1 2004-2005 Cardiovascular System Review

2 Acebutolol Sympatholytic

β1 antagonist Antihypertensive Antiarrhythmic Bronchoconstrictor

3 Acetylcholine Cholinomimetic Antigluacoma Muscle contraction (nicotinic receptor)

4 Adenosine Antiarrhythmic Miscellaneous (does not fit class I-IV organization)

5 Albuterol Sympathomimetic

β2 adrenergic Short acting Used in

6 Amiodarone Class I/III antiarrhythmic Na+ and K+ channel blocker (inactivated channels)

7 Indirect sympathomimetic of abuse ADD treatment

8 Amyl nitrite Vasodilator Antianginal Aerosol

9 Angiotensin II Autacoid

1 Vasoconstrictor

10 Atenolol Sympatholytic

β1 adrenergic antagonist Antihypertensive Antiarrhythmic Antianginal Bronchoconstrictor

11 Atorvastatin Antihyperlipidemic HMG-CoA reductase inhibitor

12 Atropine Antimuscarinic Treatment for bradycardia, diarrhea, cholinesterase poisoning

13 Betaxolol Sympatholytic

β1 adrenergic antagonist Antihypertensive Glaucoma Bronchoconstrictor

14 Bethanecol Cholinomimetic Muscarinic agonist Induces defecation and urination Bronchoconstrictor

15 Biltolterol Sympathomimetic

β2 adrenergic agonist Bronchodilator

16 Bretylium Sympatholytic Class III antiarrhythmic K+ channel blocker

17 Candesartan Antihypertensive Angiotensin receptor blocker (ARB)

2 18 Captopril Antihypertensive Converting enzyme inhibitor failure treatment Angioedema producer

19 Cholestyramine Antihyperlipidemic Bile acid binding resin (BABR)

20 Clofibrate Antihyperlipidemic Lipoprotein lipase activator

21 Clonidine Sympatholytic

α2 adrenergic agonist Antihypertensive

22 Colestipol Antihyperlipidemic Bile acid binding resin (BABR)

23 Diazoxide Vasodilator Antihypertensive

24 Digitalis Antiarrhythmic Na+/K+ ATPase inhibitor Positive inotrope Miscellaneous (does not fit class I-IV organization)

25 Digitoxin Cardiac glycoside Antiarrhythmic Na+/K+ ATPase inhibitor Positive inotrope Miscellaneous (does not fit class I-IV organization)

26 Digoxin Cardiac glycoside Antiarrhythmic Na+/K+ ATPase inhibitor

3 Positive inotrope Miscellaneous (does not fit class I-IV organization)

27 DIG-specific antibody fragments Cardiac glycoside poisoning

28 Diltiazem Class IV antiarrhythmic Antihypertensive Ca2+ channel blocker

29 Disopyramide Class I antiarrhythmic Na+ channel blocker (activated channels)

30 Dobutamine Sympathomimetic

β1 adrenergic agonist Inotrope

31 Dofetilide Class III antiarrhythmic K+ channel blocker

32 Dopamine Sympathomimetic Inotrope Vasodilator

33 Doxazosin Sympatholytic

α1 adrenergic antagonist Antihypertensive

34 Ecothiophate Anticholinesterase Vasodilator Bronchoconstrictor Glaucoma treatment

35 Edrophonium Anticholinesterase Vasodilator Diagnostic for myaesthenia gravis Bronchoconstrictor

4 36 Enalapril Antihypertensive Converting enzyme inhibitor Angioedema producer

37 Indirect sympathomimetic Vasoconstrictor Bronchodilator

38 Sympathomimetic α and β adrenergic agonist Vasoconstrictor Bronchodilator

39 Eprosartan Antihypertensive Angiotensin receptor blocker (ARB)

40 Esmolol Sympatholytic

β1 adrenergic antagonist Class II Antiarrhythmic Antihypertensive Bronchoconstrictor

41 Ezitimibe Antihyperlipidemic Cholesterol absorption inhibitor

42 Fenofibrate Antihyperlipidemic Lipoprotein lipase activator

43 Flecainide Class I antiarrhythmic Na+ channel blocker

44 Fluvastatin Antihyperlipidemic HMG-CoA Reductase Inhibitor

45 Fosinopril

5 Antihypertensive Converting enzyme inhibitor

46 Gemfibrozil Antihyperlipidemic Lipoprotein lipase activator

47 Guanabenz Sympatholytic Antihypertensive

48 Guanadrel Sympatholytic Antihypertensive

49 Guanethidine Sympatholytic Antihypertensive

50 Guanfacine Sympatholytic

α2 adrenergic agonist Antihypertensive

51 Hydralazine Vasodilator Antihypertensive

52 Ibutilide Class III antiarrhythmic K+ channel blocker

53 Imipramine Indirect sympathomimetic Tricyclic (TCA) Antimicturant

54 Isoproterenol Sympathomimetic β adrenergic agonist Vasodilator Bronchodilator

55 Isosorbide dinitrate Venodilator Used to treat CHF

6 56 Lidocaine Class I antiarrhythmic Local anaesthetic Na+ channel blocker (activated and inactivated channels)

57 Lisinopril Antihypertensive Converting enzyme inhibitor Heart failure treatment Angioedema producer

58 Losartan Antihypertensive Angiotensin receptor blocker (ARB)

59 Lovastatin Antihyperlipidemic HMG-CoA reductase inhibitor

60 Malathion Anticholinesterase Vasodilator Bronchoconstrictor

61 Metaproterenol Sympathomimetic

β2 adrenergic agonist Bronchodilator Used in asthma

62 Methacholine Cholinomimetic Bronchoconstrictor

63 Sympathomimetic

α1 adrenergic agonist Vasoconstrictor

64 Methydopa Sympatholytic

α2 adrenergic agonist Antihypertensive

7 65 Methylphenidate Indirect of abuse ADD treatment Stimulant

66 Metoprolol Sympatholytic

β1 adrenergic antagonist Antihypertensive Heart failure medication Bronchoconstrictor

67 Mexilitine Class I antiarrhythmic Na+ channel blocker (activated and inactivated channels)

68 Minoxidil Vasodilator Antihypertensive

69 Moezipril Antihypertensive Converting enzyme inhibitor

70 Moricizine Class I antiarrhythmic Na+ channel blocker

71 Nadolol Sympatholytic β adrenergic antagonist Antihypertensive

72 Neostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Promotes defecation and urination Bronchoconstrictor

73 Nicotine Cholinomimetic Drug of abuse Nicotinic receptor agonist ( contraction)

8 Stimulant Smoking cessation medication

74 Nicotinic acid Antihyperlipidemic Inhibition of VLDL secretion (?)

75 Nifedipine Antihypertensive Antianginal

76 Nitroglycerine Venodilator Antianginal

77 Nitroprusside Vasodilator Antihypertensive

78 Sympathomimetic Vasoconstrictor

79 Perindopril Antihypertensive Converting enzyme inhibitor

80 Phenoxybenzamine Sympatholytic α adrenergic antagonist Antihypertensive

81 Phentolamine Sympatholytic α adrenergic antagonist Antihypertensive

82 Sympathomimetic

α1 adrenergic agonist Vasoconstrictor Nasal decongestant

83 Phenytoin Class I antiarrhythmic

9 Na+ channel blocker (inactivated channels)

84 Physostigmine Anticholinesterase Bradycardic Vasodilator Bronchoconstrictor

85 Pilocarpine Cholinomimetic Muscarinic agonist Antiglaucoma Bronchoconstrictor

86 Pindolol Sympatholytic β adrenergic antagonist Antihypertensive Bronchoconstrictor

87 Pravastatin Antihyperlipidemic HMG-CoA reductase inhibitor

88 Prazosin Sympatholytic

α1 adrenergic antagonist Antihypertensive

89 Propranolol Sympatholytic β adrenergic antagonist Class II antiarrhythmic Antihypertensive Bronchoconstrictor

90 Sympathomimetic α and β adrenergic agonist Vasoconstrictor Nasal decongestant

91 Pyridostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis

10 Bronchoconstrictor

92 Quinapril Antihypertensive Converting enzyme inhibitor

93 Quinidine Antimalarial Protein and nucleic acid synthesis inhibitor

Class I antiarrhythmic Intercalates in DNA Binds to ferriprotoporphyrin Na+ channel blocker

94 Ramipril Antihypertensive Converting enzyme inhibitor

95 Reserpine Sympatholytic Antihypertensive

96 Sildenafil Vasodilator Promotes erection

97 Simvastatin Antihyperlipidemic HMG-CoA reductase inhibitor

98 Sotolol Class II antiarrythmic Sympatholytic β adrenergic antagonist

99 Terazosin Sympatholytic

α1 adrenergic antagonist Antihypertensive Treatment for benign prostatic hypertrophy

100 Sympathomimetic

β2 adrenergic agonist Short acting bronchodilator

11 Tocolytic Uterine relaxant

101 Timolol Sympatholytic β adrenergic antagonist Antihypertensive Glaucoma treatment Anti-anginal Bronchoconstrictor

102 Tocainide Class I antiarrhythmic Na+ channel blocker (activated channels)

103 Trandopril Antihypertensive Converting enzyme inhibitor

104 Trimethaphan Sympatholytic Anticholinergic Nicotinic antagonist Antihypertensive

105 Tyramine Indirect sympathomimetic Vasoconstrictor Vasopressor

106 Valsartan Antihypertensive Angiotensin receptor blocker (ARB)

107 Verapamil Class IV antiarrhythmic Antihypertensive L-type Ca2+ channel blocker Antianginal

12