING IN/PCT/2002/00724/DEL 24-07-2002 246366 25-02-2011 A TWO COMPONENT EFFERVESCENT DENTIFRICE COLGATE-PALMOLIVE COMPANY COMPOSITION AND METHOD THEREOF 263/CHENP/2006 20-01-2006 246396 25-02-2011 HEPARIN-DERIVED OLIGOSACCHARIDE MIXTURES, AVENTIS PHARMA S.A. PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID MIXTURES IN/PCT/2002/00262/MUM 04-03-2002 246466 28-02-2011 A GRANULE FORMULATION AND A PROCESS FOR ASTRAZENECA AB PREPARING THE SAME 1515/DELNP/2005 15-04-2005 246467 01-03-2011 A BAICALEIN DERIVATIVE JENKEN BIOSCIENCES,INC. 250/DELNP/2005 24-01-2005 246481 01-03-2011 HETERO BIARYL COMPOUNDS WARNER-LAMBERT COMPANY LLC 1376/DELNP/2005 05-04-2005 246487 01-03-2011 A COMPOUND N-ALKYNYL-2-ALKOXY-2-(SUBSTITUTED SYNGENTA LIMITED PHENOXY ALKYLAMIDES) OF GENERAL FORMULA (I) AND PHARMACEUTICAL COMPOSITION THEREOF

208/DELNP/2005 19-01-2005 246494 01-03-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL CRUX DDS PTY. LTD. DELIVERY OF PHYSIOLOGICALLY ACTIVE AGENT

1025/DEL/2003 19-08-2003 246484 01-03-2011 A NOVEL CONTROLLED RELEASE FORMULATION OF NATIONAL INSTITUTE OF AZITHROMYCIN PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) 1201/CHENP/2006 06-04-2006 246515 02-03-2011 METHYLPHENIDATE SOLUTION AND ASSOCIATED MALLINCKRODT INC. METHODS OF ADMINISTRATION AND PRODUCTION

917/CHE/2006 29-05-2006 246524 02-03-2011 2-(2-AMINO-1, 6-DIHYDRO-6-OXO-PURIN-9-YL) F. Hoffmann-La Roche AG METHOXY-1, 3-PROPANEDIOL DERIVATIVE 1399/DELNP/2003 01-09-2003 246558 04-03-2011 A DELAYED RELEASE ORAL SOLID COMPOSITION PENWEST PHARMACEUTICALS CO. 2849/DELNP/2004 23-09-2004 246560 04-03-2011 A B-AMINO ACID OF FORMULA IA AND COMPOSITIONS WARNER-LAMBERT COMPANY LLC THEREOF 3160/DELNP/2004 13-10-2004 246574 04-03-2011 SUSTAINED RELEASE COMPOSITION FOR TREATING APOTEX INC IRON INDUCED CARDIAC DISEASE 2720/DELNP/2004 15-09-2004 246581 04-03-2011 COMPOUND OF FORMULA (I) AS TROPANE PFIZER INC. DERIVATIVES IN/PCT/2002/00135/DEL 31-01-2002 246584 07-03-2011 PHENOXYPROPIONIC ACID ALKOXYCARBONYL ANILID DONBU HANNONG CHEMICAL CO.,LTD COMPOUNDS AND PREPARATION THEREOF 3401/KOLNP/2006 17-11-2006 246620 08-03-2011 COMPOUNDS FOR TREATING DYSLIPIDEMIA ELI LILLY AND COMPANY 1327/CHENP/2007 30-03-2007 246642 08-03-2011 2-AMINOPYRIDINE COMPOUNDS USEFUL AS BETA- MERCK & CO INC SECRET ASE INHIBITORS FOR THE TREATMENT OF ALZHEMER'S DISEASE 1363/DELNP/2005 05-04-2005 246655 09-03-2011 ALKENYL ESTERS OF AMINO SUBSTITUTED ALKONIC YEDA RESEARCH AND DEVELOPMENT ACID CO. LTD. 766/CHENP/2007 22-02-2007 246671 10-03-2011 ACIDIC SOLID ORAL COMPOSITIONS WITHOUT EROSIVE TOMS GRUPPEN A/S POTENTIAL IN SALIVA AND METHOD FOR REDUCTION OF EROSIVE POTENTIAL IN SALIVA 647/KOLNP/2003 20-05-2003 246761 15-03-2011 AEROGEL POWDER AND A PROCESS FOR ASPEN AEROGELS, INC. MANUFACTURING IT 423/KOLNP/2003 08-04-2003 246771 15-03-2011 A METHOD OF PREPARING A COMPOSITION OF CEPHALON INC PARTICLES, AND THE COMPOSITION THEREOF 1256/DEL/2005 16-05-2005 246763 15-03-2011 NEW PYROOLIDINE AND THIAZOLIDINE COMPOUNDS, A LES LABORATOIRES SERVIER PROCES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

1034/KOLNP/2006 21-04-2006 246789 16-03-2011 BENZIMIDAZOLE DERIVATIVES : PREPARATION AND S*BIO PTE LTD. PHARMACEUTICAL APPLICATIONS 1826/KOLNP/2006 30-06-2006 246799 16-03-2011 A SOFT CAPSULE OF BUTYLPHTHALIDE SHIJIAZHUANG PHARMA. GROUP ZHONGQI PHARMACEUTICAL TECHNOLOGY (SHIJIAZHUANG) CO., LTD. 1411/CHENP/2005 24-06-2005 246807 16-03-2011 1,2,4-TRIAMINOBENZENE DERIVATIVES USEFUL FOR H. LUNDBECK A/S TREATING DISORDERS OF THE CENTRAL NERVOUS SYSTEM 115/KOL/2008 16-01-2008 246818 16-03-2011 PHARMACEUTICAL COMPOSITION FOR THE DEVELOPMENT CENTER FOR TREATMENT OF RHEUMATOIDARTHRITIS BIOTECHNOLOGY 1885/CHENP/2006 29-05-2006 246853 17-03-2011 ANGIOGENIC PEPTIDES RAMOT AT TEL AVIV UNIVERSITY LTD. 6802/DELNP/2006 15-11-2006 246923 22-03-2011 2-PYRIDYL SUBSTITUTED IMIDAZOLE COMPOUND AS SK CHEMICALS CO.LTD ALK5 ALK4 INHIBITORS AND A COMPOSITION THEREOF

01281/DELNP/2003 13-08-2003 246948 22-03-2011 CIS-1(5-CYANO-PYRIDIN-2-YL)-3-(4,7-DIFLUORO- MEDIVIR AB 1,1A,2,7B-TETRAHYDRO CYCLOPROPA[C]CHROMEN-1- YL)-UREA OF FORMULA 1 2098/DELNP/2005 17-05-2005 246952 23-03-2011 A PHARMACEUTICAL COMPOSITION COMPRISING BIOMARIN PHARMACEUTICAL INC. PRECURSOR HUMAN N-ACETYLGALACTOSAMINE-4- SULFATASE 1759/DELNP/2004 21-06-2004 246961 23-03-2011 ORAL PHARMACEUTICAL COMPOSITION FOR UCB FARCHIM SA IMPROVING PALATABILITY AND AVOIDING UNDESIRED REACTION PRODUCTS CONTAINING AT LEAST TWO SEPARATE FORMULATIONS 796/KOLNP/2006 03-04-2006 246966 23-03-2011 FUSED PENTACYCLIC POLYETHERS UNIVERSITY OF NORTH CAROLINA AT WILMINGTON 719/DELNP/2005 22-02-2005 247029 25-03-2011 PHARMACEUTICAL FORMULATION COMPRISING PATEL SATISHCHANDRA CYCLOSPORIN PROPYLENE GLYCOL ESTER AND NON- PUNAMBHAI,27 YALE IONIC SURFACTANT COURT,LIVINGSTON,NEW JERSEY 07039,U.S.A 1133/CHENP/2006 03-04-2006 247041 25-03-2011 DRUG CONTAINING (2R)-2-PROPYLOCTANOIC ACID AS ONO PHARMACEUTICAL CO., LTD. THE ACTIVE INGREDIENT 1511/MUM/2006 21-09-2006 247054 26-03-2011 SUSTAINED RELEASE ANTI-EPILEPTIC COMPOSITIONS INVENTIA HEALTHCARE PRIVATE LIMITED 3511/KOLNP/2006 24-11-2006 247064 28-03-2011 GLUCAGON RECEPTOR ANTAGONISTS AND ELI LILLY AND COMPANY PHARMACEUTICAL COMPOSITION THEREOF 1099/KOLNP/2004 03-08-2004 247070 28-03-2011 A 2,4,6 - TRIAMINE-1,3,5-TRIAZINE ASTELLAS PHARMA INC. 2906/DELNP/2006 22-05-2006 247072 28-03-2011 IMIDAZOLE DERIVATIVES UCB S.A 210/DELNP/2005 19-01-2005 247093 28-03-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL ACRUX DDS PTY. LTD. DELIVERY RATE CONTROL OF PHYSIOLOGICALLY ACTIVE AGENT USING AMORPHOUS DEPOSIT

1990/DELNP/2005 10-05-2005 247096 28-03-2011 A PHARMACEUTICAL COMPOUND FOR TREATING TARO PHARMACEUTICAL INDUSTRIES MOVEMENT DISORDERS LIMITED 811/KOLNP/2005 04-05-2005 247104 28-03-2011 N-SUBSTITUTED CARBAMATE META-BIPHENYL ESTER THE REGENTS OF THE UNIVERSITY OF AS NOVEL FATTY ACID AMIDE HYDROLASE INHIBITORS CALIFORNIA

1885/KOLNP/2006 06-07-2006 247116 28-03-2011 DERIVATIVES OF N-' (1,5-DIPHENYL-1 H-PYRAZOL-3-YL) SANOFI-AVENTIS SUPHONAMIDE WITH CB1 RECEPTOR AFFINITY 2621/KOLNP/2005 19-12-2005 247151 29-03-2011 AN ORAL PHARMACEUTICAL COMPOSITION UNITED THERAPEUTICS CORPORATION 6026/DELNP/2005 23-12-2005 247176 29-03-2011 A CONJUGATE MOLECULE CONSISTING OF AN OLIGO- INSTITUT PASTEUR OR POLYSACCHARIDE 978/DEL/2004 28-05-2004 247177 29-03-2011 AN AZITHROMYCIN COMPOSITION PFIZER PRODUCTS INC. 2347/DELNP/2006 27-04-2006 247226 30-03-2011 SPIROCYCLIC HETEROCYLIC COMPOUND ADOLOR CORPORATION 2103/MUM/2006 22-12-2006 247344 31-03-2011 ( 1-H-PYRAZOL-1-YL)ALKYLAMINE COMPOUNDS OF AVENTIS PHARMA S.A. FORMULA (III) 1279/MUM/2005 11-10-2005 247285 31-03-2011 NOVEL ANTI-MALARIAL COMBINATION AND METHODS IPCA LABORATORIES LTD. OF FORMULATION 83/MUM/2006 18-01-2006 247313 31-03-2011 MODIFIED RELEASE ORAL DOSAGES FORM USING CO- ASTRON RESEARCH LIMITED POLYMER OF POLYVINYI ACETATE 1125/MUM/2004 20-10-2004 247325 31-03-2011 DRUGS LOADED INTRANASAL NASOADHESIVE AMBIKANANDAN MISRA MICROEMULSIONS FOR BRAIN TARGETED DELIVERY IN MIGRAINE 1269/CHENP/2006 13-04-2006 247373 04-04-2011 A COMPOSITION FOR ASSISTING MUCUS CLEARANCE IN VECTURA LIMITED THE RESPIRATORY TRACT 00590/DELNP/2004 09-03-2004 247381 04-04-2011 A NOVEL COMPOUND OF FORMULA (1) BRISTOL - MYERS SQUIBB COMPANY 1882/KOLNP/2006 06-07-2006 247403 05-04-2011 SUBSITUTED PIPERAZINES CHEMOCENTRYX, INC. 1921/DELNP/2005 06-05-2005 247426 06-04-2011 DERMASTICK THICKENED OINTMENT JAGOTEC AG 3762/KOLNP/2006 13-12-2006 247490 12-04-2011 CAPSULES COMPRISING A MICRO-ORGANISM, A FIRMENICH SA MATRIX COMPONENTS AND AT LEAST ONE ENCAPSULATABLE MATERIAL AND PROCESS FOR ITS PREPARATION 1208/KOLNP/2006 09-05-2006 247495 12-04-2011 PYRAZOLYL DERIVATIVES IN THE FORM OF DRUGS FOR AVENTIS PHARMA S.A. TREATING ACUTE OR CHRONIC NEURONAL REGRESSIONS 3481/KOLNP/2006 22-11-2006 247501 12-04-2011 PROPANE-1,3-DIONE DERIVATIVE OR SALT THEREOF ASTELLAS PHARMA INC.

132/KOLNP/2007 10-01-2007 247503 12-04-2011 2-(PYRIDIN-2-YL)-PYRIMIDINES AND THEIR USE FOR BASF AKTIENGESELLSCHAFT CONTROLLING HARMFUL FUNGI 2286/KOLNP/2006 10-08-2006 247504 12-04-2011 TRIAZOLOPYRIMIDINES BASF AKTIENGESELLSCHAFT 405/DELNP/2005 02-02-2005 247532 18-04-2011 AZABICYCLO DERIVATIVES AS MUSCARINIC RECEPTOR RANBAXY LABORATORIES LIMITED ANTAGONISTS 1406/DELNP/2005 07-04-2005 247540 18-04-2011 A PHARMACEUTICAL COMPOSITION COMPRISING AN OREXO AB ACID SUSCEPTIBLE PROTON PUMP INHIBITOR AND AN H2 RECEPTOR ANTAGONIST 2482/CHENP/2006 06-07-2006 247551 19-04-2011 TETRAPEPTIDE LYSYL-GLUTAMYL-ASPARTYL- ACCESS BIOSCIENCE CJSC TRYPTOPHANE AMIDE 233/MUM/2003 27-02-2003 247575 25-04-2011 HERBAL SKIN-CARE COMPOSITION THE KELKAR EDUCATION TRUST'S SCIENTIFIC RESEARCH CENTRE 1411/MUM/2006 04-09-2006 247582 25-04-2011 A SYSTEM FOR SPATIALLY AND TEMPORALLY PANACEA BIOTEC LTD. PROGRAMMABLE DELIVERY OF AN ACTIVE AGENT 4915/DELNP/2005 26-10-2005 247600 26-04-2011 MAYTANSINOID CELL-BINDING CONJUGATES AND THE IMMUNOGEN , INC. PREPARATION THEREOF 1310/CHENP/2006 17-04-2006 247612 27-04-2011 - MASKED FORMULATION COMPRISING NOVARTIS AG CLARITHROMYCIN 858/DEL/2004 11-05-2004 247615 27-04-2011 A POLYHERBAL COMPOSITION FOR THE TREATMENT OF OHARI, VIJAY KUMAR VIRAL HEPATITIS 2954/KOLNP/2006 12-10-2006 247675 02-05-2011 COMBINATION OF PENTRAXIN PTX3 AND AN SIGMA-TAU INDUSTRIE ANTIFUNGAL AGENT FARMACEUTICHE RIUNITE S.P.A. IN/PCT/2002/00585/DEL 06-06-2002 247731 09-05-2011 A COMPOSITION USEFUL FOR TREATING OR CHEMGEN CORPORATION AMELIORATING THE RISK OF DIGESTIVE TRACT INFECTION 156/MUM/2005 14-02-2005 247743 10-05-2011 WATER SOLUBLE ANTI-DANDRUDFF COMPOUNDS AND GALAXY SURFACTANTS LIMITED COMPOSITIONS THEREOF 2576/DELNP/2006 08-05-2006 247748 11-05-2011 PHARMACEUTICAL COMPOSITION COMPRISING RIEMSER ARZNEIMITTEL AG. OXOPLATIN, THE SALTS AND DERIVATIVES THEREOF 1388/DEL/1999 20-10-1999 247750 11-05-2011 A SUSTAINED-RELEASE FORMULATION FOR ORAL PFIZER RESEARCH AND DEVELOPMENT ADMINISTRATION FOR THE TREATMENT OR COMPANY, N.V./S.A., PREVENTION OF SEXUAL DYSFUNCTION 187/DEL/2002 01-03-2002 247754 11-05-2011 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDE JANSSEN PHARMACEUTICA N.V COMPOUNDS 462/MUM/2004 16-04-2004 247764 16-05-2011 ANTIINFECTIVE QUINOLONE COMPOUNDS AND CADILA HEALTHCARE LIMITED PROCESS FOR PREPARATION THEREOF 3818/KOLNP/2006 18-12-2006 247808 24-05-2011 A COMPOSITION FOR TREATING AND PREVENTING BRIGHT FUTURE PHARMACEUTICAL SLEEP DISORDER LABORATORIES LIMITED 52/DELNP/2006 03-01-2006 247821 25-05-2011 6-(1,1-DIFLUOROALKYL)-4-AMINOPICOLINATES AND DOW AGROSCIENCES LLC THEIR USE AS HERBICIDES 179/DELNP/2006 10-01-2006 247860 27-05-2011 ISETHIONATE SALT OF A SELECTIVE CDK4 INHIBITOR WARNER-LAMBERT COMPANY LLC,

6241/DELNP/2006 25-10-2006 247890 31-05-2011 AN ORAL MODIFIED RELEASE PHARMACEUTICAL ASTRAZENECA AB COMPOSITION 971/MUMNP/2006 21-08-2006 247891 31-05-2011 ENTERIC COATINGS FOR ORALLY INGESTIBLE BPSI HOLDINGS,INC. SUBSTRATES 2478/KOLNP/2006 22-08-2006 247909 01-06-2011 A FLUORO SUBSTITUTED COMPOUND OF FORMULA ELI LILLY AND COMPANY (1A) USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS AND PHARMACEUTICAL COMPOSITION THEREOF 485/CAL/2001 29-08-2001 247910 01-06-2011 A STERILE OPHTHALMIC DROP PREPARATION DR. GERHARD MANN CHEMISCH- PHARMAZEUTISCHE FABRIK GMBH 922/MUM/2002 23-10-2002 247913 02-06-2011 NOVEL TRICYCLIC COMPOUNDS AS PDE4 INHIBITORS GLENMARK PHARMACEUTICALS LIMITED 811/MUMNP/2003 28-08-2003 247914 02-06-2011 A COMPOUND OF FORMULA I AND BAYER HEALTHCARE LLC PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF IN TREATING RAF MEDIATED DISEASES 5515/DELNP/2005 29-11-2005 247944 06-06-2011 STABILIZED PHARMACEUTICAL PEPTIDE NOVO NORDISK A/S COMPOSITIONS. 2479/KOLNP/2006 31-08-2006 247943 06-06-2011 A BENZAZEPINE COMPOUND ELI LILLY AND COMPANY 3137/DELNP/2005 14-07-2005 247967 07-06-2011 ORAL CARE COMPOSITION COLGATE-PALMOLIVE COMPANY 13/MUMNP/2007 02-01-2007 247984 08-06-2011 CRYSTALLINE FORM OF A TRIAZOLO (4,5-D)PYRIMIDINE ASTRAZENECA AB COMPOUND 1891/MUM/2006 15-11-2006 248024 09-06-2011 A LIQUID FORMULATION FOR HYGIENE AND JOSHI, VINAYAK NARAHAR TREATMENT OF AILMENTS OF THROAT AND MOUTH

890/MUM/2004 16-08-2004 248023 09-06-2011 A CONTROLLED RELEASE ANTIDIABETIC FORMULATION IPCA LABORATORIES LIMITED COMPRISING GLICLAZIDE 1112/DEL/2002 06-11-2002 248025 09-06-2011 NOVEL 4-ETHYL-5ALKOXYPRIMAQUINE COMPOUNDS NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) 844/DELNP/2005 04-03-2005 248026 09-06-2011 S-(-)- AMLODIPINE NICOTINATE AND PROCESS FOR THE HANLIM PHARMACEUTICAL CO., LTD. PREPARATION THEREOF 456/DEL/2000 25-04-2000 248090 16-06-2011 GLUCOCORTICOID RECEPTOR MODULATORS PFIZER PRODUCTS IN 58/MUM/2005 19-01-2005 248096 16-06-2011 HERBAL CONTRACEPTIVE FORMULATIONS SINGH KAMALINDER KAUR 02044/DELNP/2003 28-11-2003 248107 17-06-2011 PHARMACEUTICAL FORMULATION FOR THE EFFICIENT AXON BIOCHEMICALS B.V. ADMINISTRATION OF APOMORPHINE 6AR-(-)-N-PROPYL- NORAPOMORPHINE AND THEIR DERIVATIVES AND PRO- DRUGS THEREOF 768/DELNP/2005 25-02-2005 248186 27-06-2011 A HEMIACETAL COMPOUND KISSEI PHARMACEUTICAL CO.,LTD., 1556/KOLNP/2006 06-06-2006 248227 28-06-2011 PYRAZINES VERTEX PHARMACEUTICALS INCORPORATED 1193/KOLNP/2003 18-09-2003 248253 29-06-2011 AN INVITRO ASSAY FOR IDENTIFYING A CANDIDATE CHIRON CORPORATION AGENT THAT REDUCES GROWTH OF A CANCEROUS CELL IN/PCT/2002/00769/DEL 06-08-2002 248284 01-07-2011 AN AQUEOUS PREPARATION OF PROPOFOL WITH MAELOR PHARMACEUTICALS LIMITED IMPROVED SOLUBILITES 1891/DELNP/2004 01-07-2004 248287 01-07-2011 PURIFICATION OF ONIUM HYDROXIDES BY SACHEM, INC ELECTRODIALYSIS 666/DELNP/2005 21-02-2005 248348 06-07-2011 A SUBSTITUTED PYRAZOLE COMPOUND AND KISSEI PHARMACEUTICAL CO. LTD PHARMACEUTICAL COMPOSITION THEREOF 2248/KOLNP/2006 08-08-2006 248349 06-07-2011 NOVEL COMPOUNDS AS FAAH INHIBITORS SANOFI AVENTIS 1334/DELNP/2005 04-04-2005 248353 06-07-2011 A SPOT-ON FORMULATION USEFUL FOR THE MERIAL LIMITED TREATMENT OF PARASITE INFESTATION 6786/DELNP/2006 15-11-2006 248361 07-07-2011 A PHARMACEUTICAL COMPOSITION FOR EFFECTIVE WARNER CHILCOTT COMPANY,LLC ABSORPTION 1135/CHENP/2006 03-04-2006 248395 12-07-2011 PYRAZOLO AND IMIDAZO-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG

2240/KOLNP/2006 08-08-2006 248401 12-07-2011 THIOAMIDES AND SALTS THEREOF AND CYTOKINE ISHIHARA SANGYO KAISHA, LTD. PRODUCTION INHIBITORS CONTAINING BOTH 491/DELNP/2007 18-01-2007 248459 18-07-2011 A COMPOUND REPRESENTED BY FORMULA (I) MEIJI SEIKA KAISHA  LTD. 583/MUMNP/2004 19-10-2004 248542 25-07-2011 PHARMACEUTICAL FORMULATION COMPRISING NEURIM PHARMACEUTICALS (1991) MELATONIN LTD. 5666/DELNP/2006 28-09-2006 248545 25-07-2011 FLAVOPEREIRINE DERIVATIVES FOR CANCER THERAPY DABUR PHARMA LTD

2504/DEL/2004 16-12-2004 248560 25-07-2011 ANTICIGARETTE HERBAL FORMULATION AS AN ANTI- COUNCIL OF SCIENTIFIC & INDUSTRIAL DOTE TO RESEARCH 327/DELNP/2004 12-02-2004 248615 28-07-2011 A COSMETIC COMPOSITION HAVING A SKIN LVMH RECHERCHE TIGHTENNING EFFECT 1480/MUM/2005 29-11-2005 248622 28-07-2011 PREPARATION OF DIGESTIVE ENZYMES CONTAINING MERCURY LABORATORIES LIMITED DRY SYRUP 3239/DELNP/2005 21-07-2005 248632 29-07-2011 AZABICYCLIC HETEROCYCLIC COMPOUND NOVEXEL 539/DELNP/2004 04-03-2004 248635 29-07-2011 BENZOTHIAZEPINE AND BENZOTHIADIAZEPINE ASTRAZENECA AB DERIVATIVES WITH LLEAL BILE ACID TRANSPORT (IBAT) INHIBITORY ACTIVITY FOR THE TREATMENT OF HYPERLIPIDAEMIA 685/DEL/2002 26-06-2002 248660 02-08-2011 A SYNERGISTIC PHARMACEUTICAL COMPOSITION OF NATIONAL INSTITUTE OF CELECOXIB WITH IMPROVED AQUEOUS SOLUBILITY PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) 583/MUM/2007 29-03-2007 248729 12-08-2011 MODIFIED DOSAGE FORMS OF TACROLIMUS PANACEA BIOTEC LIMITED 775/MUM/2004 21-07-2004 248777 24-08-2011 PHARMACEUTICAL COMPOSITION CONTAINING MACLEODS PHARMACEUTICALS COMBINATION OF PROTON PUMP INHIBITOR WITH LIMITED MODIFIED RELEASE DOMPERIDONE 2507/DEL/2004 16-12-2004 248784 24-08-2011 DEVELOPMENT OF HARBAL NUTRITIOUS CHOCAEATE COUNCIL OF SCIENTIFIC AND AND ITS PROCESSING INDUSTRIAL RESEARCH 4656/DELNP/2005 13-10-2005 248794 25-08-2011 A COMPOSITION CONTAINING L-LACTIC ACID OR L- INNOGENE KALBIOTECH PTE LTD LACTATE AND USES THEREOF 1535/DEL/2004 18-08-2004 248796 25-08-2011 AN ANALGESIC PREPARATION CONTAINING MORPHINE ALL INDIA INSTITUTE OF MEDICAL AND NIMODIPINE AND A PROCESS FOR PREPARATION SCIENCE THEREOF 2426/DEL/2005 09-09-2005 248802 25-08-2011 A SUSTAINED RELEASE MULTILAYERED TABLET DELHI INSTITUTE OF PHARMACEUTICAL COMPOSITION FOR UNSTABLE DRUG SCIENCES & RESEARCH

147/DEL/2005 24-01-2005 248830 29-08-2011 A RELEASE PHARMACEUTICAL PREPARATION FOR JAMIA HAMDARD (HAMDARD COLON DELIVERY UNIVERSITY) 2403/KOLNP/2006 24-08-2006 248843 30-08-2011 ANTITHROMBOTIC COMPOUND SANOFI-AVENTIS 74/MUM/2005 24-01-2005 248852 31-08-2011 NOVEL OPTHALMIC COMBINATION OF GATIFLOXACIN CIPLA LIMITED AND PREDNISOLONE 1197/MUM/2006 28-07-2006 248853 31-08-2011 TOPICAL COMPOSITION FOR MINIMIZING HAIR LOSS HINDUSTAN UNILEVER LIMITED

1643/DELNP/2005 21-04-2005 248867 02-09-2011 AMIDE COMPOUNDS OF GENERAL FORMULA I AS MCH BOEHRINGER INGELHEIM PHARMA ANTAGONISTS GMBH & CO. KG. 3162/DELNP/2007 27-04-2007 248904 07-09-2011 QUINOLINE DERIVATIVES. F.HOFFMANN-LA ROCHE AG 1353/MUM/2006 28-08-2006 248977 19-09-2011 LIPIDIC NANOPARTICULATE BASED DOSAGE FORMS OF PATRAVALE VANDANA BHARAT ANTIPARASITICS AND ANTIINFECTIVES 2669/KOLNP/2007 18-07-2007 248983 19-09-2011 A SUBSTITUTED THIAZOLOPYRIDINONE COMPOUND ELI LILLY AND COMPANY USEFUL AS MELANIN CONCENTRATING HERMONE (MCH) ANTAGONISTS AND PHARMACEUTICAL COMPOSITION THEREOF 3008/DELNP/2007 23-04-2007 248995 20-09-2011 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR WAKUNAGA PHARMACEUTICAL CO., SALTS THEREOF LTD 2282/KOLNP/2006 10-08-2006 248998 20-09-2011 DERIVATIVES OF ALKYLPIPERAZINE- AND SANOFI-AVENTIS ALKYLHOMOPIPERAZINE- CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS 4047/DELNP/2004 20-12-2004 249008 21-09-2011 A PHARMACEUTICAL COMPOSITION COMPRISING A PFIZER PRODUCTS INC. TABLET CORE OR CAPSULE FILL 2997/KOLNP/2006 17-10-2006 249090 29-09-2011 PIPERAZINYLPIPERIDINE DERIVATIVES AS CYTOKINE INCYTE CORPORATION RECEPTOR ANTAGONISTS 3884/DELNP/2005 31-08-2005 249112 30-09-2011 AN ORALLY ADMINISTERED PHARMACEUTICAL MCNEIL AB FORMULATION 478/MUM/2006 29-03-2006 249133 03-10-2011 HERBAL COMPOSITION COMPRISING EXTRACT OF ROOT PIRAMAL LIFE SCIENCES LIMITED OF MURRAYA KOENIGII FOR TREATMENT OF INFECTIONS CAUSED BY DERMATOPHYTES 4188/DELNP/2005 16-09-2005 249157 05-10-2011 OXIDATIVE REDUCTIVE POTENTIAL WATER SOLUTION OCULUS INNOVATIVE SCIENCES, INC. AND PROCESSES FOR PRODUCING SAME 3208/DELNP/2006 05-06-2006 249171 10-10-2011 A PHARMACEUTICAL FORMULATION ADAPTED FOR BIONUMERIK PHARMACEUTICALS, INC. ADMINISTRATION TO HUMAN PATIENTS 1698/MUM/2007 05-09-2007 249181 10-10-2011 STABLE SOLID ORAL PHARMACEUTICAL COMPOSITIONS IPCA LABORATORIES LIMITED OF ISOTRETINOIN AND PROCESS THEREOF

4048/DELNP/2005 09-09-2005 249175 10-10-2011 AN ORAL PHARMACEUTICAL PREPARATION PIERRE FABRE MEDICAMENT 688/MUM/2005 08-06-2005 249183 10-10-2011 A TOPICAL SEMISOLID SILVER NANOPARTICLE SANJEEV KHANDELWAL DISPERSION FORMULATION 215/DEL/2006 25-01-2006 249180 10-10-2011 A HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR NAZFUDDAM AND A PROCESS FOR THE PREPARATION RESEARCH IN UNANI MEDICINE THEREOF" 218/DEL/2006 25-01-2006 249186 10-10-2011 A NOVEL HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR CORYZA AND A PROCESS FOR PREPARING THEREOF RESEARCH IN UNANI MEDICINE

1230/MUM/2006 03-08-2006 249226 12-10-2011 ION EXCHANGE RESIN BASED EXTENDED RELEASE AMIN, PURNIMA DHANRAJ GASTRO-RETENTIVE DOSAGE FORMS 5691/DELNP/2006 29-09-2006 249232 12-10-2011 MICROFLUIDIZED OIL-IN-WATER EMULSIONS AND PFIZER PRODUCTS INC. VACCINE COMPOSITIONS 1012/MUM/2006 27-06-2006 249243 12-10-2011 THE THROMBOCHEK TEST KIT DILIP SHRINIVAS VELASKAR 2128/MUM/2006 26-12-2006 249299 17-10-2011 A SYNERGISTIC HERBAL FORMULATION FOR THE PATANKAR SURESH TREATMENT OF RENAL CONDITION 2114/MUM/2006 22-12-2006 249293 17-10-2011 A MEDICAMENT FOR THE TREATMENT OF HIV SAYYED BAWA ABDUL KAREEM INFECTION, 3734/DELNP/2005 23-08-2005 249316 17-10-2011 AN AMINO-PYRIDINE COMPOUND OF FORMULA I SUGEN, INC., 2254/DELNP/2003 24-12-2003 249325 17-10-2011 A COMPOUND OF FORMULA (I) BAOSHUN LIU 515/MUMNP/2007 09-04-2007 249345 18-10-2011 CONVENIENTLY IMPLANTABLE SUSTAINED RELEASE RAMSCOR INC. DRUG COMPOSITIONS 2492/KOLNP/2006 31-08-2006 249558 25-10-2011 PHYSIOLOGICAL COOLING COMPOSITIONS CONTAINING MILLENNIUM SPECIALTY CHEMICALS HIGHLY PURIFIED ETHYL ESTER OF N-[[5-METHYL-2-(1- METHYLETHYL)CYCLOHEXYL)CARBONYL]GLYCINE

3827/KOLNP/2006 19-12-2006 249525 25-10-2011 NOVEL ARYLAMIDINE COMPOUND HAVING M/S TOYAMA CHEMICAL CO., LTD. ANTIFUNGAL AND ANTIPROTOZOAL ACTIVITY 1961/KOLNP/2006 12-07-2006 249527 25-10-2011 A PHARMACEUTICAL COMPOSITION RICHTER GEDEON VEGYESZETI GYAR RT

7358/DELNP/2006 06-12-2006 249562 27-10-2011 A FORMULATION PROVIDING ENHANCED ULTRASOUND ACUSPHERE  INC CONTRAST IMAGES AND A METHOD FOR MAKING THE SAME 4201/CHENP/2006 14-11-2006 249605 31-10-2011 A COMPOUND OF FORMULA I AS PPAR MODULATORS IRM LLC

1054/KOLNP/2007 26-03-2007 249614 31-10-2011 OPTICALLY ACTIVE 4,4-DI-SUBSTITUTED OXAZOLIDINE SANKYO COMPANY LIMITED DERIVATIVE AND PROCEDURES FOR THEIR PREPARATION 497/KOLNP/2006 03-03-2006 249626 31-10-2011 A NON-TRANSLUCENT OIL IN WATER EMULSION FOAMIX LTD. 1944/KOLNP/2006 11-07-2006 249627 31-10-2011 ARYLOXYALKYLCARBAMATE COMPOUNDS, SANOFI-AVENTIS PREPARATION METHOD THEREOF AND COMPOSITION COMPRSING THEM 1290/CHENP/2006 13-04-2006 249666 01-11-2011 IMIDAZOPYRAZINE TYROSINE KINASE INHIBITORS OSI PHARMACEUTICALS, INC. 2932/KOLNP/2006 11-10-2006 249679 02-11-2011 THIOAMIDE DERIVATIVES AS PROGESTERONE WYETH RECEPTOR MODULATORS 2938/KOLNP/2006 11-10-2006 249735 08-11-2011 CYANOPYRROLE CONTAINING CYCLIC CARBAMATE AND WYETH THIOCARBAMATE BIARYLS AND METHODS FOR PREPARING THE SAME 8001/DELNP/2006 29-12-2006 249742 08-11-2011 2-QUINAZOLINYLAMINOC1-6ALKANEDIYL COMPOUND JANSSEN PHARMACEUTICA N.V. AS PARP INHIBITORS 3206/KOLNP/2006 02-11-2006 249747 08-11-2011 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS ARENA PHARMACEUTICALS, INC. MODULATORS OF METABOLISM AND THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO.

2984/KOLNP/2006 16-10-2006 249754 08-11-2011 PURIFICATION OF PROGESTERONE RECEPTOR WYETH MODULATORS 1960/KOLNP/2006 12-07-2006 249758 08-11-2011 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB 4509/DELNP/2005 04-10-2005 249774 09-11-2011 A TWO-PART BICARBONATE CONTAINING SOLUTION. BAXTER INTERNATIONAL INC.

1960/MUM/2006 29-01-2007 249777 10-11-2011 PHARMACEUTICAL DERMAL COMPOSITION USEFUL IN VLIFE SCIENCES TECHNOLOGIES PVT. TREATMENT OF DIABETIC COMPLICATIONS LTD. 404/KOLNP/2007 05-02-2007 249810 14-11-2011 ACID AMIDE DERIVATIVE AND FUNGICIDAL ISHIHARA SANGYO KAISHA, LTD. COMPOSITION COMPRISING IT 194/KOLNP/2007 16-01-2007 249822 15-11-2011 N-(1H-INDOLYL)-1H-INDOLE-2-CARBOXAMIDE SANOFI-AVENTIS DERIVATIVES AND THEIR PREPARATION 1517/CHENP/2006 03-05-2006 249834 16-11-2011 STABLE PHARMACEUTICAL COMPOSITION COMPRISING LEK PHARMACEUTICALS d.d. GRANULOCYTE-COLONY STIMULATING FACTOR

1080/DELNP/2006 01-03-2006 249872 17-11-2011 MELT-FORMULATED, MULTIPARTICULATE ORAL GRUNENTHAL GMBH DOSAGE FORM IN/PCT/2000/322/KOL 18-09-2000 249892 21-11-2011 INHIBITORS OF CASPASES VERTEX PHARMACEUTICALS INCORPORATED 1963/KOLNP/2006 13-07-2006 249917 23-11-2011 NOVEL FUSED PYRROLOCARBAZOLES CEPHALON, INC 3798/KOLNP/2006 18-12-2006 249919 23-11-2011 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED 2761/KOLNP/2006 21-09-2006 249922 23-11-2011 NON-CYCLIC KETONES AND PERFUMING COMPOSITION FIRMENICH S.A. COMPRISING THEM 385/MUM/2007 28-02-2007 249929 23-11-2011 NOVEL COSMETIC CREAM COMPOSITIONS HINDUSTAN UNILEVER LIMITED 2544/DELNP/2004 31-08-2004 249968 25-11-2011 ACYLAMINOPIPERIDINE-1-CARBOXAMIDINE KALVISTA PHARMACEUTICALS LIMITED COMPOUND OF FOUMULA 1 5385/DELNP/2005 23-11-2005 250040 30-11-2011 A PHARMACEUTIACAL COMPOSITION OF PHARMA MAR S.A.U. ECTEINASCIDIN 743 (ET-743) IN COMBINATION WITH A PLATINUM COMPOUND WITHOUT INCREASING THE TOXICITY OF EACH DRUG 144/DELNP/2007 05-01-2007 250050 30-11-2011 AN ENANTIOMERICALLY PURE AMINOPYRIDINE PFIZER INC COMPOUND OF FORMULA (I) 3494/DELNP/2006 19-06-2006 250055 01-12-2011 AN OPHTHALMICALLY ACCEPTABLE COMPOSITION ALLERGAN, INC. 6179/DELNP/2006 23-10-2006 250059 01-12-2011 ”BIOCOMPATIBLE COMPOSITE PARTICLE OR NANOBIOTIX NANOPARTICLE AGGREGATE CAPABLE OF GENERATING FREE RADICALS OR HEAT” 1375/MUMNP/2006 16-11-2006 250088 05-12-2011 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES WITH ZENTARIS GMBH IMPROVED BIOLOOGICAL ACTION AND IMPROVED SOLUBILITY AS LIGANDS FOR G-PROTEIN COUPLED RECEPTORS (GPCRS) 2121/MUM/2007 26-10-2007 250095 07-12-2011 A STABLE ORAL FORMULATION CONTAINING A PROTON CADILA HEALTHCARE LIMITED PUMP INHIBITOR 2150/DELNP/2004 23-07-2004 250133 09-12-2011 A 4-(ARYLMETHYLOXY)-PYRIDIN-2-ONE COMPOUND" PHARMACIA CORPORATION 1340/MUM/2007 12-07-2007 250130 09-12-2011 A SUSTAINED RELEASE ANTIMALARIAL TABLET IPCA LABORATORIES LIMITED COMPOSITION COMPRISING PRIMAQUINE PHOSPHATE AND A PROCESS FOR PREPARING THE SAME

1233/KOLNP/2006 11-05-2006 250181 14-12-2011 MODULATORS OF CELLULAR ADHESION SARCODE CORPORATION 580/MUM/2003 06-06-2003 250249 19-12-2011 MODIFIED RELEASE PHARMACEUTICAL FORMULATION CADILA HEALTHCARE LIMITED CONTAINING FLUVASTATIN SODIUM

3348/DELNP/2007 04-05-2007 250251 20-12-2011 EYE DROP COMPRISING HOMOPIPERAZINE AND KOWA CO.,LTD PHOSPHORIC ACID OR THEIR SALTS THEREOF 2140/DELNP/2006 19-04-2006 250309 22-12-2011 COMPOUND USEFUL AS CCR-2 ANTAGONIST SALT MERCK SHARP & DOHME CORP. 4311/DELNP/2006 26-07-2006 250334 27-12-2011 AN AMINE SALT OF A 2-QUINOLINE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD 6170/DELNP/2007 07-08-2007 250384 30-12-2011 RINSE-OFF/WIPE-OFF SKIN CLEANSING COMPOSITION THE PROCTER & GAMBLE COMPANY

5178/DELNP/2007 05-07-2007 250392 30-12-2011 N-[(1S)-2-(DMETHYLAMINO)-1-PHENYLETHYL]-6,6- PFIZER INC. DIMITHYL-3-[(2-METHYLTHIENO[3,2-D]PYRIMDIN-4- YL)AMINO]-4,6-DIHYDROPYRROLO[3,4-C]PYRAZOLE- 5(1H) CARBOXAMIDE 3130/KOLNP/2006 27-10-2006 250430 03-01-2012 AMIDO COMPOUNDS AND THEIR USE AS INCYTE CORPORATION PHARMACEUTICALS 2112/KOLNP/2006 26-07-2006 250432 03-01-2012 FUSED CYCLIC SYSTEMS USEFUL AS INHIBITORS OF TEC VERTEX PHARMACEUTICALS FAMILY PROTEIN KINASES INCORPORATED 3348/KOLNP/2006 14-11-2006 250453 04-01-2012 PYRROLE COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED 2395/KOLNP/2006 23-08-2006 250461 04-01-2012 LYSINE BASED COMPOUNDS AMBRILIA BIOPHARMA INC. 3049/KOLNP/2006 20-10-2006 250462 04-01-2012 SUBSTITUTED AZEPINE DERIVATIVES AS ATHERSYS, INC. RECEPTOR MODULATORS 2683/KOLNP/2005 23-12-2005 250464 04-01-2012 ABUSE RESISTANT AMPHETAMINE COMPOUNDS NEW RIVER PHARMACEUTICALS INC 4483/KOLNP/2007 21-11-2007 250478 05-01-2012 PHARMACEUTICAL COMBINATION COMPRISING AN ADVANCED SCIENTIFIC DEVELOPMENTS ANTIFUNGAL AGENT AND AN ACTIVE SUBSTANCE SELECTED FROM CARVEOL, , , BORNEOL, , AND ALPHA- AND BETA- IONONES 3074/DELNP/2004 07-10-2004 250486 05-01-2012 " AND ADHYPERFORIN DERIVATIVES FOR INDENA S.P.A USE IN THE TREATMENT OF DEPRESSION AND ALZHEIMER'S DISEASE" 5093/DELNP/2007 02-07-2007 250488 05-01-2012 "2-CYCLOPENTEN-1-ONE OXIME DERIVATIVES AMOREPACIFIC CORPORATION INHIBITING PRODUCTION OF TNF-ALPHA" 2498/DEL/2006 20-11-2006 250538 09-01-2012 "A NOVEL HETEROCYCLEC CMPOUND XANTHONOXY HAMDARD UNIVERSITY PROPANOLAMINES" 6487/DELNP/2006 02-11-2006 250549 10-01-2012 "INDENE DERIVATIVES AND PROCESS FOR THE KOREA RESEARCH INSTITUTE OF PREPARATION THEREOF" CHEMICAL TECHNOLOGY 2027/KOLNP/2005 17-10-2005 250551 10-01-2012 NOVEL PHOSPHONIC ACID COMPOUNDS AS INHIBITORS ORTHO-MCNEIL PHARMACEUTICAL, OF SERINE PROTEASES INC. 3178/KOLNP/2006 31-10-2006 250552 10-01-2012 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED 2947/KOLNP/2006 12-10-2006 250556 10-01-2012 NOVEL COMPOUNDS (CAMPTOTHECIN DERIVATIVES SIGMA-TAU INDUSTRIE CONJUGATED IN POSITION 7 TO ANTI-INTEGRIN CYCLIC FARMACEUTICHE RIUNITE S.P.A. PEPTIDES) AS CYTOSTATIC AGENTS

2107/MUMNP/2008 01-10-2008 250583 11-01-2012 SUBSTITUTED PYRROLIDINONES AS INHIBITORS OF 11- ELI LILLY AND COMPANY BETA-HYDROXYSTEROID DEHYDROGENASE 1 2793/KOLNP/2006 25-09-2006 250594 11-01-2012 NOVEL COMPOUNDS AND COMPOSITION THEREOF AS ARYX T HERAPEUTICS ANTICOAGULANT 1653/DELNP/2006 27-03-2006 250598 11-01-2012 "A BODY-ABSORBABLE COMPOSITION" ORTHOCON, INC 3187/DEL/1998 29-10-1998 250614 12-01-2012 " MUTILIN 14-(EXO-8-METHYL-8-AZABICYCLO[3.2.1]OCT-SMITHKLINE BEECHAM LIMITED 3-YLSULFANYL)-ACETATE AND ITS SALT"

1343/KOLNP/2005 12-07-2005 250653 16-01-2012 HYDROXAMIC ACID COMPOUND NOVARTIS VACCINES AND DIAGNOSTICS INC. 2955/KOLNP/2006 12-10-2006 250673 18-01-2012 7-T-BUTOXYIMINOMETHYLCAMPTOTHECIN SIGMA-TAU INDUSTRIE CONJUGATED IN POSITION 20 WITH INTEGRIN FARMACEUTICHE RIUNITE S.P.A. ANTAGONISTS 6268/DELNP/2006 25-10-2006 250681 18-01-2012 "SOFTGEL ENCAPSULATED PHARMACEUTICAL THE PROCTER & GAMBLE COMPANY COMPOSITIONS COMPRISING CONCENTRATED ACTIVE INGREDIENTS" 216/DEL/2006 25-01-2006 250700 20-01-2012 ""A HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR ARTHRITIS AND TO PROCESS FOR THE PREPARATION RESEARCH IN UNANI MEDICINE THEREOF". 1321/CHENP/2007 30-03-2007 250702 20-01-2012 HYDROXYLAMINE ESTERS AS POLYMERIZATION CIBA HOLDING INC. INITIATORS 828/CAL/1999 06-10-1999 250728 23-01-2012 A COMPOUND OF PYRIDINIUM SERIES TORRENT PHARMACEUTICALS LTD. 901/MUM/2004 20-08-2004 250735 23-01-2012 NOVEL ANTIDIABETIC COMPOUNDS CADILA HEALTHCARE LIMITED 337/MUMNP/2007 06-03-2007 250747 23-01-2012 PURINE DERIVATIVES AS A3 AND A1 ADENOSINE GOVERNMENT OF THE UNITED STATES RECEPTOR AGONISTS OF AMERICA REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 406/DELNP/2005 02-02-2005 250752 24-01-2012 "3,6-DISUBSTITUTED AZABICYCLO [3.1.0]HEXANE RANBAXY LABORATORIES LIMITED DERIVATIVES USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS" IN/PCT/2001/00758/DEL 24-08-2001 250754 24-01-2012 "A PHARMACEEUTICAL COMPOSITION" TRIANGLE PHARMACEUTICALS, INC. 5055/DELNP/2006 01-09-2006 250758 24-01-2012 TETRAHYDROCARBAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG 3183/DELNP/2006 02-06-2006 250807 30-01-2012 "HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF ARRAY BIOPHARMA INC. USE THEREOF" 1511/CHENP/2006 03-05-2006 250824 31-01-2012 AQUEOUS SOLUTION OF CHROMIUM SALT AND NIPPON CHEMICAL INDUSTRIAL CO., METHOD FOR PRODUCING SAME LTD 3339/DELNP/2007 03-05-2007 250842 01-02-2012 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 SYNTA PHARMACEUTICALS CORP. ACTIVITY 2301/DELNP/2007 23-03-2007 250843 01-02-2012 "LIPOSOMAL COMPOSITIONS OF GLUCOCORTICOID YISSUM RESEARCH DEVELOPMENT AND GLUCOCORTICOID DERIVATIVES" COMPANY OF THE HERBREW UNIVERSITY OF JERUSALEM 2488/CHENP/2006 06-07-2006 250853 02-02-2012 DIAZA-SPIROPIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG 2284/DEL/2004 17-11-2004 250857 02-02-2012 "2-ETHYL-4,6-DIMETHYLPHENYL-SUBSTITUTED BAYER CROPSCIENCE AG, SPIROCYCLIC TETRAMIC ACID COMPOUNDS" 419/DEL/2002 28-03-2002 250881 03-02-2012 "A HERBAL OPHTHALMIC FORMULATION OF CURCUMA ALL INDIA INSTITUTE OF MEDICAL LONGA FOR DELAYING THE ONSET AND PROGRESSION SCIENCES, OF CATARACT" 1139/CHENP/2006 03-04-2006 250918 07-02-2012 ALKOXY SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY 2872/CHENP/2006 04-08-2006 250919 07-02-2012 MICROEMULSION FORMULATIONS COMPRISING NOVARTIS AG PARTICULAR ANTAGONISTS 3870/CHENP/2007 05-09-2007 250923 07-02-2012 ANALOGUES OF GLP-1 IPSEN PHARMA S.A.S 2395/CHENP/2007 04-06-2007 250971 14-02-2012 A COMPOSITION COMPRISING A SEQUESTERING AND A ALPHARMA, INC. THERAPEUTIC SUBUNIT 3320/CHENP/2006 13-09-2006 250977 14-02-2012 A METHOD OF DEACTIVATING DUST MITE ALLERGENS RECKITT BENCKISER (UK) LIMITED DER P AND DER F BY HOTPLATE EMANATION

2391/DEL/2004 30-11-2004 250983 14-02-2012 "A PHARMACEUTICAL COMPOSITION FOR JAMIA HAMDARD (HAMDARD TRANSDERMAL/TRANSMUCOSAL DELIVERY" UNIVERSITY) 1012/DELNP/2006 27-02-2006 251016 16-02-2012 "A PHARMACEUTICAL COMPOSITIONS SUITABLE FOR STIEFEL LABORATORIES, INC. TOPICAL ADMINISTRATION" 275/MUM/2004 07-03-2004 251029 17-02-2012 ORAL DROP FORMULATION CONTAINING SIMETHICONE SANJEEV KHANDELWAL AND CAMYLOFIN DIHYDRAOCHLORIDE

6498/DELNP/2007 22-08-2007 251035 17-02-2012 "A BENZOIMIDAZOLE COMPOUND AND DAEWOONG PHARMACEUTICAL CO., PHARMACEUTICAL COMPOSITION COMPRISING THE LTD. SAME" 1291/MUMNP/2006 03-11-2006 251055 20-02-2012 DERIVATIVES OF 14.15-DIHYDRO 20.21- BIOCORTECH DINOREBURNAMENIN-14-OL FOR TREATMENT OF DIPRESSIUON 2496/MUM/2007 18-12-2007 251063 21-02-2012 NOVEL SUBSTITUTED ARALKYL DERIVATIVES HAVING CADILA HEALTHCARE LIMITED ANTIDIABETIC HYPOLIPIDEMIC,HYPOCHOLESTEREMIC ACTIVITIES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN MEDICINE

3740/DELNP/2005 23-08-2005 251084 22-02-2012 "A PHARMACEUTICAL FORMULATION" CHIESI FARMACEUTICI S.P.A. 1117/DELNP/2006 02-03-2006 251092 22-02-2012 "A COMPOSITION OF AT LEAST TWO AMIDE-BASED NEW JAPAN CHEMICAL CO., LTD. COMPOUNDS REPRESENTED BY GENERAL FORMULA I"

1402/MUM/2006 01-09-2006 251100 22-02-2012 A NOVEL FORMULATION OF SEVELAMER USV LIMITED HYDROCHLORIDE 4715/DELNP/2007 19-06-2007 251113 24-02-2012 "MATRIX TYPE SUSTAINED-RELEASE PREPARATION EISAI R & D MANAGEMENT CO.,LTD CONTAINING BASIC DRUG OR SALT THEREOF, AND METHOD FOR MANUFACTURING THE SAME" 1867/DELNP/2007 09-03-2007 251123 24-02-2012 "A MIXTURE OF FISH OIL FATTY ACID ESTER(S) OF ENZYMOTEC LTD. PHYTOSTEROLS AND 1,3-(S) (DAG)" 745/MUM/2004 12-07-2004 251135 27-02-2012 NOVEL HETEROCYCLIC COMPOUNDS CADILA HEALTHCARE LIMITED 304/KOLNP/2007 25-01-2007 251140 27-02-2012 A COMPOSITION FOR A CAPSULE COATING WAKUNAGA PHARMACEUTICAL CO., LTD. 2013/DELNP/2007 15-03-2007 251142 27-02-2012 "A CYCLIC AMINE DERIVATIVE OR SALT THEREOF AND ASTELLAS PHARMA INC. ITS PHARMACEUTICAL COMPOSITION" 177/MUMNP/2007 05-02-2007 251154 28-02-2012 NEW SELENOHYDROXY ACIDS AND THEIR DERIVATIVES TETRAHEDRON APPLICATIONS IN NUTRITION, COSMETICS AND PHARMACEUTICS 2418/MUM/2007 10-12-2007 251161 28-02-2012 NOVEL OMEGA -3 FATTY ACID COMPOSITION WITH OMNIACTIVE HEALTH TECHNOLOGIES SIGNIFICANTLY REDUCED OFFENSIVE ODOUR AND PVT. LTD. PROCESS FOR ITS PREPARATION 1976/MUMNP/2008 16-09-2008 251162 28-02-2012 BICYCLOHETEROARYL COMPOUNDS AS P2X7 RENOVIS, INC. MODULATORS AND USES THEREOF 1378/MUMNP/2006 16-11-2006 251169 28-02-2012 GUANYLHYDRAZONE SALTS, COMPOSITIONS, CYTOKINE PHARMASCIENCES INC. PROCESSES OF MAKING AND METHODS OF USING 1638/CHENP/2006 11-05-2006 251191 29-02-2012 ORTHO-SUBSTITUTED PENTAFLUORIDE SULFANYL- SANOFI-AVENTIS DEUTSCHLAND GMBH BENZENES, METHOD FOR THE PRODUCTION THEREOF AND THE THEREOF 2118/CHENP/2006 15-06-2006 251196 29-02-2012 COMPOSITION FOR COUPLING FILLER AND ELASTOMER CIBA HOLDING INC.

610/CHE/2006 03-04-2006 251197 29-02-2012 NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITORS, MATRIX LABORATORIES LTD. PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

7041/DELNP/2007 12-09-2007 251204 29-02-2012 "A HETEROCYCLIC COMPOUND REPRESENTED BY THE OTSUKA PHARMACEUTICAL CO., LTD. FORMULA(1)" 3795/DELNP/2004 01-12-2004 251219 01-03-2012 "BASIC NON-PEPTIDE ANTAGONISTS MENARINI RICERCHE S.P.A. CONTAINING QUINOLINE AND A NITROGEN HETEROCYCLE" 1331/CHENP/2003 25-08-2003 251226 02-03-2012 SALTS OF AVERMECTINS SUBSTITUTED IN THE 4"- SYNGENTA PARTICIPATIONS AG POSITION AND HAVING PESTICIDAL PROPERTIES" 712/DELNP/2006 13-02-2006 251234 02-03-2012 "AN α-2A/α-1A SELECTIVE AGONIST, 1-(2,3- ALLERGAN, INC. DIMETHYL-PHENYL)-ETHYL-1,3-DIHYDRO-IMIDAZOLE-2- THIONE COMPOUND" 1838/CHENP/2004 18-08-2004 251236 02-03-2012 PHARMACEUTICAL FORMULATIONS OF SCHERING CORPORATION TEMOZOLOMIDE 2130/KOLNP/2007 12-06-2007 251257 05-03-2012 POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY 1734/CHE/2007 07-08-2007 251268 05-03-2012 SOLID DOSAGE FORM OF ENTERIC SOLID DISPERSION SHIN-ETSU CHEMICAL CO., LTD AND METHOD FOR PRODUCING THE SAME

1835/CHENP/2007 30-04-2007 251278 05-03-2012 PYRIMIDONE COMPOUND MITSUBISHI PHARMA CORPORATION, SANOFI- AVENTIS 1170/DEL/1998 01-05-1998 251314 06-03-2012 "PHARMACEUTICAL COMPOSITION WITH FDXED FERRER INTERNACIONAL S.A. QUANTITIES OF AN EPNALARIL AND NITRENDIPINE AND METHOD FOR OBTAINING THE SAME" 710/CHENP/2007 19-02-2007 251320 06-03-2012 3-SUBSTITUTED-5-AND 6-AMINOALKYL INDOLE-2- AVENTIS PHARMACEUTICALS, INC CARBOXYLIC ACID AMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE Ie 3006/DELNP/2004 01-10-2004 251447 16-03-2012 "A PHARMACEUTICAL COMPOSITION USEFUL FOR SINCLAIR PHARMACEUTICALS LIMITED TOPICAL ADMINISTRATION COMPRISING AS ACTIVE INGREDIENTS PROANTHOCYANIDINS" 3359/DELNP/2004 29-10-2004 251451 16-03-2012 "HYDROXAMIC ACID COMPOUNDS COMPRISING A TOPOTARGET UK (LIMITED) PIPERAZINE LINKAGE AS HDAC INHIBITORS" 1862/DEL/2006 21-08-2006 251453 16-03-2012 "A NOVEL HERBAL COMPOSITION AND A PROCESS FOR CENTRAL COUNCIL FOR RESEARCH IN PREPARATION THEREOF EFFECTIVE AGAINST UNANI MEDICINE CONSTIPATION" 15/MUMNP/2005 10-01-2005 251454 16-03-2012 FLAVONE DERIVATIVES AS INHIBITORS OF CYCLIN- NICHOLAS PIRAMAL INDIA LIMITED DEPENDENT KINASES 1374/DEL/2007 27-06-2007 251457 16-03-2012 "NAPHTHALENE COMPOUNDS OF FORMULA (I)" LES LABORATOIRES SERVIER 2269/CHENP/2006 22-06-2006 251463 19-03-2012 A PHARMACEUTICAL COMPOSITION COMPRISING AN LEK PHARMACEUTICALS D.D. ACTIVE PRINCIPLE AND SULPHOBETAINE 431/CAL/1999 10-05-1999 251480 20-03-2012 INHIBITORS OF p38 VERTEX PHARMACEUTICALS INCORPORATED 8276/DELNP/2007 26-10-2007 251484 20-03-2012 "PYRROLIDINE COMPOUND OF GENERAL FORMULA(I)" OTSUKA PHARMACEUTICAL CO., LTD.,

1850/KOLNP/2005 16-09-2005 251492 20-03-2012 A NASAL PHARMACEUTICAL FORMULATION MERCK PATENT GMBH 1192/DEL/2002 27-11-2002 251502 21-03-2012 "A COMPOSITION COMPRISING COMPONENT A AND ROHM AND HAAS COMPANY COMPONENT B" 2104/MUMNP/2008 30-09-2008 251513 21-03-2012 BIPHENYL AMIDELACTAM DERIVATIVES AS INHIBITORS ELI LILLY AND COMPANY OF 11 - BETA - HYDROXYSTEROID DEHYDROGENASE 1

1684/MUM/2008 08-08-2008 251524 21-03-2012 A NOVEL PHARMACEUTICAL COMPOSITION OF TOPICAL MRS. ANURADHA MAJUMDAR METHOTREXATE GEL IN CHRONIC INFLAMMATORY CONDITION 4926/KOLNP/2007 19-12-2007 251525 21-03-2012 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY THERAPEUTIC USES 1885/DEL/2005 20-07-2005 251564 23-03-2012 "COMPOSITIONS WITH CYCLOPROPENES AND METAL- ROHM AND HAAS COMPANY COMPLEXING AGENTS" 1796/KOLNP/2007 21-05-2007 251577 26-03-2012 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT TOYAMA CHEMICAL CO., LTD. THEREOF 3158/DEL/2005 25-11-2005 251579 26-03-2012 "NOVEL LOGANIN ANALOGUES AND A PROCESS FOR COUNCIL OF SCIENTIFIC & INDUSTRIAL THE PREPARATION THEREOF" RESEARCH 5293/DELNP/2006 13-09-2006 251580 26-03-2012 "COMPOSITIONS AND METHODS FOR REDUCING OR NESTEC S.A. PREVENTING OBESITY" IN/PCT/2002/00308/MUM 13-03-2002 251589 26-03-2012 CICLESONIDE CONTAINED PHARMACEUTICAL NYCOMED GMBH, COMPOSITION FOR APPLICATION TO MUCOSA 1770/MUM/2008 22-08-2008 251593 26-03-2012 A MICROEMULSION BASED INTRANASAL DRUG AMRITA BAJAJ DELIVERY SYSTEM AND METHOD FOR PREPARATION THEREOF 1701/MUMNP/2008 07-08-2008 251601 26-03-2012 MICROTABLET-BASED PHARMACEUTICAL PREPARATION BIOGENERICS PHARMA GMBH

2876/KOLNP/2007 07-08-2007 251605 26-03-2012 SUBSTITUTED THIOPHENES AS GLUCAGON RECEPTOR ELI LILLY AND COMPANY ANTAGONISTS 2238/CHENP/2006 21-06-2006 251654 27-03-2012 A PHARMACEUTICAL COMPOSITION AND A METHOD DAIICHI SANKYO COMPANY, LIMITED FOR PROLIFERATING CARDIOMYOCYTES 5502/DELNP/2007 17-07-2007 251668 27-03-2012 "A 4"-SUBTITUTED 8A OR 9A-LACTAM 15-MEMBERED GLAXO GROUP LIMITED. MACROLIDE COMPOUND OF FORMULA (I)"

2966/DELNP/2007 20-04-2007 251671 27-03-2012 ALKIL-PYRIDINE COMPOUNDS F.HOFFMANN-LA ROCHE AG 2626/MUMNP/2008 10-12-2008 251679 28-03-2012 HETEROCYCLIC NON-NUCLEOSIDE COMPOUNDS, SHANGHAI INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF SCIENCES 5889/DELNP/2007 27-07-2007 251739 30-03-2012 "A QUINAZOLINE DERIVATIVE" HANMI HOLDINGS CO., LTD. 2970/KOLNP/2007 14-08-2007 251793 03-04-2012 SUBSTITUTED IMIDAZO[1,2-b] PYRIDAZINE COMPOUND ELI LILLY AND COMPANY

7324/DELNP/2006 05-12-2006 251800 03-04-2012 "3-{(3R,4R)-4-METHYL-3-[METHYL-(7H-PYRROLO[2,3- PFIZER PRODUCTS INC D]PYRIMIDIN-4-YL)-AMINO]-PIPERIDIN-1-YL}-3-OXO- PROPIONITRILE MONO CITRATE SALT AND ITS METHOD OF PREPARATION" 781/DEL/2003 05-06-2003 251801 04-04-2012 "A FEXOFENADINE-CARBOMER COMPLEX" M/S. IND-SWIFT LIMITED 910/MUMNP/2008 06-05-2008 251804 04-04-2012 NERAMEXANE MODIFIED RELEASE MATRIX TABLET MERZ PHARMA GMBH & CO. KGAA 613/MUMNP/2009 30-03-2009 251805 04-04-2012 1, 5-DIPHENYL-3-PYRIDINYLAMINO-1, 5- ELI LILLY AND COMPANY DIHYDROPYRROLIDIN-2-ONE AS CB1 203/CHENP/2008 11-01-2008 251826 10-04-2012 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS F. HOFFMANN-LA ROCHE AG VIA RECEPTOR ANTAGONISTS 8313/DELNP/2007 29-10-2007 251828 10-04-2012 "MOTILIDE COMPOUNDS" PFIZER INC. 949/MUMNP/2006 10-08-2006 251841 11-04-2012 EXTENDED RELEASE COATED MINITABLETS OF ALEMBIC LIMITED HYDROCHLORIDE 2474/KOLNP/2006 30-08-2006 251854 12-04-2012 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED 1816/KOLNP/2007 22-05-2007 251857 12-04-2012 A LUBRICANT COMPOSITION HCB HAPPY CHILD BIRTH HOLDING AG.

5334/DELNP/2006 14-09-2006 251863 12-04-2012 "PHARMACEUTICAL COMPOSITION AND PROCESS FOR SOLVAY PHARMACEUTICALS GMBH. THEIR PREPARATION" 4253/CHENP/2006 17-11-2006 251875 12-04-2012 NOVEL CIS-IMIDAZOLINES HAVING ANTIPROLIFERATIVE F. HOFFMANN-LA ROCHE AG ACTIVITY IN/PCT/2000/00792/MUM 29-12-2000 251878 13-04-2012 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS IDUN PHARMACEUTICALS, INC., INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES 5209/DELNP/2007 06-07-2007 251908 17-04-2012 "SUBSTITUTED TRIAZOLE COMPOUNDS AS OXYTOCIN PFIZER LIMITED ANTAGONISTS" IN/PCT/2002/484/KOL 18-04-2002 251919 17-04-2012 QUINOLINE DERIVATIVES FOR THE TREATMENT OF ACTIVE BIOTECH AB MALIGNANT TUMORS 305/KOLNP/2007 25-01-2007 251921 17-04-2012 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR METHYLGENE, INC. SIGNALING 3362/DELNP/2007 04-05-2007 251922 17-04-2012 "A BOTANICAL DRUG SUBSTANCE OBTAINABLE FROM GW PHARMA LIMITED BOTANICAL RAW MATERIAL" 7575/DELNP/2007 03-10-2007 251929 18-04-2012 A PHARMACUTICAL COMPOSITION CONTAINING WARNER CHILCOTT COMPANY,LLC RISEDRONATE 2888/KOLNP/2006 06-10-2006 251939 18-04-2012 SUBSTITUTED ORGANOSULFUR COMPOUNDS AND ACEA BIOSCIENCES INC. PHARMACEUTICAL COMPOSITION COMPRISING THEM

4769/KOLNP/2007 10-12-2007 251944 18-04-2012 FORMULATION OF A THIENOPYRIDINE PLATELET ELI LILLY AND COMPANY AGGREGATION INHIBITOR 2052/KOLNP/2006 21-07-2006 251946 18-04-2012 NOVEL FUSED PYRROLOCARBAZOLES CEPHALON, INC. 436/KOLNP/2007 07-02-2007 251952 18-04-2012 METHOD AND COMPOSITION FOR HIGH LEVEL NANOSONICS PTY LIMITED DISINFECTION EMPLOYING QUATERNARY AMMONIUM COMPOUNDS 232/KOLNP/2007 18-01-2007 251957 18-04-2012 "NEW 4-BENZYLIDENE-PIPERIDIN DERIVATIVES" RICHTER GEDEON VEGYÉSZETI GYÁR RT.

1308/KOLNP/2008 01-04-2008 251964 18-04-2012 CYCLIC AMINE COMPOUNDS AND PESTICIDAL NIPPON SODA CO., LTD. COMPOSITION COMPRISING THEM 5059/DELNP/2006 01-09-2006 251968 18-04-2012 "A FUSED HETEROCYCLE DERIVATIVE AND KISSEI PHARMACEUTICAL CO., LTD PHARMACEUTICAL COMPOSITION COMPRISING THE SAME" 3400/DELNP/2007 07-05-2007 251979 19-04-2012 "HETEROCYCLIC COMPOUNDS SUITABLE FOR TREATING ABBOTT GMBH & CO. KG DISORDERS THAT RESPOND TO MODULATION OF THE D3 RECEPTOR" 4247/DELNP/2006 24-07-2006 251981 19-04-2012 A STABLE SOLID PHARMACEUTICAL COMPOSITION ACTIVE BIOTECH AB CONTAINING QUINOLINE COMPOUNDS AND PROCESS THEREOF 2453/KOLNP/2006 29-08-2006 251984 19-04-2012 CHEMICALLY STABLE COMPOSITIONS OF 4- HYDROXY LABORATOIRES BESINES TAMOXIFEN INTERNATIONAL 3547/DELNP/2006 20-06-2006 251990 19-04-2012 "AN AZABICYCLO-INDAZOLE COMPOUND" MEMORY PHARMACEUTICALS CORPORATION 6842/DELNP/2006 16-11-2006 252033 23-04-2012 "COMPOUNDS AND COMPOSITIONS AS PROTEIN IRM LLC KINASE INHIBITORS" 1943/KOLNP/2006 11-07-2006 252043 23-04-2012 ACYLAMINOTHIAZOLE DERIVATIVES AND USE THEREOF SANOFI-AVENTIS AS BETA-AMYLOID INHIBITORS 2332/KOLNP/2006 17-08-2006 252044 23-04-2012 "DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, SANOFI AVENTIS PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS" 2877/DELNP/2006 22-05-2006 252046 23-04-2012 "A COMPOUND OF 1-BENZYLAMINO-2CARBAMOYL- NEWRON PHARMACEUTICALS S.P.A CYELOPENTANE DERIVATIVES OF FORMULA 1" 1462/KOLNP/2005 27-07-2005 252078 25-04-2012 A MEDICAMENT FOR THE PROPHYLAXIS AND DAIICHI SANKYO COMPANY LIMITED TREATMENT OF ARTERIOSCLEROSIS AND HYPERTENSION 3325/KOLNP/2006 13-11-2006 252091 25-04-2012 PHARMACEUTICAL TABLETS HAVING A RELATIVELY ACCU-BREAK TECHNOLOGIES INC. INACTIVE SEGMENT 605/KOLNP/2007 20-02-2007 252108 25-04-2012 2-DEOXY-2-FLUORO-2-METHYL-D-RIBONOLACTONE PHARMASSET, INC. DERIVATIVES AND PROCESS FOR PREPARATION OF THE SAME 2306/KOLNP/2007 22-06-2007 252109 25-04-2012 NOVEL RECEPTOR ANTAGONISTS OF MELANIN ELI LILLY AND COMPANY CONCENTRATING HORMONE 1646/CHENP/2006 11-05-2006 252114 26-04-2012 PENTAFLUOROSULFANYL BENZOYLGUANIDINES, SANOFI-AVENTIS DEUTSCHLAND GMBH METHOD FOR THEIR PRODUCTION, THEIR USE AS MEDICAMENTS OR DIAGNOSTIC AGENTS AND MEDICAMENT CONTAINING THE SAME 2774/DELNP/2006 17-05-2006 252120 26-04-2012 "NOVEL PHENOL DERIVATIVES AND ARIGEN PHARMACEUTICALS INC., ANTITRYPANOSOMA PREVENTIVE/THERAPEUTIC AGENT COMPRISING THE SAME AS ACTIVE INGREDIENT"

1825/MUMNP/2009 01-10-2009 252131 27-04-2012 TRIAZOLYL AMINOPYRIMIDINE COMPOUNDS ELI LILLY AND COMPANY 7959/DELNP/2006 28-12-2006 252132 27-04-2012 "A SUBSTITUTED 2-ALKYL QUINAZOLINONE DERIVATIVE JANSSEN PHARMACEUTICA N.V OF FORMULA (I)" 702/MUMNP/2009 13-04-2009 252133 27-04-2012 TETRAHYDROCYCLOPENTA[B] INDOLE COMPOUNDS AS ELI LILLY AND COMPANY ANDROGEN RECEPTOR MODULATORS

2825/DELNP/2004 22-09-2004 252137 27-04-2012 "THIOXANTHINE DERIVATIVES AS MYELOPEROXIDASE ASTRAZENECA AB INHIBITORS" 4429/DELNP/2006 01-08-2006 252144 30-04-2012 "N-DEACETYLTHIOCOLCHICINE DERIVATIVES, THEIR USE INDENA S.P.A. AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM" 4298/DELNP/2005 22-09-2005 252150 30-04-2012 "PYRROLE COMPOUNDS AS MODULATORS OF MERCK & CO. INC. METABOTROPIC GLUTAMATE RECEPTOR-5" 5054/DELNP/2006 01-09-2006 252159 30-04-2012 PYRAZOLYL INDOLYL COMPOUNDS F. HOFFMANN-LA ROCHE AG 1863/DEL/2006 21-08-2006 252163 30-04-2012 "A NOVEL HERBAL COMPOSITION AND A PROCESS FOR CENTRAL COUNCIL FOR RESEARCH IN PREPARATION THEREOF EFFECTIVE AGAINST UNANI MEDICINE ABDOMINAL WORM ." 2724/DEL/2005 10-10-2005 252167 30-04-2012 OXY SUBSTITUTED CHALCONES AS COUNCIL OF SCIENTIFIC AND ANTIHYPERGLYCEMIC AND ANTIDYSLIPIDEMIC AGENTS INDUSTRIAL RESEARCH

1518/DELNP/2005 15-04-2005 252201 01-05-2012 "A PHARMACEUTICAL COMPOSITION" FICAAR INC. 3229/CHENP/2006 05-09-2006 252203 01-05-2012 DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 F. HOFFMANN-LA ROCHE AG ANTAGONISTS 2452/CHENP/2006 05-07-2006 252204 01-05-2012 POLYPEPTIDES OF ALICYCLOBACILLUS SP NOVOZYMES A/S 649/MUMNP/2006 06-06-2006 252206 01-05-2012 PHARMACEUTICAL COMPOSITION CONTAINING Senju Pharmaceutical Co.Ltd. PROSTAGLANDIN 3263/DEL/2005 05-12-2005 252211 01-05-2012 "NATURAL CALCLUM CARBONATE TOOTHPOWDER COLGATE-PALMOLIVE COMPANY COMPOSITIONS" 188/DELNP/2003 19-02-2003 252221 02-05-2012 " HARD CAPSULE PREPARED FROM POLYMERIZABLE NISSHIN KASEI CO., LTD., VINYL MONOMER OF FORMULA H2C=C(R1)-COOR2 "

1473/KOLNP/2006 31-05-2006 252229 02-05-2012 NOVEL NITROPHENYL AND AUCKLAND UNISERVICES LIMITED NITROPHENYLAZIRIDINE ALCOHOLS AND THEIR CORRESPONDING PHOSPHATES AND THEIR USE AS TARGETED CYTOTOXIC AGENT 3549/DELNP/2006 20-06-2006 252268 04-05-2012 "COBALAMINE DERIVATIVES USEFUL FOR DIAGNOSIS SOLIDAGO AG. AND TREATMENT OF ABNORMAL CELLULAR PROLIFERATION " 2201/CHENP/2006 19-06-2006 252274 04-05-2012 IMMUNOSTIMULANT COMPOSITION COMPRISING AT SANOFI PASTEUR LEAST ONE TOLL-LIKE RECEPTOR 7 OR TOLL-LIKE RECEPTOR 8 AGONIST AND A TOLL-LIKE RECEPTOR 4 AGONIST 1267/CHENP/2006 13-04-2006 252299 08-05-2012 AMINOALKANOL DERIVATIVES NOVARTIS AG 1661/KOLNP/2006 15-06-2006 252305 08-05-2012 A PHARMACEUTICAL COMPOSITION MERCK EPROVA AG 1295/KOLNP/2007 12-04-2007 252311 08-05-2012 NOVEL COMPOUNDS AS BRADYKININ RECEPTOR ISTITUTO LUSO FARMACO D'ITALIA ANTAGONIST AND COMPOSITION THEREFROM S.P.A. 3127/DEL/2005 23-11-2005 252316 08-05-2012 "A HERBAL HEALTH FORMULATION" Three-N-Products Pvt. Ltd. 1980/KOLNP/2007 01-06-2007 252351 09-05-2012 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AND FERRER INTERNACIONAL S.A. COMPOSITIONS 352/CHENP/2008 22-01-2008 252366 10-05-2012 IMPROVED POLYSACCHARIDE-BASED SOLID GRANULES RHODIA OPERATIONS

1724/CHENP/2006 17-05-2006 252367 10-05-2012 DIPEPTIDYL PEPTIDASE IV INHIBITORS COMPOSITION NOVARTIS AG

2319/DELNP/2007 26-03-2007 252371 10-05-2012 INDOZOLONE DERIVATIVES AS 11B-HSD 1 INHIBITORS H.HOFFMANN-LA ROCHE AG

3432/CHENP/2006 19-09-2006 252374 11-05-2012 A PEPTIDE COMPOSITION FOR IMMUNE DIAGNOSTIC ISTITUTO NAZIONALE PER LE MALATTIE ASSAY TO DIAGNOSE AND MONITOR TUBERCULOSIS INFETTIVE "LAZZARO SPALLANZANI" INFECTION IRCCS 2247/KOLNP/2006 08-08-2006 252397 14-05-2012 NOVEL COMPOUNDS FOR INHIBITING FAAH ENZYME, SANOFI AVENTIS PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME 3563/KOLNP/2006 28-11-2006 252407 14-05-2012 SUBSTITUTED INDAZOLES, COMPOSITIONS AVENTIS PHARMA SA CONTAINING SAME, PREPARATION AND USE IN/PCT/2001/31/KOL 09-01-2001 252425 15-05-2012 QUINOLINE DERIVATIVES ACTIVE BIOTECH AB 506/MUMNP/2009 12-03-2009 252432 15-05-2012 SUBSTITUTED THIAZOLE PYRAZOLOPYRIMIDINE ELI LILLY AND COMPANY COMPOUNDS AS CRF1 RECEPTOR ANTAGONISTS 499/MUMNP/2009 09-03-2009 252439 16-05-2012 “THIOPHENE PYRAZOLOPYRIMIDINE COMPOUNDS” ELI LILLY AND COMPANY

380/MUMNP/2009 18-02-2009 252441 16-05-2012 “COMBINATION OF MODAFINIL AND AN ANTAGONIST BIOPROJET OR INVERSE AGONIST OF THE H3 RECEPTOR”

3557/DELNP/2006 20-06-2006 252445 16-05-2012 "PHOSPHONATES, MONOPHOSPHONAMIDATES, GILEAD SCIENCES, INC. BISPHOSPHONAMIDATES FOR THE TREATMNET OF VIRAL DISEASES " 1282/MUMNP/2007 22-08-2007 252449 16-05-2012 COMPOSITION FOR REDUCING THE EXUDATION OF THE CHOI SEONG-HYUN SERUM PROTEINS 3624/DELNP/2006 23-06-2006 252466 16-05-2012 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE NOVO NORDISK A/S ACTIVATORS 2448/DEL/2005 12-09-2005 252478 17-05-2012 "SUSTAINED RELEASE SYRUP COMPOSITION AND DELHI INSTITUTE OF PHARMACEUTICAL PROCESS THEREOF" SCIENCES & RESEARCH

3854/DELNP/2006 05-07-2006 252483 17-05-2012 "MICROCYCLIC PROLINE ANALOGUES AS HCV NS-3 MEDIVIR AB SERINE PROTEASE INHIBITORS" 7656/DELNP/2007 05-10-2007 252486 17-05-2012 "THE COMPOUND OF 1-METHYL-1H-IMIDAZOLE-4- PFIZER PRODUCTS INC. CARBOXYLIC ACID (3-AZA-BICYCLO[3.1.0]HEX-6- YLMETHYL)-(3-CHLORO-4-FLUORO-BENZYL)-AMIDE" 2978/DELNP/2008 10-04-2008 252491 18-05-2012 "IONTOPHORETIC PREPARATION FOR TREATMENT OF KOWA CO. , LTD. BREAST CANCER AND/OR MASTITIS" 697/DELNP/2004 18-03-2004 252493 18-05-2012 "A COMPOSITION COMPRISING AN ISOMERIC MEXTURE PALADIN LABS INC. OF A CYCLOSPORINE ANALOGUE' 2702/DELNP/2004 14-09-2004 252499 18-05-2012 "A SUBSTITUTED BENZIMIDAZOLE SULFONAMIDE TIBOTEC PHARMACEUTICALS LTD COMPOUND AND A PHARMACEUTICAL COMPOSITION COMPRISING THE SAME" 4837/DELNP/2007 22-06-2007 252509 21-05-2012 PHARMACEUTICAL , THERAPEUTIC, AND DIETARY RENAISSANCE HERBS, INC. COMPOSITIONS DERIVED FROM LEAVES OF LAGERSTROEMIA SPECIOSAL I. PLANT 7590/DELNP/2006 15-12-2006 252518 21-05-2012 "AMINOCYCLOHEXANES AS DIPEPTIDYL PEPTIDASE-IV MERCK SHARP & DOHME CORP. INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES" 1521/DELNP/2007 26-02-2007 252533 21-05-2012 INDOLE COMPOUNDS COMRISING AN ACETYLENE F. HOFFMANN-LA-ROCHE AG GROUP AS PPAR ACTIVATORS 8778/DELNP/2007 15-11-2007 252535 21-05-2012 "PHARMACEUTICAL COMPOSITION COMPRISING AN ADVANCED SCIENTIFIC DEVELOPMENTS ANTIVIRAL AGENT, AN ANTITUMORAL AGENT OR AN ANTIPARASITIC AGENT, AND AN ACTIVE AGENT SELECTED AMONG CARVEOL, THYMOL, EUGENOL, BORNEOL AND CARVACROL" 9905/DELNP/2007 20-12-2007 252541 21-05-2012 "MAO-B INHIBITORS USEFUL FOR TREATING OBESITY" JENRIN DISCOVERY

963/MUMNP/2009 14-05-2009 252549 22-05-2012 “IMIDAZOLIDINONYL AMINOPYRIMIDINE ELI LILLY AND COMPANY COMPOUNDS" 855/MUM/2006 01-06-2006 252567 23-05-2012 A PROCESS FOR PREPARATION OF A POLYHERBAL CHARAK PHARMA PRIVATE LIMITED COMPOSITION AND THE PRODUCT THEREOF 1931/MUMNP/2008 08-09-2008 252574 23-05-2012 CAMPTOTHECIN DERIVATIVES SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES 1/DEL/2004 01-01-2004 252589 23-05-2012 "SOLID PHASE BENZOPYRAN COMPOSITION, PROCESS INTERNATIONAL FLAVORS & FOR PREPARING SAME" FRAGRANCES INC. 1314/DEL/2004 16-07-2004 252592 23-05-2012 A TOPICAL FORMULATION FOR PREVENTION AND THE DIRECTOR GENERAL MANAGEMENT OF PERIPHERAL VASCULAR DISEASES AND A PROCESS OF PREPARATION THEREOF

5248/DELNP/2007 06-07-2007 252599 23-05-2012 "ORAL COMPOSITIONS CONTAINING BIPHENOL COLGATE-PALMOLIVE COMPANY ANTIBACTERIAL COMPOUNDS" 6544/DELNP/2006 06-11-2006 252605 23-05-2012 "A 2-PYRROLIDIN-OR-2-PIPERIDINONE DERIVATIVE OF JANSSEN PHARMACEUTICA N.V., FORMULA (I)" 26/MUMNP/2009 02-01-2009 252606 23-05-2012 GLUCOCORTICOID RECEPTOR MODULATOR ELI LILLY AND COMPANY 3402/DELNP/2004 02-11-2004 252607 23-05-2012 "HYDROXY TETRAHYDRO-NAPHTHALENYLUREA XENTION LIMITED., DERIVATIVES" 2936/CHENP/2006 10-08-2006 252617 24-05-2012 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG 999/DELNP/2006 24-02-2006 252629 24-05-2012 "HETEROARYL-TETRAHYDROPIPERIDYL COMPOUNDS EUROCELTIQUE S. A. USEFUL FOR TREATING OR PREVENTING PAIN"

3727/DELNP/2006 28-06-2006 252647 25-05-2012 "A COMPOSITION CONTAINING A LYOPHILISATE OF BIOTECHMARINE. DEDIFFERENTIATED PLANT CELLS FOR SKIN DEPIGMENTATION" 4015/DELNP/2004 16-12-2004 252658 25-05-2012 " A PHARMACEUTICAL COMPOSITION FOR THE FIDELINE TREATMENT OF STRESS IN AN AVIAN" 7188/DELNP/2006 29-11-2006 252687 28-05-2012 "A PHARMACEUTICAL COMPOSITION COMPRISING M3 ALMIRALL S.A. ANTAGONIST AND B2-AGONIST FOR USE IN THE RESPIRATORY DISORDERS" 272/MUMNP/2006 08-03-2006 252689 28-05-2012 6-CYCLOAMINO-2-QUINOLINONE DERIVATIVES AS LIGAND PHARMACEUTICALS ANDROGEN RECEPTOR MODULATOR COMPOUNDS INCORPORATED 3341/DELNP/2004 27-10-2004 252695 28-05-2012 A COMPOSITION FOR THE TREATMENT OF OBESITY DUKE UNIVERSITY 705/DELNP/2006 13-02-2006 252720 29-05-2012 " CARBONATE GRANULATION" DELAVAU L.L.C 1848/CHENP/2006 25-05-2006 252776 30-05-2012 COMPOUNDS WITH SUBSTITUTED IMIDAZO RING 3M INNOVATIVE PROPERTIES SYSTEMS COMPANY 951/MAS/2002 18-12-2002 252779 30-05-2012 NOVEL TETRACYCLIC 3-SUBSTITUTED INDOLES HAVING SUVEN PHARMACEUTICALS LTD SEROTONIN RECEPTOR AFFINITY AND PROCESS FOR THEIR PREPARATION 332/KOLNP/2007 29-01-2007 252786 30-05-2012 "THIENOPYRAZOLE DERIVATIVE HAVING PDE7 DAIICHI SANKYO CO., LTD. INHIBITORY ACTIVITY" 2501/DELNP/2004 26-08-2004 252787 30-05-2012 "PHARMACEUTICAL AEROSOL FORMULATION OF CHIESI FARMACEUTICI S.p.A. FORMOTEROL FUMARATE TO BE ADMINISTERED BY A PRESSURIZED METERED DOSE INHALER" 2010/DEL/2004 15-10-2004 252796 31-05-2012 "AMIDE DERIVATIVES" ASTRAZENECA AB 1820/DELNP/2006 03-04-2006 252801 31-05-2012 AN ANTHRAPYRIDONE OF THE FORMULA (I) SABIC INNOVATIVE PLASTICS IP B.V. 778/DELNP/2007 31-01-2007 252825 01-06-2012 ARYL-PYRIDINE COMPOUNDS F. HOFFMANN-LA ROCHE AG 607/DELNP/2007 23-01-2007 252833 04-06-2012 "TRIAZOLOPYRIDINYLSULFANYL DERIVATIVES AS P38 PFIZER INC MAP KINASE INHIBITORS" 9927/DELNP/2007 20-12-2007 252838 04-06-2012 "SULFONAMIDE DERIVATIVES USEFUL AS LIVER F. HOFFMANN-LA ROCHE AG CARNITINE PALMITOYL TRANSFERASE (L-CPT1) INHIBITORS" 498/MUMNP/2009 09-03-2009 252845 04-06-2012 “COMPOSITIONS OF CHK1 INHIBITORS” ICOS CORPORATION 381/KOLNP/2007 02-02-2007 252855 05-06-2012 "THIENOPYRIMIDINES USEFUL AS AURORA KINASE SUNESIS PHARMACEUTICALS, INC. INHIBITORS". 1767/KOLNP/2006 23-06-2006 252877 06-06-2012 "STEREOISOMERIC COMPOUNDS AND METHODS FOR ARYX THERAPEUTICS THE TREATMENT OF GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS" 510/MUMNP/2009 13-03-2009 252901 07-06-2012 “ORAL RECOMBINANT HELICOBACTER PYLORI VACCINE CHONGQING KANG WEI AND PREPARING METHOD THEREOF” BIOTECHNOLOGY CO. LTD. 489/MUMNP/2007 04-04-2007 252902 07-06-2012 PHARMACEUTICAL COMPOSITION COMPRISING AN CIPLA LIMITED ISOMER OF A BETAMIMETIC AGENT AND AN ANTI- CHOLINERGIC AGENT 2916/CHENP/2007 02-07-2007 252910 08-06-2012 BORON-CONTAINING MOLECULAR SIEVE CHA CHEVRON U.S.A INC. 3646/KOLNP/2006 05-12-2006 252936 11-06-2012 COMPOSITIONS AND METHODS TO PREVENT AAV GENZYME CORPORATION VECTOR AGGREGATION 2089/CHENP/2006 12-06-2006 252964 12-06-2012 SPIROINDOLINE DERIVATIVES HAVING INSECTICIDAL SYNGENTA PARTICIPATIONS AG PROPERTIES 1268/DEL/2003 14-10-2003 252981 13-06-2012 "TRICYCLIC COMPOUNDS HAVING ANTIOXIDANT NATIONAL INSTITUTE OF PROPERTIES" PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) 3429/DELNP/2006 14-06-2006 252982 13-06-2012 "PYRAZOLE DERIVATIVES AS PROTEIN KINASE ASTEX THERAPEUTICS LIMITED MODULATORS" 2451/KOLNP/2006 28-08-2006 252989 13-06-2012 2H OR 3H-BENZO[E]INDAZOL-1-YLE CARBAMATE SANOFI AVENTIS DERIVATIVES, AND THEIR PREPARATION 1851/CHENP/2006 26-05-2006 252990 13-06-2012 NOVEL ANALGESIC COMPOUNDS, EXTRACTS GRIFFITH UNIVERSITY CONTAINING SAME AND METHODS OF PREPARATION

2888/DELNP/2006 22-05-2006 253024 15-06-2012 "A COMPOSITION, FOR THE TREATMENT OF AN INDENA S.P.A. AFECTION OF THE ORAL CAVITY AND UPPER RESPIRATORY TRACT" 1939/MUM/2006 24-11-2006 253029 15-06-2012 CCR5 MODULATOR COMPOUNDS PHIVCO-1 LLC 443/MUMNP/2006 18-04-2006 253030 15-06-2012 SUBSTITUTED DIAZABICYCLOALKANE DERIVATIVES AS LIGANDS AT ALPHA 7 NICOTINIC ACETY LCHOLINE RECEPTORS. 2180/DELNP/2007 21-03-2007 253033 18-06-2012 "A COMPOSITION FOR PREVENTING OR IMPROVING OTSUKA PHARMACEUTICAL CO., LTD., PIGMENTATION" 4720/DELNP/2006 17-08-2006 253042 19-06-2012 "A DIKETOPIPERAZINE" NEREUS PHARMACEUTICALS, INC. 145/CHENP/2008 09-01-2008 253053 20-06-2012 COMPOUND EXHIBITING GLUCOKINASE ACTIVATION MITSUBISHI TANABE PHARMA AND ITS PREPARATION THEREOF CORPORATION 1331/CAL/1998 29-07-1998 253099 25-06-2012 4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b] INDOLE-1- SANOFI AVENTIS ACETAMIDE-DEIVATIVES 393/MUMNP/2008 29-02-2008 253106 26-06-2012 A COMPOSITION COMPRISING PHARMACEUTICAL- GLOBOASIA LLC GRADE FERRIC CITRATE EFFECTIVE IN REDUCING SERUM PHOSPHATE LEVEL 3268/KOLNP/2006 08-11-2006 253108 26-06-2012 AZASUGAR DERIVATIVES, HEPARANASE INHIBITORS SANOFI-AVENTIS AND PHARMACEUTICAL COMPOSITIONS THEREOF 4470/DELNP/2006 02-08-2006 253109 26-06-2012 "TETRAZOLE COMPOUND AND COMPOSITION ASTRAZENECA AB THEREOF" 3685/CHENP/2006 05-10-2006 253139 27-06-2012 HYALURONIC ACID-METHOTREXATE CONJUGATE DENKI KAGAKU KOGYO KABUSHIKI KAISHA 571/DEL/2007 16-03-2007 253149 28-06-2012 "A COMPOUND USEFUL AS PHARMACEUTICALS, WHITE FLOWER ASSOCIATES LLP AVERSIVE AGENTS AND/OR ANTIFOULANTS" 5184/DELNP/2006 08-09-2006 253159 28-06-2012 "A COMPOSITION COMPRISING GLYPHOSPHATE AND FMC CORPORATION AT LEAST ONE TAURATE SALT" 2120/DELNP/2006 19-04-2006 253168 29-06-2012 "SOLID PHARMACEUTICAL COMPOSITION" BAYER ANIMAL HEALTH GMBH 4557/DELNP/2005 06-10-2005 253179 29-06-2012 "ORAL FORMULATIONS OF CLADRIBINE" ARES TRADING S.A., 644/KOLNP/2007 22-02-2007 253193 04-07-2012 COMPOUND OF FORMULA (I) FOR TREATMENT OF IVAX DRUG RESEARCH INSTITUTE LTD. INFLAMMATORY DISEASES OF THE AIRWAY 764/CHENP/2008 14-02-2008 253217 04-07-2012 PIPERIDINE AND PIPERAZINE DERIVATIVES AS P2X3 F. HOFFMANN-LA ROCHE AG ANTAGONISTS 2870/DELNP/2006 19-05-2006 253261 09-07-2012 PYRAZOLE DERIVATIVES AS INHIBITORS OF RECEPTOR ASTRAZENECA AB TYROSYNE KINASES 511/KOLNP/2007 12-02-2007 253273 10-07-2012 SUBSTITUTED QUINOLONES AICURIS GMBH & CO. KG, 982/KOLNP/2007 20-03-2007 253276 10-07-2012 POLYPHOSPHATE DERIVATIVE OF A 1,3,5-TRIAZINE CHEMISCHE FABRIK BUDENHEIM KG. COMPOUND, A PROCESS FOR THE PRODUCTION THEREOF 3937/KOLNP/2006 28-12-2006 253283 10-07-2012 "TRICYCLIC INDENO-PYRROLE DERIVATIVES AS ATHERSYS, INC. SEROTONIN RECEPTOR MODULATORS" 1484/KOLNP/2007 25-04-2007 253285 10-07-2012 COMPOSITION COMPRISING AN ACTIVE CORE CADBURY ADAMS USA LLC. ENCAPSULATED BY MATRIX INCLUDING POLYMER AND SUCRALOSE AND METHOD OF PREPARATION THEREOF

2681/DELNP/2006 12-05-2006 253290 11-07-2012 "A SUBSTITUTED AMIDE DERIVATIVE HAVING POTENT ASTRAZENECA AB CYTOKINE INHIBITORY ACTIVITY" 2698/KOLNP/2007 20-07-2007 253297 11-07-2012 TRIOXEPANE COMPOSITION AND PROCESS FOR AKZO NOBEL N.V. PREPARING TRIOXEPANE COMPOSITION 1574/KOLNP/2006 07-06-2006 253308 11-07-2012 A COMBINATION OF DEXAMETHASONE AND 4-AMINO- NOVARTIS VACCINES & 5-FLUORO-3-[6-(4-METHYLPIPERAZIN-1-YL)-1H- DIAGNOSTICS S.R.L., BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE A TAUTOMER OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 2096/MUMNP/2007 10-12-2007 253338 13-07-2012 PYRIMIDINE COMPOUNDS TAIGEN BIOTECHNOLOGY CO., LTD. 3684/CHENP/2006 05-10-2006 253384 17-07-2012 4-BENZYL-[1,2,4]THIADIAZOLIDINE-3,5-DIONE NOSCIRA S A DERIVATIVES AS GSK-3 INHIBITORS 4138/DELNP/2007 31-05-2007 253414 18-07-2012 "A PIPERIDINYL INDOLE COMPOUND" EURO-CELTIQUE, S.A 621/KOLNP/2007 20-02-2007 253465 24-07-2012 "VACCINE FOR PREVENTION AND TREATMENT OF HIV- GLAXOSMITHKLINE BIOLOGICALS S.A. INFECTION" 144/KOLNP/2007 11-01-2007 253477 25-07-2012 SUBSTITUTED IMIDAZOLE DERIVATIVES NOVARTIS VACCINES AND DIAGNOSTICS, INC. 953/DELNP/2008 04-02-2008 253482 25-07-2012 BIS (THIO-HYDRAZIDE AMIDE) FORMULATION SYNTA PHARMACEUTICALS CORP. 3323/KOLNP/2006 13-11-2006 253493 25-07-2012 IMMEDIATE RELEASE PHARMACEUTICAL TABLETS WITH ACCU-BREAK TECHNOLOGIES INC. HEIGHT GREATER THAN WIDTH 931/DELNP/2007 05-02-2007 253503 26-07-2012 "A 6-CYCLOPENTYL 4-HYDROXY-5,6-DIHYDRO-2-ONE PFIZER INC. COMPOUND AND A PHARMACEUTICAL COMPOSITION THEREOF" 444/KOLNP/2007 07-02-2007 253517 26-07-2012 BIVALENT LINKERS AND CONJUGATES THEREOF ENDOCYTE, INC. 388/KOLNP/2007 05-02-2007 253519 26-07-2012 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY THERAPEUTIC USES 1476/CHENP/2008 26-03-2008 253552 31-07-2012 OXADIAZOLYL PYRAZOLO-PYRIMIDINES AS MGLUR2 F. HOFFMANN-LA ROCHE AG ANTAGONISTS 2692/DELNP/2006 12-05-2006 253571 01-08-2012 INJECTABLE SUSTAINED RELEASE IMPLANT HAVING A PSIVIDA INC. BIOERODIBLE MATRIX CORE AND A BIOERODIBLE SKIN

3768/CHENP/2006 11-10-2006 253575 01-08-2012 TETRAHYDROPYRIDOINDOLE DERIVATIVES PHARMACEUTICALS LTD 4136/DELNP/2007 31-05-2007 253581 02-08-2012 "A PIPERIDINYL CYANOIMINO-BENZIMIDAZOLE EURO-CELTIQUE, S.A. COMPOUND OF FORMULA (IV)" 5205/DELNP/2006 11-09-2006 253587 03-08-2012 "COMPOSITION FOR ORAL ADMINISTRATION OF HANMI PHARM. CO., LTD. TAMSULOSIN HYDROCHLORIDE" 2931/DELNP/2006 22-05-2006 253605 06-08-2012 2-PHENOXY PROPIONIC ACID COMPOUNDS AS PPAR F. HOFFMANN-LA ROCHE AG AGONISTS 4625/KOLNP/2007 29-11-2007 253606 06-08-2012 HETEROAROYL-SUBSTITUTED SERINE AMIDES BASF AKTIENGESELLSCHAFT 3287/KOLNP/2006 09-11-2006 253619 07-08-2012 "TETRAHYDROISOQUINOLINE SULFONAMIDE SANOFI-AVENTIS DERIVATIVES, THE PREPARATION THEREOF, AND THE USE OF THE SAME IN THERAPEUTICS" 3518/CHENP/2006 25-09-2006 253630 08-08-2012 NOVEL ADENINE COMPOUND AND A PROCESS FOR DAINIPPON SUMITOMO PHARMA CO PREPARING THE SAME LTD 9790/DELNP/2007 18-12-2007 253642 08-08-2012 "PHARMACEUTICAL COMPOSITION COMPRISING 2,3- OTSUKA PHARMACEUTICAL CO.,LTD. DIHYDRO-6-NITROIMIDAZO[2,1-B]OXAZOLE DERIVATIVES" 6872/DELNP/2006 17-11-2006 253644 08-08-2012 4-AMINO-5-CYANOPYRIMIDINE DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD 1223/KOLNP/2007 09-04-2007 253645 08-08-2012 A SUBSTITUTED CHROMAN DERIVATIVE MARSHALL EDWARDS, INC 690/MUMNP/2009 09-04-2009 253661 09-08-2012 A PHARMACEUTICAL FORMULATION BEN-GURION UNIVERSITY OF THE NEGEV RESEACH AND DEVELOPMENT AUTHORITY 3430/CHENP/2006 19-09-2006 253671 10-08-2012 PHARMACEUTICAL COMPOSITION COMPRISING A ARROW THERAPEUTICS LIMITED BENZODIAZEPINE DERIVATIVE AND AN INHIBITOR OF THE RSV FUSION PROTEIN 1046/MUMNP/2007 12-07-2007 253681 13-08-2012 TETRAHYDROQUINOLINE ANALOGUES ACADIA PHARMACEUTICALS INC 1522/MUMNP/2007 24-09-2007 253716 16-08-2012 SUBSTITUTED PYRIDINES AND PYRIDAZINES WITH BAYER CORPORATION ANGIOGENESIS INHIBITING ACTIVITY 538/MUM/2006 05-04-2006 253721 17-08-2012 LIQUID ORAL FORMULATION CONTAINING STRIDES ARCOLAB LIMITED FEXOFINADINE 952/KOLNP/2007 19-03-2007 253742 22-08-2012 MODULATORS OF MUSCARINIC RECEPTORS VERTEX PHARMACEUTICALS INCORPORATED 7514/DELNP/2006 12-12-2006 253747 22-08-2012 "SUBSTITUTED HYDANTION COMPOUNDS FOR THE ASTRAZENECA AB TREATMENT OF OBSTRUCTIVE AIRWAY DISEASE" 751/KOLNP/2007 01-03-2007 253750 22-08-2012 4-((PHENOXYALKYL) THIO)-PHENOXYACETIC ACIDS AND JANSSEN PHARMACEUTICA N.V. ANALOGS 2579/KOLNP/2007 10-07-2007 253754 22-08-2012 N-(HETEROARYL)-1H-INDOLE-2-CARBOXAMIDE SANOFI AVENTIS DERIVATIVES AND THEIR USE AS VANILLOID TRPV 1 RECEPTOR LIGANDS. 1443/KOLNP/2006 29-05-2006 253756 22-08-2012 QUINOLINES USEFUL IN TREATING CARDIOVASCULAR WYETH DISEASE 637/KOLNP/2007 21-02-2007 253761 22-08-2012 "5-[3-(4-BENZYLOXYPHENYLTHIO)-FUR-2-YL]- QUEST PHARMACEUTICAL SERVICES IMIDAZOLIDIN-2,4-DIONES (QPS) 2287/KOLNP/2006 10-08-2006 253771 23-08-2012 5,6-DIALKYL-7- AMINOTRIAZOLOPYRIMIDINES, THEIR BASF AKTIENGESELSCHAFT PREPARATION AND COMPOSITIONS COMPRISING THESE COMPOUNDS 461/MUMNP/2009 04-03-2009 253776 23-08-2012 KINASE INHIBITIRS USEFUL FOR THE TREATMENT OF DECIPHERA PHARMACEUTICALS LLC PROLIFERATIVE DISEASES 2775/DELNP/2004 20-09-2004 253805 27-08-2012 "ORALLY ADMINISTRABLE COMPOSITION FOR THE SOCIETE DES PRODUITS NESTLE S.A PHOTOPROTECTION OF THE SKIN" 2552/KOLNP/2007 09-07-2007 253821 28-08-2012 3, 5-DISUBSTITUTED AND 3,5,7-TRISUBSTITUTED-3H- ANADYS PHARMACEUTICALS, INC. OXAZOLO AND 3H-THIAZOLO [4,5-D] PYRIMIDIN-2-ONE COMPOUNDS AND PRODRUGS THEREOF

2595/DELNP/2006 09-05-2006 253825 28-08-2012 "N,2-DIMETHYL-{[7-(2-MORPHOLIN-4- PFIZER INC. YLETHOXY)QUINOLIN-4-YL]OXY}-1-BENZOFURAN-3- CARBOXAMIDE" 4841/DELNP/2007 22-06-2007 253890 30-08-2012 "TRANSDERMAL THERAPEUTIC SYSTEM (TTS), LTS LOHMANN THERAPIE-SYSTEME AG COMPRISING A FIRST COMPARTMENT AND A SECOND COMPARTMENT" 3059/CHENP/2006 22-08-2006 253897 31-08-2012 IMMUNOSUPPRESSANT COMPOUNDS IRM LLC 7158/DELNP/2007 17-09-2007 253900 31-08-2012 "BISHETEROCYCLE TANDEM COMPOUNDS USEFUL AS SHANGHAI INSTITUTE OF MATERIA ANTIVIRAL AGENTS" MEDICA, CHINESE ACADEMY OF SCIENCES 1892/DEL/2006 22-08-2006 253901 31-08-2012 "A NOVEL CYCLIC DONOR-ACCEPTOR COUNCIL OF SCIENTIFIC & INDUSTRIAL CONJUGATE,PROCESS AND A SUPRAMOLECULAR RESEARCH FLUORESCENT MARKER THEREOF" 3450/DEL/1997 01-12-1997 253903 31-08-2012 "1-ARYL-4-CYCLOPROPYLPYRAZOLE COMPOUNDS" PFIZER INC., 1151/MUMNP/2009 16-06-2009 253922 03-09-2012 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS ELI LILLY AND COMPANY FOR THE TREATMENT OF CANCER 2485/KOLNP/2008 19-06-2008 253930 04-09-2012 3-(4-{[4-(4-{[3-(3,3-DIMETHYL-1-PIPERIDINYL) GLAXO GROUP LIMITED PROPYL]0XY} PHENYL)-1-PIPERIDINYL] CARBONYL}-1- NAPTHALENYL) PROPANOIC OR PROPENOIC ACID AS H1 AND H3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY AND/OR ALLERGIC DISORDERS

198/DEL/2008 24-01-2008 253942 05-09-2012 "A COMPOSITION COMPRISING METHYL N-(2,6- SYNGENTA PARTICIPATIONS AG DIMETHYLPHENYL)-N-(METHOXYACETYL)-DL- ALANINATE AND 3-ANILINO-5-METHYL-5-(4- PHENOXYPHENYL)-1,3-OXAZOLIDINE-2,4-DIONE" 880/MUM/2004 13-08-2004 253950 06-09-2012 DISPERSIBLE SUSTAINED RELEASE PHARMACEUTICAL SINGH, KAMALINDER KAUR COMPOSITIONS 4742/DELNP/2005 18-10-2005 253962 06-09-2012 "DELAYED RELEASE TABLET WITH DEFINED CORE JAGOTEC AG GEOMETRY" 704/DEL/2005 30-03-2005 253965 07-09-2012 " ANTIFUNGAL STEROIDAL DIMERS, N1, N3- COUNCIL OF SCIENTIFIC & INDUSTRIAL DIETHYLENETRIAMINE BIS [ CHOLIC ACID AMIDE] " RESEARCH 1020/CHENP/2008 29-02-2008 253968 07-09-2012 DIAMINOPYRIMIDINES AS P2X3 AND P3X2/3 F. HOFFMANN-LA ROCHE AG MODULATORS 1195/DEL/2001 29-11-2001 253983 11-09-2012 AN ANTI BACTERIAL COMPOSITION COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH 2733/DELNP/2007 12-04-2007 253993 12-09-2012 "PYROZOLO (1,5-ALPHA), PYRIMIDINYL COMPOUND" SMITHKLINE BEECHAM (CORK) LIMITED

2115/DELNP/2006 19-04-2006 253996 12-09-2012 "NOVEL 17B HYDROSYSTEROID DEHYDROGENASE TYPE SOLVAY PHARMACEUTICALS GMBH 1 INHIBITORS" 3157/CHENP/2006 31-08-2006 254003 12-09-2012 IMIDAZO[1,2-C]PYRIMIDINYLACETIC ACID DERIVATIVES ACTIMIS PHARMACEUTICALS, INC.

674/KOLNP/2007 23-02-2007 254012 12-09-2012 NOVEL BENZO-FUSED HETEROARYL SULFAMIDE JANSSEN PHARMACEUTICA N.V. DERIVATIVES USEFUL AS ANTICONVULSANT AGENTS 3767/DEL/1998 16-12-1998 254063 18-09-2012 "2,4-DUSULFONYL PHENYL BUTYL NITRONE" OKLAHOMA MEDICAL RESEARCH FOUNDATION 2981/KOLNP/2006 16-10-2006 254073 18-09-2012 NOVEL COMPOUNDS AS OPIOID RECEPTOR JANSSEN PHARMACEUTICA N.V MODULATORS 3074/KOLNP/2006 24-10-2006 254078 18-09-2012 TETRAHYDRO-INDAZOLE CANNABINO ID MODULATORS JANSSEN PHARMACEUTICA N.V.

2719/KOLNP/2007 23-07-2007 254080 18-09-2012 PEPTIDIC COMPOUNDS UNIVERSITY OF WOLLONGONG 1838/DELNP/2007 08-03-2007 254115 20-09-2012 "A COMPOUND 1-(4-BENZOYLPIPERAZIN-1-YL)-2-(4- BRISTOL-MYERS SQUIBB COMPANY METHOXY-7-(3-METHYL-1H-1,2,4-TRIAZOL-1-YL)-1H- PYRROLO[2,32-C]PYRIDIN-3-YL)ETHANE-1,2-DIONE"

3013/DEL/2005 10-11-2005 254119 21-09-2012 A NOVEL PYRROLO[2,1-C) [1,4]BENZODIAZEPINE COUNCIL OF SCIENTIFIC AND HYBRIDS AND A PROCESS FOR PREPARATION THEREOF INDUSTRIAL RESEARCH

1162/DEL/1999 30-08-1999 254130 21-09-2012 "A PIPERAZINE OF THE FORMULA I" ASTRAZENECA UK LTD., 42/MUMNP/2009 05-01-2009 254149 24-09-2012 IMPROVEMENTS RELATING TO PHARMACEUTICAL UNILEVER PLC COMPOSITIONS 1568/MUM/2008 23-07-2008 254150 24-09-2012 NOVEL ANTICANCER HYDRAZINO DERIVATIVE OF INDIAN INSTITUTE OF TECHNOLOGY, AND PROCESS FOR PREPARATION THEREOF BOMBAY

5560/DELNP/2006 25-09-2006 254165 25-09-2012 "A PHARMACEUTICAL COMPOSITION FOR TREATING BRISTOL-MYERS SQUIBB COMPANY HIV INFACTION" 2157/CHENP/2004 28-09-2004 254167 25-09-2012 5-SUBSTITUTED 1, 1-DIOXO-1,2,5-THIAZOLIDINE-3-ONE NOVARTIS AG DERIVATIVES AS PTPASE IB INHIBITORS 4597/CHENP/2007 16-10-2007 254174 26-09-2012 SPIRO-OXINDOLE COMPOUNDS XENON PHARMACEUTICALS INC. 95/CHENP/2008 07-01-2008 254184 28-09-2012 A COMPOSITION FOR TOPICAL USE FIDIA FARMACEUTICI S.P.A 2225/CHENP/2006 21-06-2006 254201 01-10-2012 NOVEL THIAZOLIDIN-4-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD 706/MUM/2006 05-05-2006 254202 01-10-2012 NOVEL INTERMEDIATES, PROCESS FOR THEIR PIRAMAL HEALTHCARE LIMITED PREPARATION AND PROCESS FOR THE PREPARATION OF CoQ10 EMPLOYING THE SAID NOVEL INTERMEDIATES 2788/DELNP/2008 03-04-2008 254214 03-10-2012 "5-(4-{[(2-FLUOROPHENYL)METHYL} PHENYL)- GLAXO GROUP LIMITED PROLINAMIDE OF FORMULA (I) AND PROCESS OF PREPARING THE SAME" 2892/KOLNP/2007 08-08-2007 254225 04-10-2012 HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLE AICURIS GMBH & CO. KG. COMPOUNDS AND METHOD OF PREPARATION THEREOF 757/DELNP/2006 15-02-2006 254229 04-10-2012 "LIQUID, AQUEOUS, PHARMACEUTICAL COMPOSITIONS NOVO NORDISK HEALTH CARE AG OF FACTOR VII POLYPEPTIDES." 383/DEL/2006 13-02-2006 254250 09-10-2012 NOVEL BIS-PYRROLO[2,1-C][1,4] BENZODIAZEPINE- COUNCIL OF SCIENTIFIC AND ANTHRAQUINONE CONJUGATES AND A PROCESS FOR INDUSTRIAL RESEARCH THE PREPARATION THEREOF 3061/KOLNP/2006 23-10-2006 254255 10-10-2012 PROCESS AND INTERMEDIATE COMPOUNDS USEFUL IN REDX PHARMA LIMITED THE PREPARATION OF STATINS, PARTICULARLY ROSUVASTATIN 1725/CHENP/2006 17-05-2006 254261 10-10-2012 A PHARMACEUTICAL COMPOSITION COMPRISING A SANOFI PASTEUR VACCINE ANTIGEN AND A PHOSPHORIC ESTER DERIVATIVE OF PHOSPHATIDYLCHOLINE 6256/DELNP/2006 25-10-2006 254265 11-10-2012 "AN ADHESIVE PATCH FOR TREATMENT AND HUNTER-FLEMING LIMITED COMPOSITION THEREOF" 1525/MUMNP/2007 24-09-2007 254285 17-10-2012 AN AQUEOUS DISINFECTANTS OR STERILANT SOLUTIONS BIOMED LLC COMPOSITION 1030/KOLNP/2007 23-03-2007 254307 18-10-2012 BUTYLPHTHALIDE SELF-EMULSIFYING DRUG DELIVERY SHIJIAZHUANG PHARMA GROUP SYSTEM, ITS PREPARATION METHOD AND APPLICATION ZHONGQI PHARMACEUTICAL TECHNOLOGY (SHIJIAZHUANG) CO., LTD. 259/DELNP/2005 24-01-2005 254316 18-10-2012 BROADSPECTRUM 2-AMINO-BENZOTHIAZOLE TIBOTEC PHARMACEUTICALS LTD. SULFONAMIDE HIV PROTEASE INHIBITORS" 6180/DELNP/2007 08-08-2007 254349 27-10-2012 "A SUBSTITUTED ECTEINASCIDIN COMPOUND" PHARMA MAR, S.A. 481/DELNP/2008 17-01-2008 254354 29-10-2012 "A COMPOUND, WHICH IS N-(3-FLUOROPHENYL)-1-[(4- GLAXO GROUP LIMITED {[(-3S)-3-METHYL-1- PIPERAZINYL]METHYL}PHENYL)ACETYL]-4- PIPERIDINAMINE ANA PHARMACEUTICALLY ACCEPTABLE SALT THEREOF" 5546/CHENP/2007 03-12-2007 254362 29-10-2012 A PHARMACEUTICAL FORMULATION FOR TREATING SCHERING CORPORATION HCV INFECTION 2824/DELNP/2006 18-05-2006 254363 29-10-2012 "A TRIAZOLE COMPOUND OF FORMULA (I) AND PFIZER INC COMPOSITION COMPRISING THE SAME" 529/DEL/2006 28-02-2006 254367 29-10-2012 "5-[2-(2,6,6,-TRIMENTHYL-CYCLOHEX-2-ENYL)- COUNCIL OF SCIENTIFIC & INDUSTRIAL ENTHENYL]-ISOXAAZOLES" RESEARCH 977/CHE/2007 08-05-2007 254378 30-10-2012 A STABLE CONTROLLED RELEASE ORAL SOLID DOSAGE MEDREICH LIMITED FORM COMPOSITION AND A PROCESS THEREOF

3715/DELNP/2007 18-05-2007 254427 02-11-2012 "A PHARMACEUTICAL COMPOSITION" ENDORECHERCHE, INC 7676/DELNP/2006 18-12-2006 254439 05-11-2012 HETEROCYCLE-SUBSTITUTED PYRROLIDINE AND , INC. PIPERIDINE 2041/DELNP/2006 13-04-2006 254443 05-11-2012 "PELLETS CONTAINING VENLAFAXINE HYDROCHLORIDE" EGIS GYOGYSZERGYAR RT

3155/CHENP/2006 31-08-2006 254449 05-11-2012 HETEROARYL PIPERIDINE GLYCINE TRANSPORTER MERCK SHARP & DOHME CORP. INHIBITORS 1565/MUM/2008 23-07-2008 254454 06-11-2012 STABLE INJECTABLE OIL-IN-WATER NANOEMULSION BHARAT SERUMS AND VACCINES LTD 3513/CHENP/2006 25-09-2006 254466 06-11-2012 PROGESTERONE RECEPTOR MODULATORS MSD Oss B.V. 2926/CHENP/2006 09-08-2006 254469 06-11-2012 COMPOUNDS AND COMPOSITIONS AS LXR IRM LLC MODULATORS 2755/DEL/2005 13-10-2005 254474 07-11-2012 "A SUSTAINED RELEASE MONOTHILIC FORMULATION NATIONAL INSTITUTE OF OF ROPINIROLE" PHARMACEUTICAL EDUCATION AND RESEARCH 433/DELNP/2007 17-01-2007 254484 07-11-2012 "PYRIMIDINE DERIVATIVES" F. HOFFMANN-LA ROCHE AG 4535/DELNP/2006 04-08-2006 254505 09-11-2012 "A MICROEMULSION PREPARATION OF HIGH BIOAVAILABILITY INC CONCENTRATION PROPOFOL FOR ANESTHETIC USES"

520/CHENP/2008 31-01-2008 254533 12-11-2012 ANTITUMORAL BIOCONJUGATES OF HYALURONIC ACID FIDIA FARMACEUTICI S.P.A OR ITS DERIVATIVES 1623/DELNP/2006 24-03-2006 254541 15-11-2012 PRESERVATIVES AND METHODS OF THE PROCTER & GAMBLE COMPANY THEIR USE 3149/DELNP/2007 26-04-2007 254551 17-11-2012 "ß-L-2'-DEOXY-NUCLEOSIDES FOR THE TREATMENT OF IDENIX (CAYMAN) LIMITED HEPATITIS B" 3094/KOLNP/2006 25-10-2006 254567 20-11-2012 IMIDAZOLE COMPOUNDS. JANSSEN PHARMACEUTICA N.V. 1253/CHE/2006 19-07-2006 254572 20-11-2012 OXAZOLIDINONE DERIVATIVES ORCHID RESEARCH LABORATORIES LTD

1855/DELNP/2006 04-04-2006 254576 21-11-2012 "MORPHOLINE DERIVATIVES AS ELI LILLY AND COMPANY LIMITED INHIBITORS" 5080/DELNP/2006 04-09-2006 254601 23-11-2012 NITROGENOUS FUSED-RING COMPOUND" KISSEI PHARMACEUTICAL CO., LTD. 2910/DELNP/2005 29-06-2005 254616 26-11-2012 "COMPOSITION HAVING ACTION PREVENTING OR SUNTORY HOLDINGS LIMITED., ALLEVIATING SYMPTOMS OR DISEASES DUE TO AGING OF BLOOD VESSELS" 520/CHE/2005 02-05-2005 254638 29-11-2012 A PEPTIDE AND A METHOD THEREOF INDIAN INSTITUTE OF SCIENCE 4024/CHENP/2006 01-11-2006 254662 03-12-2012 A COMPOSITION FOR TREATING HYPERLIPAEMIA LUNAN PHARMACEUTICAL GROUP CORPORATION 2300/CHENP/2006 23-06-2006 254675 05-12-2012 CONTROLLED-RELEASE PHARMACEUTICAL LEK PHARMACEUTICALS D.D. FORMULATION 3843/DELNP/2004 03-12-2004 254678 05-12-2012 "A STABLE FENOFIBRATE COMPOSITION FOR ORAL ELAN PHARMA INTERNATIONAL, LTD ADMINISTRATION" 2763/MAS/1998 09-12-1998 254706 07-12-2012 EPLERENONE COMPOSITIONS GD SEARLE & CO 5/CHE/2004 02-01-2004 254714 10-12-2012 "NOVEL INDENO [2,1A] INDENE AND ISOINDOLO [2,1-A] SUVEN LIFE SCIENCES LIMITED INDOLES AS 5-HT 6 RECEPTORS 3601/KOLNP/2006 01-12-2006 254726 11-12-2012 AMIDO COMPOUNDS AND THEIR USE AS INCYTE CORPORATION PHARMACEUTICALS 1424/CHENP/2008 24-03-2008 254730 12-12-2012 NOVEL PYRIDINE AND PYRIMIDINE COMPOUNDS EISAI R&D MANAGEMENT CO, LTD 372/MUMNP/2008 27-02-2008 254746 14-12-2012 NOVEL TRIAZOLE DERIVATIVES RECEPTORS AETERNA ZENTARIS GMBH 5303/DELNP/2006 13-09-2006 254758 14-12-2012 COMPOSITION COMPRISING AN HDAC INHIBITOR IN DSM IP ASSET B.V. COMBINATION WITH A RETINOID 1350/KOLNP/2007 17-04-2007 254759 14-12-2012 HYDROXYBENZOATE SALT OF A METANICOTINE TARGACEPT, INC. COMPOUND,PROCESS FOR ITS PREPARATION AND COMPOSITION COMPRISING IT 1255/KOLNP/2006 12-05-2006 254788 18-12-2012 A TOCOPHEROL MODIFIED COMPOUND SONUS PHARMACEUTICALS, INC. 00558/DELNP/2003 16-04-2003 254813 21-12-2012 "CRYSTALLINE TIOTROPIUM BROMIDE MONOHYDRATE BOEHRINGER INGELHEIM PHARMA AND PROCESS THEREOF " GMBH & CO. KG 3841/DELNP/2008 06-05-2008 254830 24-12-2012 "COMPOUNDS AS GLUCAGON RECEPTOR ELI LILLY AND COMPANY ANTAGONISTS" 106/DELNP/2008 03-01-2008 254839 26-12-2012 "POLYMORPHIC FORMS OF RIFAXIMIN, PROCESSES FOR ALFA WASSERMANN S. P. A. THEIR PRODUCTION AND USE THEREOF IN MEDICINAL PREPARATIONS" 439/MUMNP/2007 26-03-2007 254845 26-12-2012 PRODRUGS CONTAINING NOVEL BIO-CLEAVABLE PIRAMAL ENTERPRISES LIMITED LINKERS 4346/CHENP/2006 27-11-2006 254919 04-01-2013 BINDING MOLECULES CAPABLE OF NEUTRALIZING CRUCELL HOLLAND B.V RABIES VIRUS 4727/CHENP/2006 22-12-2006 254921 04-01-2013 HETEROCYCLIC CARBOXAMIDES WITH MICROBIOCIDAL SYNGENTA PARTICIPATIONS AG ACTIVITY 5185/CHENP/2007 16-11-2007 254930 07-01-2013 STREPTOGRAMINDERIVATIVES, THEIR PREPARATION AVENTIS PHARMA S.A AND COMPOSITIONS WHICH CONTAIN THEM

5355/DELNP/2006 15-09-2006 254948 07-01-2013 A COMPOUND OF FORMULA I BRISTOL-MYERS SQUIBB COMPANY. 1046/CHENP/2006 27-03-2006 254955 08-01-2013 SUBSTITUTED THIENO [2,3-D] PYRIMIDINES AS HSP 90 M/S. VERNALIS (CAMBRIDGE) Ltd INHIBITORS 1582/MUMNP/2008 25-07-2008 254957 09-01-2013 ACYLOXYALKYL CARBAMATE PRODUCTS, XENOPORT, INC. 1550/CHE/2006 29-08-2006 254994 11-01-2013 NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITOR ORCHID CHEMICALS & PHARMACEUTICALS LTD 2064/DELNP/2004 19-07-2004 255028 16-01-2013 A CONTROLLED RELEASE PHARMACEUTICAL GLAXO GROUP LIMITED FORMULATION 438/MUM/2008 03-03-2008 255029 16-01-2013 THIENO[2,3-D]-PYRIMIDINE-4(3H)-ONE COMPOUNDS NATIONAL CHEMICAL LABORATORY AND PROCESS THEREOF 2163/MUMNP/2008 10-10-2008 255039 16-01-2013 COSMETIC COMPOSITION WITH SOFT FOCUS HINDUSTAN UNILEVER LIMITED PROPERTIES 1589/KOLNP/2006 08-06-2006 255081 21-01-2013 AN ANTIBODY GLAXO GROUP LIMITED 5707/DELNP/2006 29-09-2006 255083 21-01-2013 COMPRESSED PHARMACEUTICAL COMPOSITIONS NORGINE B.V COMPRISING PEG AND ELECTROLYTES 2046/DELNP/2003 12-02-2003 255111 23-01-2013 A PHARMACEUTICAL COMPOSITION FOR HF ARZNEIMITTELFORSCHUNG GMBH PHARMACOLOGICAL ADDICTIVE SUBSTANCE OR INTOXICANT THERAPY 1747/MUM/2006 20-10-2006 255115 23-01-2013 STABLE AEROSOL FORMULATION CIPLA LIMITED 4322/CHENP/2006 24-11-2006 255153 30-01-2013 THERAPEUTIC ENZYME FORMULATIONS AND USES THE BOARD OF TRUSTEES OF THE THEREOF LELAND STANFORD JUNIOR UNIVERSITY

1276/CHENP/2008 14-03-2008 255154 30-01-2013 4-AMINO-THIENO[3,2-c]PYRIDINE-7-CARBOXYLIC ACID F. HOFFMANN-LA ROCHE AG COMPOUNDS 1217/CHE/2006 12-07-2006 255172 31-01-2013 2-SUBSTITUTED METHYL PENAM DERIVATIVES ORCHID CHEMICALS & PHARMACEUTICALS LTD 1904/DELNP/2005 05-05-2005 255194 01-02-2013 NOVEL BENZOXAZOCINES COMPOUNDS ARAKIS LTD 1607/DEL/1996 19-07-1996 255196 01-02-2013 A CONTROLLED RELEASE AND DELAYED RELEASE SMITHKLINE BEECHAM P.L.C. FORMULATION 1514/DEL/1999 30-11-1999 255203 02-02-2013 FAST DISSOLVING PHARMACEUTICAL COMPOSITIONS IN PANACEA BIOTEC LIMITED SOLID FORM WITH PROLONGED SWEET TASTE AND A PROCESS FOR THE MANUFACTURE THEREOF

169/DELNP/2007 05-01-2007 255207 04-02-2013 SALTS OF BENZIMIDAZOLE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD. 1726/KOLNP/2007 15-05-2007 255232 05-02-2013 PROCESS FOR PREPARING 4-(N-ALKYLAMINO)-5, 6- RAGACTIVES, S.L. DIHYDRO-4H-THEINO-[2,3-B]-THIOPYRANS 3577/DELNP/2006 21-06-2006 255243 06-02-2013 A COMPOUND DENOTED 4-(((6-(3-((1S,1AR,7BR)-4,7- MEDIVIR AB. DIFLUORO-1,1A,2,7B- TETRAHYDROCYCLOPROPA[C]CHROMEN-1- YL)UREIDO)PYRIDIN-3-YL)OXY)BENZENESULFONAMIDE

40/DEL/2006 04-01-2006 255262 07-02-2013 ORAL FORMULATIONS FOR ENAHANCING GASTRIC DIRECTOR GENERAL , DEFENCE EMPTYING AND SPHINCTER RELAXATION INSTANTLY RESEARCH & DEVELOPMENT AND A PROCESS OF PREPARTATION THEREOF ORGANISATION

2792/MUMNP/2008 30-12-2008 255273 08-02-2013 FLUOROALKYLOXYCOMBRETASTATIN DERIVATIVES, ZHEJIANG DADE PHARMACEUTICAL METHODS FOR PRODUCING SAME GROUP CO. LTD. 1636/CHENP/2007 20-04-2007 255279 08-02-2013 (BIPHENYL)CARBOXYLIC ACIDS AND DERIVATIVES CELLZOME LIMITED THEREOF 2725/DELNP/2006 16-05-2006 255287 09-02-2013 3- AMINOPYRROLIDONE DERIVATIVES NEWRON PHARMACEUTICALS S.p.A 6210/DELNP/2007 09-08-2007 255288 09-02-2013 A CYCLOHEPTA[B] PYRIDINE-3-CARBONYLGUANIDINE TOA EIYO LTD. COMPOUND 7764/DELNP/2006 20-12-2006 255289 09-02-2013 PHARMACEUTICAL COMPOSITION COMPRISING A PFIZER PRODUCTS, INC TABLET CORE OR CAPSULE FILL AND OPACIFYING COAT AND POLISH COAT 3810/DELNP/2004 01-12-2004 255299 11-02-2013 COMPOSITION BASED ON SUBSTITUTED 1,3- GENFIT DIPHENYLPROP-2-EN-1-ONE DERIVATIVES 3458/CHENP/2006 21-09-2006 255301 11-02-2013 INHIBITORS OF DIPEPTIDYLPEPTIDASE IV FOR TRUSTEES OF TUFTS COLLEGE REGULATING METABOLISM 592/KOLNP/2007 16-02-2007 255313 12-02-2013 A STAIN REMOVING ORAL COMPOSITION KRAFT FOODS GLOBAL BRANDS, LLC 1724/KOLNP/2007 15-05-2007 255543 01-03-2013 PYRAZOLO[1,5-A]PYRIMIDINES USEFUL AS INHIBITORS VERTEX PHARMACEUTICALS OF PROTEIN KINASES INCORPORATED 17/MUM/2006 04-01-2006 255544 01-03-2013 PROCESS AND INTERMEDIATES FOR PREPARATION OF CIPLA LIMITED DONEPEZIL HYDROCHLORIDE 4408/CHENP/2006 30-11-2006 255582 06-03-2013 3-AMINO-1-ARYLPROPYL INDOLES AS MONOAMINE F.HOFFMANN-LA ROCHE AG 1733/CHE/2005 25-11-2005 255642 12-03-2013 SYNERGISTIC ANTIBACTERIAL COMPOSITION OF SRINIVAS JEGANNATHAN CEFIXIME AND CLOXACILLIN / DICLOXACILLIN SODIUM OR ANY OTHER OXACILLIN WITH CLAVULANIC ACID

533/DELNP/2007 19-01-2007 255673 14-03-2013 COMPOSITION COMPRISING ASPARTATE AND VITAMIN N.V. NUTRICIA B12 OR BIOTIN FOR REGULATING KETONE BODIES

3141/DEL/2005 23-11-2005 255703 15-03-2013 A COMPOUND OF PROTECTED 4-AMINOMETHYLENE- LG LIFE SCIENCES LTD. PYRROLIDIN-3-ONE 5661/DELNP/2007 23-07-2007 255745 20-03-2013 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 750/KOLNP/2007 01-03-2007 255776 21-03-2013 4-(( PHENOXYALKYL)THIO) -PHENOXYACETIC ACIDS AND JANSSEN PHARMACEUTICA N.V. ANALOGS 353/CHENP/2008 22-01-2008 255868 26-03-2013 AMPHOLYTIC COPOLYMER AND PRODUCTION THEREOF BASF AKTIENGESELLSCHAFT

119/KOLNP/2008 08-01-2008 255840 26-03-2013 SUBSTITUTED IMIDAZOLE COMPOUNDS AS KSP NOVARTIS AG INHIBITORS 2353/CHENP/2008 12-05-2008 255979 12-04-2013 SUSTAINED RELEASE FILM FORMULATION FOR HEALING DAEWOONG CO., LTD WOUND COMPRISING EPIDERMAL GROWTH FACTOR

4551/CHENP/2006 12-12-2006 255986 15-04-2013 SUBSTITUTED N-PHENYL BENZAMIDES PROTEOTECH INC. 7341/DELNP/2006 05-12-2006 255984 15-04-2013 "3-(HETEROARYL-OXY)-2-ALKYL-1-AZA-BICYCLOALKYL NOVARTIS AG, DERIVATIVES AS ALPHA, 7-NACHR LIGANDS FOR THE TREATMENT OF CNS DISEASES" 3035/DELNP/2007 23-04-2007 255996 17-04-2013 A COMPOUND 3'-{N'-[1-3,5-DIMETHYL-PHENYL)-6- LIGAND PHARMACEUTICALS,INC TRIFLUOROMETHYL-2-OXO-1,2-DIHYDRO-INDOL-3- YLIDENE]-HYDRAZINO}-2'-HYDROXY-BIPHENYL-3- CARBOXYLIC ACID AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, FOR MODULATING THROMBOPOIETIN ACTIVITY 2461/DEL/2004 10-12-2004 256010 18-04-2013 "PHARMACEUTICAL COMPOSITION FOR IMPROVING COUNCIL OF SCIENTIFIC & INDUSTRIAL PALATABILITY OF DRUGS AND PROCESS FOR RESEARCH PREPARATION THEREOF" 1302/CHE/2005 15-09-2005 256019 19-04-2013 PYRIMIDINE CARBOXIMIDES ORCHID RESEARCH LABORATORIES LTD

26/DELNP/2008 01-01-2008 256021 19-04-2013 "HELIX 12 DIRECTED NON-STEROIDAL ENDORECHERCHE, INC. ANTIANDROGENS" 1665/MUMNP/2008 04-08-2008 256023 22-04-2013 DEUTERATED CATECHOLAMINE DERIVATIVES AND BIRDS PHARMA GMBH BEROLINA MEDICAMENTS COMPRISING SAID COMPOUNDS INNOVATIVE RESEARCH & DEVELOPMENT SERVICES 5815/DELNP/2005 13-12-2005 256025 22-04-2013 "THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM XENTION DISCOVERY LIMITED CHANNEL INHIBITORS" 6550/DELNP/2007 23-08-2007 256032 22-04-2013 "OPTHALMOLOGIC COMPOSITIONS" LABORATOIRES THEA 4284/KOLNP/2007 07-11-2007 256041 23-04-2013 GLP-1 PEGYLATED COMPOUNDS ELI LILLY AND COMPANY 5224/DELNP/2006 11-09-2006 256046 24-04-2013 "COMPOUNDS USEFUL FOR INHIBITING MACROPHAGE CYTOKINE PHARMASCIENCES, INC. MIGRATION INHIBITORY FACTOR" 1339/DEL/2005 25-05-2005 256052 26-04-2013 "A LIPOSOMAL FORMULATION AND USE THEREOF" COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH 7052/DELNP/2006 23-11-2006 256066 29-04-2013 ANTIBODY DRUG CONJUGATES AND METHODS. GENENTECH, INC. 3073/DELNP/2004 07-10-2004 256069 29-04-2013 "NOVEL PYRAZOLO [4,3-D]PYRIMIDINES, PROCESSES USTAV EXPERIMENTALNI BOTANIKY AV FOR THEIR PREPARATION AND METHODS FOR CR (INSTITUTE OF EXPERIMENTAL THERAPY" BOTANY ACADEMY OF SCIENCES OF THE CZECH REPUBLIC) 2449/DEL/2005 12-09-2005 256107 02-05-2013 "SUSTAINED RELEASE COMPOSITION" DELHI INSTITUTE OF PHARMACEUTICAL SCIENCES & RESEARCH

32/KOLNP/2008 02-01-2008 256108 02-05-2013 N-(ARYLALKYL)-1H-PYRROLOPYRIDINE-2-CARBOXAMIDE SANOFI-AVENTIS DERIVATIVES, PREPARATION AND THERAPEUTIC COMPOSITION THEREOF 2192/DEL/2006 05-10-2006 256122 05-05-2013 A FORMULATION FOR THE STABILIZATION OF COUNCIL OF SCIENTIFIC & INDUSTRIAL ALLERGENIC EXTRACTS USED IN DIAGNOSIS AND RESEARCH THERAPY OF ALLERGY. 2335/DELNP/2007 26-03-2007 256125 06-05-2013 "NOVEL PYRAZOLE DERIVATIVE" KISSEI PHARMACEUTICAL CO.LTD. 2726/KOLNP/2007 24-07-2007 256132 07-05-2013 PROTEASOME INHIBITORS AND METHODS OF USING CEPHALON, INC THE SAME 4247/CHENP/2006 17-11-2006 256182 13-05-2013 A MEDICAMENT COMPRISING GLYCOPYRROLATE AND NOVARTIS AG (R)- 5-[2-(5,6-DIETHYL-INDAN-2-YLAMINO)-1-HYDROXY- ETHYL]-8-HYDROXY-1H-QUINOLIN-2-ONE MALEATE

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