Detergents Enzyme Inhibitors Immunosuppressants Ionophores Molecular Biology Tools Protein Purification Reagents Stem Cell Research Tools

Activators/Inducers, Agonists, etc. Antibiotics Anticancer Agents Antioxidants Apoptosis Inducers Apoptosis Inhibitors Buffers Detergents Enzyme Inhibitors Immunosuppressants Ionophores Molecular Biology Tools Protein Purification Reagents Stem Cell Research Tools ..... and more Order Instructions & Warranty Information

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2 Printed December,Tech help: 2011 [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Table of Contents

Activators/Inducers, Agonists, etc...... 04

Antibiotics ...... 06

Anticancer Agents ...... 07

Antioxidants ...... 08

Apoptosis Inducers ...... 09

Apoptosis Inhibitors ...... 10

Buffers ...... 10

Calcium Modulators ...... 10

Detergents ...... 10

Dyes/Stains, Probes, Substrates, etc...... 11

Enzyme Inhibitors ...... 15

Immunosuppressants ...... 36

Ionophores ...... 37

Molecular Biology Tools ...... 37

Other Biochemicals ...... 38

Protein Purification Reagents...... 38

Stem Cell Research Tools ...... 40

Product Index ...... 44

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 3 Activators/Inducers, Agonists.. Biochemicals Activators/Inducers, Agonists, etc. ► Adenylase Cyclase Activators

Product Name Catalog # Size Forskolin 1531-5 5 mg

► Autophagy Inducers

Product Name Catalog # Size Amiodarone Hydrochloride 1828-100 100 mg 1828-500 500 mg Rottlerin 1827-10 10 mg SMER28 1856-5 5 mg 1856-25 25 mg

► Hedgehog Signaling Pathway Agonists

Product Name Catalog # Size Purmorphamine 1672-5 5 mg Smo Agonist, SAG 1939-500 500 µg 1939-1000 1 mg

► p53 Activators

Product Name Catalog # Size NSC 146109 hydrochloride 1907-5 5 mg

► PPAR Activators

Product Name Catalog # Size Ciglitazone 1695-5 5 mg Pioglitazone 1877-5 5 mg 1877-25 25 mg 1877-100 100 mg Rosiglitazone 1559-5 5 mg 1559-50 50 mg 1559-100 100 mg Troglitazone 1696-5 5 mg

► Pro-caspase Activators

Product Name Catalog # Size PAC-1 1654-10 10 mg

4 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Activators/Inducers, Agonists..

► Protein Kinase Activators Product Name Catalog # Size 8-Br-cAMP 1837-5 5 mg 1837-25 25 mg 8-Br-cGMP 1838-5 5 mg 1838-25 25 mg A-769662 1719-5 5 mg AICAR 1687-50 50 mg Anisomycin 1549-10 10 mg Arachidonic Acid 1505-100 100 mg Aurintricarboxylic acid 1506-1000 1 g bpV(phen) 1793-5 5 mg bpV(pic) 1794-5 5 mg Metformin, Hydrochloride 1691-5G 5 g Phenformin hydrochloride 1889-100 100 mg 1899-1000 1 g Phorbol-12-myristate 13-acetate (PMA) 1544-5 5 mg PS48 1869-5 5 mg 1869-25 25 mg 1869-100 100 mg

► ROR Ligands

Product Name Catalog # Size SR1001 1902-5 5 mg 1902-25 25 mg

► Sirtuin Activators

Product Name Catalog # Size Resveratrol 1758-100 100 mg 1758-500 500 mg

► TGR5 Receptor Agonist

Product Name Catalog # Size Betulinic acid 1552-25 25 mg 1552-100 100 mg Oleanolic Acid 1731-100 100 mg 1731-500 500 mg TGR5 Receptor Agonist 1722-5 5 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 5 Antibiotics Biochemicals

► Toll-Like Receptor (TLR) Agonists Product Name Catalog # Size Imiquimod 1698-100 100 mg Pam3Cys-Ser-(Lys)4, Trihydrochloride 1700-100 100 µg Resiquimod 1699-5 5 mg

Antibiotics Product Name Catalog # Size A23187 1501-10 10 mg Anisomycin 1549-10 10 mg Ascomycin 1573-2 2 mg Blasticidin S Hydrochloride 1859-25 25 mg 1859-100 100 mg Brefeldin A 1560-5 5 mg Cycloheximide 1041-1G 1 g Cycloheximide (100 mM) 1041-1 1 ml Cyclosporine A 1522-100 100 mg 1522-1G 1 g Daunorubicin.HCl 1524-10 10 mg 1524-50 50 mg 1524-500 500 mg Doxorubicin.HCl 1527-5 5 mg G418 Sulfate (siRNA Vector Approved) 1557-1000 1 g 1557-5G 5 g 1557-25G 25 g Geldanamycin 1564-1 1 mg Ionomycin (Calcium salt) 1566-5 5 mg Ionomycin (free acid) 1565-5 5 mg Puromycin Dihydrochloride 1860-25 25 mg 1860-100 100 mg 1860-250 250 mg 1860-500 500 mg 1860-1000 1 g EZSolution™ Puromycin Dihydrochloride 1861-100 100 mg Staurosporine 1048-100 100 µg 1048-1 1 mg EZSolution™ Staurosporine 1745-01 100 µg Streptozocin 1930-100 100 mg 1930-500 500 mg 1930-1000 1 g Teicoplanin 1756-100 100 mg 1756-1G 1 g

6 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Anticancer Agents

Antibiotics Continued... Product Name Catalog # Size Tigecycline 1956-5 5 mg 1956-25 25 mg Thapsigargin 1558-1 1 mg Trichostatin A 1606-1 1 mg

Anticancer Agents Product Name Catalog # Size (R,S)-Lenalidomide 1862-25 25 mg 1862-100 100 mg Betulinic acid 1552-25 25 mg Bexarotene 1575-5 5 mg 1575-50 50 mg Brefeldin A 1560-5 5 mg Capecitabine 1741-100 100 mg 1741-1000 1 g Carboplatin 1553-100 100 mg Cisplatin 1550-100 100 mg 1550-1000 1 g CP-31398 Dihydrochloride 1815-5 5 mg 1815-25 25 mg Cyclopamine 1578-5 5 mg Daunorubicin.HCl 1524-10 10 mg 1524-50 50 mg 1524-500 500 mg Doxorubicin.HCl 1527-5 5 mg Fludarabine Phosphate 1763-10 10 mg 1763-50 50 mg Geldanamycin 1564-1 1 mg Gemcitabine Hydrochloride 1759-25 25 mg 1759-100 100 mg Genistein 1533-10 10 mg Jasplakinolide, jaspis johnstoni 1689-05 5 µg Mitoxantrone 1885-50 50 mg 1885-250 250 mg Naringenin 1772-250 250 mg 1772-1000 1 g Nedaplatin 1576-5 5 mg Nimbolide 1891-5 5 mg 1891-25 25 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 7 Antioxidants Biochemicals Anticancer Agents Continued... Product Name Catalog # Size Oridonin 1730-5 5 mg 1730-25 25 mg Oxaliplatin 1577-25 25 mg Paclitaxel 1567-25 25 mg Pifithrin-ɑ 1554-10 10 mg Piperlongumine 1919-10 10 mg 1919-50 50 mg Pixantrone maleate 1958-5 5 mg 1958-25 25 mg Rapamycin 1568-5 5 mg EZSolution™ Rapamycin 1746-5 5 mg Tamoxifen citrate 1551-1000 1 g Vinblastine Sulfate 1959-5 5 mg 1959-25 25 mg Vinorelbine Tartrate 1957-5 5 mg 1957-25 25 mg

Antioxidants Product Name Catalog # Size Celastrol 1940-5 5 mg 1940-25 25 mg Deferoxamine Mesylate 1883-500 500 mg 1883-1000 1 g (-)-Epigallocatechin gallate 1841-50 50 mg IPAM 1817-100 100 mg 1817-500 500 mg 1817-1000 1 g Naringenin 1772-250 250 mg 1772-1000 1 g Quercetin, Dihydrate 1773-250 250 mg 1773-1000 1 g Reduced Glutathione (GSH) 1242-1 1 g Resveratrol 1758-100 100 mg 1758-500 500 mg Rosmarinic Acid 1843-50 50 mg 1843-250 250 mg Tiliroside 1879-1 1 mg 1879-5 5 mg

8 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Apoptosis Inducers Apoptosis Inducers Product Name Catalog # Size Actinomycin D 1036-5MG 5 mg 1036-50MG 50 mg Actinomycin D (10 mM) 1036-50 50 µl Anisomycin 1549-10 10 mg Berberine Chloride 1830-100 100 mg 1830-500 500 mg Betulinic acid 1552-25 25 mg Brefeldin A 1560-5 5 mg Cerulenin 1579-5 5 mg 1579-50 50 mg Camptothecin 1039-50MG 50 mg 1039-500MG 500 mg Camptothecin (2 mM) 1039-1 1 ml Colchicine 1519-1000 1 g Cycloheximide 1041-1G 1 g Cycloheximide (100 mM) 1041-1 1 ml Daunorubicin.HCl 1524-10 10 mg Dexamethasone 1042-1G 1 g 1042-10G 10 g Doxorubicin.HCl 1527-5 5 mg Etoposide 1043-250MG 250 mg 1043-25MG 25 mg Etoposide (100 mM) 1043-100 100 µl Staurosporine 1048-01 100 µg 1048-1 1 mg Tamoxifen citrate 1551-1000 1 g

Etoposide A topoisomerase II inhibitor. A derivative of podophyllotoxin that has major activity against a number of tumors, including germ cell neo- plasms, small cell lung cancer, and malignant lymphoma. Induces apoptosis in human T cells, mouse thymocytes, and HL-60 human leukemia cells . Appearance: White solid

Molecular Formula: C22H29FO5 Molecular Weight: 588.56 Purity: >98% by HPLC

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 9 Apoptosis Inhibitors Biochemicals Apoptosis Inhibitors ► Caspase & Granzyme B Inhibitors (see page 16) Buffers Product Name Catalog # Size EDTA Solution (pH 8.0) 2103-100 100 ml ( 1 M) Imidazole, MegaPure™ 1802-25G 25 g 1802-100G 100 g PBS Tablets 2129-10 10 Tablets 2129-100 100 Tablets PBS-Tween® Tablets 2130-10 10 Tablets 2130-100 100 Tablets Phosphate Buffered Saline (PBS) 2113-500 500 ml (10X) RIPA Buffer 2114-100 100 ml 2114-500 500 ml 3X SDS-PAGE Loading Buffer 2108-10 5 x 2 ml

SDS Solution (10% in H2O) 2102-100 100 ml Tris-HCl (pH 6.8) 2106-100 100 ml (1 M) Tris-HCl (pH 8.8) 2107-100 100 ml (1.5 M)

Calcium Modulators Product Name Catalog # Size 2-APB 1798-100 100 mg Calcitriol 1880-50 50 µg 1880-250 250 µg Pamidronate disodium 1884-50 50 mg 1884-250 250 mg Thapsigargin 1558-1 1 mg

Detergents Product Name Catalog # Size ASB-14 1738-5G 5 g 1738-25G 25 g CHAPS, High Purity 1545-10G 10 g 1545-50G 50 g 1545-100G 100 g 1545-500G 500 g 1545-1Kg 1 Kg n-Octyl-β-D-glucopyranoside 1646-5G 5 g 1646-25G 25 g 1646-50G 50 g

NP-40 (10% in H2O) 2111-100 100 ml

10 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Detergents Detergents Continued... NP-40 Substitute, MegaPure™ Detergent, 10% 2127-50 50 ml Solution 2127-100 100 ml 2127-500 500 ml Octyl-β-D-thioglucopyranoside 1782-1G 1 g 1782-5G 5 g 1782-50G 50 g 1782-100G 100 g

SDS Solution (10% in H2O) 2102-100 100 ml Sulfobetaine 3-16 1777-5G 5 g 1777-25G 25 g

Triton® X-100 Solution (10% in H2O) 2104-100 100 ml Triton® X-100, MegaPure™ Detergent, 10% 2124-50 50 ml Solution 2124-100 100 ml 2124-500 500 ml

Tween® 20 Solution (10% in H2O) 2109-100 100 ml Tween® 20, MegaPure™ Detergent, 10% 2125-50 50 ml Solution 2125-100 100 ml 2125-500 500 ml Tween® 80, MegaPure™ Detergent, 10% 2126-50 50 ml Solution 2126-100 100 ml 2126-500 500 ml

Dyes/Stains, Probes and Substrates ► Dyes/Stains, etc.

Product Name Catalog # Size Ethidium Bromide 1203-10 10 ml Propidium Iodide 1056-1 1 ml Trypan Blue (0.4%) 1209-10 10 ml

► Probes

Product Name Catalog # Size Calcein AM 1755-50 50 µg 1755-250 5 x 50 µg Jasplakinolide, jaspis johnstoni 1689-05 50 µg JC-1 1130-5 5 mg OxiRed™ Probe 1572-5 5 mg 1572-10-5 10 x 5 mg 1572-20-5 20 x 5 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 11 D/S,Probes,Substrates Biochemicals

► Substrates Calpain Substrate

Product Name Catalog # Size Suc-Leu-Leu-Val-Tyr-AMC 1833-5 5 mg

Caspase Substrates

Caspase-1 Substrates

Product Name Catalog # Size Caspase-1 Substrate YVAD-AFC 1103-200 200 assays 1103-1000 1000 assays Caspase-1 Substrate YVAD-pNA 1104-200 200 assays 1104-1000 1000 assays

Caspase-2 Substrates

Product Name Catalog # Size Caspase-2 Substrate VDVAD-AFC 1071-200 200 assays 1071-1000 1000 assays Caspase-2 Substrate VDVAD-pNA 1072-200 200 assays 1072-1000 1000 assays

Caspase-3 Substrates

Product Name Catalog # Size Caspase-3 Substrate DEVD-AFC 1007-200 200 assays 1007-1000 1000 assays Caspase-3 Substrate DEVD-pNA 1008-200 200 assays 1008-1000 1000 assays

Caspase-4 Substrates

Product Name Catalog # Size Caspase-4 Substrate LEVD-AFC 1109-200 200 assays 1109-1000 1000 assays Caspase-4 Substrate LEVD-pNA 1110-200 200 assays 1110-1000 1000 assays

12 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals D/S,Probes,Substrates

Caspase-5 Substrates

Product Name Catalog # Size Caspase-5 Substrate WEHD-AFC 1101-200 200 assays 1101-1000 1000 assays Caspase-5 Substrate WEHD-pNA 1102-200 200 assays 1102-1000 1000 assays

Caspase-6 Substrates

Product Name Catalog # Size Caspase-6 Substrate VEID-AFC 1069-200 200 assays 1069-1000 1000 assays Caspase-6 Substrate VEID-pNA 1070-200 200 assays 1070-1000 1000 assays

Caspase-8 Substrates

Product Name Catalog # Size Caspase-8 Substrate IETD-AFC 1062-200 200 assays 1062-1000 1000 assays Caspase-8 Substrate IETD-pNA 1063-200 200 assays 1063-1000 1000 assays

Caspase-9 Substrates

Product Name Catalog # Size Caspase-9 Substrate LEHD-AFC 1075-200 200 assays 1075-1000 1000 assays Caspase-9 Substrate LEHD-pNA 1076-200 200 assays 1076-1000 1000 assays

Caspase-10 Substrates

Product Name Catalog # Size Caspase-10 Substrate AEVD-AFC 1113-200 200 assays 1113-1000 1000 assays Caspase-10 Substrate AEVD-pNA 1114-200 200 assays 1114-1000 1000 assays

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 13 D/S,Probes,Substrates Biochemicals

Caspase-12 Substrate

Product Name Catalog # Size Caspase-12 Substrate ATAD-AFC 1117-200 200 assays 1117-1000 1000 assays

Caspase-13 Substrate

Product Name Catalog # Size Caspase-13 Substrate LEED-AFC 1116-200 200 assays 1116-1000 1000 assays

Pan Caspase Substrates

Product Name Catalog # Size Caspase Colorimetric Substrate Set K132-7-25 7 x 25 assays Caspase Colorimetric Substrate Set II K134-9-25 9 x 25 assays Caspase Colorimetric Substrate Set II Plus K138-9-25 9 x 25 assays Caspase Colorimetric Substrate Set Plus K136-7-25 7 x 25 assays Caspase Fluorometric Substrate Set K131-7-25 7 x 25 assays Caspase Fluorometric Substrate Set II K133-9-25 9 x 25 assays Caspase Fluorometric Substrate Set II Plus K137-9-25 9 x 25 assays Caspase Fluorometric Substrate Set Plus K135-7-25 7 x 25 assays

HRP Substrates

Product Name Catalog # Size ABTS™ 1212-100 100 ml TMB, High Kinetics 1216-100 100 ml

Luciferase Substrate

Product Name Catalog # Size StayBrite™ D-Luciferin, Sodium Salt 7902-100 100 mg 7902-1G 1 g 7902-10G 10 g

14 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Enzyme Inhibitors

Ubiquitin Proteasome Pathway Substrates

Product Name Catalog # Size NEDD8-AMC 4843-25 25 μg Proteasome Substrate, Fluorogenic 1832-1 1 mg 1832-5 5 mg Suc-Leu-Leu-Val-Tyr-AMC 1833-5 5 mg Ubiquitin-AMC 4842-25 25 μg

Other Related Products

Product Name Catalog # Size 7-Amino-4-methylcoumarin 1844-25 25 mg 1844-100 100 mg AFC (7-amino-4-trifluoromethyl-coumarin) 1077-100 100 mg pNA (p-nitroaniline) 1078-100 100 mg

Enzyme Inhibitors ► ACC2 Inhibitors

Product Name Catalog # Size ACC2 Inhibitor 1717-1 1 mg

► ATPase Inhibitors

Product Name Catalog # Size Bafilomycin A1 1829-50 50 µg 1829-250 250 µg

► Calpain Inhibitors

Product Name Catalog # Size Calpain Inhibitor I, ALLN 1834-5 5 mg 1834-25 25 mg Calpain Inhibitor II, ALLM 1835-5 5 mg 1838-25 25 mg Calpain Inhibitor Z-LLY-FMK 1125-20C 20 µl (10 mM) PD 150,606 1906-5 5 mg 1906-25 25 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 15 Enzyme Inhibitors Biochemicals

► Caspase & Granzyme B Inhibitors

Product Name Catalog # Size Biotin-DEVD-FMK 1124-20C 20 µl (10 mM) Biotin-IETD-FMK 1121-20C 20 µl (10 mM) Biotin-VAD-FMK 1123-20C 20 µl (10 mM) Boc-D-FMK 1160-1 1 mg 1160-5 5 mg Caspase Inhibitor Boc-D-FMK 1120-20C 20 µl (10 mM) Caspase-1 Inhibitor Z-YVAD-FMK 1012-100 100 µl (2 mM) 1012-20C 20 µl (10 mM) Caspase-2 Inhibitor Z-VDVAD-FMK 1073-100 100 µl (2 mM) 1073-20C 20 µl (10 mM) Caspase-3 Inhibitor Z-DEVD-FMK 1009-100 100 µl (2 mM) 1009-20C 20 µl (10 mM) Caspase-4 Inhibitor Z-LEVD-FMK 1108-100 100 µl (2 mM) 1108-20C 20 µl (10 mM) Caspase-5 Inhibitor Z-WEHD-FMK 1100-100 100 µl (2 mM) 1100-20C 20 µl (10 mM) Caspase-6 Inhibitor Z-VEID-FMK 1011-100 100 µl (2 mM) 1011-20C 20 µl (10 mM) Caspase-8 Inhibitor Z-IETD-FMK 1064-100 100 µl (2 mM) 1064-20C 20 µl (10 mM) Caspase-9 Inhibitor Z-LEHD-FMK 1074-100 100 µl (2 mM) 1074-20C 20 µl (10 mM) Caspase-10 Inhibitor AEVD-FMK 1112-100 100 µl (2 mM) 1112-20C 20 µl (10 mM) Caspase-12 Inhibitor Z-ATAD-FMK 1079-100 100 µl (2 mM) 1079-20C 20 µl (10 mM) Caspase-13 Inhibitor LEED-FMK 1115-100 100 µl (2 mM) 1115-20C 20 µl (10 mM) Caspase-Family Inhibitor Set K107-5-25 5 x 25 µl Caspase-Family Inhibitor Set II K108-7-25 7 x 25 µl Caspase-Family Inhibitor Set III K210-8-25 8 x 25 µl Caspase-Family Inhibitor Set IV K220-12-25 12 x 25 µl Caspase-Family Inhibitor Z-VAD-FMK 1010-100 100 µl 1010-20C 20 µl EMAP-II Inhibitor Z-ASTD-FMK 1127-20C 20 µl (10 mM) FMK Negative Control 1122-100 100 µl (2 mM) 1122-20C 20 µl (10 mM) Granzyme B Inhibitor Ac-IEPD-CHO 1119-1 1 mg

Granzyme B Inhibitor Z-AAD-CH2Cl 1128-20C 20 µl (10 mM) Q-VD-OPh 1170-1 1 mg

16 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Enzyme Inhibitors

► Caspase & Granzyme B Inhibitors Continued... Product Name Catalog # Size Q-VD-OPh 1170-3 3 mg 1170-5 5 mg EZSolution™ Q-VD-OPh 1173-1 1 mg Q-VD-OPh Negative Control 1171-1 1 mg 1171-3 3 mg 1171-5 5 mg EZSolution™ Q-VD-OPh, Negative Control 1174-1 1 mg Z-ATAD-FMK 1152-1 1 mg 1152-5 5 mg Z-DEVD-FMK 1143-1 1 mg 1143-5 5 mg Z-IETD-FMK 1148-1 1 mg 1148-5 5 mg Z-LEHD-FMK 1149-1 1 mg 1149-5 5 mg Z-LEVD-FMK 1144-1 1 mg 1144-5 5 mg Z-VAD-FMK 1140-1 1 mg 1140-5 5 mg Z-VDVAD-FMK 1142-1 1 mg 1142-5 5 mg Z-VEID-FMK 1146-1 1 mg 1146-5 5 mg Z-YVAD-FMK 1141-1 1 mg 1141-5 5 mg

► Cathepsin Inhibitor

Product Name Catalog # Size Cathepsin B&L Inhibitor Z-Phe-Phe-FMK 1126-20C 20 µl (10 mM)

► CDc42 Inhibitor

Product Name Catalog # Size MLS-573151 1929-5 5 mg 1929-25 25 mg

► Cyclooxygenase (COX) Inhibitor

Product Name Catalog # Size Celecoxib 1574-100 100 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 17 Enzyme Inhibitors Biochemicals

► Dipeptidyl peptidase-4 (DPP-4) Inhibitor

Product Name Catalog # Size DPP IV Inhibitor, K 579 1963-1 1 mg 1963-5 5 mg DPP IV Inhibitor, NVP DPP 728 1964-1 1 mg 1964-5 5 mg Sitagliptin Phosphate Monohydrate 1757-100 100 mg 1757-1G 1 g

► DUB Inhibitor

Product Name Catalog # Size USP14 Inhibitor, IU1 1845-5 5 mg 1845-25 25 mg

► FAAH Inhibitor

Product Name Catalog # Size FAAH Inhibitor, PF-622 1928-5 5 mg 1928-25 25 mg

► Fatty Acid Synthase (FAS) Inhibitors

Product Name Catalog # Size Cerulenin 1579-5 5 mg 1579-50 50 mg FAS Inhibitor, C75 1547-1 1 mg

► GST Inhibitors

Product Name Catalog # Size GST Inhibitor-1 (Cibacron Blue 3G-A, Sodium Salt) 1555R-1000 1 g GST Inhibitor-2 (Ethacrynic acid) 1556-1000 1 g

► Heat Shock Protein (Hsp) Inhibitors

Product Name Catalog # Size 17-AAG 1774-1 1 mg 1774-5 5 mg 17-DMAG 1776-1 1 mg 1776-5 5 mg Geldanamycin 1564-1 1 mg 1564-5 5 mg NVP-AUY922 1591-1 1 mg 1591-5 5 mg

18 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Enzyme Inhibitors

► Hedgehog (Hh) Signaling Pathway Antagonists

Product Name Catalog # Size Cyclopamine 1578-5 5 mg Cyclopamine-KAAD 1910-50 50 µg DiscoveryPak™ Hedgehog (Hh) Signaling Pathway K868-6 6 antagonists Inhibitors Set GANT58 1812-5 5 mg 1812-25 25 mg GANT61 1892-5 5 mg GDC-0449 1890-5 5 mg 1890-25 25 mg Hh Signaling Pathway Antagonist 1659-1 1 mg JK 184 1726-1 1 mg Robotnikinin 1923-1 1 mg Tomatidine hydrochloride 1893-25 25 mg

► Histone Acetyltransferase (HAT) Inhibitors

Product Name Catalog # Size Anacardic Acid 1849-5 5 mg 1849-25 25 mg Curcumin, Curcuma longa (High Purity) 1850-10 10 mg 1850-50 50 mg

► Histone Deacetylase (HDAC) Inhibitors

Product Name Catalog # Size Apicidin 1601-1 1 mg C646, p300/CBP Inhibitor 1948-1 1 mg 1948-5 5 mg CI-994 1742-10 10 mg 1742-50 50 mg DiscoveryPak™ HDAC Inhibitor Set K851-6 6 inhibitors M344 1607-1 1 mg MS-275 (Entinostat, SNDX-275) 1590-1 1 mg 1590-5 5 mg Panobinostat (LBH589) 1612-1 1 mg 1612-5 5 mg SAHA 1604-1 1 mg Sodium 4-phenylbutyrate 1608-100 100 mg 1608-1000 1 g Sodium butyrate 1609-1000 1 g

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► Histone Deacetylase (HDAC) Inhibitors Continued...

Product Name Catalog # Size Splitomicin 1610-5 5 mg Trichostatin A 1606-1 1 mg Tubastatin A 1724-1 1 mg 1724-5 5 mg Valproic Acid, Sodium Salt 1647-200 200 mg

► HMG-CoA Inhibitors

Product Name Catalog # Size Lovastatin 1692-50 50 mg 1692-250 250 mg Mevastatin 1694-50 50 mg 1694-250 250 mg Rosuvastatin 1955-5 5 mg 1955-25 25 mg Simvastatin 1693-50 50 mg 1693-250 250 mg

► KMO (Kynurenine 3-monoxygenase) Inhibitors

Product Name Catalog # Size JM6 1913-5 5 mg 1913-25 25 mg Ro 61-8048 1912-5 5 mg 1912-25 25 mg

JM6 Cell-permeable. A slow-release prodrug version of Ro 61-8048 (Cat. No. 1912-5, 25), an inhibitor of KMO (kynurenine 3-monoxygenase), the enzyme that controls the kynurenine pathway, long believed to be implicated in neu- rodegeneration. JM6 reverses and prevents symptoms of neurodegenerative diseases like Alzheimer’s and Huntington’s in animal models. JM6 does not penetrate into the brain, but works by inhibiting KMO in the blood. Appearance: Off-white solid

Molecular Formula: C22H26N4O6S2 Molecular Weight: 518.61 Purity: ≥98% by HPLC

► Matrix Metalloproteinase (MMP) Inhibitors

Product Name Catalog # Size Batimastat (MMP Inhibitor) 1704-1 1 mg GM 6001 1799-1 1 mg Marimastat 1790-1 1 mg 1790-5 5 mg

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► Methyltransferase Inhibitors

Product Name Catalog # Size 5-Aza-2’-deoxycytidine 1754-10 10 mg 1754-50 50 mg AMI-1 1943-5 5 mg 1943-25 25 mg BIX 01294 1678-5 5 mg 1678-25 25 mg RG 108 1679-10 10 mg 1679-30 30 mg UNC0638 1933-1 1 mg 1933-5 5 mg

► Necroptosis Inhibitors

Product Name Catalog # Size Necrostatin-1 1864-5 5 mg 1864-25 25 mg Necrostatin-5 1865-5 5 mg 1865-25 25 mg Necrostatin-7 1866-5 5 mg 1866-25 25 mg

► NF-KB Pathway Inhibitors

Product Name Catalog # Size BAY 11-7082 1867-10 10 mg 1867-50 50 mg Celastrol 1940-5 5 mg 1940-25 25 mg Honokiol 1762-10 10 mg 1762-50 50 mg IKK-ε Kinase Inhibitor I 1810-1 1 mg 1810-5 5 mg IKK-ε Kinase Inhibitor II 1811-1 1 mg 1811-5 5 mg Parthenolide 1868-10 10 mg 1868-50 50 mg PDTC 1676-100 100 mg Rocaglamide 1863-100 100 μg Triptolide 1761-1 1 mg 1761-5 5 mg

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► Nuclear Export Inhibitors

Product Name Catalog # Size Leptomycin B 1814-025 25 µg

► p53 Inhibitors

Product Name Catalog # Size Nutlin-3 1842-1 1 mg 1842-5 5 mg Pifithrin-ɑ 1554-10 10 mg

► Phosphatase Inhibitors

Product Name Catalog # Size bpV(phen) 1793-5 5 mg bpV(pic) 1794-5 5 mg Calyculin A 1562-025 25 µg Cyclosporine A 1522-100 100 mg EZBlock™ Phosphatase Inhibitor Cocktail I (50X) K273-1 1 ml K273-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail II K275-1 1 ml K275-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail III K276-1 1 ml K276-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail IV K282-1 1 ml K282-1EA 1 set (5 x 1 ml) EZBlock™ Universal Protease and Phosphatase Inhibitor K283-1 1 ml Cocktail K283-1EA 1 set (5 x 1 ml) EZBlock™ Universal Protease and Phosphatase Inhibitor K284-1 1 ml Cocktail , EDTA-Free K284-1EA 1 set (5 x 1 ml) FK-506 1563-1 1 mg 1563-10 10 mg IQ-1 1663-1 1 mg Microcystin-LR 1840-100 100 µg 1840-500 500 µg Okadaic acid 1543-025 25 µg Okadaic acid, Ammonium Salt 1766-025 25 µg Okadaic acid, Potassium Salt 1765-025 25 µg Okadaic acid, Sodium Salt 1764-025 25 µg

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► Phosphodiesterase (PDE) Inhibitors

Product Name Catalog # Size IBMX 1714-100 100 mg Zaprinast 1715-25 25 mg

► Poly (ADP-ribose) Polymerase (PARP) Inhibitors

Product Name Catalog # Size ABT-888 1620-1 1 mg 1620-5 5 mg DPQ 1899-1 1 mg 1899-5 5 mg DR2313 1771-1 1 mg 1771-5 5 mg Olaparib 1952-5 5 mg 1952-25 25 mg

► PPAR Antagonists

Product Name Catalog # Size GW 9662 1697-5 5 mg

► Protease Inhibitors

Product Name Catalog # Size AEBSF.HCl 1644-200 200 mg 1644-1000 1 g Aprotinin 4690-5 5 mg 4690-100 100 mg 4690-1000 1 g Batimastat (MMP Inhibitor) 1704-1 1 mg Bestatin 1733-25 25 mg 1733-100 100 mg Clasto-Lactacystin β-lactone 1710-100 100 µg E-64 1739-5 5 mg 1739-25 25 mg Elastase Inhibitor 1922-5 5 mg Elastase Inhibitor, SPCK 1921-5 5 mg EZBlock™ Protease Inhibitor Cocktail II K277-1EA 1 set (5 x 1 ml) EZBlock™ Protease Inhibitor Cocktail III K278-1EA 1 set (5 x 1 ml)

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► Protease Inhibitors Continued...

Product Name Catalog # Size EZBlock™ Protease Inhibitor Cocktail IV K279-1 1 ml K279-1EA 1 set (5 x 1 ml) EZBlock™ Protease Inhibitor Cocktail, EDTA-Free K272-1 1 ml K272-5 5 ml EZBlock™ Universal Protease and Phosphatase K283-1 1 ml Inhibitor Cocktail K283-1EA 1 set (5 x 1 ml) EZBlock™ Universal Protease and Phosphatase Inhibitor K284-1 1 ml Cocktail , EDTA-Free K284-1EA 1 set (5 x 1 ml) GGACK Dihydrochloride 1847-5 5 mg Lactacystin (Synthetic) 1709-200 200 µg Leupeptin, hemisulfate (Microbial) 1648-25 25 mg 1648-50 50 mg 1648-100 100 mg MG-132 1703-5 5 mg EZSolution™ MG-132 1791-5 5 mg Nafamostat Mesylate 1760-10 10 mg 1760-50 50 mg Pepstatin A 1732-25 25 mg 1732-100 100 mg PMSF 1548-5 5 g PPACK Dihydrochloride 1848-5 5 mg Protease Inhibitor Cocktail K271-500 1 kit Vicriviroc Malate 1599-1 1 mg 1599-5 5 mg

► Proteasome Inhibitors

Product Name Catalog # Size Celastrol 1940-5 5 mg 1940-25 25 mg Clasto-Lactacystin β-lactone 1710-100 100 µg (-)-Epigallocatechin gallate 1841-50 50 mg Lactacystin (Synthetic) 1709-200 200 µg MG-115 1831-1 1 mg 1831-5 5 mg MG-132 1703-5 5 mg EZSolution™ MG-132 1791-5 5 mg PS-341 1846-1 1 mg 1846-5 5 mg

24 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Enzyme Inhibitors Biochemicals Enzyme Inhibitors ► Protein Kinase Inhibitors Akt Inhibitors

Product Name Catalog # Size Akt Inhibitor 1701-1 1 mg Akt Inhibitor, Isozyme-Selective 1708-1 1 mg MK-2206 1888-500 500 µg 1888-1000 1 mg Perifosine (KRX-0401) 1592-5 5 mg 1592-25 25 mg SC66 1870-10 10 mg 1870-50 50 mg SH-5 1818-500 500 µg SH-6 1819-500 500 µg Triciribine 1701-1 1 mg

AMPK Inhibitor

Product Name Catalog # Size Dorsomorphin 1686-5 5 mg

ATM Kinase Inhibitor

Product Name Catalog # Size ATM Kinase Inhibitor 1685-5 5 mg

Aurora Kinase Inhibitors

Product Name Catalog # Size Aurora Kinase B Inhibitor (AZD1152-HQPA) 1583-5 5 mg 1583-25 25 mg Reversine 1851-1 1 mg 1851-5 5 mg Tozasertib (VX-680, MK-0457, VX6) 1595-25 25 mg 1595-100 100 mg EZSolution™ Tozasertib 1803-25 25 mg

CaM Kinase Inhibitor

Product Name Catalog # Size KN-93, Water-Soluble 1909-1 1 mg 1909-5 5 mg

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Casein kinase (CK) Inhibitor

Product Name Catalog # Size D4476 1770-1 1 mg 1770-5 5 mg

CDK Inhibitors

Product Name Catalog # Size Alsterpaullone 1897-1 1 mg 1897-5 5 mg Butyrolactone I 1690-200 200 µg Kenpaullone 1904-1 1 mg Roscovitine 1950-1 1 mg 1950-5 5 mg TG003 1905-5 5 mg 1905-25 25 mg

Chk Kinase Inhibitor

Product Name Catalog # Size Chk2 Inhibitor 1702-1 1 mg

DNA-PK Inhibitor

Product Name Catalog # Size Compound 401 1657-5 5 mg

GSK Inhibitors

Product Name Catalog # Size 1-Azakenpaullone 1944-1 1 mg 1944-5 5 mg Alsterpaullone 1897-1 1 mg 1897-5 5 mg Bisindolylmaleimide I 1945-1 1 mg 1945-5 5 mg Bisindolylmaleimide I hydrochloride 1947-1 1 mg 1947-5 5 mg BIO 1673-1 1 mg CHIR 99021 1677-5 5 mg 1677-25 25 mg EZSolution™ CHIR99021 1748-5 5 mg GSK-3 Inhibitor, AR-A014418 1953-2 2 mg 1953-5 5 mg

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GSK Inhibitors Continued...

Product Name Catalog # Size GSK-3β Inhibitor, TWS119 1655-2 2 mg Kenpaullone 1904-1 1 mg Ro 31-8220 methanesulfonate 1946-1 1 mg 1946-5 5 mg SB 216763 1769-1 1 mg 1769-5 5 mg

JAK Inhibitors

Product Name Catalog # Size CP-690550 1622-5 5 mg 1622-25 25 mg PathwayReady™ JAK/STAT Signaling Inhibitor Panel K864-8 8 inhibitors MS-1020 1911-1 1 mg Tyrphostin AG 490 1570-5 5 mg WHI-P131 1853-5 5 mg 1853-25 25 mg WP1066 1809-5 5 mg 1809-25 25 mg

JNK Inhibitors

Product Name Catalog # Size L-JNK Peptide Inhibitor I 7011-50 50 µl L-JNKI1 Negative Control Peptide 7021-50 50 µl SP600125 1669-5 5 mg

MAP Kinase/MEK Inhibitors

Product Name Catalog # Size Doramapimod 1954-5 5 mg 1954-25 25 mg GSK-1120212 1960-1 1 mg 1960-5 5 mg PathwayReady™ MAP Kinase Signaling Inhibitor Panel K862-7 7 inhibitors PD 98059 1666-2 5 mg EZSolution™ PD 98059 1783-5 5 mg PD-0325901 1643-2 2 mg 1643-5 5 mg 1643-25 25 mg

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MAP Kinase/MEK Inhibitors Continued...

Product Name Catalog # Size PD184352 1585-1 1 mg 1585-5 5 mg

EZSolution™ PD184352 1871-1 1 mg SB 203580 1712-1 1 mg 1712-5 5 mg EZSolution™ SB 203580 1786-1 1 mg Sorafenib 1594-25 25 mg 1594-100 100 mg 7,3’,4’-Trihydroxyisoflavone 1886-25 25 mg 1886-100 100 mg U0126 1668-5 5 mg VX-702 1598-1 1 mg 1598-5 5 mg

mTOR Inhibitors

Product Name Catalog # Size BEZ235 (NVP-BEZ235) 1626-5 5 mg 1626-25 25 mg BI-D1870 1924-1 1 mg 1924-5 5 mg Deforolimus 1587-5 5 mg 1587-25 25 mg Everolimus 1917-5 5 mg 1917-25 25 mg GSK-2126458 1960-1 1 mg 1960-5 5 mg mTOR Inhibitor, Ku-0063794 1779-1 1 mg 1779-5 5 mg DiscoveryPak™ PI 3-Kinase Inhibitor Set K856-5 5 inhibitors PP242 1658-1 1 mg Rapamycin 1568-5 5 mg 1568-50 50 mg EZSolution™ Rapamycin 1746-5 5 mg Temsirolimus (CCI-779, Torisel) 1600-5 5 mg 1600-25 25 mg

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PI 3-Kinase Inhibitors

Product Name Catalog # Size BEZ235 (NVP-BEZ235) 1626-5 5 mg 1626-25 25 mg GDC-0941 1623-1 1 mg 1623-5 5 mg GSK-2126458 1960-1 1 mg 1960-5 5 mg IC87114 1661-1 1 mg LY 294002 1667-5 5 mg 1667-25 25 mg EZSolution™ LY294002 1747-5 5 mg PI-103 1728-1 1 mg 1728-5 5 mg PathwayReady™ PI3-K/Akt/mTOR Signaling Inhibitor K857-11 11 inhibitors Panel DiscoveryPak™ PI 3-Kinase Inhibitor Set K856-5 5 inhibitors PI3-Kɣ Inhibitor, AS-605240 1780-1 1 mg 1780-5 5 mg PX-866 1965-1 1 mg 1965-5 5 mg TGX-115 1660-1 1 mg TGX-221 1781-1 1 mg 1781-5 5 mg Wortmannin, Penicillium funiculosum 1670-1 1 mg

PIM1 Kinase Inhibitor

Product Name Catalog # Size Quercetin, Dihydrate 1773-250 250 mg 1773-1000 1 g

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Protein Kinase A (PKA) Inhibitors

Product Name Catalog # Size Fasudil, Monohydrochloride 1787-10 10 mg 1787-50 50 mg H-89 Dihydrochloride 1768-1 1 mg 1768-5 5 mg

Protein Kinase C Inhibitors

Product Name Catalog # Size Bisindolylmaleimide I 1945-1 1 mg 1945-5 5 mg Bisindolylmaleimide I hydrochloride 1947-1 1 mg 1947-5 5 mg Enzastaurin (LY317615) 1619-1 1 mg 1619-5 5 mg Gö 6976 1711-500 500 µg EZSolution™ Gö 6976 1785-500 500 µg Ro 31-8220 methanesulfonate 1946-1 1 mg 1946-5 5 mg Staurosporine 1048-01 100 µg 1048-1 1 mg EZSolution™ Staurosporine 1745-01 100 µg Tamoxifen citrate 1551-1000 1 g

Protein Tyrosine Kinase Inhibitors

Product Name Catalog # Size A 83-01 1725-1 1 mg ABT-869 1615-1 1 mg 1615-5 5 mg AG 1478 1800-5 5 mg 1800-25 25 mg Axitinib (AG-013736) 1581-5 5 mg 1581-25 25 mg Bay 61-3606 Hydrochloride 1796-1 1 mg 1796-5 5 mg BIBW2992 (Tovok) 1616-1 1 mg 1616-5 5 mg BMS-599626 1614-1 1 mg 1614-5 5 mg

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Protein Tyrosine Kinase Inhibitors Continued...

Product Name Catalog # Size Bosutinib (SKI-606) 1584-5 5 mg 1584-25 25 mg Canertinib (CI-1033, PD-183805) 1617-5 5 mg 1617-50 50 mg Carbozantinib 1935-5 5 mg 1935-25 25 mg Cediranib (AZD2171) 1613-1 1 mg 1613-5 5 mg CP-690550 1622-5 5 mg 1622-25 25 mg Crizotinib 1934-5 5 mg 1934-25 25 mg Dasatinib (BMS-354825, Sprycel) 1586-25 25 mg 1586-100 100 mg PathwayReady™ EGFR Signaling Inhibitor Panel K863-14 14 inhibitors DiscoveryPak™ EGFR Tyrosine Kinase Inhibitor Set K858-5 5 inhibitors Emodin 1875-25 25 mg 1875-100 100 mg Erlotinib, Hydrochloride Salt 1588-100 100 mg 1588-1000 1 g Fostamatinib Disodium 1936-1 1 mg 1936-5 5 mg Gefitinib 1589-5 5 mg 1589-25 25 mg Genistein 1533-10 10 mg 1533-100 100 mg Genistin 1535-10 10 mg GW2580 1740-5 5 mg 1740-25 25 mg Imatinib Mesylate (CGP-57148B, STI-571) 1625-100 100 mg 1625-1000 1 g PathwayReady™ JAK/STAT Signaling Inhibitor Panel K864-8 8 inhibitors Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) 1624-25 25 mg 1624-100 100 mg Nilotinib 1750-25 25 mg 1750-100 100 mg NVP-TAE684 1683-5 5 mg Pazopanib 1916-5 5 mg 1916-25 25 mg PD 153035 Hydrochloride 1656-2 2 mg

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Protein Tyrosine Kinase Inhibitors Continued...

Product Name Catalog # Size PD 173074 1675-1 1 mg PP1 1927-1 1 mg 1927-5 5 mg PP2 1767-1 1 mg 1767-5 5 mg PP3 1797-10 10 mg 1797-50 50 mg DiscoveryPak™ Receptor Tyrosine Kinase (RTK) Inhibitor K859-8 8 inhibitors Set Saracatinib (AZD0530) 1582-5 5 mg 1582-25 25 mg SB-431542 1674-1 1 mg EZSolution™ SB-431542 1872-1 1 mg Sorafenib 1594-25 25 mg 1594-100 100 mg SU 11274 1938-5 5 mg 1938-25 25 mg SU 1498 1836-1 1 mg 1836-5 5 mg SU 6668 1931-5 5 mg 1931-25 25 mg SU-5402 1645-05 500 µg Sunitinib Malate (Sutent) 1611-25 25 mg 1611-100 100 mg 1611-1000 1 g EZSolution™ Sunitinib Malate 1804-25 25 mg TAK 165 1951-5 5 mg 1951-25 25 mg Tyrphostin AG 1295 1571-5 5 mg Tyrphostin AG 490 1570-5 5 mg Vandetanib 1751-25 25 mg 1751-100 100 mg WHI-P131 1853-5 5 mg 1853-25 25 mg

Raf Kinase Inhibitor

Product Name Catalog # Size ZM 336372 1789-1 1 mg 1789-5 5 mg

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Rho Kinase (ROCK) Inhibitors

Product Name Catalog # Size Fasudil, Monohydrochloride 1787-10 10 mg 1787-50 50 mg Y-27632 1596-1 1 mg 1596-5 5 mg 1596-50 50 mg EZSolution™ Y-27632 1784-5 2 mg

Y-27632 Selective inhibitor of the Rho-associated protein kinase p160ROCK. Ki val- ues are 0.14, 26, 25 and >250 µM for p160ROCK, PKC, cAMP-dependent protein kinase and myosin light-chain kinase, respectively. Prevents apoptosis as well as enhance the survival and cloning efficiency of dissociated human embryonic stem cells (hES) without affecting their pluripotency. Appearance: White solid

Molecular Formula: C14H21N3O.2HCl Molecular Weight: 320.26 Purity: ≥99% by HPLC

► PTEN Inhibitors

Product Name Catalog # Size bpV(phen) 1793-5 5 mg bpV(pic) 1794-5 5 mg VO-OHpic, Trihydrate 1801-5 5 mg 1801-25 25 mg

► Rac1 Inhibitor

Product Name Catalog # Size NSC 23766 1941-1 1 mg 1941-5 5 mg

► SCD1 Inhibitor

Product Name Catalog # Size SCD1 Inhibitor 1716-1 1 mg 1716-5 5 mg

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► Secretase Inhibitors

Product Name Catalog # Size β-Secretase Inhibitor I 7501-1 1 mg β-Secretase Inhibitor II 7502-1 1 mg Compound 34 1898-200 200 µg 1898-1000 1 mg Compound E 1949-250 250 µg 1949-1000 1 mg DAPT 1855-5 5 mg L-685, 458 1713-250 250 µg

► SIRT Inhibitors Product Name Catalog # Size Cambinol 1653-10 10 mg Salermide 1873-5 5 mg 1873-25 25 mg SIRT1 Inhibitor, EX-527 1652-10 10 mg SIRT2 Inhibitor 1857-5 5 mg 1857-25 25 mg SIRT2 Inhibitor, AGK2 1651-10 10 mg Suramin Hexasodium Salt 1874-50 50 mg 1874-250 250 mg

► Stat Inhibitors

Product Name Catalog # Size PathwayReady™ JAK/STAT Signaling Inhibitor Panel K864-8 8 inhibitors Lestaurtinib 1805-500 500 µg 1805-1000 1 mg LLL12 1792-5 5 mg 1792-25 25 mg MS-1020 1911-1 1 mg Niclosamide 1826-100 100 mg 1826-500 500 mg Pimozide 1887-50 50 mg 1887-250 250 mg Stat3 Activation Inhibitor, SPI 1813-2 2 mg Stat3 Inhibitor I, S3I-201 1775-5 5 mg 1775-25 25 mg Stat3 Peptide Inhibitor, Cell-Permeable 1778-1 1 mg 1778-5 5 mg

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► Topoisomerase Inhibitors

Product Name Catalog # Size Camptothecin 1039-50MG 50 mg 1039-500MG 500 mg Doxorubicin.HCl 1527-5 5 mg Epirubicin Hydrochloride 1753-5 5 mg 1753-25 25 mg Etoposide 1043-25MG 25 mg 1043-250MG 250 mg Irinotecan Hydrochloride 1752-50 50 mg 1752-250 250 mg Mitoxantrone 1885-50 50 mg 1885-250 250 mg

► Ubiquitin Activating Enzyme E1 Inhibitor

Product Name Catalog # Size PYR-41 1925-5 5 mg 1925-25 25 mg

► Wnt Signaling Inhibitors

Product Name Catalog # Size CRT Inhibitor, iCRT5 1896-5 5 mg 1896-25 25 mg IQ-1 1663-1 1 mg IWP-2 1962-5 5 mg 1962-25 25 mg QS11 1680-5 5 mg XAV939 1727-1 1 mg

CRT Inhibitor, iCRT5 Cell-permeable. A potent inhibitor of the β-catenin-responsive transcrip- tion (CRT) in the nucleus. iCRT5 inhibits Wnt responsive STF16 luciferase

(STF16-Luc) with an IC50 of 18 nM. It acts by disrupting the interaction be- tween β-catenin and TCF4, possibly by direct binding to β-catenin. However, it displays minimal or less prominent effect on non-canonical Wnt signaling and other pathways such as Hh, JAK/STAT, and Notch signaling. Appearance: Yellow solid

Molecular Formula: C16H17NO5S2 Molecular Weight: 367.44 Purity: ≥98% by HPLC

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► Other Inhibitors Product Name Catalog # Size Betulin 1942-5 5 mg 1942-25 25 mg Catharanthine 1749-100 100 mg 1749-1000 1 g DBeQ 1858-5 5 mg 1585-25 25 mg Dynasore 1900-5 5 mg 1900-25 25 mg FK-866 1914-1 1 mg 1914-5 5 mg Ganciclovir 1918-50 50 mg 1918-250 250 mg 1918-1000 1 g GYY 4137 1908-5 5 mg 1908-25 25 mg MIF-Antagonist, ISO-1 1895-5 5 mg Mifepristone 1561-50 50 mg Pimecrolimus 1593-5 5 mg 1593-25 25 mg Tenofovir disoproxil fumarate 1920-5 5 mg 1920-25 5 mg Tetrahydrouridine 1671-10 10 mg 1671-25 25 mg Thapsigargin 1558-1 1 mg Tranilast 1876-10 10 mg 1876-50 50 mg

Immunosuppressants Product Name Catalog # Size Ascomycin 1573-2 2 mg Cyclosporine A 1522-100 100 mg 1522-1G 1 g Fingolimod (FTY-720A, FTY720) 1618-5 5 mg 1618-25 25 mg FK-506 1563-1 1 mg 1563-10 10 mg (R,S)-Lenalidomide 1862-25 25 mg 1862-100 100 mg

36 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com EnzymeIonophores Inhibitors Biochemicals Molecular Biology Tools Immunosuppressants Continued.. Product Name Catalog # Size Mycophenolic Acid 1882-50 50 mg 1882-250 250 mg Rapamycin 1568-5 5 mg 1568-50 50 mg Rocaglamide 1863-100 100 μg

Ionophores Product Name Catalog # Size A23187 1501-10 10 mg Ionomycin (Calcium salt) 1566-5 5 mg Ionomycin (free acid) 1565-5 5 mg Monensin Methyl Ester 1808-50 50 mg 1808-250 250 mg

Molecular Biology Tools Product Name Catalog # Size Blasticidin S Hydrochloride 1859-25 25 mg 1859-100 100 mg Cycloheximide 1041-1G 1 g Cycloheximide (100 mM) 1041-1 1 ml DTT 1201-1 1 ml (1 M) G418 Sulfate (siRNA Vector Approved) 1557-1000 1 g IPTG, Animal-Free (Dioxane-Free) 1649-1G 1 g 1649-5G 5 g 1649-50G 50 g Puromycin Dihydrochloride 1860-25 25 mg 1860-100 100 mg 1860-250 250 mg 1860-500 500 mg 1860-1000 1 g EZSolution™ Puromycin Dihydrochloride 1861-100 100 mg Streptozocin 1930-100 100 mg 1930-500 500 mg 1930-1000 1 g TCEP.HCl 1202-1ML 1 ml (1 M) 1202-10G 10 g

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 37 Protein Purification Reagents Biochemicals Other Biochemicals Other Biochemicals Product Name Catalog # Size AEC 2122-10 10 ml GSNO 1580-25 25 mg 1580-100 100 mg Obestatin (Human) 1705-500 500 µg

Protein Purification Reagents Product Name Catalog # Size AEBSF.HCl 1644-200 200 mg 1644-1000 1 g Aprotinin 4690-5 5 mg 4690-100 100 mg 4690-1000 1 g ASB-14 1738-5G 5 g 1738-25G 25 g Bestatin 1733-25 25 mg 1733-100 100 mg Calyculin A 1562-025 25 µg CHAPS, High Purity 1545-10G 10 g 1545-50G 50 g 1545-100G 100 g 1545-500G 500 g 1545-1Kg 1 Kg DTT 1201-1 1 ml (1 M) E-64 1739-5 5 mg 1739-25 25 mg Leupeptin, hemisulfate (Microbial) 1648-25 25 mg 1648-50 50 mg 1648-100 100 mg

NP-40 (10% in H2O) 2111-100 100 ml NP-40 Substitute, MegaPure™ Detergent, 10% 2127-50 50 ml Solution 2127-100 100 ml 2127-500 500 ml n-Octyl-β-D-glucopyranoside 1646-5G 5 g 1646-25G 25 g 1646-50G 50 g Octyl-β-D-thioglucopyranoside 1782-1G 1 g 1782-5G 5 g 1782-50G 50 g 1782-100G 100 g

38 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Enzyme Inhibitors Biochemicals Protein Purification Reagents Protein Purification Reagents Continued... Product Name Catalog # Size Pepstatin A 1732-25 25 mg 1732-100 100 mg EZBlock™ Phosphatase Inhibitor Cocktail I (50X) K273-1 1 ml K273-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail II K275-1 1 ml K275-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail III K276-1 1 ml K276-1EA 1 set (5 x 1 ml) EZBlock™ Phosphatase Inhibitor Cocktail IV K282-1 1 ml K282-1EA 1 set (5 x 1 ml) PMSF 1548-5 5 g Protease Inhibitor Cocktail K271-500 1 kit EZBlock™ Protease Inhibitor Cocktail II K277-1EA 1 set (5 x 1 ml) EZBlock™ Protease Inhibitor Cocktail III K278-1EA 1 set (5 x 1 ml) EZBlock™ Protease Inhibitor Cocktail IV K279-1 1 ml K279-1EA 1 set (5 x 1 ml) EZBlock™ Protease Inhibitor Cocktail, EDTA-Free K272-1EA 1 set K272-1 1 ml K272-5 5 ml EZBlock™ Universal Protease and Phosphatase K283-1 1 ml Inhibitor Cocktail K283-1EA 1 set (5 x 1 ml) EZBlock™ Universal Protease and Phosphatase Inhibitor K284-1 1 ml Cocktail , EDTA-Free K284-1EA 1 set (5 x 1 ml)

SDS Solution (10% in H2O) 2102-100 100 ml Sulfobetaine 3-16 1777-5G 5 g 1777-25G 25 g TCEP.HCl 1202-1ML 1 ml (1 M) 1202-10G 10 g

Triton® X-100 Solution (10% in H2O) 2104-100 100 ml Triton® X-100, MegaPure™ Detergent, 10% 2124-50 50 ml Solution 2124-100 100 ml 2124-500 500 ml

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 39 Stem Cell Research Tools Biochemicals Stem Cell Research Tools ► Stem Cell Fate Regulators Differentiation

Product Name Catalog # Size Cardiogenol C hydrochloride 1926-5 5 mg 1926-25 25 mg Compound 1 1688-5 5 mg Cyclopamine 1578-5 5 mg Cyclosporine A 1522-100 100 mg 1522-1G 1 g Cyclopamine-KAAD 1910-50 50 µg DAPT 1855-5 5 mg Dexamethasone 1042-1G 1 g 1042-10G 10 g Forskolin 1531-5 5 mg GANT58 1812-5 5 mg 1812-25 25 mg GANT61 1892-5 5 mg GDC-0449 1890-5 5 mg 1890-25 25 mg Geldanamycin 1564-1 1 mg 1564-5 5 mg Hh Signaling Pathway Antagonist 1659-1 1 mg IWP-2 1962-5 5 mg 1962-25 25 mg JK 184 1726-1 1 mg Kenpaullone 1904-1 1 mg MoTP 1852-5 5 mg 1852-25 25 mg Neuropathiazol 1903-5 5 mg 1903-25 25 mg Purmorphamine 1672-5 5 mg Rapamycin 1568-5 5 mg 1568-50 50 mg EZSolution™ Rapamycin 1746-5 5 mg Reversine 1851-1 1 mg 1851-5 5 mg Robotnikinin 1923-1 1 mg SB-431542 1674-1 1 mg EZSolution™ SB-431542 1872-1 1 mg

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Differentiation Continued...

Product Name Catalog # Size Shz-1 1915-1 1 mg 1915-5 5 mg Smo Agonist, SAG 1939-500 500 µg 1939-1000 1 g Sodium butyrate 1609-1000 1 g Stauprimide 1743-500 500 µg Tomatidine hydrochloride 1893-25 25 mg Trichostatin A 1606-1 1 mg U0126 1668-5 5 mg WHI-P131 1853-5 5 mg 1853-25 25 mg

Induced Pluripotent Stem (iPS) cells and Reprogramming

Product Name Catalog # Size 5-Azacytidine 1854-50 50 mg 1854-250 250 mg 8-Br-cAMP 1837-5 5 mg 1837-25 25 mg (+-)-Bay K 8644 1682-5 5 mg BIX 01294 1678-5 5 mg 1678-25 25 mg PS48 1869-5 5 mg 1869-25 25 mg 1869-100 100 mg StemBoost™ Reprogramming Cocktail Set I (1000X), K869-1ML 1 ml Sterile-Filtered K869-5ML 5 ml K869-1set 5 x 1 ml StemBoost™ Reprogramming Cocktail Set II (1000X), K870-1ML 1 ml Sterile-Filtered K870-5ML 5 ml K870-1set 5 x 1 ml RepSox 1894-5 5 mg 1894-25 25 mg RG 108 1679-10 10 mg 1679-30 30 mg Sodium butyrate 1609-1000 1 g Thiazovivin 1681-1 1 mg 1681-5 5 mg EZSolution™ Thiazovivin 1736-1 1 mg

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 41 Stem Cell Research Tools Biochemicals Induced Pluripotent Stem (iPS) cells and Reprogramming Continued...

Product Name Catalog # Size Tranylcypromine Hemisulfate 1816-25 25 mg 1816-100 100 mg UNC0638 1933-1 1 mg 1933-5 5 mg Valproic Acid, Sodium Salt 1647-200 200 mg StemBoost™ YPAC Cocktail Set (1000X), Sterile-Filtered K871-1ML 1 ml K871-5ML 5 ml K871-1set 5 x 1 ml

Self-Renewal and Survival

Product Name Catalog # Size A 83-01 1725-1 1 mg BIO 1673-1 1 mg CHIR 99021 1677-5 5 mg 1677-25 25 mg EZSolution™ CHIR99021 1748-5 5 mg GSK-3β Inhibitor, TWS119 1655-2 2 mg Heparin-Binding Peptide I 1821-5 5 mg 1821-25 25 mg Heparin-Binding Peptide II 1822-5 5 mg 1822-25 25 mg Heparin-Binding Peptide III 1823-5 5 mg 1823-25 25 mg Integrin Ligand peptide 1824-5 5 mg 1824-25 25 mg IQ-1 1663-1 1 mg PD 173074 1675-1 1 mg PD 98059 1666-5 5 mg EZSolution™ PD 98059 1783-5 5 mg PD-0325901 1643-2 2 mg 1643-5 5 mg 1643-25 25 mg PD184352 1585-1 1 mg 1585-5 5 mg 1585-25 25 mg EZSolution™ PD184352 1871-1 1 mg Pifithrin-ɑ 1554-10 10 mg Pyrintegrin 1729-1 1 mg 1729-5 5 mg

42 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Biochemicals Stem Cell Research Tools Self-Renewal and Survival Continued...

Product Name Catalog # Size EZSolution™ Pyrintegrin 1737-1 1 mg QS11 1680-5 5 mg SU-5402 1645-05 500 µg Thiazovivin 1681-1 1 mg 1681-5 5 mg EZSolution™ Thiazovivin 1736-1 1 mg XAV939 1727-1 1 mg Y-27632 1596-1 1 mg 1596-5 5 mg 1596-50 50 mg EZSolution™ Y-27632 1784-5 5 mg

Stem Cell Fate Regulator Sets

Product Name Catalog # Size DiscoveryPak™ Stem Cell Fate Regulator Set I K852-3 3 inhibitors DiscoveryPak™ Stem Cell Fate Regulator Set II K853-8 8 Modulators DiscoveryPak™ Stem Cell Fate Regulator Set III K854-3 3 Modulators DiscoveryPak™ Stem Cell Fate Regulator Set IV K855-3 3 Modulators DiscoveryPak™ Stem Cell Fate Regulator Set V K865-5 5 Modulators DiscoveryPak™ Stem Cell Fate Regulator Set VI K866-5 5 Modulators DiscoveryPak™ Stem Cell Fate Regulator Set VII K867-10 10 Modulators

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 43 Product Index

||| A ||| Biotin-IETD-FMK...... 16 Caspase-2 Inhibitor Z-VDVAD- CHAPS, High Purity...... 10, 38 FMK...... 16 A 83-01 ...... 30, 42 Biotin-VAD-FMK...... 16 CHIR 99021...... 26, 42 Caspase-2 Substrate VDVAD- EZSolution™ CHIR99021.....26, 42 A23187 ...... 6, 37 Bisindolylmaleimide I...... 26, 30 AFC...... 12 Chk2 Inhibitor...... 26 A-769662...... 5 Bisindolylmaleimide I Caspase-2 Substrate VDVAD- hydrochloride...... 26, 30 17-AAG...... 18 pNA...... 12 CI-994...... 19 BIX 01294...... 21, 41 ABT-869...... 30 Caspase-3 Inhibitor Z-DEVD- Ciglitazone...... 4 Blasticidin S Hydrochloride.....6, 37 FMK...... 16 ABT-888...... 23 Cisplatin...... 7 BMS-599626 ...... 30 Caspase-3 Substrate DEVD- ABTS...... 14 AFC...... 12 Clasto-Lactacystin β-lactone...... 23 Boc-D-FMK...... 16 ACC2 Inhibitor...... 15 Caspase-3 Substrate DEVD- Colchicine...... 9 Bosutinib (SKI-606)...... 31 pNA...... 12 Actinomycin D ...... 9 Compound 1...... 40 8-Br-cAMP...... 41, 5 Caspase-4 Inhibitor Z-LEVD- Actinomycin D (10 mM)...... 9 Compound E...... 34 8-Br-cGMP...... 5 FMK...... 16 AEBSF.HCl...... 23, 38 Compound 34...... 34 bpV(phen)...... 5, 22, 33 Caspase-4 Substrate LEVD- AEC...... 38 AFC...... 12 Compound 401...... 26 bpV(pic)...... 5, 22, 33 AFC...... 15 Caspase-4 Substrate LEVD- CP-31398 Dihydrochloride...... 7 Brefeldin A...... 6, 7, 9 pNA...... 12 AG 1478...... 30 CP-690550...... 27, 31 Butyrolactone I...... 26, 41 Caspase-5 Inhibitor Z-WEHD- Crizotinib...... 31 AICAR...... 5 FMK...... 16 ||| C ||| CRT Inhibitor, iCRT5...... 35 Akt Inhibitor...... 25 Caspase-5 Substrate WEHD- C646, p300/CBP Inhibitor...... 19 Akt Inhibitor, Isozyme-Selective..25 AFC...... 13 Curcumin, Curcuma longa (High Pu- Calcein AM...... 11 rity)...... 19 Alsterpaullone...... 26 Caspase-5 Substrate WEHD- Calcitriol...... 10 pNA...... 13 Cycloheximide...... 6, 9, 37 AMI-1...... 21 Calpain Inhibitor I, ALLN...... 15 Caspase-6 Inhibitor Z-VEID- Cycloheximide (100 mM)....6, 9, 37 7-Amino-4-methylcoumarin...... 15 FMK...... 16 Calpain Inhibitor II, ALLM...... 15 Cyclopamine...... 7, 19 Amiodarone Hydrochloride...... 4 Caspase-6 Substrate VEID- Calpain Inhibitor Z-LLY-FMK...... 15 Cyclopamine-KAAD...... 19 Anacardic Acid...... 19 AFC...... 13 Calyculin A...... 22 Cyclosporine A...... 6, 22, 36, 38 Anisomycin...... 5, 6, 9 Caspase-6 Substrate VEID- Cambinol...... 34 pNA...... 13 ||| D ||| 2-APB...... 10 Camptothecin...... 9, 35 Caspase-8 Inhibitor Z-IETD- D4476...... 26 Apicidin...... 19 FMK...... 16 Camptothecin (2 mM)...... 9 DAPT...... 34, 40 Aprotinin...... 23, 38 Caspase-8 Substrate IETD- Canertinib (CI-1033, PD-183805) Dasatinib (BMS-354825, Arachidonic Acid...... 5 AFC...... 13 ...... 31 Sprycel)...... 31 ASB-14...... 10, 38 Caspase-8 Substrate IETD- Capecitabine...... 7 pNA...... 13 Daunorubicin.HCl...... 6, 7, 9 Ascomycin...... 6, 36 Carboplatin...... 7 Caspase-9 Inhibitor Z-LEHD- DBeQ...... 36 ATM Kinase Inhibitor...... 25 FMK...... 16 Carbozantinib...... 31 DPP IV Inhibitor, K 579...... 18 Aurintricarboxylic acid...... 5 Caspase-9 Substrate LEHD- Cardiogenol C hydrochloride...... 40 DPP IV Inhibitor, NVP DPP 728..18 AFC...... 13 Aurora Kinase B Inhibitor Caspase Colorimetric Substrate Deferoxamine Mesylate...... 8 (AZD1152-HQPA)...... 25 Caspase-9 Substrate LEHD- Set ...... 14 pNA...... 13 Deforolimus...... 28 Axitinib (AG-013736)...... 30 Caspase Colorimetric Substrate Caspase-10 Inhibitor AEVD- Dexamethasone...... 9, 40 5-Azacytidine...... 41 Set II ...... 14 FMK...... 16 17-DMAG...... 18 5-Aza-2’-deoxycytidine ...... 21 Caspase Colorimetric Substrate Caspase-10 Substrate AEVD- Set II Plus ...... 14 Doramapimod...... 27 1-Azakenpaullone...... 26 AFC...... 13 Caspase Colorimetric Substrate Dorsomorphin...... 25 Caspase-10 Substrate AEVD- ||| B ||| Set Plus...... 14 pNA...... 13 Doxorubicin.HCl...... 6, 7, 9, 35 Bafilomycin A1...... 15 Caspase Fluorometric Substrate Caspase-12 Inhibitor Z-ATAD- DPQ...... 23 Set ...... 14 Batimastat (MMP Inhibitor)....20, 23 FMK...... 16 DR2313...... 23 Caspase Fluorometric Substrate (±)-Bay K 8644...... 41 Caspase-12 Substrate ATAD- Set II...... 14 AFC...... 14 DTT...... 37, 38 BAY 11-7082...... 21 Caspase Fluorometric Substrate Caspase-13 Inhibitor LEEF Dynasore...... 36 Bay 61-3606 Hydrochloride...... 30 Set II Plus ...... 14 MK...... 16 ||| E ||| Caspase Fluorometric Substrate Berberine Chloride...... 9 Caspase-13 Substrate LEED- Set Plus ...... 14 E-64...... 23, 38 Bestatin...... 23, 38 AFC...... 14 Caspase-Family Inhibitor EDTA Solution (pH 8.0)...... 10 Caspase-Family Inhibitor Z-VAD- Betulin...... 36 Set IV...... 16 FMK...... 16 DiscoveryPak™ EGFR Tyrosine Betulinic acid...... 5, 7, 9 Caspase Inhibitor Boc-D- Kinase Inhibitor Set...... 31 Catharanthine...... 36 FMK...... 16 Bexarotene...... 7 Elastase Inhibitor...... 23 Cathepsin B&L Inhibitor Z-Phe- Caspase-1 Inhibitor Z-YVAD- BEZ235 (NVP-BEZ235)...... 28, 29 Phe-FMK...... 17 Elastase Inhibitor, SPCK...... 23 FMK...... 16 BI-D1870...... 28 Cediranib (AZD2171)...... 31 EMAP-II Inhibitor Z-ASTD- Caspase-1 Substrate YVAD- FMK...... 16 BIBW2992 (Tovok)...... 30 AFC...... 12 Celastrol...... 8, 21 Emodin...... 31 BIO...... 26, 42 Caspase-1 Substrate YVAD- Celecoxib...... 17 pNA...... 12 Enzastaurin (LY317615)...... 30 Biotin-DEVD-FMK...... 16 Cerulenin...... 9

44 Tech help: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com Product Index

(-)-Epigallocatechin gallate.....8, 24 DiscoveryPak™ Hedgehog (Hh) Marimastat...... 20 Pam3Cys-Ser-(Lys)4, Signaling Pathway Inhibitors Trihydrochloride...... 6 Metformin, Hydrochloride...... 5 Epirubicin Hydrochloride...... 35 Set...... 19 Pamidronate disodium...... 10 Mevastatin...... 20 Erlotinib, Hydrochloride Salt...... 31 Heparin-Binding Peptide I...... 42 Panobinostat (LBH589)...... 19 MG-115...... 24 Ethidium Bromide...... 11 Heparin-Binding Peptide II...... 42 Parthenolide...... 21 MG-132...... 24 Etoposide...... 9, 35 Heparin-Binding Peptide III...... 42 PathwayReady™ EGFR Signaling EZSolution™ MG-132...... 24 Etoposide (100 mM)...... 9 Hh Signaling Pathway Inhibitor Panel...... 31 Antagonist...... 19, 40 Microcystin-LR...... 22 Everolimus...... 28 PathwayReady™ JAK/STAT Sig- ||| F ||| Honokiol...... 21 MIF-Antagonist, ISO-1...... 36 naling Inhibitor Panel...... 27, 31, 34 Mifepristone...... 36 PathwayReady™ MAP Kinase FAAH Inhibitor, PF-622...... 48 ||| I ||| Signaling Inhibitor Panel...... 27 Mitoxantrone...... 7, 35 FAS Inhibitor, C75...... 48 IBMX...... 23 PathwayReady™ PI3-K/Akt/mTOR MK-2206...... 25 Fasudil, Monohydrochloride.30, 33 IC87114...... 29 Signaling Inhibitor Panel...... 29 MLS-573151...... 17 Fingolimod (FTY-720A, FTY720)36 IKK-ε Kinase Inhibitor I...... 21 Pazopanib...... 31 Monensin Methyl Ester...... 37 FK-506...... 22, 36 IKK-ε Kinase Inhibitor II...... 21 PBS Tablets...... 10 MoTP...... 40 FK-866...... 36 Imatinib Mesylate (CGP-57148B, PBS-Tween® Tablets...... 10 STI-571)...... 31 MS-1020...... 27, 34 Fludarabine Phosphate...... 7 PD 150,606...... 15 Imidazole, MegaPure™...... 10 MS-275 (Entinostat, FMK Negative Control...... 16 PD 153035 Hydrochloride...... 31 Imiquimod...... 6 SNDX-275)...... 19 Forskolin...... 4, 40 PD 173074...... 32 Integrin Ligand peptide...... 42 mTOR Inhibitor, Ku-0063794...... 28 Fostamatinib Disodium...... 31 PD 98059...... 27 Ionomycin (Calcium salt)...... 6, 37 Mycophenolic Acid...... 37 ||| G ||| EZSolution™ PD 98059...... 27, 42 Ionomycin (free acid)...... 6, 37 ||| N ||| G418 Sulfate (siRNA Vector Appro PD-0325901...... 27 IPAM...... 8 Nafamostat Mesylate...... 24 ved)...... 6, 37 PD184352...... 28 IPTG, Animal-Free (Dioxane- Naringenin...... 7, 8 Ganciclovir...... 36 Free)...... 37 EZSolution™ PD184352...... 28, 42 Necrostatin-1...... 21 GANT58...... 19, 40 IQ-1...... 22, 35 PDTC...... 21 Necrostatin-5...... 21 GANT61...... 19, 40 Irinotecan Hydrochloride...... 35 Pepstatin A...... 24, 39 Necrostatin-7...... 21 GDC-0449...... 19, 40 IWP-2...... 35, 40 Perifosine (KRX-0401)...... 25 Nedaplatin...... 7 GDC-0941...... 29 Phenformin hydrochloride...... 5 ||| J ||| NEDD8-AMC...... 15 Gefitinib...... 31 Jasplakinolide, jaspis Phorbol-12-myristate 13-acetate Neuropathiazol...... 40 Geldanamycin...... 6, 7, 18 johnstoni...... 7, 11 (PMA)...... 5 Niclosamide...... 34 Gemcitabine Hydrochloride...... 7 JC-1...... 11 Phosphate Buffered Saline Nilotinib...... 31 (PBS)...... 10 Genistein...... 17, 31 JK 184...... 19, 40 Nimbolide...... 7 EZBlock™ Phosphatase Inhibitor Genistin...... 31 JM6...... 20 Cocktail I (50X)...... 22, 39 NP-40 (10% in H O)...... 10, 38 GGACK Dihydrochloride...... 24 ||| K ||| 2 EZBlock™ Phosphatase Inhibitor NP-40 Substitute, MegaPure™ GM 6001...... 20 Cocktail II...... 22, 39 Kenpaullone...... 26, 27, 40 Detergent, 10% Solution...... 11, 38 Gö 6976...... 30 EZBlock™ Phosphatase Inhibitor KN-93, Water-Soluble...... 25 NSC 146109 hydrochloride...... 4 Cocktail III...... 22, 39 EZSolution™ Gö 6976...... 30 ||| L ||| NSC 23766...... 33 EZBlock™ Phosphatase Inhibitor Granzyme B Inhibitor Cocktail IV...... 22, 39 Nutlin-3...... 22 Ac-IEPD-CHO...... 16 L-685, 458...... 34 PI-103...... 29 NVP-AUY922...... 18 Granzyme B Inhibitor Lactacystin (Synthetic)...... 24 PI3-Kɣ Inhibitor, AS-605240...... 29 Z-AAD-CH2Cl...... 16 Lapatinib Ditosylate (Tykerb, NVP-TAE684...... 31 GSK-3β Inhibitor, TWS119....27, 42 Tyverb, GW-572016)...... 31 DiscoveryPak™ PI 3-Kinase Inhibi- ||| O ||| tor Set...... 25, 28, 29 GSNO...... 38 (R,S)-Lenalidomide...... 7, 36 Obestatin (Human)...... 38 Pifithrin-ɑ...... 8, 22, 42 GSK-1120212...... 27 Leptomycin B...... 22 Octyl-β-D-thioglucopyranoside...38 Pimecrolimus...... 36 GSK-2126458...... 28, 29 Lestaurtinib...... 34 n-Octyl-β-D-glucopyranoside...... 38 Pimozide...... 34 GSK-3 Inhibitor, AR-A014418...... 26 Leupeptin, hemisulfate (Microbial)...... 24, 38 Okadaic acid...... 22 Piperlongumine...... 8 GST Inhibitor-1 (Cibacron Blue 3G- Okadaic acid, Ammonium Salt....22 A, Sodium Salt)...... 18 L-JNK Peptide Inhibitor I...... 27 Pioglitazone...... 4 Okadaic acid, Potassium Salt.....22 GST Inhibitor-2 (Ethacrynic L-JNKI1 Negative Control Pixantrone maleate...... 8 Peptide...... 27 acid)...... 18 Okadaic acid, Sodium Salt...... 22 PMSF...... 24, 39 LLL12...... 34 GW2580...... 31 Olaparib...... 23 pNA (p-nitroaniline)...... 15 Lovastatin...... 20 GW 9662...... 23 Oleanolic Acid...... 5 PP1...... 32 StayBrite™ D-Luciferin, GYY 4137...... 36 Oridonin...... 8 PP2...... 32 Sodium Salt...... 14 Oxaliplatin...... 8 PP242...... 28 ||| H ||| LY 294002...... 29 H-89 Dihydrochloride...... 30 OxiRed™ Probe...... 11 PP3...... 32 EZSolution™ LY294002...... 29 DiscoveryPak™ HDAC Inhibitor ||| P ||| PPACK Dihydrochloride...... 24 Set...... 19 ||| M ||| PAC-1...... 4 Propidium Iodide...... 11 M344...... 19 Paclitaxel...... 8 Protease Inhibitor Cocktail...... 24

Ordering: [email protected] | Tel: 800.891.9699 | Web: www.biovision.com 45 Product Index EZBlock™ Protease Inhibitor Rottlerin...... 4 SU 6668...... 32 ||| V ||| Cocktail II...... 23, 39 ||| S ||| Suc-Leu-Leu-Val-Tyr-AMC....12, 15 Valproic Acid, Sodium Salt....20, 42 EZBlock™ Protease Inhibitor Cocktail III...... 23, 39 SAHA...... 19 Sulfobetaine 3-16...... 11, 39 Vandetanib...... 32 EZBlock™ Protease Inhibitor Salermide...... 34 Sunitinib Malate (Sutent)...... 32 Vicriviroc Malate...... 24 Cocktail IV...... 34, 39 Saracatinib (AZD0530)...... 32 EZSolution™ Sunitinib Malate....32 Vinblastine Sulfate...... 8 EZBlock™ Protease Inhibitor SB 203580...... 28 Suramin Hexasodium Salt...... 34 Vinorelbine Tartrate...... 8 Cocktail, EDTA-Free...... 23 EZSolution™ SB 203580...... 28 ||| T ||| VO-OHpic, Trihydrate...... 33 EZBlock™ Universal Protease and Phosphatase Inhibitor Cocktail...22 SB 216763...... 27 TAK 165...... 32 VX-702...... 28 EZBlock™ Universal Protease and SB-431542...... 32, 40 Tamoxifen citrate...... 8, 9 ||| W ||| Phosphatase Inhibitor Cocktail , EZSolution™ SB-431542.....32, 40 TCEP.HCl...... 37 EDTA-Free...... 22, 24 WHI-P131...... 27, 32, 41 SC66...... 25 Teicoplanin...... 6 Proteasome Substrate, Wortmannin, Penicillium Fluorogenic...... 15 SCD1 Inhibitor...... 33 Temsirolimus (CCI-779, Torisel)..28 funiculosum...... 29 PS-341...... 24 3X SDS-PAGE loading buffer...... 10 Tenofovir disoproxil fumarate...... 36 WP1066...... 27

PS48...... 5, 41 SDS Solution (10% in H2O)...11, 37 Tetrahydrouridine...... 36 ||| X ||| Purmorphamine...... 4, 40 β-Secretase Inhibitor I...... 34 TG003...... 26 XAV939...... 35, 43 Puromycin Dihydrochloride.....6, 37 β-Secretase Inhibitor II...... 34 TGR5 Receptor Agonist...... 5 ||| Y ||| EZSolution™ Puromycin SH-5...... 25 TGX-115...... 29 Y-27632...... 33, 43 Dihydrochloride...... 6, 37 SH-6...... 25 TGX-221...... 29 EZSolution™ Y-27632...... 33 PX-866...... 29 Shz-1...... 41 Thapsigargin...... 7, 10, 36 StemBoost™ YPAC Cocktail Set PYR-41...... 35 Simvastatin...... 20 Thiazovivin...... 41, 43 (1000X), Sterile-Filtered...... 42 Pyrintegrin...... 42 SIRT1 Inhibitor, EX-527...... 34 EZSolution™ Thiazovivin...... 41, 43 ||| Z ||| EZSolution™ Pyrintegrin...... 43 SIRT2 Inhibitor...... 34 Tigecyclin...... 7 Z-ATAD-FMK...... 17 ||| Q ||| SIRT2 Inhibitor, AGK2...... 34 Tiliroside...... 8 Z-DEVD-FMK...... 17 QS11...... 35, 43 Sitagliptin Phosphate TMB, High Kinetics...... 14 Z-IETD-FMK...... 17 Quercetin, Dihydrate...... 8, 29 Monohydrate...... 18 Tomatidine hydrochloride...... 19, 41 Z-LEHD-FMK...... 17 Q-VD-OPh...... 16 SMER28...... 4 Tozasertib (VX-680, MK-0457, Z-LEVD-FMK...... 17 Smo Agonist, SAG...... 4, 41 VX6)...... 25 EZSolution™ Q-VD-OPh...... 17 Z-VAD-FMK...... 17 Sodium 4-phenylbutyrate...... 19 EZSolution™ Tozasertib...... 25 QVD-OPh Negative Control...... 16 Z-VDVAD-FMK...... 17 Sodium butyrate...... 19, 41 Tranilast...... 36 EZSolution™ Q-VD-OPh, Negative Z-VEID-FMK...... 17 Control...... 16 Sorafenib...... 28, 32 Tranylcypromine Hemisulfate.....42 Z-YVAD-FMK...... 17 ||| R ||| SP600125...... 27 Trichostatin A...... 7, 20 Zaprinast...... 23 Rapamycin...... 8, 28, 37, 40 Splitomicin...... 20 Triciribine...... 25 ZM 336372...... 32 EZSolution™ Rapamycin.8, 28, 40 SR1001...... 5 7,3’,4’-Trihydroxyisoflavone...... 28 DiscoveryPak™ Receptor Tyrosine Stat3 Activation Inhibitor, SPI.....34 Triptolide...... 21 Kinase (RTK) Inhibitor Set...... 32 Stat3 Inhibitor I, S3I-201...... 34 Tris-HCl (pH 6.8)...... 10 Reduced Glutathione (GSH)...... 8 Stat3 Peptide Inhibitor, Cell-Per- Tris-HCl (pH 8.8)...... 10 StemBoost™ Reprogramming meable...... 34 Cocktail Set I (1000X), Triton® X-100 Solution (10% in Staurosporine...... 6, 9, 30, 41 Sterile-Filtered...... 41 H2O)...... 11, 38 StemBoost™ Reprogramming EZSolution™ Staurosporine...6, 30 Triton® X-100, MegaPure™ Detergent, 10% Solution...... 11, 38 Cocktail Set II (1000X), DiscoveryPak™ Stem Cell Fate Sterile-Filtered...... 41 Regulator Set I...... 43 Troglitazone...... 4 RepSox...... 41 DiscoveryPak™ Stem Cell Fate Trypan Blue (0.4%)...... 11 Regulator Set II...... 43 Resiquimod...... 6 Tubastatin A...... 20 Resveratrol...... 5, 8 DiscoveryPak™ Stem Cell Fate Regulator Set III...... 43 Tween® 20 Solution Reversine...... 25, 40 (10% in H2O)...... 11, 38 DiscoveryPak™ Stem Cell Fate RG 108...... 21, 41 Regulator Set IV...... 43 Tween® 20, MegaPure™ Detergent, 10% Solution...... 11, 39 RIPA Buffer...... 10 DiscoveryPak™ Stem Cell Fate Regulator Set V...... 43 Tween® 80, MegaPure™ Ro 31-8220 methanesulfonate....30 Detergent, 10% Solution...... 11, 39 DiscoveryPak™ Stem Cell Fate Ro 61-8048...... 20 Regulator Set VI...... 43 Tyrphostin AG 1295...... 32 Robotnikinin...... 19, 40 DiscoveryPak™ Stem Cell Fate Tyrphostin AG 490 ...... 32 Rocaglamide...... 21, 37 Regulator Set VII...... 43 ||| U ||| Roscovitine...... 26 Streptozocin...... 6, 37 U0126...... 28, 41 Rosiglitazone...... 4 SU 11274...... 32 Ubiquitin-AMC...... 15 Rosmarinic Acid...... 8 SU 1498...... 32 UNC0638...... 21, 42 Rosuvastatin...... 20 SU-5402...... 32, 43 USP14 Inhibitor, IU1...... 18

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Customer Service [email protected] Technical Support [email protected] www.biovision.com To Place an Order USA [email protected] BioVision, Inc. 155 South Milpitas Blvd. OEM or Bulk Order Inquiries Milpitas, CA 95035 [email protected] Phone: 800-891-9699