<<

• Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Anti-Cancer Compound Library (96-well)

Product Details:

Catalog Number: CS-L025

Formulation: A collection of 4779 anti-cancer compounds supplied as pre-dissolved Solutions or Solid

Container: 96- or 384-well Plate with Peelable Foil Seal; 96-well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode

Storage: -80°C

Shipping: Blue ice

Packaging: Inert gas

Plate layout: CS-L025-1

1 2 3 4 5 6 7 8 9 10 11 12

SKF-96365 Fumarate MRT68921 a Empty (hydrochlorid ML162 ML-210 hydratase-IN- (dihydrochlori Peretinoin SR-3029 CBR-5884 Mivebresib AZD0156 Empty e) 1 de)

HLCL-61 b Empty BAY-876 BAY1125976 BAY-1436032 Tomivosertib LY3177833 (hydrochlorid PQR620 AT-130 NSC 663284 MK-4101 Empty e)

Flavopiridol c Empty Flavopiridol (Hydrochlorid SNS-032 Ko 143 KNK437 TA-02 Mitoquinone AZD-5438 R547 4-IBP Empty e) (mesylate)

d Empty SAR-020106 HUHS015 SMER28 A-196 TPEN CP21R7 HC-067047 EAI045 RSL3 GSK6853 Empty

IQ-1S (free Rho-Kinase- e Empty CZ415 SANT-1 ME0328 acid) GSK591 Madrasin SZL P1-41 IN-1 Nutlin-3a 9-amino-CPT Empty

MELK-8a f Empty GNE-495 EPI-001 CA-074 BI-7273 BI-9564 CL-82198 MS049 Remetinostat (hydrochlorid MRK-016 Empty methyl ester e)

SHP099 g Empty Nigericin BH3I-1 SHP099 (hydrochlorid (S)- NVP- F16 PF-04979064 Nevanimibe CFMTI Empty (sodium salt) e) ML753286 BAW2881 hydrochloride

h Empty Ro 67-7476 GNF-6231 PHCCC FCCP Linaprazan UKI-1 BFH772 CPI-455 KDM5-IN-1 CAN508 Empty

Plate layout: CS-L025-2

1 2 3 4 5 6 7 8 9 10 11 12

αvβ1 integrin- TM5275 a Empty CCF642 IMR-1 IMR-1A PACMA 31 PD-161570 HA15 WYE-132 IN-1 (TFA) (sodium) AEE788 Empty

REV7/REV3L b Empty TCS-OX2-29 HO-3867 Plerixafor TPI-1 -IN-1 NSC781406 ZYZ-488 CPI-637 A-804598 TAK-243 Empty

Rilmenidine c Empty Bay 59-3074 TBHQ (hemifumarat Rilmenidine Fisogatinib BP-1-102 SH5-07 GSK2256098 Tyrphostin M2698 Empty e) (phosphate) AG 528

GSK484 d Empty CID5721353 GLPG0187 Avadomide ITSA-1 NPS-1034 RAF709 (hydrochlorid NVS-PAK1-1 Aprepitant GKI-1 Empty e)

e Empty FMK 9a ML385 LRE1 XMU-MP-1 PD150606 CD437 DTP3 DTP3 (TFA) Golgicide A INH6 Empty

D-α- GSK-LSD1 Cyclo(RGDyK f Empty Hydroxyglutar FLLL32 (dihydrochlori GSK621 (S)-Crizotinib Tie2 kinase SecinH3 Tempol ) SGC2085 Empty ic acid de) inhibitor 1 (trifluoroaceta

Cl-amidine g Empty Necrosulfona (hydrochlorid Acriflavine NH125 AGK2 Ferrostatin-1 (-)-(S)-Equol (±)-Equol Splitomicin SirReal2 Empty mide e)

Sodium h Empty Nicaraven stibogluconat Urolithin A HJC0152 BMS453 CaCCinh-A01 AS1517499 BVT948 WNK463 APS-2-79 Empty e hydrochloride

Plate layout: CS-L025-3

1 2 3 4 5 6 7 8 9 10 11 12

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

AZD5153 (6- Empty Ticagrelor Axitinib Hydroxy-2- Mycro 3 Y-33075 L002 JTE-013 CGS 15943 GSK2837808 MS-444 Empty a naphthoic A

Y-33075 b Empty ML390 Propyl (dihydrochlori Lin28-let-7a SYP-5 TPOP146 NSC632839 Y-27632 Eganelisib GNE-272 Empty pyrazole triol de) antagonist 1

Histone c Empty GSK9311 Cambinol Acetyltransfer ML348 ML349 RA190 TPCA-1 S63845 GNE-140 (R)-GNE-140 Empty ase Inhibitor II (racemate)

d Empty (S)-GNE-140 STF-62247 PSB-12379 CXD101 STAT3-IN-1 FUBP1-IN-1 Toxoflavin HTHQ CHS-828 Ciliobrevin A Empty

NSC23005 Teglarinad e Empty (sodium) URB602 (chloride) Futibatinib 3-AP BGP-15 NCB-0846 UNC3866 GS-444217 JQEZ5 Empty

TAK-659 f Empty IWP-O1 BRCA1-IN-2 (hydrochlorid Navitoclax WT-161 KRIBB11 Bisantrene GGTI298 GCN2-IN-1 Zibotentan Empty e)

W-7 g Empty Acelarin BAY1082439 Simurosertib MX69 SAR-20347 OGT 2115 ML364 (hydrochlorid ML-9 MY-5445 Empty e)

ATM-3507 h Empty CCCP CEP-40783 (trihydrochlori Beaucage (E)-AG 99 HA-100 10074-G5 Nrf2-IN-1 CCT251236 GSK 4027 Empty de) reagent

Plate layout: CS-L025-4

1 2 3 4 5 6 7 8 9 10 11 12

ZK756326 a Empty GSK4028 ZINC1346675 LOM612 Sarcosine (dihydrochlori AG-494 D-erythro- Src Inhibitor 1 Kinetin TOFA Empty 1 de) Sphingosine riboside

Acetylcholine b Empty Monastrol Salermide LY294002 NSC 228155 SKL2001 (iodide) CeMMEC13 RHPS4 AS-605240 KYA1797K Empty

(2- Empty Importazole PD-1-IN-17 IC-87114 Hydroxypropy AR7 TG100-115 PF-06840003 EED226 666-15 TP-3654 Empty c l)-β-

PI-103 Naltrindole d Empty PNU-74654 TGX-221 PGMI-004A SF2523 PI-103 (Hydrochlorid 2- (hydrochlorid Tesmilifene Ecteinascidin Empty e) Iodomelatonin e) (fumarate) 770

Tin- e Empty protoporphyri Silodosin Agmatine XMD16-5 ZINC0088152 RPI-1 L-732138 ODQ YKL-5-124 YKL-5-124 Empty n IX (sulfate) 4 (TFA)

Milademetan f Empty Barasertib- (tosylate CHMFL-BMX- Barasertib STK16-IN-1 GDC-0326 EMT inhibitor- Thiomyristoyl ZM-447439 DMU2105 Empty HQPA hydrate) 078 1

Veliparib 3- g Empty DMU2139 Veliparib Iberdomide Pan-RAS-IN- PD-166866 (dihydrochlori R-IMPP Hesperin Harmane (Methylthio)pr Empty 1 de) opionic acid

N-(5- SI-2 h Empty Aminopentyl) L-DABA RG14620 RG13022 Trolox (R)-Trolox (hydrochlorid PF-6274484 PBIT Ceefourin 1 Empty acetamide e)

Plate layout: CS-L025-5

1 2 3 4 5 6 7 8 9 10 11 12

IT1t Trilaciclib a Empty SR0987 (dihydrochlori RAD51 (hydrochlorid (±)- Zanubrutinib Dihydromund LF3 GZD856 LY3214996 Empty de) Inhibitor B02 e) Zanubrutinib uletone (formic)

MT-DADMe- Polyoxyethyle b Empty ImmA Pico145 F1063-0967 A-395 eIF4A3-IN-1 Cdc7-IN-1 TC13172 ne stearate AZD-5991 MRX-2843 Empty

Elimusertib c Empty HI-TOPK-032 Linrodostat Avapritinib GDC-0077 GSK3326595 JNJ- Elimusertib (hydrochlorid BMS-986158 Roblitinib Empty 64619178 e)

Nilotinib Empty Darovasertib Bosutinib Nilotinib NVX-207 (monohydroc Tozasertib MSC2530818 Olaparib Recilisib Ilaprazole Empty d hloride

UAMC00039 e Empty LTURM34 Oxyphenisati IMD-0354 TM5441 PRN1371 (dihydrochlori BTB-1 CSF1R-IN-1 ML311 PHA-680632 Empty n acetate de)

ZM223 Dasatinib f Empty EDO-S101 eIF4A3-IN-2 Danusertib (hydrochlorid NCGC002445 MLN8054 SK1-IN-1 Dasatinib (hydrochlorid CHIR-99021 Empty e) 36 e)

CHIR-99021 CHIR-99021 EIPA g Empty (monohydroc (trihydrochlori DKM 2-93 dBET1 EIPA (hydrochlorid ML-18 FITM AX-15836 Fasentin Empty hloride) de) e)

N6-(2- LYN-1604 h Empty STAT5-IN-1 Phenylethyl)a TG 100801 AU1235 Linsitinib Heparan NVP-TAE 684 Autophinib (dihydrochlori CM-272 Empty denosine Sulfate de)

Plate layout: CS-L025-6 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

1 2 3 4 5 6 7 8 9 10 11 12

Sepantronium a Empty KDM4D-IN-1 CU-CPT17e AZD-1480 hVEGF-IN-1 TNP-470 (bromide) BTK IN-1 LY 345899 SMI-16a AD80 Empty

CB-1158 IACS-9571 b Empty SPI-112 NCT-503 Wortmannin AZ PFKFB3 Selitrectinib CPI-444 (dihydrochlori AZD4635 BMS-754807 (hydrochlorid Empty 26 de) e)

Tandutinib c Empty Rucaparib Sorafenib BMS-1166 6-Biopterin Sorafenib Tandutinib A2A receptor FX1 KY1220 (hydrochlorid Empty (Camsylate) (Tosylate) antagonist 1 e)

KDOAM-25 d Empty Linperlisib Oxamflatin CDK9-IN-8 OSI-930 (citrate) STAT5-IN-2 Cediranib WM-1119 MOZ-IN-2 Amuvatinib Empty

Retaspimycin e Empty WM-8014 Dovitinib Pazopanib SAFit2 2OH-BNPP1 JPM-OEt Masitinib Masitinib (Hydrochlorid Tanespimycin Empty (lactate) (mesylate) e)

f Empty BIIB021 Luminespib Everolimus Rapamycin Vorinostat Ixabepilone CUDC-101 Panobinostat Belinostat Bortezomib Empty

Motesanib BRAF AKT Kinase NVP- g Empty Motesanib (Diphosphate) Midostaurin Saracatinib inhibitor RAF265 GSK-690693 Inhibitor ADW742 AG1024 Empty

SB 203580 h Empty PD0325901 Sunitinib SB 203580 (hydrochlorid BAY 11-7085 Vandetanib Afatinib Afatinib BMS-536924 SB 202190 Empty e) (dimaleate)

Plate layout: CS-L025-7

1 2 3 4 5 6 7 8 9 10 11 12

(+)-BAY- (±)-BAY- (-)-BAY- a Empty Omipalisib GSK-923295 HSF1A HMN-154 Gusacitinib 1251152 1251152 1251152 BAY-1816032 LY3200882 Empty

BET EHNA b Empty Repotrectinib PIK-294 bromodomain Diethyl- T-3775440 E7046 R162 PU02 inS3-54A18 (hydrochlorid Empty inhibitor pythiDC hydrochloride e)

5'-N- Empty Ethylcarboxa Proxalutamid Doramapimod PD173074 Falnidamol D4476 Ro 90-7501 TCPOBOP Toyocamycin CL-387785 Empty c midoadenosin e

Regorafenib d Empty TC ASK 10 GW788388 BAI1 PD176252 JNJ-7706621 Toceranib Toceranib Regorafenib Calmidazoliu (monohydrate Empty (phosphate) m chloride )

1- e Empty BMS-690514 PETCM CA-074 Proglumide Brivanib Brivanib Foretinib Aminobenzotr KW-2449 Methylmaloni Empty (sodium) (alaninate) iazole c acid

Tirbanibulin Fasudil f Empty Tirbanibulin (dihydrochlori Tirbanibulin (Hydrochlorid Enzastaurin Sotrastaurin AZD 6482 ARP-100 G15 PHTPP Empty de) (Mesylate) e)

5'- MK-2206 g Empty AV-412 Fluoroindirubi AV-412 (free JNJ0966 PI-273 Takinib AKT inhibitor (dihydrochlori DUPA(OtBu)- LCL521 Empty noxime base) VIII de) OH

LCL521 4,4'- PROTAC PROTAC Amifostine (2R)-Octyl-α- (2S)-Octyl-α- h Empty dihydrochlorid Dimethoxybe PKM2-IN-1 CDK9 BET thiol hydroxyglutar hydroxyglutar GW779439X K00546 Empty e nzil Degrader-1 Degrader-1 (dihydrochlori ate ate

Plate layout: CS-L025-8

1 2 3 4 5 6 7 8 9 10 11 12

Fmoc-1,6- IPN60090 Canertinib a Empty Tetraphenylp BI-78D3 MAK683 diaminohexan STING 2-HBA Canertinib IPN60090 (dihydrochlori (dihydrochlori Empty orphyrin e agonist-3 de) de)

Samuraciclib b Empty PF-06726304 NAZ2329 CD73-IN-1 PTC-028 Gardiquimod iCRT3 ROC-325 Pim1/AKK1- IBR2 (hydrochlorid Empty (diTFA) IN-1 e)

Samuraciclib c Empty (trihydrochlori Seclidemstat Ensartinib PP121 Semaxinib PD173955 Emricasan CTS-1027 BAY-320 BAY-524 Empty de) hydrochloride

Fmoc-Ser(O- Empty α-D- Asciminib NecroX-5 Losmapimod L-Kynurenine PH-797804 IDH-305 Cintirorgon MKC8866 Vorasidenib Empty d GalNAc(OAc)

Naphthol AS- e Empty Pamiparib QC6352 Lanifibranor Talmapimod 1A-116 Theliatinib E SU 5402 LG-100064 Fedratinib Empty

Fedratinib f Empty (hydrochlorid TG101209 AZ960 kinase AZD-8055 OSI-027 Milciclib A-443654 XCT790 SB-431542 Empty e hydrate) inhibitor

Dapagliflozin Empty Vismodegib Pralatrexate Capsaicin Capsaicin Dapagliflozin ((2S)-1,2- Canagliflozin Ixazomib Ixazomib Delanzomib Empty g (purity>99%) propanediol, citrate

SCH- Empty PF-562271 PF-562271 PF-573228 Torkinib AM580 1473759 Pevonedistat Dinaciclib SC75741 BMS-794833 Empty h (besylate) (hydrochlorid hydrochloride

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Plate layout: CS-L025-9

1 2 3 4 5 6 7 8 9 10 11 12

Melflufen Pimonidazole a Empty Lexibulin SU14813 (hydrochlorid SU14813 Tipifarnib Tipifarnib (S Orteronel BI-D1870 AR-A014418 (hydrochlorid Empty e) (maleate) enantiomer) e)

BMS-345541 b Empty BX795 Orantinib (Z)-Orantinib (hydrochlorid BMS-345541 CGP 57380 GSK1904529 Telatinib Tasquinimod Betulinic acid Empty e) A

Tariquidar Empty Varlitinib ARRY-380 Eniluracil Evofosfamide GW 5074 Tariquidar (methanesulf CYC-116 Nelotanserin IMD-0560 Empty c (analog ) onate,

Y-27632 d Empty Nevirapine Efavirenz PD 169316 Pluripotin GSK 3 Flurbiprofen (dihydrochlori Valproic acid Valproic acid 5-Azacytidine Empty Inhibitor IX de) (sodium salt)

Rucaparib e Empty BIX-01294 TWS119 IQ 1 Lobaplatin Zamicastat Liarozole A-966492 (phosphate) PMX-53 Rucaparib Empty

Niraparib GW3965 DL- L-Buthionine- DL- f Empty Niraparib (hydrochlorid Niraparib Niraparib (R- T0901317 (hydrochlorid LXR-623 Buthionine- (S,R)- Buthionine- Empty e) (tosylate) enantiomer) e) (S,R)- sulfoximine (S,R)-

L-Buthionine- Chloroquinox Peldesine g Empty (S,R)- Tefinostat Neticonazole Mitoguazone aline MK-6892 PKI-402 (dihydrochlori S 3304 Ningetinib Empty sulfoximine sulfonamide de) Tosylate

h Empty Ningetinib PZ-128 PF-AKT400 G-1 β-Elemene AZD4205 CH7057288 MTX-211 PQR530 SGN-2FF Empty

Plate layout: CS-L025-10

1 2 3 4 5 6 7 8 9 10 11 12

Epertinib 6-Bromo-2- a Empty (hydrochlorid hydroxy-3- Uridine Benzo[a]pyre Epristeride UK 356618 CD3254 B I09 Proteasome SR11237 Empty e) methoxybenz triphosphate ne inhibitor IX

I-BET762 N- PROTAC b Empty NU6140 BAY-299 Oxythiamine LE135 carboxylic Deshydroxyet BET-binding SLF-amido- OSS_128167 A-485 Empty acid hyl Dasatinib moiety 1 C2-COOH

JNK Inhibitor Guggulsteron Duocarmycin c Empty (E/Z)-AG490 GSK8573 A 1070722 Garcinol VIII GYY4137 DC_AC50 MIF-1 (TFA) e TM Empty

SCR7 5- d Empty Fluensulfone LLY-283 PF-9366 BI-882370 (Z)-JIB-04 pyrazine Fluorouridine Isosulfan blue LSN 3213128 FT671 Empty

Aminooxyacet Delphinidin 3- e Empty GNE-6776 EG00229 ic acid CADD522 CCT 137690 glucoside GNE-493 Pemetrexed Pemetrexed Raltitrexed Empty (hemihydrochl (chloride) (disodium)

6- 6-Diazo-5- f Empty (R)- Mogroside II- Promestriene GC7 Sulfate Aminochryse ABL127 Brequinar SB-633825 oxo-L-nor- PDD Empty Bicalutamide A2 ne Leucine 00017273

Talazoparib g Empty CCG-203971 GW 501516 tosylate (R)-Equol WHI-P258 GNE-049 Pretomanid WS-12 Delamanid Ro 08-2750 Empty

Nolatrexed RS-25344 h Empty Ro5-3335 CU-CPT22 Loxoribine dihydrochlorid TMPyP4 LAT1-IN-1 NSC 95397 WAY 316606 (hydrochlorid BYK204165 Empty e tosylate e)

Plate layout: CS-L025-11

1 2 3 4 5 6 7 8 9 10 11 12

AZ10606120 a Empty PhiKan 083 PhiKan 083 CMPD1 (dihydrochlori PF-06465469 GNE-781 PT2399 (Rac)-PT2399 ML-792 BI-3802 Empty hydrochloride de)

N-Desethyl Lavendustin b Empty GeA-69 TDCPP Sunitinib LRRK2-IN-1 Clotrimazole JWG-071 B GlyRS-IN-1 JFD00244 Rosiptor Empty

Parsaclisib c Empty Tucidinostat Vorolanib Adavivint Alobresib Lazertinib (hydrochlorid Ralaniten Vecabrutinib Belvarafenib Conteltinib Empty e)

Fosifloxuridin Empty Pemigatinib Tegatrabetan Telratolimod Valemetostat e Danicamtiv GW2580 Giredestrant Rezivertinib Zandelisib Empty d (tosylate) nafalbenamid

Calf thymus Cerivastatin 5α-Pregnane- e Empty UNC0224 UNC0321 Pifithrin-μ VER-155008 VER-82576 GNF-7 SMER3 3β,6α-diol-20- Empty DNA (sodium) one

D4- Momelotinib f Empty ASTX660 AZD1390 Raf inhibitor 2 IRAK4-IN-7 RG7112 Momelotinib abiraterone sulfate Vadimezan SB-590885 Empty

Obatoclax Lenvatinib Pomalidomid ENMD-2076 g Empty (Mesylate) Alisertib MK-0752 Tivozanib Lenvatinib (mesylate) Amonafide e (Tartrate) ENMD-2076 Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Trametinib h Empty MGCD-265 AZD-7762 Adavosertib KHS101 Ibrutinib Ibrutinib Trametinib (DMSO GSK429286A PHA-793887 Empty analog hydrochloride (Racemate) solvate)

Plate layout: CS-L025-12

1 2 3 4 5 6 7 8 9 10 11 12

(Z)- a Empty CP-466722 GW843682X AZ 628 BX-912 TBCA KU-57788 Guggulsteron GNF-2 TNP CGP60474 Empty e

Furamidine b Empty A-484954 AS601245 TDZD-8 DSR-6434 NU9056 (dihydrochlori UNC3230 SP-141 SPP-86 R-7050 Empty de)

SNT-207858 VUF11207 c Empty BRD9876 Tilfrinib ML334 GN44028 Apcin SNT-207707 (free base) (fumarate) WAY-262611 CU-T12-9 Empty

PKI-179 Alendronate 2,2,5,7,8- d Empty Capzimin GNE-477 Fingolimod PKI-179 (hydrochlorid (sodium RO4929097 Pentamethyl- Corin Pilaralisib Empty e) hydrate) 6-Chromanol analogue

3- e Empty JNJ- Nintedanib PHA-665752 R406 (free Resatorvid AZ1495 FL-411 LDH-IN-1 EZM 2302 Methyltoxofla Empty 38877618 esylate base) vin

(E/Z)- f Empty JT010 CZC-8004 PIK-108 IPR-803 GSK5182 HAMNO HDAC8-IN-1 ONC212 FT827 FN-1501 Empty

SEL120-34A g Empty NMDI14 BI-3812 E-7386 IDF-11774 (monohydroc SR-4370 MK-8353 EOAI3402143 ATX inhibitor EBI-2511 Empty hloride) 1

1- 1,4- h Empty CBP/p300-IN- PLX51107 BDP9066 SSE15206 Ethynylnapht Chrysenequin CeMMEC1 AHR GSK2643943 Porcn-IN-1 Empty 1 halene one antagonist 1 A

Plate layout: CS-L025-13

1 2 3 4 5 6 7 8 9 10 11 12

DIM-C- RGX-104 a Empty SM 16 AZD-0364 GDC-0927 INCB-057643 LSZ-102 pPhOCH3 RGX-104 (free Acid) Y06036 Y06137 Empty

PDGFRα b Empty NAcM-OPT kinase PI3K/mTOR GSTO1-IN-1 MAGL-IN-1 IDO1-IN-5 (Rac)-IDO1- (S)-IDO1-IN-5 M1001 Bragsin1 Empty inhibitor 1 Inhibitor-2 IN-5

Bobcat339 SAHA 5-Aza-7- c Empty FT113 TAS0728 (hydrochlorid BDP-13176 chloroalkane Melengestrol BTR-1 DC661 deazaguanin PluriSIn #2 Empty e) T1 acetate e

Epsilon- 3- EML4-ALK d Empty momfluorothri Methylcytidin Gboxin S-Gboxin VL285 kinase WDR5-IN-4 BLM-IN-1 NRX-252262 FASN-IN-1 Empty n e inhibitor 1 (TFA)

CBP/p300-IN- HO-1-IN-1 e Empty AZD-7648 4 CSF1R-IN-2 Subasumstat M3258 ACY-1083 HO-1-IN-1 hydrochloride TH34 VH032 thiol Empty

ZZW-115 PROTAC 5-Iodo- D-Ala-Lys- f Empty (hydrochlorid RIPK SNIPER(ABL) indirubin-3'- GSK8612 GSK3145095 AMCA IACS-010759 Unesbulin Aminomalonic Empty e) degrader-6 -020 monoxime (hydrochlorid acid

Saccharin 1- N-Bis(2- g Empty DIM-C- DIM-C- methylimidaz CIL56 SHIN1 (S,R,S)- BAY885 hydroxypropyl AZD4573 LXH254 Empty pPhOH pPhCO2Me ole AHPC-Me )nitrosamine

Chitosan h Empty ABBV-744 eCF506 E260 oligosacchari SLV-2436 AGI-24512 MAT2A TAO Kinase JH-VIII-157- FLT3-IN-3 Empty de inhibitor 1 inhibitor 1 02

Plate layout: CS-L025-14

1 2 3 4 5 6 7 8 9 10 11 12

EG01377 GDC-0575 a Empty (dihydrochlori MS4078 NSC139021 Branebrutinib PRN1008 GDC-0575 dihydrochlorid KO-947 UM-164 ARQ 531 Empty de) e

Lerociclib GW806742X b Empty MIK665 D-Lin-MC3- CDK12-IN-3 (dihydrochlori M443 TNF-α-IN-1 ERK1/2 C188-9 IDH889 (hydrochlorid Empty DMA de) inhibitor 1 e)

trans- NCGC002477 (R)- (Rac)- c Empty T025 TAS6417 Pralsetinib Pralsetinib AZ32 Ripretinib 43 BAY1238097 BAY1238097 BAY1238097 Empty

Aurora kinase EGFR/ErbB- d Empty SJ000291942 MZP-54 MZP-55 AZD4320 2/ErbB-4 CE-245677 ETC-206 Sirt2-IN-1 HJB97 Empty inhibitor-2 inhibitor-2

PNU112455A α-2,3- e Empty MF-094 AZD3458 SGC3027 (hydrochlorid NAV-2729 PRL-3 RS-246204 INCB054329 GSTO-IN-2 sialyltransfera Empty e) Inhibitor I se-IN-1

H3B-6545 9- f Empty MAT2A CC-90003 MC3482 dBET6 H3B-6545 (hydrochlorid Tubulin CF53 H3B-5942 Methoxycanth Empty inhibitor 2 e) inhibitor 1 in-6-one

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

V-9302 N-alpha- PROTAC g Empty BAY-2402234 CG-806 GCN2iB V-9302 (hydrochlorid CA-5f CCR6 LV-320 Tosyl-L-lysine BET Empty e) inhibitor 1 chloromethyl Degrader-10

4'- h Empty BRD 4354 FDI-6 Sparfosic acid Methylchryso Hexadimethri BN82002 (+)-JQ1 PA DK419 AZD3229 AZD3229 Empty (trisodium) eriol ne bromide Tosylate

Plate layout: CS-L025-15

1 2 3 4 5 6 7 8 9 10 11 12

Almonertinib a Empty SGC-iMLLT KAN0438757 ALK2-IN-2 S130 ON-013100 Almonertinib (hydrochlorid TVB-2640 MBQ-167 TL02-59 Empty e)

diABZI Empty VU0661013 nor-NOHA UT-155 (R)-UT-155 IITZ-01 UAMC-3203 Grp94 mTOR STING DT-061 Empty b (acetate) hydrochloride Inhibitor-1 inhibitor-1 agonist-1

N1- 1- N2,N2- Estrone 10Z- c Empty (1S,2S,3R)- GNE-6640 ChX710 Urocanic acid Acetylspermid Methylguanos Dimethylguan sulfate FAPy- Nonadecenoi Empty DT-061 ine ine osine (potassium) adenine c acid

Stachyose ERRα LPA2 (S)-PF- d Empty (tetrahydrate) 9-ING-41 Actinonin antagonist-1 antagonist 2 trans-AUCB VTP50469 2-D08 WRG-28 06873600 Empty

BI-9321 PROTAC Se- e Empty GW284543 (trihydrochlori MRK-740 Olutasidenib BET USL311 Methylseleno LY3295668 NXT629 Sotorasib Empty de) degrader-2 cysteine

FGFR1/DDR2 NQO1 MARK4 Glutaminase- DS-1205b f Empty CCB02 COH000 inhibitor 1 MD-224 substrate inhibitor 1 IN-1 CDK4/6-IN-2 HS-1371 (free base) Empty

SRI 31215 HDACs/mTO g Empty ONO-7475 (TFA) Selpercatinib SHP394 BAY-293 TD-106 GB1107 CCI-006 R Inhibitor 1 GS-626510 Empty

AP1867-2- h Empty (carboxymeth P110δ-IN-1 MRTX-1257 INH14 AES-135 ULK-101 Rineterkib GSK547 NSAH LY2452473 Empty oxy)

Plate layout: CS-L025-16

1 2 3 4 5 6 7 8 9 10 11 12

Camptothecin Pyridoxal a Empty Benproperine -20(S)-O- SJ572403 isonicotinoyl Fluzoparib SLF SLF (TFA) DDAO KEA1-97 Fluorizoline Empty (phosphate) propionate

BCI b Empty JNJ- 1V209 G5-7 UBCS039 EB-3D CLK-IN-T3 MF-766 BCI (hydrochlorid NAE-IN-M22 Empty 63576253 e)

8- c Empty K-Ras-PDEδ- GW406108X MALAT1-IN-1 Pitstop 2 ML-180 KS15 ILK-IN-3 Azaadenosin Glumetinib RMC-4550 Empty IN-1 e

5-Fluoro-2'- (S)-(?)-Perillyl PIN1 inhibitor d Empty SRS11-92 Ceranib-2 deoxycytidine 1G244 VPC-14449 Bigelovin alcohol MAZ51 API-1 GSK467 Empty

MLS0005322 e Empty PFM01 BRD0705 BRD5648 SRPKIN-1 ANI-7 JI051 23 INH154 PKI-166 FzM1.8 Empty

S55746 f Empty CDK12-IN-E9 Diallyl NCT-502 AZD7507 AZ304 JG-98 (S)-JQ-35 S55746 (hydrochlorid USP25/28 Empty Trisulfide e) inhibitor AZ1

CM-579 g Empty NGI-1 ALLO-2 trihydrochlorid CDK2-IN-4 UNC569 AUT1 SPHINX31 I-191 BJE6-106 HJC0197 Empty e

SK1-?I h Empty SU4984 BTdCPU Clitocine 4-MMPB Tyrphostin Coralyne Vacuolin-1 (hydrochlorid RU-301 MS7972 Empty AG30 (chloride) e)

Plate layout: CS-L025-17

1 2 3 4 5 6 7 8 9 10 11 12

a Empty Halopemide Laminaran NSC-60339 CCT020312 K777 Apratastat SX-682 ODM-203 UPGL00004 FLTX1 Empty

Xanthopterin Tyrphostin b Empty Camalexin AZ9482 (hydrate) Hematein AG1433 Trofosfamide RIPK1-IN-7 CHDI-390576 MC180295 JND3229 Empty

SNS-314 Fingolimod Erlotinib Pazopanib c Empty Caracemide AG490 MS402 WZ-3146 (hydrochlorid TVB-3664 TJ191 (Hydrochlorid (Hydrochlorid Empty (mesylate) e) e) e)

BMS-599626 PD153035 d Empty (Hydrochlorid HA14-1 Metarrestin SB 216763 (Hydrochlorid CMP-5 SU11274 EC359 MST-312 Iniparib Empty e) e)

PF-04217903 Vatalanib 3- e Empty KU-55933 PF-04217903 (methanesulf (dihydrochlori SGX-523 TW-37 BI8626 XY018 VH032 Aminobenza Empty onate) de) mide

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Alvespimycin 2- f Empty GTx-007 (hydrochlorid Serdemetan WZ4002 SMAP-2 PD98059 PIK-90 U0126-EtOH AG14361 Methoxyestra Empty e) diol

T-1101 Rigosertib g Empty WYE-354 AMG-208 BI-1347 (tosylate) GSK1059615 (sodium) Ki8751 Lyn-IN-1 TVB-3166 UC-514321 Empty

Cabozantinib Chelerythrine h Empty Elesclomol KDM5-C70 SP600125 Pimasertib SB 525334 (S-malate) HMN-214 PIK-93 Ponatinib (chloride) Empty

Plate layout: CS-L025-18

1 2 3 4 5 6 7 8 9 10 11 12

N- GB-110 a Empty CCT129202 CP-673451 Acetyltyramin (hydrochlorid Vinorelbine Hesperadin KBU2046 BIX02188 BIX02189 Vemurafenib Empty e e) (ditartrate)

AT7867 BMS-1001 b Empty TH1338 AZD8330 AT7867 VERU-111 (dihydrochlori KRN-633 KU-60019 PD318088 PHT-427 (hydrochlorid Empty de) e)

SB-743921 LDN193189 c Empty R406 SSTC3 PI3K-IN-1 (hydrochlorid MSAB DPH (Tetrahydroch TCH-165 LY2109761 BMS 777607 Empty e) loride)

d Empty CMC2.24 ARN-3236 MRT199665 BI8622 BCI-215 Chrysene Oprozomib Droloxifene L-Albizziin 1,4-DPCA Empty

Mepazine Vofopitant e Empty BI-167107 (hydrochlorid Poloxin Purpurogallin Volasertib dihydrochlorid (E/Z)-IT-603 CAY10404 PS210 Entinostat Empty e) e

Prinomastat Aliskiren f Empty Quinoclamine (5Z,2E)-CU-3 Mocetinostat Marimastat (hydrochlorid CCG-222740 Aliskiren (hemifumarat SHP836 FW1256 Empty e) e)

BPK-29 g Empty TAK-901 MEK inhibitor JR-AB2-011 PFK-158 PFK-015 (hydrochlorid Omaveloxolo ML-60218 CDDO-EA Lorlatinib Empty e) ne

OTS186935 h Empty (hydrochlorid SGC-GAK-1 ML367 MM-102 AC-73 BAY-8002 PI-3065 IWR-1 CID755673 AZ82 Empty e) (TFA)

Plate layout: CS-L025-19

1 2 3 4 5 6 7 8 9 10 11 12

Glabrescione a Empty Telaglenastat Retro-2 B PTUPB TRPM4-IN-1 DPA-714 SPOP-IN-6b Mcl1-IN-8 TH-257 Ciliobrevin D Empty

Deltasonamid Mefuparib b Empty Deltasonamid e 2 (hydrochlorid sAJM589 CCI-007 SEC inhibitor GOT1 STL127705 DMH-1 ML347 Empty e 2 (TFA) (hydrochlorid e) KL-1 inhibitor-1

Umbralisib c Empty FR 180204 MALT1 AZ191 δ-Tocotrienol Umbralisib (hydrochlorid THZ2 FPH2 HLY78 bpV(phen) Empty inhibitor MI-2 e) (trihydrate)

RAS inhibitor d Empty Serabelisib AZ12601011 PI-1840 Abd-7 ZT-12-037-01 YH239-EE MKK7-COV-9 HOIPIN-1 Defactinib E64FC26 Empty

Defactinib e Empty (E/Z)- (hydrochlorid TK216 (-)-TK216 HG6-64-1 RIPGBM Borussertib IM-12 LY2857785 Sulfatinib Empty E64FC26 e)

8-Bromo- f Empty WH-4-023 Kenpaullone IOX1 AS1708727 Q-VD-OPh BTSA1 Adenosine cAMP sodium (S,R,S)- AKI603 Empty dialdehyde salt AHPC-Boc

20(S)- g Empty Hydroxychole FTI-2153 FTI-2153 GSK2194069 SM-276001 AZD8186 KRCA-0008 G-749 HTH-01-015 UNC0379 Empty sterol (TFA)

UNC2025 Mozavaptan h Empty GK921 ETP-46321 ML216 UNC2025 (hydrochlorid OUL35 Enocitabine SB-3CT (hydrochlorid TH1834 Empty e) e)

Plate layout: CS-L025-20

1 2 3 4 5 6 7 8 9 10 11 12

TH1834 CDK5 a Empty (dihydrochlori Supinoxin C75 trans-C75 Namodenoso MCP110 inhibitor 20- NMS-P715 FEN1-IN-1 KPT-6566 Empty de) n 223

Ralaniten LIN28 LIN28 SEC inhibitor b Empty RK-287107 inhibitor LI71 JMS-17-2 ZLDI-8 RTC-5 ζ-Stat CTPI-2 Empty triacetate inhibitor LI71 enantiomer KL-2

c Empty MKC9989 Mps1-IN-3 SRT 1460 TAS-114 6H05 (TFA) PFI-3 ML132 DS-437 WYC-209 E7449 Empty

JNJ- Voruciclib (2S,3R)- 42-(2- d Empty BMS-983970 47117096 BET-BAY 002 (hydrochlorid Voruciclib TAS-115 Zotarolimus Tetrazolyl)rap Gilteritinib PIP-199 Empty hydrochloride e) (hydrochlorid mesylate amycin

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Gilteritinib e Empty hemifumarate INT-767 BDP5290 G007-LK Y15 BTYNB CDKI-73 Crenigacestat Chiauranib DM4 Empty

AMXT-1501 f Empty OBI-3424 Minnelide PTC299 DI-591 tetrahydrochl IPI-9119 DB2313 WJ460 Z-Ile-Leu- HSP27 Empty oride aldehyde inhibitor J2

OTS964 BMP g Empty Z-DEVD-FMK (hydrochlorid A-1210477 D-I03 signaling TBOPP p32 Inhibitor hSMG-1 KY-05009 Mutant IDH1- Empty e) agonist sb4 M36 inhibitor 11j IN-1

hSMG-1 Rheb inhibitor SAR405 R h Empty inhibitor 11e SW106065 NR1 SAR405 enantiomer COH-SR4 iGOT1-01 CMLD-2 BMH-21 STD1T Empty

Plate layout: CS-L025-21

1 2 3 4 5 6 7 8 9 10 11 12

Malic enzyme LY-2584702 a Empty SC99 inhibitor ME1 LY2510924 (6R)-FR054 VER-246608 (tosylate salt) LDC1267 APS6-45 β-NETA CTPB Empty

b Empty TRi-1 Bozitinib CFM-2 LCH-7749944 Samotolisib AA92593 DB04760 NSC 185058 OF-1 Oltipraz Empty

CFTR c Empty PF-06380101 MS645 TED-347 Pyridoclax Ro-3306 Velpatasvir DRF-1042 SEC corrector 2 NP-G2-044 Empty

3- Alpha- MS31 (S,S,S)- d Empty LY3009120 Phenyltoxofla BI-3406 Cytidine-5'- A-366 Naphthoflavo GMB-475 (trihydrochlori AHPC Ginsenoside Empty vin triphosphate ne de) (hydrochlorid F2

ZM39923 VH032- e Empty Thiamet G (hydrochlorid cyclopropane Allocholic HM03 URMC-099 AZD5582 Bractoppin DFP00173 WS-383 Empty e) -F acid

JAK/HDAC- PKC-iota Tankyrase- f Empty IN-1 inhibitor 1 J22352 TAM-IN-2 HSP70-IN-1 ON123300 CDC25B-IN-1 BI-2852 IN-2 CDK9-IN-7 Empty

ERK1/2 g Empty BI-4916 BI-4924 HSD1590 GNE-618 inhibitor 2 c-Fms-IN-10 SU5204 GNE 2861 EGFR-IN-8 SP2509 Empty

PROTAC (S,R,S)- Rhosin h Empty ERRα ligand CDDO-2P-Im Kansuinine A Acalisib AHPC- Thalidomide- (hydrochlorid Telomerase- FASN-IN-4 Y16 Empty 2 propargyl propargyl e) IN-2 (tosylate)

Plate layout: CS-L025-22

1 2 3 4 5 6 7 8 9 10 11 12

LSN3106729 Succinyl a Empty (hydrochlorid MPI-0479605 AMG PERK Entrectinib CCT251545 Glutaminase BPTES phosphonate Mitapivat KSI-3716 Empty e) 44 C-IN-1 (trisodium

Bromocriptine FMF-04-159- Genz-123346 b Empty (mesylate) FB23-2 2 NDI-091143 ML324 Liproxstatin-1 EPZ015666 (free base) DC-05 DC_517 Empty

YHO-13351 c Empty AZD3965 ML228 ML141 YHO-13177 (free base) CARM1-IN-1 QS11 GNE-317 BLZ945 IC261 Empty

Iadademstat 5-(N,N- d Empty (dihydrochlori L-779450 Vps34-IN-1 AG1557 Hexamethyle Acifluorfen STF-118804 EHop-016 Autotaxin TH588 Empty de) ne)-amiloride modulator 1

Thienopyrido e Empty ne BLU9931 BHPI IMB-XH1 KH-CB19 M-110 Autogramin-2 ERK5-IN-2 PK68 FGTI-2734 Empty

Neticonazole SAG SAG f Empty FGTI-2734 (hydrochlorid Mirk-IN-1 UC-112 Allyl methyl CCT196969 SAG (hydrochlorid (dihydrochlori ARS-1323- Empty (mesylate) e) sulfide e) de) alkyne

TAS4464 g Empty Antineoplasto Lys05 GSK503 Brigatinib FLT3-IN-6 Empesertib TAS4464 (hydrochlorid Mevociclib STAT3-IN-3 Empty n A10 e)

MD2-TLR4- Legumain Larotrectinib h Empty BAY1217389 PHT-7.3 IN-1 XY101 CB-5083 inhibitor 1 Brilanestrant Larotrectinib sulfate PT-2385 Empty

Plate layout: CS-L025-23

1 2 3 4 5 6 7 8 9 10 11 12

AZD9496 Atuveciclib GSK3368715 a Empty Bimiralisib PGAM1-IN-1 PGAM1-IN-2 AZD-8835 BpV(HOpic) AZD9496 (dihydrochlori Atuveciclib Empty (maleate) (Racemate) de)

Atuveciclib S- DNA2 K-Ras G12C- b Empty Enantiomer Nazartinib inhibitor C5 RBC8 CASIN BQU57 SIAIS178 M2N12 IN-4 WEHI-9625 Empty

cIAP1 ligand CBP/p300-IN- Pyropheopho c Empty DBPR112 PK11007 IWP-4 1 Coenzyme A bio-THZ1 3 SKI-178 SKI V rbide-a Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

N- Abemaciclib AP1867-3- CC-90011 d Empty Iobenguane TFMB-(R)-2- Desmethylta XY028-133 CCT369260 ASLAN003 AGX51 metabolite (aminoethoxy (benzenesulf Empty (sulfate) HG moxifen M20 ) onate)

Benzyl-α- e Empty GalNAc Orelabrutinib CC-92480 Metoprine GNE-3511 TC11 AMG319 Enpp-1-IN-1 R-268712 DS-1001b Empty

Asperphenam MCL-1/BCL- MCL-1/BCL- MCL-1/BCL- f Empty ate SKLB4771 MYCi361 MYCi975 Dubermatinib SGI-7079 S49076 2-IN-1 2-IN-2 2-IN-3 Empty

EPZ020411 N1,N8- g Empty (hydrochlorid Nampt-IN-1 PRT-060318 AZ6102 Pimozide LDN-91946 Spautin-1 Diacetylsper Quizartinib Torin 2 Empty e) midine

Alectinib h Empty Torin 1 Maraviroc PF-3758309 Alectinib (Hydrochlorid RepSox MRTX849 Cabozantinib MRT67307 GSK1838705 Empty e) A

Plate layout: CS-L025-24

1 2 3 4 5 6 7 8 9 10 11 12

CC-401 a Empty Thiodigalacto (hydrochlorid S516 Rebastinib GCN2-IN-6 SR-4835 DS18561882 IRAK4-IN-6 Src Inhibitor 3 Idelalisib Empty side e)

Palbociclib- (R)-(-)-JQ1 GSK Molibresib b Empty HIF-2α-IN-2 DAPT propargyl (+)-JQ-1 Enantiomer Molibresib 525768A (besylate) CDK-IN-2 Gandotinib Empty

IBT6A Fostamatinib c Empty (Rac)-IBT6A IBT6A (hydrochlorid Fostamatinib Fostamatinib (disodium Cediranib Sapitinib Cdc7-IN-5 Ro-0335 Empty e) Disodium hexahydrate) (maleate)

1- Daunorubicin d Empty Naphthohydr Telotristat Telotristat O6BTG- DCZ0415 DT2216 Nampt-IN-5 Daun02 EGFR-IN-11 (hydrochlorid Empty oxamic acid etiprate ethyl octylglucoside e)

Cobimetinib e Empty Cobimetinib (hemifumarat Isobavachalc TL12-186 Tripterin Golvatinib MDM2-IN-1 TD-165 Cenisertib VO-Ohpic Empty e) one (trihydrate)

FKBP12 N-piperidine Androgen f Empty Cobimetinib TLR7/8 CC-90009 DBCO-PEG4- PROTAC HS-27 Thalidomide- EED226- Ibrutinib receptor Empty (racemate) agonist 3 Biotin RC32 O-C8-COOH COOH (hydrochlorid antagonist 1

SHP2-IN-6 Desmorpholin g Empty Taletrectinib KCC-07 EMI48 EMI56 (hydrochlorid BD750 Thalidomide- yl Navitoclax- DM-01 Lenalidomide Empty e) O-C8-Boc NH-Me -I

DOTA- h Empty tris(tBu)ester Pirtobrutinib SP-96 Syk-IN-4 mTOR PI3Kα-IN-4 (S)-PI3Kα-IN- PD-1/PD-L1- Nur77 KB02-COOH Empty NHS ester inhibitor-8 4 IN-NP19 modulator 1

Plate layout: CS-L025-25

1 2 3 4 5 6 7 8 9 10 11 12

1- Thalidomide- a Empty Ethynylpyren SR-717 (+)-JQ-1- FGFR4-IN-5 NH-CH2- MLT-231 POMHEX JAK2-IN-7 CPL304110 CD73-IN-4 Empty e aldehyde COOH

(E)-2- (Z)-2- CK2 inhibitor b Empty T0070907 NVP-TAE 226 Decenoic acid Decenoic acid Avasimibe Pyroxamide M4205 AZD5305 2 JMJD7-IN-1 Empty

Necrostatin- Talabostat c Empty SJ6986 UNC5293 34 Crenolanib Galunisertib SD-208 YM-201636 PF-9363 BOC-D-FMK (mesylate) Empty

A-674563 d Empty I-BET151 Ralimetinib Taladegib Apitolisib Silvestrol MK-5108 AMG 900 A-674563 (hydrochlorid TAME Empty dimesylate aglycone e)

Desmethyl Empty TAME Erlotinib Desmethyl Thiazovivin NVP-BHG712 NVP-BHG712 CCT128930 A66 CHIR-124 Degrasyn Empty e hydrochloride (hydrochlorid Erlotinib isomer

BS-181 Tubastatin A PIK-75 f Empty (hydrochlorid Droxinostat ABT-751 (Hydrochlorid Tubastatin A Dacomitinib (hydrochlorid GANT 58 Ki16425 SGI-1776 Empty e) e) e)

MK-8033 g Empty KN-62 Vinpocetine PYR-41 PYZD-4409 Mps1-IN-1 MK-8033 (hydrochlorid SR-3677 M8891 SAR439859 Empty e)

CP-547632 Regorafenib 5-ALA benzyl h Empty Myristyl CKI-7 (free (hydrochlorid LY2874455 VHL Ligand 8 JK184 CCR7 Ligand (Hydrochlorid BAY-474 ester Empty nicotinate base) e) 1 e) (hydrochlorid

Plate layout: CS-L025-26

1 2 3 4 5 6 7 8 9 10 11 12

Lenalidomide a Empty Infigratinib BAY-985 6RK73 MS1943 XL888 SJF620 Tesevatinib -OH JNK-IN-8 Pracinostat Empty

CX-5461 b Empty CX-5461 dihydrochlorid Bardoxolone ASP3026 Sapanisertib AZD4547 BGT226 Imisopasem ZM 336372 PF-8380 Empty e methyl (maleate) manganese

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

MLS0005444 Aminohexylge (Rac)- c Empty 60 HBC514 WF-47-JS03 RET-IN-3 VII-31 ldanamycin MS117 Indoximod NVS-PI3-4 SIRT-IN-3 Empty

Dorsomorphin d Empty Capmatinib Gossypol AICAR (dihydrochlori Dorsomorphin Zebularine Tenovin-1 RITA Deguelin MEISi-2 Empty (phosphate) de)

Allitinib Ionomycin AZD3839 e Empty Roxadustat tosylate Tubacin KU-0060648 Nanatinostat ICCB280 (calcium) (free base) AMG 511 NHWD-870 Empty

LDN-192960 653-47 PHA-767491 GSK- f Empty TAK-733 BAY 11-7082 IMT1 CID 2011756 (hydrochlorid PF-5274857 (hydrochlorid (hydrochlorid LY-364947 3/CDK5/CDK Empty e) e) e) 2-IN-1

g Empty ALK-IN-1 5-Ph-IAA UZH1 UZH1a KW-2478 Debio 0932 GSK126 EN4 Indophagolin USP7-IN-8 Empty

USP7/USP47 h Empty MD-222 AZ506 Mito-LND STM2457 inhibitor RMC-0331 WM-3835 GNF-5837 AC710 ML281 Empty

Plate layout: CS-L025-27

1 2 3 4 5 6 7 8 9 10 11 12

Mitoxantrone a Empty VT107 NY2267 GSK343 J14 Mubritinib Mitoxantrone (dihydrochlori Epothilone A PIK-293 M344 Empty de)

GSK- b Empty Lumiracoxib Dot1L-IN-4 U-104 TG 100713 CB-103 3484862 ONC206 Sirtinol Aloperine Piceatannol Empty

AV-153 (free DB04760 c Empty (-)-Cedrene Nocodazole SB-505124 base) Fimepinostat PAC-1 NL-1 MMP-9-IN-1 OXFBD04 analog 1 Empty

(R)-Verapamil (S)-Verapamil d Empty AG-1478 YO-01027 CH6953755 CAY10505 AS-604850 NBDHEX AS-252424 (hydrochlorid (hydrochlorid Abarelix Empty e) e) (Acetate)

ATN-161 ADH-1 Amsacrine e Empty (trifluoroaceta AZD-2461 BPR1J-097 Gemcitabine (1S,2S)- (trifluoroaceta Tretazicar Amsacrine Wnt pathway (hydrochlorid Empty te salt) Hydrochloride (elaidate) Bortezomib te) activator 1 e)

Banoxantrone Belotecan f Empty β-Lapachone AVN-944 AZM475271 (dihydrochlori Batabulin Batabulin Batimastat (hydrochlorid SR-318 hnRNPK-IN-1 Empty de) (sodium) e)

Betamethaso DB1976 g Empty TD52 Betamethaso ne Brivudine Macropa-NH2 (dihydrochlori Budesonide (Rac)-JBJ-04- Mobocertinib Mobocertinib Empty ne dipropionate diester de) 125-02 (succinate)

MSC2360844 SIRT7 h Empty Carbendazim Necroptosis- MSC2360844 (hemifumarat BAY 2416964 AHR CM10 Carmustine CG347B inhibitor Empty IN-1 e) antagonist 2 97491

Plate layout: CS-L025-28

1 2 3 4 5 6 7 8 9 10 11 12

PDK4-IN-1 a Empty CK2/ERK8- Piclidenoson 3,4-Dehydro Chlorambucil Chrysophanol CDDO-3P-Im (hydrochlorid Cisatracurium BO-264 Valecobulin Empty IN-1 Cilostazol e) (besylate)

Valecobulin Cytarabine b Empty DCLK1-IN-1 (hydrochlorid Cladribine Crolibulin Cyproterone Cytarabine iFSP1 (hydrochlorid Dacinostat IM156 Empty e) acetate e)

Tubulin Efaproxiral c Empty inhibitor 6 H3B-120 Dutasteride VH032-OH TNO155 RBN-2397 SNDX-5613 Efaproxiral SRX3207 (sodium) Empty

Epirubicin Estramustine d Empty Resveratrol OT-82 PF-06952229 (hydrochlorid BSJ-03-204 BSJ-04-132 AZD-9833 DCC-3014 (phosphate ATR inhibitor Empty analog 1 e) sodium) 2

NHS-PEG1- e Empty Etalocib Etoposide Etoposide SS-PEG1- Exatecan Dxd Exemestane SETD2-IN-1 Ezatiostat TLK117 Empty phosphate NHS (mesylate) (TFA)

Melanin f Empty Finasteride BRD9500 Fulvestrant MI-3454 ARRY-382 CID44216842 GDC-0152 AZA1 probe-1 RG108 Empty

β-catenin-IN- Encequidar Pentagamavu g Empty JCN037 BC-DXI-843 MYLS22 ASP4132 2 (mesylate) HMN-176 non-1 Incyclinide Empty

(-)- h Empty FEN1-IN-3 FEN1-IN-4 Indibulin Indisulam CIL62 RA-9 Epigallocatec SR18662 RET V804M- LQZ-7I Empty hin Gallate IN-1

Plate layout: CS-L025-29

1 2 3 4 5 6 7 8 9 10 11 12

Z-Ala-Ala- a Empty Stafia-1 WYC-210 TBAP-001 GSK778 ERK-IN-3 DGY-06-116 Lansoprazole Asn-AMC BCL6-IN-4 SC-43 Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

6- b Empty Levoleucovori Lomeguatrib BrBzGCp2 Lomustine LW6 LY2334737 Goserelin Maytansine Megestrol Mercaptopuri Empty n (Calcium) (acetate) acetate ne

6- PJ34 c Empty BCL6-IN-5 Mercaptopuri BDTX-189 Mesna Meisoindigo Mifepristone Miltefosine PQ401 (hydrochlorid PJ34 Empty ne hydrate e)

d Empty Go 6983 AZ12672857 Mitotane MSA-2 NEO2734 Methionine MSX-122 OP-5244 RBN012759 Nelarabine Empty

Nimustine e Empty Nilutamide (hydrochlorid SN-38 CAY10471 IMT1B IACS-13909 FB23 Oleandrin Phenoxodiol HPPH Empty e) (Racemate)

Pirarubicin Phosphorami Quinacrine Raloxifene f Empty 1,4-DPCA (Hydrochlorid Pixantrone de mustard (Hydrochlorid PX-12 (dihydrochlori R1530 TAS-119 (hydrochlorid Empty ethyl ester e) (dimaleate) (cyclohexana e) de) e)

Sardomozide KB-0742 g Empty Resiquimod Rubitecan Senaparib Venadaparib Vodobatinib AG-636 ARN-21934 dihydrochlorid RBPJ (dihydrochlori Empty e Inhibitor-1 de)

Tacrolimus h Empty Silibinin KRAS Ebselen XST-14 MKI-1 (R)- (monohydrate Tamoxifen CC-90010 Tamoxifen Empty inhibitor-9 Sulforaphane ) (Citrate)

Plate layout: CS-L025-30

1 2 3 4 5 6 7 8 9 10 11 12

TAS-103 Topotecan a Empty (dihydrochlori WSF1-IN-1 Teniposide Tetrandrine 6- BMS-P5 (free Tirapazamine (Hydrochlorid Ursodiol Valrubicin Empty de) Thioguanine base) e)

Zoledronic Pemetrexed Empty Motolimod SBP-7455 XL019 acid Vinblastine (disodium Tenofovir BIBF0775 ZM 306416 DMU-212 Empty b (monohydrate (sulfate) hemipenta Disoproxil

Tazemetostat c Empty SC-514 Tazemetostat (hydrobromid PP1 CRBN PP2 XL388 UNC0646 UNC 0631 BMS-833923 Empty e) modulator-1

d Empty α-NETA PR-619 JKE-1674 NU6027 Stattic MK-8745 GSK2656157 SKI II C646 WEE1-IN-3 Empty

PD-1/PD-L1- e Empty DTHIB MR837 CDK7-IN-3 BPTU YUM70 PLX647 IN 7 BX517 NF-κB-IN-1 AKR1C3-IN-4 Empty

2'-O-Me- 2'-OMe- 2'-OMe-A(Bz) DMT-dA(PAc) DMT-dG(dmf) DMT-dC(ac) 5-O-TBDMS- f Empty PAR-2-IN-1 K-975 C(Bz) G(ibu) Phosphorami Phosphorami Phosphorami Phosphorami N4-Benzoyl- 5'-O-TBDMS- Empty Phosphorami Phosphorami dite dite dite dite 2- Bz-dA

5'-O-DMT- 5'-O-DMT- 5'-O-DMT- 5'-O-DMT-3'- 5'-O-DMT-2'- g Empty 5'-O-TBDMS- 5'-O-TBDMS- 5'-O-TBDMS- N4-Bz-5-Me- N4-Ac-2'-F- N4-Bz-2'-F- 5'-O-DMT-rU 5'-O-DMT-Bz- O-TBDMS- O-TBDMS- Empty dT dG dA dC dC dC rC Ac-rC Ac-rC

AST5902 NCGC003784 Ro 31-8220 Bisindolylmal h Empty AI-10-47 LOX-IN-3 (trimesylate) AG-270 PF-4989216 ARV-110 P 22077 30 (mesylate) eimide I Empty

Plate layout: CS-L025-31

1 2 3 4 5 6 7 8 9 10 11 12

FTO-IN-1 Tyrphostin a Empty XL092 XL177A AES-350 (TFA) AG1296 XY028-140 WHI-P154 PD168393 CNX-2006 Taselisib Empty

Hydroxyfasud Empty GANT 61 BSJ-4-116 Flumatinib Flumatinib SU0268 TCS 359 RGFP966 Hydroxyfasud il IWP-2 Empty b (mesylate) il (hydrochlorid

PND-1186 c Empty NS-398 MAT2A Roniciclib UMB298 NiCur NSC348884 PND-1186 (hydrochlorid Napabucasin BMS-986242 Empty inhibitor 3 e)

1-Naphthyl Empty PD0166285 GW0742 SCR130 Miquelianin CL4H6 1-Naphthyl PP1 1-NM-PP1 CNX-774 NVP 231 Empty d PP1 (hydrochlorid

Angiotensin II e Empty BML-277 Angiotensin II human SRPIN340 JIB-04 Pioglitazone MS436 GSK1324726 GLPG0634 SGI-1027 Empty human (acetate) A analog

Mutant IDH1 Mutant EGFR NVP- f Empty ZCL278 JW 55 inhibitor DDR1-IN-1 UNC0642 JSH-23 IDO-IN-7 inhibitor TNKS656 CCG-1423 Empty

Rimonabant Fmoc-L- g Empty Mps1-IN-2 (Hydrochlorid Asn(beta-D- GSK-3β WSB1 Zileuton MK-886 Bexarotene Raf inhibitor 1 VX-11e Empty e) GlcNAc(Ac)3) inhibitor 3 Degrader 1

Amiodarone Siramesine Fadrozole h Empty Macitentan (hydrochlorid (hydrochlorid (hydrochlorid Fadrozole Letrozole Bicalutamide Febuxostat Anastrozole Trilostane Empty e) e) e)

Plate layout: CS-L025-32

1 2 3 4 5 6 7 8 9 10 11 12

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Elagolix a Empty Cimetidine PD153035 EBE-A22 sodium CB30865 PF-3845 LP-261 Emodin TBB Indomethacin Empty

Indomethacin b Empty (sodium Celecoxib ERK5-IN-1 SR1078 4E1RCat ICG-001 Pyridone 6 MP7 XMD8-92 Plinabulin Empty hydrate)

Fatostatin c Empty Fatostatin (hydrobromid TPh A Onalespib UPF 1069 AF-353 YK-4-279 Aminopterin Methotrexate Methotrexate Empty e) (disodium)

d Empty Pelitrexol Sertindole Amisulpride E7820 PF-03814735 Palomid 529 Irosustat Chrysin Tectochrysin Empty

Pioglitazone e Empty Diethylstilbest Rosiglitazone (hydrochlorid Tramiprosate Clioquinol [6]-Gingerol Shogaol Paradol Empty rol (maleate) e)

Necrostatin 2 f Empty Zingerone Necrostatin 2 Necrostatin 2 (S (-)-DHMEQ Dexamethaso Dexamethaso Retinoic acid Tamibarotene Aspirin Empty (racemate) enantiomer) ne ne acetate

CCT241533 g Empty Sulfasalazine Thalidomide Dabrafenib Dabrafenib Fluvastatin CP-724714 Refametinib AZ3146 Reversine (hydrochlorid Empty (Mesylate) (sodium) e)

Resminostat NVP-BSK805 Anamorelin h Empty (hydrochlorid RO4987655 Rabusertib (dihydrochlori VE-821 Anamorelin (hydrochlorid Rolapitant Salirasib Bentamapimo Empty e) de) e) d

Plate layout: CS-L025-33

1 2 3 4 5 6 7 8 9 10 11 12

Inolitazone Givinostat a Empty Monepantel Levomefolic (R)-Elagolix (dihydrochlori Palifosfamide Tasisulam Tosedostat Adarotene Karenitecin (hydrochlorid Empty acid de) e

Homoharringt Cevipabulin b Empty Litronesib Verubulin Bardoxolone Lificiguat Prinaberel Succinobucol Elacytarabine onine Cevipabulin fumarate Empty

R1487 BAY 61-3606 c Empty Dalcetrapib Ulipristal NSC 66811 (E)-Akt (Hydrochlorid GSK2334470 (dihydrochlori StemRegenin AST 487 ATH686 Empty inhibitor-IV e) de) 1

5- d Empty AUZ 454 Sildenafil Sildenafil Aminosalicylic Naproxen Naproxen ELN-441958 NU1025 INO-1001 DNQX Empty (citrate) Acid (sodium)

Purmorphami Sinomenine 9-cis-Retinoic e Empty MKT-077 Myricetin Apoptozole MK-0429 ne Sinomenine hydrochloride acid Lonafarnib Staurosporine Empty

Doxorubicin SBE13 TAK-960 f Empty (hydrochlorid Trichostatin A XAV-939 Bemcentinib NG 52 MLN0905 (Hydrochlorid Cyclapolin 9 TAK-960 (dihydrochlori Empty e) e) de)

Icotinib Glyoxalase I Pyridostatin g Empty Ro3280 Monomethyl (Hydrochlorid Icotinib Zotiraciclib Glyoxalase I inhibitor (free Dactolisib (hydrochlorid PF-04691502 Empty auristatin E e) inhibitor base) (Tosylate) e)

Buparlisib Collagen Ipatasertib h Empty (Hydrochlorid proline Nirogacestat Ipatasertib (dihydrochlori Filanesib (R)-Filanesib NVP-HSP990 Sabutoclax GSK 650394 Empty e) hydroxylase de)

Plate layout: CS-L025-34

1 2 3 4 5 6 7 8 9 10 11 12

Dimethylcurc Menin-MLL a Empty EMD638683 umin TAK-285 Agerafenib Binimetinib Ganetespib CHR-6494 inhibitor MI-2 MI-3 PCI-34051 Empty

AZ505 EPZ004777 b Empty AZ505 (ditrifluoroace EPZ004777 (hydrochlorid RX-3117 Geldanamyci SL 0101-1 c-Kit-IN-1 NVP-LCQ195 Alpelisib Empty tate) e) n

XL413 c Empty GSK2636771 TAK-580 Vistusertib GDC-0349 Reparixin Reparixin (L- Tiplaxtinin (hydrochlorid SRT 2104 BMS-911543 Empty lysine salt) e)

Nelfinavir d Empty WYE-687 WAY-600 UNC0638 L-798106 BMS-265246 Epothilone D E-64 Nelfinavir (Mesylate) AIM-100 Empty

CBB1007 PRT062607 e Empty CZC24832 Eltrombopag Eltrombopag Ivermectin WP1066 (trihydrochlori RI-1 AMG 487 Etoricoxib (Hydrochlorid Empty (Olamine) de) e)

Copanlisib f Empty Nutlin-3b AG 555 Hesperidin TG003 CVT-313 BAM7 CEP-33779 (dihydrochlori ALK inhibitor ALK inhibitor Empty de) 1 2

Atrasentan ML-7 g Empty Forskolin GW6471 Fenretinide Tazarotene Lucitanib (hydrochlorid HhAntag KB-R7943 (hydrochlorid BML-190 Empty e) (mesylate) e)

5- PF-543 Selisistat S- h Empty Iodotubercidin (Citrate) Capivasertib Quisinostat NG25 SL327 Tezacaftor Kaempferide Selisistat enantiomer Empty

Plate layout: CS-L025-35 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

1 2 3 4 5 6 7 8 9 10 11 12

(R)-(-)- a Empty Selisistat R- Devimistat Xevinapant NVP-BVU972 Triciribine SAR131675 Cabazitaxel Imatinib Gossypol (S)-Gossypol Empty enantiomer acetic acid (acetic acid)

KN-93 ZM323881 b Empty KN-93 (hydrochlorid KN-93 CH5132799 (hydrochlorid IOX2 MLN120B UK-5099 WZ811 TTP 22 Empty e) (phosphate) e)

Pifithrin-α c Empty NSC 42834 D-64131 DY131 (hydrobromid Salubrinal Scriptaid PF-670462 Picropodophy RGB-286638 RGB-286638 Empty e) llin (free base)

Tenovin-6 OTSSP167 Merestinib d Empty RWJ-67657 TAK-593 JANEX-1 Tenovin-6 (Hydrochlorid Tyrphostin A9 (hydrochlorid TC-DAPK 6 Merestinib dihydrochlorid Empty e) e) e

KN-92 Braco-19 e Empty KN-92 (hydrochlorid LCL161 CGK733 ETP-46464 (trihydrochlori kb NB 142-70 CID-2858522 Venetoclax SCH900776 Empty (phosphate) e) de)

Hoechst Empty SCH900776 DMAT FRAX597 FRAX486 Podofilox EPZ005687 AZ20 33258 NU6102 EI1 Empty f (S-isomer) (trihydrochlori

Taltobulin Taltobulin g Empty GSK3787 Taltobulin (trifluoroaceta (hydrochlorid L67 L189 AZ-23 Pinometostat 360A (iodide) Salinomycin Empty te) e)

MPTP SC144 h Empty SSR128129E AZD1208 Encorafenib WEHI-539 (hydrochlorid AZD-3463 GDC-0623 Maritoclax SC144 (hydrochlorid Empty hydrochloride e) e)

Plate layout: CS-L025-36

1 2 3 4 5 6 7 8 9 10 11 12

DMA meta- LY 303511 a Empty TIC10 JNK-IN-7 Methylproami DMA (trihydrochlori iodoHoechst Capsazepine (hydrochlorid Tyrphostin 23 UNC1999 Empty ne de) 33258 e)

GSK-J4 Ceritinib b Empty BRD9539 GSK-J1 GSK-J2 GSK-J4 (hydrochlorid UNC1215 SGC0946 Ceritinib dihydrochlorid GSK2801 Empty e) e

GZD824 PI4KIII beta c Empty Wnt-C59 IPA-3 XMD17-109 GZD824 (dimesylate) P005091 KP372-1 Idasanutlin inhibitor 3 Senexin A Empty

Puromycin CRT0066101 (Z)- d Empty TTNPB IDO5L Epacadostat SMIP004 aminonucleos dihydrochlorid PluriSIn 1 Leukadherin- ADH-503 HJC0350 Empty ide e 1

NSC 23766 e Empty LH846 NMS-873 NMS-859 Kobe0065 Kobe2602 NU 7026 FH535 (trihydrochlori CDDO-Im Afuresertib Empty de)

Afuresertib f Empty (hydrochlorid Rociletinib Rociletinib Poziotinib Lucidin AGI-6780 c-Met inhibitor DB07268 GNF-5 Ansamitocin Empty e) hydrobromide 1 P-3

Ellipticine 3,3'- g Empty Birabresib LY255283 Deltarasin XL228 (hydrochlorid CGP37157 RKI-1447 SJB2-043 Diindolylmeth Necrostatin-1 Empty e) ane

A 419259 GNE-617 Tirabrutinib h Empty (trihydrochlori GNE-617 (hydrochlorid TAK-632 Ilomastat WHI-P180 Tirabrutinib (hydrochlorid Osimertinib Osimertinib Empty de) e) e) mesylate

Plate layout: CS-L025-37

1 2 3 4 5 6 7 8 9 10 11 12

Ribociclib K145 a Empty PF-4708671 Arginase Ribociclib Ribociclib Ribociclib succinate (hydrochlorid TAS-116 UNC2250 HG-14-10-04 Empty inhibitor 1 hydrochloride succinate hydrate e)

Ulixertinib b Empty WZ4003 XMD8-87 Bromosporine Ulixertinib (hydrochlorid CAY10566 IWP L6 SGC-CBP30 NSC 405020 NMS- Empty e) 1286937

c Empty GSK 2830371 CUDC-427 BAY 87-2243 SAR-260301 ID-8 UNC 669 YLF-466D CEP-37440 SF1670 AG-825 Empty

AP-III-a4 GGTI298 FTI-277 d Empty STF-083010 CPI-203 CW-069 (hydrochlorid FLI-06 Targapremir- HS-173 Inauhzin (Trifluoroacet (hydrochlorid Empty e) 210 ate) e)

e Empty FTI 276 (TFA) BTB06584 LDC000067 CCT007093 TCS JNK 5a Mdivi-1 MG 149 PTC-209 C-7280948 CK-636 Empty

5(6)- f Empty DMOG LDN-212854 Voxtalisib 5-BrdU Carboxyfluore DBeQ Ravoxertinib Ravoxertinib Kif15-IN-1 Kif15-IN-2 Empty scein hydrochloride

NVP- g Empty ML167 NVP- CGM097 CPI-360 CPI-169 CPI-169 VBY-825 Savolitinib Antitumor Uprosertib Empty CGM097 (sulfate) (racemate) agent-3

GSK2110183 Seviteronel h Empty analog 1 Entospletinib Sal003 VER-50589 VER-49009 SM-164 SM-164 Citarinostat Seviteronel (R Empty (hydrochlorid Hydrochloride enantiomer)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Plate layout: CS-L025-38

1 2 3 4 5 6 7 8 9 10 11 12

Cerdulatinib Ilorasertib Acolbifene a Empty Cerdulatinib (hydrochlorid Domatinostat A-385358 (hydrochlorid (hydrochlorid Acolbifene (Rac)- EOC317 Ricolinostat Empty e) e) e) Acolbifene

Hexaminolev Tucatinib b Empty ulinate Arglabin Apalutamide Tucatinib (hemiethanol AT13148 AZD3514 BI 99179 Talazoparib BMS-214662 Empty (hydrochlorid ate)

CAL-130 Carboxyamid D-3263 c Empty BNC105 (Hydrochlorid otriazole Carboxyamid Cilengitide Cilengitide (hydrochlorid Degarelix DMAPT EL-102 Empty e) (Orotate) otriazole (TFA) e)

Forodesine Kevetrin L-778123 d Empty ELR510444 Ethynylcytidin (hydrochlorid FX-11 Gadoxetate Genz-644282 GGTI-2418 JI-101 (hydrochlorid (hydrochlorid Empty e e) (Disodium) e) e)

Abemaciclib e Empty Osilodrostat APTO-253 LY2090314 (methanesulf Abemaciclib Minodronic N3PT Nimorazole NKP-1339 NVP-QAV- Empty onate) acid 572

Phenformin f Empty Briciclib CP-609754 Pacritinib Pasireotide PCI-27483 Glasdegib (hydrochlorid Pipobroman RG2833 RRx-001 Empty (acetate) e)

CNDAC Trifluridine/tipi g Empty Sapacitabine (hydrochlorid SAR125844 CDK9-IN-2 Relugolix racil Temoporfin Tolrestat Transcrocetin Treosulfan Empty e) hydrochloride ate disodium

Ulipristal Riviciclib h Empty acetate UNBS5162 UNC926 Upamostat VAL-083 Vitamin CK3 Pilaralisib YF-2 Butein hydrochloride Empty

Plate layout: CS-L025-39

1 2 3 4 5 6 7 8 9 10 11 12

Irinotecan 10- Irinotecan a Empty Camptothecin Resveratrol Irinotecan (hydrochlorid Narciclasine Deacetylbacc (hydrochlorid Colchicine TCS-PIM-1- GW9662 Empty e) atin III e trihydrate) 4a

Sonidegib b Empty (diphosphate) Sonidegib VS-5584 PFI-1 Oligomycin A X-376 Birinapant Brefeldin A CNX-1351 SIRT-IN-2 Empty

Z-VAD(OMe)- Skp2 Inhibitor c Empty Folic acid Apabetalone FMK Z-VAD-FMK EHT 1864 INH1 C1 Oncrasin-1 SJ-172550 iCRT 14 Empty

CID d Empty 3CAI HLM006474 Mcl1-IN-1 AGN 195183 BAMB-4 MIM1 16020046 kb-NB77-78 Nexturastat A PNU-159682 Empty

Pifithrin-β Remodelin Amiselimod e Empty BV6 (hydrobromid ESI-09 BRD4770 (hydrobromid USP7-IN-1 SB225002 LDN-214117 Indoximod (hydrochlorid Empty e) e) e)

Pexidartinib f Empty Pexidartinib (hydrochlorid Fevipiprant Entasobulin Pexmetinib Veledimex AI-10-49 Rolipram RI-2 WIKI4 Empty e)

Heptamidine 4- (E/Z)-4- g Empty MC1568 (dimethanesul MI-503 CK-666 CK-869 Cytochalasin ISA-2011B Hydroxytamo Hydroxytamo ARV-825 Empty fonate) B xifen xifen

CC-115 h Empty CC-223 Sitravatinib CC-115 (hydrochlorid GW627368 TH287 SBI-0206965 SR9243 SH-4-54 GDC-0339 Empty e)

Plate layout: CS-L025-40

1 2 3 4 5 6 7 8 9 10 11 12

EPZ011989 SR9011 a Empty Darolutamide EPZ011989 (trifluoroaceta IDO-IN-3 SR9011 (hydrochlorid SR9009 OICR-9429 OICR-0547 Itacitinib Empty te) e)

Dexmedetomi Empty Itacitinib RO8994 Tolvaptan Saquinavir Saquinavir Dofequidar Cyclopamine Gemcitabine Epothilone B dine Empty b adipate (Mesylate) (fumarate) (hydrochlorid

Vancomycin c Empty Duvelisib Duvelisib (R BIBR 1532 Fenofibrate Deferasirox (hydrochlorid Dimethyl Temozolomid Octreotide Atazanavir Empty enantiomer) e) fumarate e (acetate) (sulfate)

Idarubicin Ranolazine d Empty Oxaliplatin Rofecoxib Ezetimibe (hydrochlorid Levomefolate Rosiglitazone Genipin Tegafur (dihydrochlori Mevastatin Empty e) (calcium) de)

4'- Mefloquine Salinomycin Sivelestat Sivelestat e Empty Limonin Acyclovir Amprenavir Demethylepip (hydrochlorid Cidofovir Sivelestat (sodium Empty odophyllotoxi e) (sodium salt) (sodium) tetrahydrate)

Fosbretabulin Parecoxib f Empty (disodium) Cilostazol Gimeracil Embelin Parecoxib (Sodium) Zafirlukast MI-773 EGFR-IN-12 Azithromycin Empty

Pantoprazole g Empty Pantoprazole (sodium Clarithromyci Gossypol Losartan Itraconazole APY29 HBX 19818 ML-323 LGK974 Empty (sodium) hydrate) n (acetic acid)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

2'- Bleomycin Berberine h Empty Folinic acid Deoxyguanos Bleomycin (hydrochlorid Atosiban Thio-TEPA (chloride Griseofulvin Chloroquine Chloroquine Empty ine (sulfate) e) (acetate) hydrate) (phosphate)

Plate layout: CS-L025-41

1 2 3 4 5 6 7 8 9 10 11 12

Bithionol Nastorazepid Tarloxotinib a Empty Bithionol (sulfoxide) Mebendazole Acalabrutinib Alofanib Amcasertib Belizatinib e (bromide) Tenalisib Empty

CEP-28122 b Empty ALW-II-41-27 PS-1145 LFM-A13 Spebrutinib (mesylate Ochromycino GSK2606414 LPA2 AGI-5198 Quercetin Empty salt) ne antagonist 1

CX-6258 CX-6258 Prexasertib c Empty TCS PIM-1 1 CX-6258 (hydrochlorid (hydrochlorid CCT241736 Prexasertib (dihydrochlori Prexasertib AZD2932 B-Raf IN 1 Empty e hydrate) e) de) (dimesylate)

Ombrabulin d Empty (hydrochlorid Berberine AZ876 Longdaysin AKT-IN-1 Purvalanol B Purvalanol A Filgotinib BMS-3 BMS-5 Empty e) (chloride)

(R)-CR8 CP-31398 e Empty SB 242235 SYN1143 GW 441756 (trihydrochlori Diflunisal (dihydrochlori Mozavaptan Indotecan mTOR TMP269 Empty de) de) inhibitor-3

RU-SKI 43 f Empty TMP195 (hydrochlorid HIF-2α-IN-3 UNC1079 Bioymifi FIIN-2 FIIN-3 PD158780 CAY10603 YL-109 Empty e)

VEGFR-2-IN- PFI-2 GSK2879552 g Empty OTS514 VI 16832 5 (hydrochlorid UMI-77 SU9516 Ro 48-8071 GSK2879552 (dihydrochlori MDK83190 Empty (hydrochlorid e) (fumarate) de)

RQ- h Empty NSC319726 Ki16198 TZ9 CWHM-12 Ro 5126766 TEPP-46 Siremadlin 00203078 PFI-4 GSK-5959 Empty

Plate layout: CS-L025-42

1 2 3 4 5 6 7 8 9 10 11 12

Enasidenib a Empty ML346 SMER18 K-Ras-IN-1 OSU-T315 ILK-IN-2 PU-WS13 Centrinone Centrinone-B Enasidenib (mesylate) Empty

Endoxifen (Z- Endoxifen b Empty AMG-337 JD-5037 BRD73954 K-Ras(G12C) Erdafitinib SCR-1481B1 BG45 Mutant IDH1- isomer (hydrochlorid Empty inhibitor 12 IN-2 hydrochloride e)

L-NAME 1400W 6-Thio-2'- c Empty Endoxifen (E- STF-31 (hydrochlorid (Dihydrochlori Lipoic acid VR23 FLT3-IN-2 Zorifertinib IN-1130 Deoxyguanos Empty isomer) e) de) ine

Indirubin d Empty Ivosidenib (R,S)- NCT-501 IDO-IN-4 IDO-IN-6 Navoximod IDO-IN-8 KC7F2 RR6 Derivative Empty Ivosidenib E804

NSC305787 e Empty BBT594 NU6300 (hydrochlorid DEL-22379 CBL0137 Alda-1 WEHI-345 Selonsertib ONO-4059 NMS-P118 Empty e) hydrochloride (analog)

AMI-1 (free Lavendustin f Empty BI-847325 Lifirafenib CCT245737 CWP232228 CHZ868 PD 407824 AMI-1 acid) A MG-101 Empty

Phorbol g Empty PF-04418948 TG4-155 Dp44mT I-BRD9 UF010 Rottlerin Decursin Anisomycin 12,13- SAR405838 Empty dibutyrate

Zinc h Empty ETC-159 CCG215022 Adjudin PLX7904 LMK-235 TCV-309 phthalocyanin LLY-507 NU2058 ITE Empty (chloride) e

Plate layout: CS-L025-43

1 2 3 4 5 6 7 8 9 10 11 12

PIM-447 a Empty MI-136 (dihydrochlori Ceralasertib (S)- SU1498 ACY-738 HA130 DASA-58 WZB117 L755507 Empty de) Ceralasertib

Pimelic b Empty BAZ2-ICR Tenovin-3 TMS Compound WDR5-0103 Diphenylamid BML-210 MN-64 T56-LIMKi Rocagloic Empty 401 e 106 acid

AEOL-10150 Pimelic c Empty Didesmethylr E3330 L-685458 Didox (pentachlorid Diphenylamid Topilutamide Maytansinol Ladarixin PF-2771 Empty ocaglamide e) e 106

d Empty ZM241385 SCH 58261 Nemiralisib NI-57 FRAX1036 GSK864 I-CBP112 Brusatol JAK3-IN-1 BAY-598 Empty

DDP-38003 MS023 e Empty SBI-0640756 JX06 NQDI-1 Peficitinib (trihydrochlori MS023 (dihydrochlori EGFR-IN-1 m-3M3FBS Branaplam Empty de) de) (TFA)

G-5555 Glesatinib f Empty NVP-ACC789 MCB-613 NSC23925 Ilginatinib Ilginatinib Ilginatinib G-5555 (hydrochlorid SW044248 (hydrochlorid Empty (maleate) hydrochloride e) e)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

(-)-p- Tauroursodeo Tauroursodeo g Empty Cariporide Bromotetrami Tauroursodeo xycholate xycholate PKR-IN-2 KIRA6 MKC3946 LJH685 LJI308 Empty sole (oxalate) xycholate (sodium) (dihydrate)

DG172 h Empty XY1 SGC707 Miransertib A-1155463 NSC59984 Olmutinib SID 3712249 NK-252 KJ Pyr 9 (dihydrochlori Empty de)

Plate layout: CS-L025-44

1 2 3 4 5 6 7 8 9 10 11 12

N- a Empty JW74 A-1331852 BMS-202 deacetylated HPOB KS176 OTX008 Sirtuin SRT 2183 RIP2 kinase Empty BMS-202 modulator 1 inhibitor 2

GSK2983559 3α- ML241 b Empty GSK1940029 BEBT-908 active amyloid P-IN- HDAC-IN-3 Aminocholest RS-1 MP-A08 ML240 (hydrochlorid Empty metabolite 1 ane e)

PI4KIIIbeta- Naquotinib Indirubin-3'- Avitinib c Empty IN-9 ML-098 (mesylate) monoxime C-DIM12 MI-463 MI-538 Olafertinib (maleate) PRT4165 Empty

d Empty 3PO 4EGI-1 (Z)-4EGI-1 SC66 Fenebrutinib AZD-5069 LTX-315 COTI-2 ASP-9521 Fruquintinib Empty

Vactosertib TAS-117 e Empty MK-1064 Vactosertib (Hydrochlorid COH29 (hydrochlorid Dimethylenas GI254023X CH5183284 (Z)-Mirin BCTC Empty e) e) tron

K858 f Empty (Racemic) ML239 YU238259 RCM-1 Eprenetapopt PRIMA-1 Derazantinib ASP5878 CCT-251921 PF-06459988 Empty

3- Pictilisib g Empty (3S,4S)-PF- BML-284 BMS-1 Bromopyruvic ML264 (dimethanesul Tyrphostin SU5205 SU5214 BCI-121 Empty 06459988 acid fonate) AG 879

5- Clemizole 3- h Empty Hydroxyflavo (±)- Thalidomide- Cycloleucine Methoxsalen (hydrochlorid Seliciclib Cot inhibitor-2 arylisoquinoli Pelitinib Empty ne Darifenacin 5-OH e) namine

Plate layout: CS-L025-45

1 2 3 4 5 6 7 8 9 10 11 12

cis-4- (S,R,S)- a Empty Neratinib Triptolide Triptonide Clofilium GSK-4716 N-Nitroso-N- Hydroxy-L- Tofacitinib Tofacitinib AHPC-Me Empty tosylate methylurea proline (citrate) (dihydrochlori

Transcrocetin PROTAC SMARCA-BD Mardepodect b Empty meglumine Ibrutinib- Tarlox-TKI Lenalidomide BET-binding ligand 1 for Navitoclax- Pictilisib (hydrochlorid GW 4064 Empty salt MPEA -Br moiety 2 Protac piperazine e)

Etomoxir JNJ- c Empty Etomoxir (sodium salt) CI-1040 AT9283 A-769662 38877605 Tivantinib Nutlin-3 BI 2536 MK-2461 Empty

Palbociclib d Empty Selumetinib Selumetinib A939572 KU-0063794 DUB-IN-1 DUB-IN-3 DUB-IN-2 Linifanib Ispinesib (monohydroc Empty (sulfate) hloride)

Silmitasertib Ruxolitinib (S Ruxolitinib Akt1 and e Empty Avagacestat SCH772984 ZSTK474 Silmitasertib (sodium salt) Ruxolitinib enantiomer) (phosphate) Akt2-IN-1 GDC-0879 Empty

Crizotinib Elacridar Gefitinib f Empty NVP- Bafetinib (E)-Daporinad GSK461364 Crizotinib (hydrochlorid Elacridar (hydrochlorid Gefitinib (hydrochlorid Empty AEW541 e) e) e)

Lapatinib ONO-AE3- Turofexorate g Empty Erlotinib Lapatinib (ditosylate) 208 Nintedanib Dovitinib ABT-737 Perifosine Temsirolimus isopropyl Empty

Plerixafor AT7519 h Empty (octahydrochl Tacedinaline Troglitazone AT7519 (Hydrochlorid Imatinib PLX-4720 CMK FMK SC-560 Empty oride) e) (Mesylate)

Plate layout: CS-L025-46

1 2 3 4 5 6 7 8 9 10 11 12

2-O- Enzalutamide Carboxypepti p53 and a Empty Maleic 6-FITC Methylcytosin Enzalutamide N-desmethyl carboxylic dase G2 Galeterone Abiraterone MDM2 Empty e Enzalutamide acid (CPG2) proteins-

p53 and Empty MDM2 GSK- TCS7010 Pevonedistat Buparlisib D609 CCG-63802 CCG-63808 Abiraterone (-)-Menthol Empty b proteins- 1070916 acetate

Azetidine-2- Methyl Cyclo(Ala- Chenodeoxyc TAK1/MAP4K (E)-[6]- 9-Dihydro-13- c Empty carboxylic Etodolac Bergaptol Poloxime Dehydropara acetylbaccati Empty acid vanillate Gly) holic Acid 2 inhibitor 1 dol n III

Benzyl JQ-1 Ibrutinib d Empty Cephalomann Cysteamine isothiocyanat Ibuprofen (R)-(-)- MNS A 77-01 CDK-IN-6 (carboxylic deacryloylpip Empty ine hydrochloride e Ibuprofen acid) eridine

THZ1 e Empty Mutated Osimertinib IDO-IN-1 Glutaminase- BMX-IN-1 SJB3-019A THZ1 (Hydrochlorid 5-Fluorouracil ent-Tadalafil Empty EGFR-IN-1 (dimesylate) IN-3 e)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Darifenacin f Empty Lenalidomide Lenalidomide Decitabine Clofarabine Pentostatin (hydrobromid Ramelteon Bazedoxifene Bazedoxifene Malotilate Empty (hemihydrate) e) (acetate)

Tipiracil Procainamide Nitroprusside g Empty Trifluridine (hydrochlorid Palbociclib Aurothiogluco Liothyronine Liothyronine (hydrochlorid (hydrochlorid Tunicamycin (disodium Empty e) (isethionate) se (sodium) e) e) dihydrate)

Buclizine Gadopentetat Methyl Gemcitabine h Empty Plicamycin Alizapride (dihydrochlori e Regadenoson aminolevulina Bupranolol Pentagastrin (hydrochlorid Empty hydrochloride de) (phosphate) (dimeglumine te e)

Plate layout: CS-L025-47

1 2 3 4 5 6 7 8 9 10 11 12

Toremifene Docetaxel Pamidronic a Empty (citrate) Carvedilol Sulindac Docetaxel (Trihydrate) acid Paclitaxel Capecitabine Doxifluridine Flutamide Empty

Bendamustin Empty Fludarabine Gimatecan Fludarabine e Dacarbazine Leflunomide Dienogest Adapalene Artemisinin Empty b (phosphate) (hydrochlorid

Tigecycline c Empty Floxuridine Doxazosin Ketoconazole Levetiracetam Acitretin Omeprazole Omeprazole Oxcarbazepin Tigecycline (tetramesylat Empty (mesylate) (sodium) e e)

Bestatin d Empty Perindopril Bestatin (hydrochlorid Furosemide Furosemide Flucytosine Estradiol Pitavastatin Verteporfin Nicotinamide Empty (erbumine) e) (sodium) (Calcium)

L-Ascorbic Imiquimod e Empty Adenine Adenine Pravastatin acid (sodium Salicylic acid Sodium Olsalazine Imiquimod (hydrochlorid Altretamine Empty (hemisulfate) (sodium) salt) Salicylate (Disodium) e)

Lidocaine Prazosin Tizanidine f Empty Carmofur Ellagic acid Lidocaine (hydrochlorid Nafamostat (hydrochlorid (hydrochlorid Tranilast Mycophenolat Candesartan Empty e) (mesylate) e) e) e Mofetil

Ethynyl Meprednison g Empty Prednisone Estradiol Nitazoxanide Allopurinol Adenosine Estrone e Busulfan Empty

Carbamazepi Adefovir Methylprednis Enoxacin Acetylcholine h Empty ne Piroxicam dipivoxil Azathioprine olone Meloxicam Nimodipine (hydrate) Ranolazine (chloride) Empty

Plate layout: CS-L025-48

1 2 3 4 5 6 7 8 9 10 11 12

Amlodipine Amlodipine a Empty Nifedipine Flubendazole Idoxuridine Nizatidine Hydroxyurea Amlodipine (maleate) (besylate) Sulfisoxazole Empty

Argatroban Bupivacaine b Empty Triamcinolone Tolfenamic Pranoprofen Rebamipide (monohydrate Mestranol (S)-(+)- Tolbutamide (hydrochlorid Estriol Empty Acid ) Rolipram e)

Phenoxybenz Medroxyprog Paroxetine c Empty Mycophenolic Novobiocin amine Salbutamol Ciclopirox Ciclopirox Econazole esterone (hydrochlorid Empty acid (Sodium) (hydrochlorid (hemisulfate) (olamine) (nitrate) acetate e)

Ibandronate Anagrelide d Empty Niclosamide Bindarit 2-Thiouracil Moguisteine Methylthioura (Sodium Benztropine (hydrochlorid Betahistine Flumequine Empty cil Monohydrate) (mesylate) e)

(+)- e Empty Pentamidine Ouabain Nabumetone Spironolacton Sodium Deferiprone Cyclosporin A Dexrazoxane Tetrabenazin Iohexol Empty (isethionate) (Octahydrate) e nitroprusside e

S-Adenosyl- f Empty L-methionine Metformin Alendronic Triamcinolone Amifostine Isosorbide Rabeprazole Eicosapentae Tamsulosin Balsalazide Empty (tosylate) acid acetonide mononitrate (sodium) noic Acid

Eflornithine L-Eflornithine g Empty Estradiol Pirfenidone Carglumic Pentoxifylline Ingenol Ospemifene (hydrochlorid (monohydroc Ramatroban Hematoporph Empty valerianate Acid Mebutate e hydrate) hloride) yrin

LY2409881 h Empty Ibudilast Bicyclol Artemotil Teprenone Acetazolamid (trihydrochlori SU6656 Altiratinib AZ-5104 AZ7550 Empty e de) Mesylate

Plate layout: CS-L025-49

1 2 3 4 5 6 7 8 9 10 11 12 Sodium Empty MHY1485 Oxaprozin Theophylline Diuron Glyphosate Suramin Acetohexami Econazole Anethole copper Empty a (sodium salt) de chlorophyllin

Thioridazine Hexylresorcin Ascorbyl Selenomethio L- 8- b Empty Azaserine Danthron Cloxiquine (hydrochlorid SelenoMethio Hydroxyquino Quinestrol Empty e) ol palmitate nine nine line

Tilorone Tetrahydroxy c Empty Trapidil Dimesna Lanatoside C Lasalocid Lasalocid Penfluridol (dihydrochlori Estradiol Tetrahydroxy quinone Empty (sodium) de) (cypionate) quinone (monohydrate

Cefoxitin Estradiol d Empty (sodium) Triclosan L-Cycloserine Auranofin Nitroxoline Timonacic benzoate Terfenadine Histamine Urethane Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Chlormethine D-α- Citalopram Chloropyrami e Empty Anethole Metyrapone (hydrochlorid Desipramine Tocopherol (hydrobromid ne Apramycin Proglumide Perhexiline Empty trithione e) hydrochloride acetate e) hydrochloride (sulfate) maleate

Methylene Dehydroisoan Nortriptyline 9- f Empty blue Hydroxychlor D-Panthenol Dienestrol drosterone 3- (hydrochlorid Aminoacridin Benzthiazide Ethoxyquin Nifuroxazide Empty (trihydrate) oquine sulfate acetate e) e

Tolmetin 3'-Fluoro-3'- Alprenolol g Empty Licofelone 8-Azaguanine (sodium Acefylline Vitamin K4 deoxythymidi (hydrochlorid L-Canavanine Ethacrynic Methenamine Empty dihydrate) ne e) sulfate acid (hippurate)

Tetraethylam Methylprednis h Empty NSC 601980 NSC 601980 Perflubron Rotenone monium Tolmetin Forchlorfenur olone Dihydroisotan Deltamethrin Empty (analog) (chloride) on succinate shinone I

Plate layout: CS-L025-50

1 2 3 4 5 6 7 8 9 10 11 12

Buformin 2- a Empty Tiamulin (hydrochlorid Oxyphenisati Escin Tannic acid Ilaprazole Aminobenzen Menaquinone γ-Oryzanol Stearic acid Empty (fumarate) e) ne (sodium) esulfonamide -4

Malachite Tartaric acid b Empty Hinokitiol 7ACC1 green Quinizarin Fluorescein Gallein Rhodamine 7ACC2 5-IAF (disodium Empty (oxalate) 6G dihydrate)

Sodium NADPH β- c Empty orthovanadat PIPES Cy7 DiC18 Py-BODIPY- Hydrofurimazi (tetrasodium Nicotinamide Canagliflozin Regorafénib Uracil Empty e NHS ester ne salt) mononucleoti (hemihydrate) N-oxyde (M2)

(-)- d Empty (-)- Epicatechin Oridonin Curcumin Demethoxycu Bisdemethoxy Geniposidic Baohuoside I Glycitin Empty rcumin curcumin acid

e Empty Vitexin Icariin Astragalin Glycitein Bergenin Daidzein Verbascoside Arctiin Arctigenin Costunolide Empty

Ginsenoside Ginsenoside Ginsenoside Ginsenoside Ginsenoside Ginsenoside Sanguinarine f Empty Alantolactone Rb1 Rb3 Rc Rd Re Rg1 Polyphyllin I (chloride) Psoralen Empty

3,4- g Empty Osthole Chlorogenic Dicaffeoylquin Ferulic acid Ferulic acid (E)-Ferulic Punicalagin Macelignan Solasodine Solamargine Empty acid ic acid (sodium) acid

Sarsasapoge Ginkgolic Betulinaldehy Dimethylfraxe Gambogic h Empty Solasonine Crotonoside Brazilin nin Acid Betulin de tin Acid Apocynin Empty

Plate layout: CS-L025-51

1 2 3 4 5 6 7 8 9 10 11 12

Ancitabine (S)-10- Sophocarpine a Empty Schisandrin B (hydrochlorid Ipriflavone Hydroxycamp Isoliquiritigeni Sophocarpine (monohydrate Curcumol Rhein Empty e) tothecin n )

Lappaconitine Naringin b Empty Danshensu Salidroside Palmatine Dihydromyric Evodiamine Indirubin (hydrobromid Dihydrochalc Polydatin Aloin Empty (sodium salt) (chloride) etin e) one

c Empty Dioscin Diosmetin Xanthone Sclareol Tangeretin Tanshinone I Troxerutin Ursolic acid Parthenolide Phloretin Empty

Quercetin Monensin d Empty Piperine Puerarin (dihydrate) Rutaecarpine Rutin Salicin sodium salt Myricitrin Naringin Nobiletin Empty

Oleanolic Gynostemma Indole-3- e Empty Acid Oxymatrine Paeonol Luteolin Matrine Gramine Extract Hesperetin carbinol Empty

Beta- Beta- 18β- f Empty Sitosterol Sitosterol Caffeic acid Cryptotanshin Dihydroartemi Diosmin Glycyrrhetinic Fisetin Formononetin Glycyrrhizic Empty (purity>80%) (purity>98%) one sinin acid acid

4- g Empty Methylumbelli Esculin Aloe emodin Amygdalin Andrographoli Arbutin Artesunate Asiatic acid Baicalein Baicalin Empty ferone de

Nordihydrogu Atractylenolid Atractylenolid Atractylenolid Pulchinenosid Patchouli h Empty aiaretic acid e I e II e III e C alcohol Cyasterone Peiminine Dauricine Daurisoline Empty

Plate layout: CS-L025-52

1 2 3 4 5 6 7 8 9 10 11 12

(-)- Bavachalcon a Empty Avicularin Epigoitrin Epigallocatec 7-epi-Taxol Scoparone Psoralidin Bavachin Bakuchiol Corylin Empty hin e

Theaflavin-3'- Theaflavin-3- Saikosaponin Saikosaponin Saikosaponin b Empty Herbacetin Fraxinellone gallate gallate A B2 D Catharanthine Hederagenin Epimedin A1 Empty

Caffeic acid c Empty Cordycepin Tetramethylp Echinocystic Brassinolide phenethyl Aconine Cardamonin Corosolic acid Daphnetin Esculetin Empty yrazine acid ester

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Lycorine 5- d Empty Isoimperatori Lycorine (hydrochlorid Mangiferin Oleuropein Protocatechu Stachydrine Aminolevulini Emodin-8- Mollugin Empty n e) aldehyde c acid glucoside

(E)-Ethyl p- e Empty Salvianolic alpha- Momordin Ic Ziyuglycoside Ziyuglycoside Eugenol Farrerol methoxycinna p-Coumaric (+)- Empty acid C Mangostin I II mate acid hydrate

18α- f Empty (-)-Catechin Columbianadi Sennoside B Trans- Linalool Bergapten Pachymic Glycyrrhetinic Liquiritin Liquiritigenin Empty gallate n Anethole acid acid

g Empty Galangin Lappaconitine Glabridin Wogonoside Wogonin Artemether Orientin Picroside II Daucosterol Trigonelline Empty

Trigonelline Cucurbitacin Cucurbitacin Sophoricosid Astragaloside h Empty chloride B E Cinobufagin e Obacunone Diosbulbin B IV Progesterone Pimpinellin Empty

Plate layout: CS-L025-53

1 2 3 4 5 6 7 8 9 10 11 12

Sinapine L-Chicoric a Empty Asiaticoside Neferine 8-Gingerol 10-Gingerol (thiocyanate) Acacetin Hypericin Acid Corilagin Geraniin Empty

Reserpine b Empty Reserpine (hydrochlorid Phillyrin Liensinine Vincristine α-Lipoic Acid Nitidine Cyanidin Mogroside III Mogroside V Empty e) (sulfate) (chloride) (Chloride)

(-)- c Empty Lovastatin Astilbin Aristolochic Loganin Erianin Calycosin (-)- (+)- Gallocatechin Gallic acid Empty acid A Gallocatechin Gallocatechin gallate

Gallic acid Rosmarinic Calceolariosid α-Angelica Wedelolacton d Empty (hydrate) Ethyl gallate acid Xylitol e B Cynaroside Allantoin lactone e Escin IA Empty

5,15-Diacetyl- 23- 9- e Empty Oroxylin A Lathyrol 3- Notopterol Hydroxybetuli Hydroxysafflo Hydroxytyros Hydroxycamp Umbelliferone Pinocembrin Empty benzoyllathyr nic acid r yellow A ol tothecin

Apigenin 7- Hydrocortison Demethylzeyl Dehydrocostu Ginsenoside Ginsenoside Ginsenoside f Empty glucoside Fraxetin e asteral s Lactone Genistin Panaxadiol F1 Rf Rg2 Empty

20(S)- g Empty Ginsenoside Ginsenoside trans- Cinnamic acid Sucralose Morin Morusin Alpinetin Kaempferitrin Maslinic acid Empty Rg3 Rh2 Cinnamic acid

α-L- h Empty Eriocitrin Rhamnose Carnosol Carnosic acid Dicoumarol Narcissin L-Serine Usnic acid (+)-Usnic acid Amentoflavon Empty monohydrate e

Plate layout: CS-L025-54

1 2 3 4 5 6 7 8 9 10 11 12

Dehydrocoryd Kalii a Empty Aucubin Stevioside Tenacissosid Rhapontin Dehydrocoryd aline Dehydroandr Dehydrograp Icaritin Retinyl Empty e H aline (chloride) ographolide holidi acetate

b Empty α-Vitamin E Vindoline Schisandrin C Schisandrin Schisandrol B Schisandrin A Crocin Crocin II (-)-Asarinin Curculigoside Empty

Berbamine Glucosamine c Empty Gracillin (S)-Indoximod Coumarin Carvacrol Berbamine (dihydrochlori Neobavaisofl Neochlorogen Dracorhodin (hydrochlorid Empty de) avone ic acid perchlorate e)

Leonurine d Empty Phellodendrin Coptisine Stachydrine Leonurine (hydrochlorid Senkyunolide Oxysophocar Oxypeucedan Monocrotaline Empty e (chloride) (chloride) hydrochloride e) A pine in

8-?O- e Empty Scutellarin Scutellarein Eupalinolide Rhoifolin Bornyl ?Acetylharpa Angelicin Isoorientin Isopimpinellin Isoliensinine Empty B acetate gide

Isorhamnetin- Empty Isorhamnetin 3-O- Isosilybin Isoalantolacto Linderalacton Eupatilin Ginkgolide B Lupeol Tectoridin Tectorigenin Empty f neohespeidos ne e

(20S)- g Empty Protopine Proanthocyan Procyanidin Protopanaxad Protodioscin Protosappani Swertiamarin Camphor Timosaponin Timosaponin Empty idins B2 iol n B AIII BII

Resibufogeni Lithospermosi h Empty n Polyphyllin VI Raddeanin A Catalpol de Shikonin Corynoline Pterostilbene Palmitic acid Jaceosidin Empty

Plate layout: CS-L025-55

1 2 3 4 5 6 7 8 9 10 11 12

Pulsatilla Cephalotaxin Epibrassinolid Methyl Macranthoidin a Empty saponin D Jervine Veratramine e Bruceantin e Schisanhenol Harringtonine protodioscin B Empty

Desacetylcino Gamabufotali b Empty Ingenol Isosteviol Arenobufagin Bufalin Bufotalin Cinobufotalin bufotalin n Ginkgetin Tubeimoside I Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Tubeimoside Tetrahydrocur Ginsenoside Ginsenoside Hexahydrocur c Empty II AKBA cumin Catechin (-)-Catechin Corynoxine Corynoxine B Rg6 Rg5 cumin Empty

Santacruzam beta- Sophoraflava d Empty ate A Coixol Mangostin Manool Xanthohumol Tricin Apigenin none G Scabertopin Salvigenin Empty

(20R)- 2- (20R)- e Empty Isoscopoletin Herniarin Fangchinoline Sophoridine Ginsenoside (E)- Periplocin 10- Methoxybenz Ginsenoside Empty Rg3 Cardamonin Deacetyltaxol oic acid Rh1

20(R)- trans- Rhamnose Glycodeoxych f Empty Ginsenoside Trimethoxyre Triacetylresve Noricaritin Sesamol Rhamnose (monohydrate Glycocholic olic acid Citric acid Empty Rh2 sveratrol ratrol ) acid (monohydrate

Methyl p- Hydroxygenk Complanatusi Sodium Ganoderic g Empty coumarate Oroxin B wanin Koumine de Isoquercetin Oleic acid oleate acid A Betulonic acid Empty

14-Deoxy- Empty Hypocrellin B Apigenin-7- Isoschaftosid Aristolone Levistolide A Picfeltarraeni Heterophyllin Ursonic acid Oleanonic 11,12- Empty h glucuronide e n IA B acid didehydroand

Plate layout: CS-L025-56

1 2 3 4 5 6 7 8 9 10 11 12

Halofuginone (2S)-2'- 3',4'- 3,4- (E)-3,4- a Empty Plumbagin Ganoderic Ponicidin Halofuginone (hydrobromid Methoxykurari Dihydroxyace Dimethoxycin Dimethoxycin Danshensu Empty acid D e) none tophenone namic acid namic acid

5-O- b Empty Dihydrocoum Epifriedelanol Pristimerin Demethylnobi Ailanthone Nerolidol Hispidulin Artemisic acid Cucurbitacin Cucurbitacin Empty arin letin D IIa

3-O- Higenamine (20R)- 11-?Keto- c Empty Theaflavin Methylgallic Methyl gallate Anacardic Castanosper Euphorbiaster (hydrochlorid Protopanaxad ?beta- Withaferin A Empty 3,3'-digallate acid Acid mine oid e) iol ?boswellic

7- d Empty Didymin Cedrol (-)-Securinine Songorine Obtusifolin Tenacissosid Ethylcamptot Glaucocalyxin Ginkgolic acid Isoginkgetin Empty e G hecin A C17:1

3- e Empty Parishin B Flavokawain Combretastati Phorbol Cytosporone Dehydrotram Acetylshikoni Deoxyshikoni Bergamottin Pseudoginse Empty B n A4 B etenolic acid n n noside RT1

4- N- 8- f Empty Esculentoside Hydroxylonch Rotundic acid Rhapontigeni ?Feruloylocto Crebanine Curcumenol Geranyloxyps Deltonin Fucoxanthin Empty H ocarpin n pamine oralen

Aclacinomyci 4'- Glycochenod Glycochenod g Empty n A Mogrol Khasianine Demethylpod Piperlongumi Proscillaridin eoxycholic eoxycholic Coumestrol Procyanidin Empty hydrochloride ophyllotoxin ne A acid acid (sodium C1

27- N-Benzoyl- h Empty Procyanidin Cynaropicrin Eudesmin Chelidonine Hydroxychole Palmaturbine Eupatorin (2R,3S)-3- Pinosylvin Auraptene Empty A2 sterol phenylisoseri

Plate layout: CS-L025-57

1 2 3 4 5 6 7 8 9 10 11 12

Delphinidin Flavokawain Flavokawain β-Elemonic Desoxyrhapo a Empty Formosanin C (chloride) A [8]-Shogaol C Amarogentin Sulforaphene acid Aloesin nticin Empty

(2S)- b Empty (E)-Methyl 4- Isoliquiritin β-Boswellic Ginsenoside Gigantol Diphyllin Steviolbioside Euphorbia Hypocrellin A Isoxanthohum Empty coumarate apioside acid Rk1 Factor L1 ol

Isorhapontige Poricoic acid c Empty Irigenin Lupenone Isocorydine nin Loureirin C Ayanin Brevilin A A Britannin Bruceine D Empty

3,4- Empty Dihydroxyben Xanthatin Pinostilbene Naringenin Methyl Caryophyllen Paris saponin Deoxylapach Dihydroresver Guaiol Empty d zylamine triacetate rosmarinate e oxide VII ol atrol

5β- O- e Empty Dihydrocortis Digitonin Glucoraphani Desmethylan Thonningiani Astringin Fucosterol Hypophyllant Decursinol Wushanicariti Empty ol n golensin n A hin n

6- 3'- Pennogenin f Empty Glycycoumari Picrocrocin Isocurcumeno Demethoxyta Demethylnobi Quercetagetin Chrysophanei 3-O-beta- Licochalcone Toringin Empty n l ngeretin letin n chacotrioside D

β- 1-Methyl-6- 4- 4- g Empty Hydroxyisoval Tetrahydropip Yadanziolide oxo-1,6- Methyldaphn Methylesculet 3-Epiursolic Ethoxysangui Decursinol Euphorbia Empty erylshikonin erine A dihydropyridin etin in Acid narine angelate Factor L2

5,7- (E)- β,β- 3'- h Empty Dimethoxyflav Rosmanol Gambogenic Asiaticoside B Terrestrosin Sinapine Flavokawain Dimethylacryl Hydroxyptero Methyl Empty one acid D A shikonin stilbene caffeate

Plate layout: CS-L025-58

1 2 3 4 5 6 7 8 9 10 11 12

7-Hydroxy- a Empty (-)-Alkannin Aloin(mixture Bacopaside II Gardenin B Kamebakauri Polygalacin D Soyasapogen Pinoresinol Cafestol 4H-chromen- Empty of A&B) n ol B 4-one

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

7- 1-beta-D- 6- 6-Hydroxy-4- Diammonium b Empty Aflatoxin B1 Methoxyisofla Arabinofurano Hydroxycoum methylcoumar Calcimycin Citrinin Sonolisib Penicillic acid Glycyrrhizinat Empty vone syluracil arin in e

5,?7,?4'- 2-O-α-D- c Empty Isoeugenol Elemicin Mogroside IIe ?Trimethoxyfl Glucopyranos Arnicolide D Mogroside I Mogroside I Mogroside Groenlandicin Empty acetate avone yl-L-ascorbic E1 A1 IIA1 e

2-O-β-D- Empty Gomisin N Abietic acid Bixin Pseudolaric Prosapogenin Mogroside IV- Mogroside IV Hederacolchi Glucopyranos Lapachol Empty d Acid B A A side A1 yl-L-ascorbic

19- 4'- e Empty Ethyl Caffeate Cepharanthin Baccatin III Perillyl Hydroxybufali Hydroxychalc Sodium Citral Citropten 1,4-Cineole Empty e alcohol n one erythorbate

(E)-m- N- f Empty Thymopentin Coumaric Flavanone Norgestrel γ-Tocopherol (Rac)- Isolongifolene Hibifolin (-)-Zuonin A Nitrosodiethyl Empty (acetate) acid Hydnocarpin amine

Cyclo(- g Empty Millepachine Isoverticine Deoxylimonin Neoanhydrop Angoline Neriifolin Aprotinin Pepstatin Cyclo(- RGDfK) Empty odophyllol RGDfK) (TFA)

[D- h Empty Lecirelin Teriparatide Vapreotide Vapreotide Tyr-Gly-Gly- Ala2]leucine- Angiotensin II Z-WEHD- Disitertide DAMGO Empty (acetate) Phe-Met-OH enkephalin 5-valine FMK (TFA)

Plate layout: CS-L025-59

1 2 3 4 5 6 7 8 9 10 11 12

Kisspeptin- Protease- LSKL, NGR peptide a Empty DAMGO 10, human Activated Inhibitor of (Trifluoroacet CALP3 Epitalon Antagonist G HSDVHK- BA 1 (TFA) Empty (TFA) (TFA) Receptor-2, Thrombospon ate) (TFA) NH2

Antioxidant Angiogenin Lactoferrin RAGE b Empty Fz7-21 (TFA) peptide A (108-122) ACTH (1-17) Malantide (17-41) Lanreotide GPLGIAGQ Angstrom6 antagonist Empty (TFA) (TFA) (TFA) (acetate) (acetate) (TFA) peptide (TFA)

Protease- BIM-23190 c Empty WL47 (TFA) Activated LyP-1 (TFA) (hydrochlorid FTISADTSK ZD-4190 EF-5 GDP366 ARS-1323 ARS-1630 Empty Receptor-1, e) (acetate)

GNE 220 Protein d Empty ARS-1620 (hydrochlorid 3BDO Neoseptin 3 FASN-IN-3 kinase CTX1 PBOX 6 PK11000 ADDA 5 Empty e) inhibitors 1 hydrochloride

N-Boc-O-tosyl 1- O6- 2-Amino-5- e Empty AGN 193109 4-O-Methyl K-80003 GSK2850163 hydroxylamin Hydroxyanthr Tempo Isohomovanill Benzylguanin phenylpyridin Empty honokiol e aquinone ic acid e e

2-(4- 5- f Empty Methoxyphen Heptadecanoi Anthraflavic 5a-Pregnane- Maleimide Acridone Hydroxyindol Bropirimine 2'- Tetrac Empty yl)acetic acid c acid acid 3,20-dione e-3-acetic Deoxyinosine

Hydroxycitric Suberoyl bis- 4- 6- g Empty acid Dibenzoylmet Sinapinic acid hydroxamic Chlorophenyl Citronellol Aminonicotina Thymine SC-236 JNJ- Empty (tripotassium hane acid acetic acid mide 10198409

GPNA 8-Hydroxy-2'- 2,6- 2,2'- h Empty Phytosphingo Benzyl butyl (hydrochlorid Triglycidyl Taurolidine deoxyguanosi Dichlorodiphe Anhydrouridin Benzothiazole Isoquinoline Empty sine phthalate e) isocyanurate ne nylamine e

Plate layout: CS-L025-60

1 2 3 4 5 6 7 8 9 10 11 12

Uridine TRPM8 3- L-2- 1,4- a Empty triphosphate CPTH2 PTP inhibitor S-Allyl-L- antagonist D-Kynurenine CRT0044876 Acetamidoco Hydroxyglutar Naphthoquino Empty (trisodium 1 cysteine WS-3 umarin ic acid ne

Ethyl 3,4- Acivicin 4- D- b Empty Fumaric acid dihydroxyben Acivicin (hydrochlorid Diethylamino 5-Fluoroorotic 2- Terpinen-4-ol Ferulic acid Ribose(mixtur Empty zoate e) benzaldehyde acid Undecanone methyl ester e of isomers)

Benzamidine 4(3H)- D-Erythro- Coumarin-3- 2′-Deoxy-2′- c Empty (hydrochlorid Quinazolinon dihydrosphing carboxylic DNMDP fluoroadenosi Nifurtimox Chromomycin Chelidonic GMBS Empty e) e osine Acid ne A3 acid

2- 2- 3- 2'-O-(2- 2'-O-(2- Acriflavine d Empty Benzylsuccini Methoxycinna Methylcarbaz Methoxyethyl) Methoxyethyl) RAMB4 MT 63-78 Anticancer Thalidomide (hydrochlorid Empty c acid maldehyde ole -uridine -cytidine agent 7 5-fluoride e)

5'-O-DMT-2'- Butylated e Empty TBDMS- JSH-150 L-Norleucine Oxindole Cinchonine hydroxytoluen Farnesol Isatin Urea Dibutyl Empty Uridine e phthalate

Semicarbazid 4- β- Methyl 3,4- f Empty e DL-Serine trans- Cuminaldehy Hydroxybenz Acetamide Monomethyl Aminopropion dihydroxyben Empty Empty (hydrochlorid Chalcone de yl alcohol phthalate itrile zoate

g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected]