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Cytoskeleton Compound Library (96-well)

Product Details:

Catalog Number: CS-L060

Formulation: A collection of 823 cytoskeleton compounds supplied as pre-dissolved Solutions or Solid

Container: 96- or 384-well Plate with Peelable Foil Seal; 96-well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode

Storage: -80°C

Shipping: Blue ice

Packaging: Inert gas

Plate layout: CS-L060-1

1 2 3 4 5 6 7 8 9 10 11 12

MELK-8a a Empty AZD0156 BAY1125976 PQR620 KNK437 R547 CP21R7 CZ415 A-205804 Rho-Kinase- (hydrochlorid Empty IN-1 e)

Brevianamide αvβ1 integrin- b Empty F PF-04979064 HA15 WYE-132 IN-1 (TFA) NSC781406 GSK2256098 M2698 GLPG0187 NVS-PAK1-1 Empty

D-α- Cyclo(RGDyK Y-33075 c Empty Hydroxyglutar GSK621 ) Hispidin Y-33075 CGS 15943 MS-444 (dihydrochlori Y-27632 Eganelisib Empty ic acid (trifluoroaceta de)

W-7 ATM-3507 d Empty Toxoflavin NCB-0846 IWP-O1 KRIBB11 BAY1082439 (hydrochlorid ML-9 (trihydrochlori HA-100 CCT251236 Empty e) de)

D-erythro- e Empty Sphingosine Monastrol LY294002 SKL2001 AS-605240 KYA1797K IC-87114 TG100-115 PNU-74654 TGX-221 Empty

PI-103 f Empty SF2523 PI-103 (Hydrochlorid ZINC0088152 GDC-0326 EMT inhibitor- ZM-447439 Paprotrain LF3 GZD856 Empty e) 4 1 (formic)

Elimusertib Nilotinib g Empty GDC-0077 Elimusertib (hydrochlorid Darovasertib Bosutinib Nilotinib (monohydroc Tozasertib Recilisib LTURM34 Empty e) hloride

Dasatinib CHIR-99021 CHIR-99021 h Empty TRC051384 BTB-1 PHA-680632 Danusertib MLN8054 Dasatinib (hydrochlorid CHIR-99021 (monohydroc (trihydrochlori Empty e) hloride) de)

Plate layout: CS-L060-2

1 2 3 4 5 6 7 8 9 10 11 12

Ruboxistaurin Retaspimycin a Empty Heparan Autophinib PI3Kδ-IN-1 (hydrochlorid Wortmannin KY1220 Linperlisib Masitinib (Hydrochlorid Tanespimycin Empty Sulfate e) e)

AKT Kinase b Empty BIIB021 Luminespib Everolimus Rapamycin Midostaurin GSK-690693 Inhibitor Omipalisib GSK-923295 Empty

Tirbanibulin c Empty HSF1A PIK-294 CMPD101 ROCK-IN-2 RSVA405 Ro 90-7501 JNJ-7706621 KW-2449 Tirbanibulin (dihydrochlori Empty de)

Fasudil MK-2206 d Empty Tirbanibulin (Hydrochlorid Enzastaurin Sotrastaurin AZD 6482 PI-273 AKT inhibitor (dihydrochlori GW779439X K00546 Empty (Mesylate) e) VIII de)

PF-562271 e Empty PF-06409577 iCRT3 PP121 PD173955 Asciminib LM22B-10 AZD-8055 OSI-027 A-443654 (besylate) Empty

SCH- Y-27632 f Empty PF-562271 PF-573228 Torkinib 1473759 Lexibulin AR-A014418 BX795 CYC-116 GSK 3 (dihydrochlori Empty (hydrochlorid Inhibitor IX de)

Larazotide Arimoclomol g Empty TWS119 IQ 1 MMV390048 Rotigaptide (acetate) (maleate) PKI-402 MAP4343 PF-AKT400 MTX-211 Empty

Bisindolylmal Empty PQR530 NU6140 A 1070722 A-286982 R 59-022 Guggulsteron MK-3903 CCT 137690 GNE-493 eimide X Empty h e (hydrochlorid

Plate layout: CS-L060-3

1 2 3 4 5 6 7 8 9 10 11 12

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Parsaclisib a Empty T- C8-Ceramide DCP-LA DCPLA-ME Mavacamten Adavivint Parsaclisib (hydrochlorid Conteltinib Tegatrabetan Empty 00127_HEV1 e)

Danegaptide ENMD-2076 b Empty Danicamtiv Hydrochloride Zandelisib Pifithrin-μ VER-155008 VER-82576 GNF-7 AZD1390 Alisertib (Tartrate) Empty

(Z)- c Empty ENMD-2076 GSK429286A CP-466722 BX-912 KU-57788 Guggulsteron GNF-2 RWJ 50271 CGP60474 TDZD-8 Empty e

Metformin D6 PKI-179 d Empty BRD9876 (hydrochlorid WAY-262611 GNE-477 Fingolimod PKI-179 (hydrochlorid Pilaralisib CZC-8004 PIK-108 Empty e) e) analogue

5-Iodo- e Empty MK8722 LX2343 SSE15206 PI3K/mTOR IPI-3063 AZ2 NRX-252262 AZD-7648 SNIPER(ABL) indirubin-3'- Empty Inhibitor-2 -020 monoxime

Chitosan f Empty oligosacchari O-304 AZ32 Aurora kinase Aurora kinase UCT943 AZD3458 Tubulin UCB9608 PKC-theta Empty de inhibitor-2 inhibitor-3 inhibitor 1 inhibitor

Grp94 mTOR N-Oleoyl g Empty EX229 VTX-27 DK419 IITZ-01 Inhibitor-1 inhibitor-1 glycine 9-ING-41 LY3295668 CCB02 Empty

NV-5138 h Empty (hydrochlorid HDACs/mTO AT-1002 P110δ-IN-1 Benproperine Parbendazole EB-3D GW406108X ILK-IN-3 BRD0705 Empty e) R Inhibitor 1 (TFA) (phosphate)

Plate layout: CS-L060-4

1 2 3 4 5 6 7 8 9 10 11 12

Fingolimod a Empty BRD5648 FzM1.8 JG-98 BJE6-106 AS-041164 Vacuolin-1 Hematein ROCK SNS-314 (hydrochlorid Empty inhibitor-2 (mesylate) e)

Alvespimycin 2- b Empty SB 216763 KU-55933 (hydrochlorid PIK-90 Methoxyestra WYE-354 GSK1059615 Rigosertib Lyn-IN-1 TASP041591 Empty e) diol (sodium) 4

AT7867 c Empty PIK-93 Ponatinib Chelerythrine CCT129202 AT7867 VERU-111 (dihydrochlori KU-60019 PHT-427 Empty (chloride) (ditartrate) de)

SB-743921 d Empty SSTC3 PI3K-IN-1 (hydrochlorid MSAB DPH MRT199665 CAY10404 PS210 CCG-222740 TAK-901 Empty e)

Umbralisib e Empty JR-AB2-011 PI-3065 IWR-1 AZ82 STL127705 (hydrochlorid HLY78 bpV(phen) Serabelisib Empty e) (trihydrate)

Defactinib Cardiogenol f Empty Defactinib (hydrochlorid Arg-Gly-Asp- Borussertib IM-12 Kenpaullone AKI603 C AZD8186 HTH-01-015 Empty e) Ser (hydrochlorid

JNJ- g Empty ETP-46321 Bempedoic NMS-P715 ζ-Stat Mps1-IN-3 47117096 Carotegrast BDP5290 Y15 DM4 Empty acid hydrochloride methyl

HSP27 p32 Inhibitor hSMG-1 hSMG-1 Rheb inhibitor h Empty (R)-BRD3731 BRD3731 inhibitor J2 M36 inhibitor 11j KY-05009 inhibitor 11e NR1 SAR405 Col003 Empty

Plate layout: CS-L060-5

1 2 3 4 5 6 7 8 9 10 11 12

3- A-3 a Empty COH-SR4 LCH-7749944 Samotolisib PF-06380101 Bikinin Phenyltoxofla GMB-475 (hydrochlorid HM03 GSK-3β Empty vin e) inhibitor 1

(E/Z)-GSK-3β PKC-iota b Empty inhibitor 1 inhibitor 1 HSP70-IN-1 ON123300 HSD1590 Urolithin B GNE 2861 Acalisib LX7101 MPI-0479605 Empty

c Empty PE859 CCT251545 GNE-317 Vps34-PIK-III Vps34-IN-1 Ampkinone Empesertib BAY1217389 Bimiralisib AZD-8835 Empty

VP3.15 N- d Empty BpV(HOpic) SIAIS178 IWP-4 (dihydrobromi SKI V Desmethylta KDU691 AMG319 GNF4877 Torin 2 Empty de) moxifen

Isobavachalc VO-Ohpic e Empty Torin 1 PF-3758309 DM4-SMe S516 Rebastinib one Cenisertib (trihydrate) CHIR-98014 Empty

GSK-3β AMPK mTOR (S)-PI3Kα-IN- f Empty inhibitor 2 HS-27 LP-922056 activator 4 SP-96 inhibitor-8 PI3Kα-IN-4 4 KY19382 NVP-TAE 226 Empty

A-674563 g Empty YM-201636 Apitolisib MK-5108 AMG 900 A-674563 (hydrochlorid Thiazovivin CCT128930 A66 Degrasyn Empty e)

PIK-75 h Empty ABT-751 (hydrochlorid Mps1-IN-1 SR-3677 Pyrintegrin XL888 Sapanisertib BGT226 Aminohexylge NVS-PI3-4 Empty e) (maleate) ldanamycin

Plate layout: CS-L060-6 Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

1 2 3 4 5 6 7 8 9 10 11 12

Dorsomorphin GSK- a Empty Integrin AICAR (dihydrochlori Dorsomorphin Deguelin KU-0060648 Ionomycin AMG 511 3/CDK5/CDK BC1618 Empty modulator 1 (phosphate) de) (calcium) 2-IN-1

Mitoxantrone b Empty KW-2478 Debio 0932 Tau tracer 2 (dihydrochlori A PIK-293 TG 100713 Nocodazole Fimepinostat Empty de)

ATN-161 MSC2360844 c Empty CAY10505 AS-604850 AS-252424 (trifluoroaceta Wnt pathway Batabulin Batabulin TD52 MSC2360844 (hemifumarat Empty te salt) activator 1 (sodium) e)

Valecobulin Estramustine d Empty Valecobulin (hydrochlorid Crolibulin IM156 Tubulin FIDAS-3 SRX3207 (phosphate ATR inhibitor ASP4132 Empty e) inhibitor 6 sodium) 2

β-catenin-IN- e Empty 2 Indibulin PQR626 Maytansine Miltefosine Go 6983 TML-6 TAS-119 Teplinovivint Vodobatinib Empty

Tamoxifen f Empty SAR502250 (Citrate) Tamoxifen (sulfate) XL388 Blebbistatin KY02111 NU6027 MK-8745 Empty

Hydroxy- Ro 31-8220 g Empty SKI II DTHIB YUM70 BX517 PS47 RO0270608 AZD1080 Dynasore PF-4989216 (mesylate) Empty

Hydroxyfasud PND-1186 h Empty Bisindolylmal Taselisib Flumatinib Flumatinib Hydroxyfasud il IWP-2 PND-1186 (hydrochlorid Indirubin-3′- Empty eimide I (mesylate) il (hydrochlorid e) oxime

Plate layout: CS-L060-7

1 2 3 4 5 6 7 8 9 10 11 12

GSK-3 GSK-3β Omecamtiv a Empty DDO-5936 inhibitor 1 Mps1-IN-2 inhibitor 3 mecarbil GSK-25 LP-261 ICG-001 MP7 Plinabulin Empty

Apilimod b Empty Onalespib E7820 PF-03814735 Palomid 529 [6]-Gingerol Apilimod (mesylate) AZ3146 Reversine VE-821 Empty

1- c Empty Litronesib Litronesib Carotegrast Deoxynojirimy Tideglusib Verubulin Prinaberel Cevipabulin Cevipabulin Firategrast Empty (Racemate) cin fumarate

5- d Empty (E)-Akt GSK2334470 EMD534085 AST 487 Aminosalicylic MKT-077 Apoptozole MK-0429 Staurosporine (hydrochlorid Empty inhibitor-IV Acid e)

Buparlisib Ipatasertib e Empty XAV-939 Dactolisib PF-04691502 (Hydrochlorid Ipatasertib (dihydrochlori Filanesib (R)-Filanesib NVP-HSP990 Tonabersat Empty (Tosylate) e) de)

Geldanamyci f Empty Ganetespib n GSK2636771 Vistusertib GDC-0349 WYE-687 WAY-600 Epothilone D CZC24832 Empty

Copanlisib ML-7 g Empty Dynasore Belumosudil (dihydrochlori BIO- ALK inhibitor ALK inhibitor Chroman 1 (hydrochlorid Capivasertib SB 415286 Empty de) acetoxime 1 2 e)

OTSSP167 h Empty Triciribine Imatinib CH5132799 YS-49 D-64131 RGB-286638 RGB-286638 (hydrochlorid CGK733 Empty (free base) e)

Plate layout: CS-L060-8

1 2 3 4 5 6 7 8 9 10 11 12

Taltobulin Taltobulin a Empty ETP-46464 FRAX597 FRAX486 Podofilox GSK269962A AZ20 Taltobulin (trifluoroaceta (hydrochlorid Salinomycin Empty te) e)

SAR407899 b Empty Wnt-C59 IPA-3 GZD824 GZD824 KP372-1 PI4KIII beta Ripasudil (hydrochlorid SAR407899 Leukadherin- Empty (dimesylate) inhibitor 3 e) 1

H-1152 Afuresertib c Empty NU 7026 (dihydrochlori FH535 Afuresertib (hydrochlorid GNF-5 Ansamitocin XL228 RKI-1447 AZD2858 Empty de) e) P-3

d Empty TR-14035 TAS-116 WZ4003 SAR-260301 YLF-466D CEP-37440 SF1670 CW-069 HS-173 Mdivi-1 Empty

GSK2110183 Ilorasertib e Empty CK-636 Voxtalisib Kif15-IN-1 Kif15-IN-2 Uprosertib analog 1 APY0201 VER-50589 VER-49009 (hydrochlorid Empty (hydrochlorid e)

CAL-130 Phenformin f Empty AT13148 BNC105 (Hydrochlorid Cilengitide Cilengitide ELR510444 LY2090314 NVP-QAV- (hydrochlorid Pilaralisib Empty e) (TFA) 572 e)

ZLN024 g Empty Narciclasine Colchicine VS-5584 CNX-1351 iCRT 14 3CAI BTS (hydrochlorid Seletalisib Verosudil Empty e)

CC-115 h Empty Entasobulin PKC-IN-1 WIKI4 CK-666 CK-869 Cytochalasin CC-223 CC-115 (hydrochlorid Epothilone B Empty B e)

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

Plate layout: CS-L060-9

1 2 3 4 5 6 7 8 9 10 11 12

Tirofiban 4'- Metformin a Empty Duvelisib (R (hydrochlorid Demethylepip Salinomycin Fosbretabulin (hydrochlorid Leniolisib Tenalisib Quercetin Empty enantiomer) e odophyllotoxi (sodium salt) (disodium) e)

Ombrabulin Phorbol 12- b Empty CCT241736 (hydrochlorid AKT-IN-1 mTOR CWHM-12 ML346 OSU-T315 ILK-IN-2 PU-WS13 myristate 13- Empty e) inhibitor-3 acetate

Phorbol c Empty BQR-695 CWP232228 TAS-301 Rottlerin Decursin 12,13- ETC-159 GSK180736A Ceralasertib (S)- Empty dibutyrate Ceralasertib

G-5555 d Empty Compound Lifitegrast Maytansinol PF-2771 Nemiralisib FRAX1036 G-5555 (hydrochlorid Miransertib JW74 Empty 401 e)

TAS-117 e Empty BEBT-908 PI4KIIIbeta- Indirubin-3'- SC66 (hydrochlorid Dimethylenas K858 YU238259 AKT-IN-6 BML-284 Empty IN-9 monoxime e) tron (Racemic)

Pictilisib f Empty (dimethanesul Triptonide Pictilisib AT9283 A-769662 KU-0063794 Ispinesib ZSTK474 Akt1 and Bafetinib Empty fonate) Akt2-IN-1

1- g Empty Perifosine Temsirolimus Imatinib Azakenpaullo TCS7010 Buparlisib Zaurategrast Methyl Zaurategrast Cephalomann Empty (Mesylate) ne vanillate ethyl ester ine

Docetaxel Pamidronic Cromolyn Triclabendazo h Empty (Trihydrate) acid Artemisinin Flubendazole (sodium) le Metformin (ditartrate) Empty

Plate layout: CS-L060-10

1 2 3 4 5 6 7 8 9 10 11 12

Nefopam Chloropyrami a Empty Eptifibatide Ingenol Teprenone SU6656 MHY1485 Danthron (hydrochlorid Flufenamic ne Meclofenamic Empty Mebutate e) acid hydrochloride acid (sodium)

Buformin b Empty Carbenoxolon Ethoxyquin (hydrochlorid Honokiol Oridonin Echinacoside Verbascoside Polyphyllin I (E)-Ferulic Sophocarpine Empty e (disodium) e) acid

Sophocarpine c Empty (monohydrate Cyclovirobuxi Salidroside Dihydromyric Quercetin 7-epi-Taxol Daphnetin Esculetin Paeoniflorin Pachymic Empty ) ne D etin (dihydrate) acid

Cucurbitacin Phellodendrin Astragaloside Nitidine Demethylene d Empty Gomisin J Wogonin B e I L-Leucine (sulfate) (chloride) berberine (+)-Usnic acid Empty

Specnuezhen e Empty ide Vindoline Daphnoretin Schaftoside Scutellarin Isorhamnetin Ginkgolide C Palmitic acid Ingenol Ginkgetin Empty

1,3- f Empty Fangchinoline 10- Platycodin D Dicaffeoylquin Vaccarin Oroxin B Heterophyllin Loureirin A Cucurbitacin Euphorbiaster Empty Deacetyltaxol ic acid B D oid

N- g Empty Glaucocalyxin Ginkgolic acid Combretastati Rotundic acid ?Feruloylocto Crebanine Deltonin Procyanidin L- Amarogentin Empty A C17:1 n A4 pamine A1 Quebrachitol

7- h Empty Deoxypodoph Ginsenoside Gigantol Hypocrellin A Irigenin Paris saponin Licochalcone Decursinol Nepodin Methoxyisofla Empty yllotoxin Rk1 VII E angelate vone

Plate layout: CS-L060-11

1 2 3 4 5 6 7 8 9 10 11 12

Cyclo(- a Empty Sonolisib Arnicolide D Hederacolchi Cimiracemosi Erucic acid Marein Cyclo(- RGDfK) Disitertide Gap19 (TFA) Empty side A1 de C RGDfK) (TFA) (TFA)

Pep2m, b Empty HSDVHK- myristoylated Fz7-21 (TFA) Malantide ICAM-1-IN-1 BF738735 3BDO PBOX 6 K-80003 Tetrac Empty NH2 (TFA)

Methyl c Empty Myoseverin cinnamate MT 63-78 Empty Empty Empty Empty Empty Empty Empty Empty

d Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected] • Bioactive Molecules • Building Blocks • Intermediates www.ChemScene.com

h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

Address: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USA Tel: 732-484-9848 Fax: 888-484-5008 Email: [email protected]