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DRUGS CONTRAINDICATED IN (Part 1 of 2) This chart represents information on select drugs that are contraindicated (Pregnancy category X) for women who are pregnant. This is not an inclusive list of products that carry that pregnancy category. Those drugs that are contraindicated at a certain phase of the pregnancy are listed next to the product name. For more information on specific drug monographs, see product entries or consult the manufacturer. ALLERGIC DISORDERS SSD (silver sulfadiazine) Late Macrodantin (nitrofurantoin pregnancy macrocrystals) Pregnancy at term Vistaril (hydroxyzine) Early pregnancy SSD AF (silver sulfadiazine) Late Rebetol (ribavirin) CARDIOVASCULAR SYSTEM pregnancy Rebetron (ribavirin/interferon alfa -2b) Tazorac (tazarotene) Septra (sulfamethoxazole/trimethoprim) Advicor ( ext-rel/lovastatin) Tilia Fe (norethindrone /ethinyl 3rd trimester Aggrenox (dipyridamole/aspirin) 3rd ) Sulfadiazine Pregnancy at term trimester Tri-Legest 21 (norethindrone acetate/ Tindamax (tinidazole) 1st trimester Altoprev (lovastatin) ethinyl estradiol) Urobiotic-250 (oxytetracycline HCl/ Bayer (aspirin) 3rd trimester Tri-Legest Fe (norethindrone acetate/ sulfamethizole/phenazopyridine) Late Caduet (amlodipine/atorvastatin) ethinyl estradiol) pregnancy Coumadin (warfarin sodium) Tri-previfem (/ethinyl Virazole (ribavirin) Crestor (rosuvastatin) estradiol) METABOLIC DISORDERS Ecotrin (aspirin) 3rd trimester Tri-sprintec (norgestimate/ethinyl Juvisync (sitagliptin/simvastatin) estradiol) Zavesca (miglustat) Lescol (fluvastatin) Yaz (/ethinyl estradiol) Lescol XL (fluvastatin) MUSCULOSKELETAL DISORDERS Letairis (ambrisentan) ENDOCRINE SYSTEM Advil (ibuprofen) 3rd trimester Lipitor (atorvastatin) Androderm () Aleve (naproxen sodium) 3rd trimester Livalo (pitavastatin) Androgel (testosterone) Ansaid (flurbiprofen) Late pregnancy Lovastatin tabs Android () Arava (leflunomide) Multaq (dronedarone) Axiron (testosterone) Arthrotec (diclofenac sodium/ misoprostol) Pravachol (pravastatin) Delatestryl () Bayer (aspirin) 3rd trimester Simcor (niacin ext-rel/simvastatin) Depo-testosterone (testosterone BC Arthritis Strength (aspirin/caffeine/ Tracleer (bosentan) cypionate) salicylamide) 3rd trimester Vytorin (ezetimibe/simvastatin) Egrifta (tesamorelin) Cataflam (diclofenac potassium) Late Zocor (simvastatin) pregnancy CENTRAL NERVOUS SYSTEM Fortesta (testosterone) Celebrex (celecoxib) 3rd trimester Juvisync (sitagliptin/simvastatin) Choline trisalicylate Beyaz (drospirenone/ethinyl estradiol) Lupron (leuprolide acetate) Pregnancy at term Doral (quazepam) Methitest (methyltestosterone) Dantrium (dantrolene) Estazolam Oxandrin () Daypro (oxaprozin) 3rd trimester Flurazepam Striant (testosterone) Diclofenac sodium Late pregnancy Halcion (triazolam) Supprelin LA (histrelin acetate) Diflunisal 3rd trimester Restoril (temazepam) Synarel (nafarelin) Duexis (ibuprofen/famotidine) Late Vistaril (hydroxyzine) Early pregnancy Testim (testosterone) pregnancy (≥30wks) Yaz (drospirenone/ethinyl estradiol) Testred (methyltestosterone) Ecotrin (aspirin) 3rd trimester DERMATOLOGICAL DISORDERS Virilon (methyltestosterone) Etodolac Late pregnancy Evista ( HCl) Amnesteem (isotretinoin) GASTROINTESTINAL TRACT Feldene (piroxicam) Late pregnancy Avage (tazarotene) Ibuprofen 3rd trimester Bellergal-S (phenobarbital/ergotamine Beyaz (drospirenone/ethinyl estradiol) Ketoprofen Late pregnancy tartrate) Carac (fluorouracil) Mobic (meloxicam) 3rd trimester Cytotec (misoprostol) Claravis (isotretinoin) Nabumetone 3rd trimester Efudex (fluorouracil) INFECTIONS & INFESTATIONS Nalfon (fenoprofen ) 3rd Estrostep Fe (norethindrone acetate/ trimester ethinyl estradiol) Bactrim (sulfamethoxazole/ Naprelan (naproxen) 3rd trimester Fluoroplex (fluorouracil) trimethoprim) 3rd trimester Prevacid Naprapac (lansoprazole/ Loryna (drospirenone/ethinyl estradiol) Copegus (ribavirin) naproxen) 3rd trimester Ortho Tri-Cyclen 28 (norgestimate/ Flagyl (metronidazole) 1st trimester for Probenecid + Colchicine ethinyl estradiol) trichomoniasis Prolia (denosumab) Propecia () Furadantin (nitrofurantoin) Pregnancy at Rheumatrex (methotrexate sodium) Silvadene (silver sulfadiazine) Late term Salsalate 3rd trimester pregnancy Gantrisin (sulfisoxazole) 3rd trimester Soma Compound w. Codeine Solage (mequinol/tretinoin) Grifulvin V (griseofulvin) (carisoprodol/aspirin/codeine) 3rd trimester Solaraze (diclofenac sodium) 3rd Gris-Peg (griseofulvin) Vimovo (naproxen/esomeprazole) Late trimester Macrobid (nitrofurantoin as pregnancy (≥30wks) Soriatane (acitretin) macrocrystals and monohydrate) Zipsor (diclofenac potassium) Late Sotret (isotretinoin) Pregnancy at term pregnancy (continued) DRUGS CONTRAINDICATED IN PREGNANCY (Part 2 of 2)

NEOPLASMS Flagyl (metronidazole) 1st trimester for Choline magnesium trisalicylate trichomoniasis Pregnancy at term Bexxar (tositumomab) Follistim (follitropin beta) D.H.E. 45 (dihydroergotamine Casodex () Ganirelix acetate mesylate) Delestrogen () Gonal-F (follitropin alfa) Diflunisal 3rd trimester Efudex (fluorouracil) Ibuprofen 3rd trimester) Etodolac Late pregnancy Eligard (leuprolide acetate) Lupron Depot (leuprolide acetate) Excedrin Migraine (acetaminophen/ Estrace (estradiol) Luveris (lutropin alfa) aspirin/ caffeine) 3rd trimester Evista (raloxifene HCl) Menopur (menoptropins) Fiorinal (butalbital/aspirin/caffeine) Firmagon (degarelix) Methergine (methylergonovine) 3rd trimester Fluoxymesterone Midol cramp (ibuprofen) 3rd trimester Fiorinal w. Codeine (butalbital/aspirin/ Menest (esterified ) Midol menstrual (acetaminophen/ caffeine/codeine phosphate) 3rd Revlimid (lenalidomide) caffeine/pyrilamine) 3rd trimester trimester Targretin (bexarotene) Midol PMS (acetaminophen/ Ibudone (hydrocodone bitartrate/ Thalomid () pamabrom/pyrilamine) 3rd trimester ibuprofen) 3rd trimester Trelstar (triptorelan pamoate) Midol teen (acetaminophen/pamabrom) Ketorolac Late pregnancy Trexall (methotrexate) 3rd trimester) Migranal (dihydroergotamine Vantas (histrelin acetate) Mifeprex () mesylate) Zytiga () Naprelan (naproxen) 3rd trimester Motrin Migraine Pain (ibuprofen) 3rd NUTRITION Ovidrel (choriogonadotropin alfa) trimester Ponstel (mefenamic acid) Late Nalfon (fenoprofen calcium) 3rd Didrex (benzphetamine) pregnancy trimester Fosteum (/citrated / Repronex 75 IU (follicle-stimulating Naprelan (naproxen) 3rd trimester cholecalciferol) /luteinizing hormone) Percodan (oxycodone HCl/aspirin) 3rd Megace ES () Repronex 150 IU (follicle-stimulating trimester Megace Suspension (megestrol acetate) hormone/luteinizing hormone) Ponstel (mefenamic acid) Late Xenical (orlistat) Serophene (clomiphene citrate) pregnancy OB/GYN Synarel (nafarelin acetate) Synalgos-DC (dihydrocodeine Tindamax (tinidazole) 1st trimester bitartrate/aspirin/caffeine) 3rd ALL ORAL CONTRACEPTIVES Zoladex (goserelin) trimester ALL HORMONE REPLACEMENT PAIN MANAGEMENT Vicoprofen (hydrocodone bitartrate/ THERAPY ibuprofen) 3rd trimester Advil (ibuprofen) 3rd trimester Advil (ibuprofen) 3rd trimester RESPIRATORY TRACT Aleve (naproxen sodium) 3rd trimester Advil Migraine (ibuprofen) 3rd Aygestin (norethindrone acetate) trimester None available Betadine douche (povidone-iodine) Aleve (naproxen sodium) 3rd UROGENITAL SYSTEM Bravelle (urofollitropin) trimester Cataflam (diclofenac potassium) Late Bayer (aspirin) 3rd trimester Avodart ( HCl) AVOID pregnancy BC Original Formula (aspirin/caffeine/ HANDLING CAPSULES Celebrex (celecoxib) 3rd trimester salicylamide) 3rd trimester Caverject (alprostadil) Cetrotide () Cafergot (ergotamine tartrate/ Edex (alprostadil) Clomid (clomiphene citrate) caffeine) Jalyn (dutasteride/tamsulosin HCl) Depo-subQ provera Caldolor (ibuprofen) 3rd trimester Lithostat (acetohydroxamic acid) (medroxyprogesterone acetate) Cataflam (diclofenac potassium) Late Proscar (finasteride) AVOID Endometrin (micronized progesterone) pregnancy HANDLING CRUSHED/BROKEN Ectopic pregnancy Celebrex (celecoxib) 3rd trimester TABLETS Not an inclusive list. (Rev. 5/2013)