PART ONE PREMIERE PARTIE PRIMERA PARTE ﺍﳉﺰﺀ ﺍﻷﻭﻝ 第一部分 ЧАСТЬ ПЕРВАЯ A Acetorphine - Acétorphine - Acetorfina Derivative of thebaine - Dérivé de la thébaïne - Derivado de la tebaína O H3C CO C27H35NO5 mol. wt. 453.6 O % b. anh. 100 N CH3 Sch. I, IV (1961) H3C O H C C CH CH 3 CH2 2 3 OH 3-O-acetyltetrahydro-7α-(1-hydroxy-1-methylbutyl)-6,14-endo-ethenooripavine Acétyl-O-3 (hydroxy-1-méthylbutyl)-7α endo-éthéno-6,14 tetrahydrooripavine 3-O-acetiltetrahidro-7α-(1-hidroxi-1-metilbutil)-6,14-endo-etenooripavina (6R,7R,14R)-3-O-acetyl-7,8-dihydro-7-(1-hydroxy-1-methylbutyl)-6-O-methyl-6,14-ethenomorphine [4α,5α-epoxy-7α-[(R)-2-hydroxypentan-2-yl]-6-methoxy-17-methyl-6,14-ethenomorphinan-3-yl]acetat [5α,7α(R)]-3-(acetyloxy)-4,5-epoxy-6-methoxy-α,17-dimethyl-α-propyl-6,14-ethenomorphinan-7-methanol 3-acetoxy-4,5-epoxy-6,14-endo-etheno-7α-(1-hydroxy-methylbutyl)-6-methoxy-N-methylmorphinan 3-acetoxy-4,5-epoxy-7α-(1-hydroxy-1-methyl-butyl)-6-methoxy-N-methyl-6,14-endo-aetheno-morphinan 3-O-acetyl-17-propylorvinol 3-O-acetyl-6,14-endoetheno-6,7,8,14-tetrahydro-7α-(2-hydroxy-pent-2-yl)-oripavine 3-O-acetyl-7α-[1(R)-hydroxy-1-methylbutyl]-6,14-endoethenotetrahydrooripavine 5-acetoxy-1,2,3,3a,8,9-hexahydro-2α-[1(R)-hydroxy-1-methylbutyl]-3-methoxy-12-methyl-3,9a-etheno-9,9b- iminoethanophenantrol[4,5-bcd]furan 5-acetyl-2α-(2-hydroxy-2-pentyl)-3,9a-etheno-9,9b-iminoethano-1,2,3,3a,8,9,9a,9b- octahydroiminoethanophenanthro[4,5-bcd]furan 6,7,8,14-tetrahydro-7α-[(1R)-hydroxy-1-methylbutyl]-6,14-endo-ethenooripavine-3-acetate Acetorphin, -um Acétoxy-5 [hydroxy-1(R) méthyl-1-butyl]-2α méthoxy-3 méthyl-12 éthéno-3,9a iminoéthano-9,9b hexahydro- 1,2,3,3a,8,9 phénantro[4,5-bcd] furanne Acétyl-O3 [hydroxy-1(R) méthyl-1 butyl]-7α méthyl-O6 endoéthéno-6,14 dihydro-7,8 morphine Etorphine 3-acetate Etorphine acetate O3-acetil-7,8-dihidro-7α-[1(R)-hidroxi-1-metilbutil]-O6-metil-6,14-endoetenomorfina O3-acetyl-7,8-dihydro-7α-[1(R)-hydroxy-1-methylbutyl]-O6-methyl-6,14-endoethenomorphine Acetorphine hydrochloride - Chlorhydrate d’acétorphine - Clorhidrato de acetorfina C27H35NO5 · HCl mol. wt. 490.1 % b. anh. 92.6 M 183 NIH 8074 UM 501 3 A Acetyl-alpha-methylfentanyl - Acétyl-alpha-méthylfentanyl - Acetil-alfa-metilfentanilo Synthetic substance - Substance synthétique - Sustancia sintética C22H28N2O O C CH mol. wt. 336.0 N N 3 CH % b. anh. 100 3 Sch. I, IV (l96l) N-[1-(α-methylphenethyl)-4-piperidyl]acetanilide N-[(α-méthylphénéthyl)-1 pipéridyl-4] acétanilide N-[1-(α-metilfenetil)-4-piperidil]acetanilida Acetil-alfa-metilfentanil Acetyl-α-methylfentanyl N-[1-(1-methyl-2-phenylethyl)-4-piperidinyl]-N-phenylacetamide N-phenyl-N-[1-(1-phenylpropan-2-yl)-4-piperidyl]acetamid Acetyldihydrocodeine - Acétyldihydrocodéine - Acetildihidrocodeína Derivative of codeine - Dérivé de la codéine - Derivado de la codeína H3C O C20H25NO4 mol. wt. 343.4 O N CH3 % b. anh. 100 H C C O Sch. II (l96l) 3 O (4,5α-epoxy-3-methoxy-17-methylmorphinan-6α-yl)acetat (5α,6α)-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol acetate (ester) 12-acetoxy-2-methoxy-N-methyl-1,11-epoxy-morphinan 3-methoxy-6-acetoxy-N-methyl-4,5-epoxymorphinan 3-metossi-4,5-epossi-6-acetossi-N-metilmorfinano 4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol acetat 4,5α-epoxy-3-methoxy-17-methylmorphinan-6α-yl acetate 6-acetoxy-3-methoxy-N-methyl-4,5-epoxymorphinan 6-acetoxy-4,5-epoxy-3-methoxy-N-methylmorphinan Acetilcodena Acetildiidrocodeina Acétyl-6 dihydro-7,8 codéine Acetyldihydrocodein, -one, -um Acetyldihydrokodein Acidrocodeine 4 A Acetyldihydrocodeine hydrochloride - Chlorhydrate d’acétyldihydrocodéine - Clorhidrato de acetildihidrocodeína C20H25NO4 · HCl mol. wt. 379.8 % b. anh. 90.4 Acetylcodon, -e Acetylmethadol - Acétylméthadol - Acetilmetadol Synthetic substance - Substance synthétique - Sustancia sintética O C23H31NO2 O C CH3 mol. wt. 353.5 CH CH2 CH * 3 C % b. anh. 100 * CH3 CH2 CH N CH3 Sch. I (l961) CH3 3-acetoxy-6-dimethylamino-4,4-diphenylheptane Acétoxy-3 diméthylamino-6 diphényl-4,4 heptane 3-acetoxi-6-dimetilamino-4,4-difenilheptano Because of the two asymmetric carbon atoms (marked with asterisks) six acetylmethadols are possible, as can be seen in the following diagram: Par suite de la présence de deux atomes de carbone asymétriques (marqués d’astérisques), six acétylméthadols sont possibles, ainsi qu’il ressort du diagramme suivant: Por la presencia de dos átomos de carbono asimétricos (marcados con asteriscos), son posibles seis acetilmetadoles, como puede verse en el diagrama siguiente: (Braenden, O.J., and Wolff, P. O. Bulletin of the World Health Organization – Bulletin del’Organisation mondiale de la santé, 1965, 10, 1003.) d-alphacetylmethadol Alphacetylmethadol dl-alphacetylmethadol l-alphacetylmethadol Acetylmethadol d-betacetylmethadol Betacetylmethadol dl-betacetylmethadol l-betacetylmethadol Alphacetylmethadol and betacetylmethadol (including their isomers) have been placed separately under international control (→ Alphacetylmethadol and → Betacetylmethadol). L’alphacétylméthadol et le bétacétylméthadol (avec leurs isomères) ont été placés séparément sous contrôle international (→ Alphacétylméthadol et → Bétacétylméthadol). Alfacetilmetadol y betacetilmetadol (incluyendo sus isómeros) han sido colocados separadamente bajo fiscalización internacional (→ Alfacetilmetadol y → Betacetilmetadol). (6-dimethylamino-4,4-diphenylheptan-3-yl)acetat 1-äthyl-4-dimethylamino-2,2-diphenylpentylacetat 1-ethyl-4-dimethylamino-2,2-diphenyl-pentylacetat 2-dimetilamino-4,4-difenil-3-acetoxiheptano 4,4-difenil-6-dimetilamino-3-acetoxiheptano 4,4-diphenyl-6-dimethylamino-3-acetoxyheptane 4-acetoxy-N,N,1-trimethyl-3,3-diphenyl-hexylamine 5 A 4-dimethylamino-1-ethyl-2,2-diphenylpentyl acetate 5-acetoxy-2-dimethylamino-4,4-diphenylheptane 5-acetoxy-N,N-dimethyl-4,4-diphenyl-2-heptylamine 6-(dimethylamino)-4,4-diphenyl-3-heptanol acetate (ester) 6-dimethylamino-4,4-diphenyl-3-acetoxyheptan, -e 6-dimethylamino-4,4-diphenyl-3-heptyl acetate 6-dimethylamino-4,4-diphenyl-heptan-3-ol-3-O-acetat 6-dimethylamino-4,4-diphenylheptyl-(3)-acetate Acemethadone Acéméthadone Acétate de méthadyl Acetato de metadilo Acetilmetadone Acetyldimepheptanol Acetylmetadol, -um Acetylmethadol, -e, -um Amidol acetate Benzeneethenol, β-[2-(dimethylamino)propyl]-α-ethyl-β-phenyl-, acetate (ester) Dimepheptanoacetat Diméthylamino-6 diphényl-4,4 acétoxy-3 heptane Diphényl-4,4 diméthylamino-6 acétoxy-3 heptane Methadyl acetate O-acetyl-2-dimethylamino-4,4-diphenyl-3-heptanol O-acetyl-6-dimethylamino-4,4-diphenyl-3-heptanol Race-Acetylmethadol β-[2-(dimethylamino)propyl]-α-ethyl-β-phenylbenzeneethanol acetate (ester) β-[2-(dimethylamino)propyl]-α-ethyl-β-phenylbenzeneethanolacetat NIH 2953 Alfentanil - Alfentanil - Alfentanilo Synthetic substance - Substance synthétique - Sustancia sintética C21H32N6O3 O mol. wt. 416.5 O N C CH CH % b. anh. 100 2 3 CH3 CH 2 N N CH22 CH N CH O CH N N 2 3 Sch. I (l96l) N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)ethyl]-4-(methoxymethyl)-4-piperidinyl]-N-phenylpropanamide N-[[(éthyl-4 oxo-5 dihydro-4,5 1H-tétrazolyl-1)-2 éthyl]-1 (méthoxyméthyl)-4 pipéridyl-4] propionanilide N-[1-[2-(4-etil-4,5-dihidro-5-oxo-1H-tetrazol-1-il)etil]-4-(metoximetil)-4-piperidinil]-N-fenilpropanamida Alfenta Alfentanilum N-[1-[2-(4-äthyl-5-oxo-2-tetrazolin-1-yl)-äthyl]-4-methoxymethyl-4-piperidyl]propionanilid N-[1-[2-(4-ethyl-5-oxo-2-tetrazolin-1-yl)-ethyl]-4-(methoxymethyl)-4-piperidyl]propionanilide N-[1-[2-(4-ethyl-5-oxo-2-tetrazolin-1-yl)-ethyl]-4-(methoxymethyl)-piperid-4-yl]propionanilide N-[1-[2-(4-ethyl-5-oxo-4,5-dihydro-1H-tetrazol-1-yl)ethyl]-4-methoxymethyl-4-piperidyl]-N-phenylpropanamid Propanamide, N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)-ethyl]-4-(methoxymethyl)-4-piperidinyl]-N- phenyl- ®Rapifen 6 A Alfentanil hydrochloride - Chlorhydrate d’alfentanil - Clorhidrato de alfentanilo C21H32N6O3 · HCl · H2O mol. wt. 471 % b. anh. 88.4 Monoclorhidrato de alfentanil Monoclorohidrato de N-[1-[2-(4-etil-4,5-dihidro-5-oxo-1H-tetrazol-1-il)etil]-4-(metoximetil)-4-piperidinil]-N- fenilpropanamida Monohydrochlorure de N-[[(ethyl-4 oxo-5 dihydro-4,5 1H-tétrazolyl-1)-2 éthyl]-1 (methoxymethyl)-4pipéridyl-4] propionanilide N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)ethyl]-4-(methoxymethyl)-4-piperidinyl]-N- phenylpropanamide monohydrochloride N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)ethyl]-4-(methoxymethyl)-4-piperidinyl]-N-phenyl, monohydrochloride, monohydrate N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-2-tetrazolin-1-yl)ethyl]-4-(methoxymethyl)-4-piperidyl]propionanilide monohydrochloride, monohydrate R 39209 ®Alfenta ®Brevafen ®Fentalim ®Rapifen ®Alfentanil ®Fanaxal ®Limifen Allobarbital - Allobarbital - Alobarbital Synthetic substance - Substance synthétique - Sustancia sintética C10H12N2O3 H mol. wt. 208.3 O N O HC CH CH % b. anh. 100 2 2 NH HC CH CH 2 2 Sch. IV (1971) O 5,5-diallylbarbituric acid Acide diallyl-5,5 barbiturique Ácido 5,5-dialilbarbitúrico 2,4,6(1H,3H,5H)-pyrimidinetrione, 5,5-di-2-propenyl- 5,5-di-2-propenil-2,4,6(1H,3H,5H)-pirimidintriona 5,5-di-2-propenyl-2,4,6(1H,3H,5H)-pyrimidinetrione 5,5-diallylbarbitursäure 5,5-diallylhexahydropyrimidine-2,4,6-trione Acidum diallylbarbituricum Allbarbital Allobarbital, -e, -um Allobarbitone Allylbarbitural Dialilbarbitona Dialilmal, -um Dialilmalonilurea Diallylbarbital Diallylbarbitone Diallylbarbituric acid Diallylmalonylurea Diallymal, -um 7 A NSC 9324 ®Allobital ®Curral ®Dwuallyl ®Sediomed S** ®Allylgesic* ®Diadol ®Eunalgit* ®Sedo ®Alnox ®Diafanal ®Malil, -um ®Sedormed ®Analgetico ®Diagen ®Malyl ®Soneryl ®Analgisul** ®Dial ®Novallyl ®Spasmo Plus* ®Asmac ®Diallynal ®Pannazin* ®Spasmo-Eunalgit* ®Barballyl ®Dialum ®Salsocain ®Supponeryl ®Barbidal ®Dorm ®Salso-Novakin ®Vitalgin* ®Cibalgin, -a, -e,* ®Dormallyl ®Sedaton Allobarbital-aminophenazone - Allobarbital-aminophénazone - Alobarbital-aminofenazona C10H12N2O3 · C11H13N3O mol. wt. 411.5 % b. anh. 50.6 Allopyrabital ®Pannazin* ®Vitalgin* Allylprodine – Allylprodine – Alilprodina Synthetic substance - Substance synthétique - Sustancia sintética O C18H25NO2 O C CH2 CH3 mol.